Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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Gramicidin S
CAS:<p>Gramicidin S (Gramicidin Soviet), a cationic cyclic peptide antibiotic, disrupts the membrane integrity of both Gram-positive and Gram-negative bacteria and</p>Fórmula:C60H92N12O10Pureza:98%Forma y color:SolidPeso molecular:1141.45Dc1a
<p>Dc1a, a toxin isolated from the desert bush spider Diguetia canities [1], potently facilitates the opening of the German cockroach Na v channel (BgNa v 1).</p>Fórmula:C276H414N76O84S8Pureza:98%Forma y color:SolidPeso molecular:6397.22BDBM50597431
CAS:<p>BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's disease and Parkinson's syndrome.</p>Fórmula:C27H43F3O2Pureza:98.64% - 99.28%Forma y color:SoildPeso molecular:456.62Furosemide
CAS:<p>Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chronic renal insufficiency.</p>Fórmula:C12H11ClN2O5SPureza:99.32% - 99.89%Forma y color:Crystals From Aqueous Ethanol Tasteless (Ntp 1992)Peso molecular:330.744GABAA receptor modulator-3
<p>GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.</p>Fórmula:C18H22O2Forma y color:SolidPeso molecular:270.37OD1
<p>Activates rat Nav1.7, human Nav1.4, rat Nav1.6 (EC50: 7, 10, 47 nM); minimal on Nav1.2, 1.3, 1.5 (EC50 >3 μM); blocks fast inactivation; triggers pain.</p>Fórmula:C308H466N90O95S8Pureza:98%Forma y color:SolidPeso molecular:7206.1NMDA agonist 2
<p>NMDA agonist 2 (compound 8d) effectively inhibits NMDA receptors, exhibiting an EC50 of 0.034 μM for GluN1/2C. It plays a significant role in neurological and psychiatric disorders.</p>Fórmula:C14H12BrFN2O3SForma y color:SolidPeso molecular:387.224Ebio2
<p>Ebio2 is an effective activator of KCNQ2.</p>Fórmula:C17H19F2N3O2Forma y color:SolidPeso molecular:335.349Huwentoxin I
CAS:<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Fórmula:C161H246N48O44S6Pureza:98%Forma y color:SolidPeso molecular:3750.36Mambalgin 1
CAS:<p>ASIC1a inhibitor; IC50: 192 nM (human), 72 nM (dimer); inactive channel binding; selective; pain response delay.</p>Fórmula:C272H429N85O84S10Pureza:98%Forma y color:SolidPeso molecular:6554.51BKCa activator-1
<p>BKCa activator-1 (Compound 51b) is an orally active activator of BKCa calcium-activated potassium channels with an EC50 of 2.82 μM. It promotes K+ efflux, leading to cell membrane hyperpolarization and inhibition of smooth muscle contraction. In a spontaneous hypertensive rat (SHR) model, it alleviates urinary incontinence and exhibits antitussive effects in a guinea pig cough model.</p>Fórmula:C22H23F7N2O3Forma y color:SolidPeso molecular:496.418GX 201
CAS:<p>GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.</p>Fórmula:C25H27ClF4N2O4SPureza:99.81%Forma y color:SolidPeso molecular:563N-Oleoyl Valine Ammonium salt
<p>N-Oleoyl Valine Ammonium salt is an N-acyl amide compound that is a TRPV3 antagonist and can be used to study inflammation.</p>Fórmula:C23H46N2O3Pureza:99.72%Forma y color:SolidPeso molecular:398.62Ethacrynic acid D5
CAS:<p>Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.</p>Fórmula:C13H12Cl2O4Pureza:98%Forma y color:SolidPeso molecular:308.17α5-GABAA receptor modulator 1
<p>α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.</p>Fórmula:C21H20FN3O4Forma y color:SolidPeso molecular:397.4GaTx2
CAS:<p>High-affinity ClC-2 blocker (KD ~50 pM), selective over other ClCs/CFTR/GABAC/CaCC/KV1.2; slows activation, no effect on open channels.</p>Fórmula:C125H199N39O47S6Pureza:98%Forma y color:SolidPeso molecular:3192.54AQP4 (201-220)
CAS:<p>AQP4 (201-220) is the encephalitogenic epitope of AQP-4. AQP4 (201-220) can induce experimental autoimmune encephalomyelitis (EAE), characterized by midline brain lesions, retinal lesions, and lesions at the gray matter/white matter boundary of the spinal cord. AQP-4 is the target antigen in neuromyelitis optica.</p>Fórmula:C97H143N27O27SForma y color:SolidPeso molecular:2151.4Cavα2δ-IN-1
CAS:<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Fórmula:C18H27N5OForma y color:SolidPeso molecular:329.448Tenapanor HCl
CAS:<p>Tenapanor (AZD-1722, RDX 5791) inhibits NHE3 for sodium control in the gut and kidneys.</p>Fórmula:C50H68Cl6N8O10S2Forma y color:SolidPeso molecular:1217.97Antidepressant agent 4
<p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>Fórmula:C19H38ClN5O2SForma y color:SolidPeso molecular:436.06Agitoxin-2
CAS:<p>Potent Shaker K+ channel blocker (Ki = 0.64 nM). Also inhibits Kv1.3, Kv1.6 and Kv1.1 K+ channels (Ki values are 4, 37 and 44 pM respectively).</p>Fórmula:C169H278N54O48S8Pureza:98%Forma y color:SolidPeso molecular:4090.87Huwentoxin-IV
CAS:<p>Selective NaV1.7 blocker; also inhibits NaV1.2, 1.3; less effect on NaV1.4, 1.5. Binds to neurotoxin site, traps voltage sensor. IC50: 26-338 nM.</p>Fórmula:C174H278N52O51S6Pureza:98%Forma y color:SolidPeso molecular:4106.79Withaphysalin D
CAS:<p>Withaphysalin D, from water lilies, blocks GluN2B NMDARs and is neuroprotective, crossing the blood-brain barrier.</p>Fórmula:C28H34O6Forma y color:SolidPeso molecular:466.57GDC-0334
CAS:<p>GDC-0334 is a TRPA1 antagonist useful in treatment TRPA1-mediated diseases, such as pain or asthma.</p>Fórmula:C24H19F8N5O3SForma y color:SolidPeso molecular:609.5Inaperisone
CAS:<p>Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.</p>Fórmula:C16H23NOPureza:99.48%Forma y color:SolidPeso molecular:245.36GsMTx4
CAS:<p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>Fórmula:C185H273N49O45S6Pureza:98%Forma y color:SolidPeso molecular:4095.84PNU-140975
CAS:<p>PNU-140975 is a bio-active chemical.</p>Fórmula:C3H9N5O2Forma y color:SolidPeso molecular:147.138Way 125971
CAS:<p>Way 125971 is a bioactive chemcial.</p>Fórmula:C22H28N4O5S2Forma y color:SolidPeso molecular:492.61PptT-IN-4
<p>PptT-IN-4 (Compound 3a) is a PptT inhibitor exhibiting an IC50 of 0.71 μM.</p>Fórmula:C17H23N3Pureza:98%Forma y color:SolidPeso molecular:269.38P-gp inhibitor 15
<p>P-gp Inhibitor 15 (compound 7a), a nonsubstrate inhibitor of P-glycoprotein (Pgp), inhibits Pgp-ATPase activity and interferes with Pgp-mediated Rhodamine123</p>Fórmula:C35H60N2O4Forma y color:SolidPeso molecular:572.86Isotachysterol 3
CAS:<p>Isotachysterol 3 boosts calcium transport in gut and bone mobilization in kidneyless rats.</p>Fórmula:C27H44OForma y color:SolidPeso molecular:384.64Roquefortine C
CAS:<p>Roquefortine C is a fungal cyclopeptide isolated from Penicillium roquefortii, activates P-gp and also inhibits P450-3A and other haemoproteins</p>Fórmula:C22H23N5O2Pureza:98%Forma y color:SolidPeso molecular:389.45(R)-Funapide
CAS:<p>(R)-Funapide ((R)-TV 45070), the less active R-enantiomer of Funapide, acts as a potent Nav1.7 sodium channel blocker, primarily utilized in pain research [1].</p>Fórmula:C22H14F3NO5Forma y color:SolidPeso molecular:429.35GluN2A Allosteric modulator 1
<p>GluN2A Allosteric modulator 1 (Compound 11) is an orally bioavailable compound that effectively crosses the blood-brain barrier and functions as a highly selective negative allosteric modulator of GluN2A. It exhibits an IC50 of 0.042 μM for GluN2A and 13 μM for GluN2B. This compound is useful for research in neurological disorders.</p>Fórmula:C20H16ClF2N5O2Forma y color:SolidPeso molecular:431.823Cevadine
<p>Cevadine is a natural product that can be used as a reference standard.</p>Fórmula:C32H49NO9Forma y color:SolidPeso molecular:591.742S-Sulfo-L-cysteine sodium salt
CAS:<p>S-Sulfo-L-cysteine sodium salt shows a weak affinity for mGluR1α and mGluR5a at high concentrations and has potential antioxidant activity.</p>Fórmula:C3H6NNaO5S2Pureza:99.88%Forma y color:SolidPeso molecular:223.2Sulcardine 2HCl
CAS:<p>Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.</p>Fórmula:C24H35Cl2N3O4SPureza:99.33% - 99.76%Forma y color:SoildPeso molecular:532.523AChE/Aβ-IN-1
<p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>Fórmula:C20H25BrN4Forma y color:SolidPeso molecular:401.34Trapencaine
CAS:<p>Trapencaine is a newly synthesized carbamate type local anesthetic that induces conformational changes in sodium channels on hypertrophic cell membranes.</p>Fórmula:C22H34N2O3Pureza:98.96%Forma y color:SolidPeso molecular:374.52XPO1-ligand-1
<p>XPO1-ligand-1 is a target protein ligand for XPO1, and it can be utilized in the synthesis of PROTAC XPO1 degrader-1.</p>Fórmula:C15H13ClF3N3O4Forma y color:SolidPeso molecular:391.73GYKI-47261 dihydrochloride
CAS:<p>GYKI-47261 dihydrochloride is an AMPA receptor antagonist and CYP2E1 inducer, demonstrating broad-spectrum anticonvulsant and neuroprotective activities.</p>Fórmula:C18H17Cl3N4Pureza:98.32% - 99.14%Forma y color:SolidPeso molecular:395.71Mambalgin-3
<p>Mambalgin-3, an acid-sensitive ion channel 1 (ASIC1) inhibitor, has potential applications in analgesia research [1].</p>Fórmula:C274H433N85O83S10Pureza:98%Forma y color:SolidPeso molecular:6566.54Jingzhaotoxin-X
<p>Jingzhaotoxin-X (JZTX-X) selectively inhibits Kv4.2 and Kv4.3 potassium channels, resulting in prolonged mechanical hyperalgesia [1].</p>Fórmula:C164H242N46O41S6Pureza:98%Forma y color:SolidPeso molecular:3706.35sFTX-3.3
CAS:<p>sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.</p>Fórmula:C12H29N7OForma y color:SolidPeso molecular:287.412Nicardipine-d3 hydrochloride
CAS:<p>Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.</p>Fórmula:C26H30ClN3O6Pureza:98%Forma y color:SolidPeso molecular:519Halofantrine hydrochloride
CAS:<p>Halofantrine hydrochloride (SKF-102886) is an orally administered antimalarial drug effective against drug-resistant P. falciparum and P. vivax. SKF-102886 has cardiac toxicity, inhibiting hERG and delayed rectifier potassium channel I Kr, leading to prolonged QTc and PR intervals.</p>Fórmula:C26H31Cl3F3NOPureza:98%Forma y color:SolidPeso molecular:536.89(S)-Nicardipine
CAS:<p>(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Fórmula:C26H29N3O6Forma y color:SolidPeso molecular:479.53Jedi2
CAS:<p>Jedi2 is a Piezo1 activator rather than a specific Piezo2 activator. Jedi2 binds to the mouse Piezo1 proteins with a K d of 2770 μM [1].</p>Fórmula:C10H8O3SPureza:97.85%Forma y color:SolidPeso molecular:208.23β-D-Glucopyranosyl abscisate
CAS:<p>β-D-Glucopyranosyl abscisate (ABA-GE) is a hydrolyzable conjugate of abscisic acid (ABA), which predominantly accumulates in the vacuole and likely in the</p>Fórmula:C21H30O9Forma y color:SolidPeso molecular:426.46NS-102
CAS:<p>NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2) and inhibits specific binding to the glur6 receptor.</p>Fórmula:C12H11N3O4Pureza:98.48% - 98.95%Forma y color:SolidPeso molecular:261.23Norverapamil-d7
CAS:<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Fórmula:C26H36N2O4Pureza:98%Forma y color:SolidPeso molecular:447.62Fluoroethylnormemantine hydrochloride
CAS:<p>Fluoroethylnormemantine HCl, an NMDA receptor antagonist, has anti-amnesic, neuroprotective effects, and is a PET tracer.</p>Fórmula:C12H21ClFNForma y color:SolidPeso molecular:233.764-(4-chlorophenyl)piperidin-4-ol
CAS:<p>Compound Fr13199 is a useful organic compound for research related to life sciences. The catalog number is Fr13199 and the CAS number is 39512-49-7.</p>Fórmula:C11H14ClNOPureza:99.63%Forma y color:White Slight Beige Solid Solid Particulate/PowderPeso molecular:211.688Phenazopyridine
CAS:<p>Phenazopyridine is an orally administered azo dye with local analgesic effects on urinary tract infections,. against SARM1 and TRPM8.</p>Fórmula:C11H11N5Pureza:99.98%Forma y color:SolidPeso molecular:213.24Perfluoroenanthic acid
CAS:<p>Perfluoroenanthic acid (Perfluoroheptanoic acid) is a perfluoroalkyl substance (PFAS) that negatively impacts spermatogenic development and testicular m6A RNA methylation in offspring exposed during gestation, thus impeding spermatogenesis and inducing reproductive toxicity. Additionally, in primary cortical neuron cultures, Perfluoroenanthic acid alters dendritic spine morphology and synaptogenesis, enhances neural activity and synaptic transmission, and increases the expression of excitatory synapse-associated proteins Synaptophysin and PSD95.</p>Fórmula:C7HF13O2Forma y color:SolidPeso molecular:364.06Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Fórmula:C24H34O2Pureza:99.51%Forma y color:SolidPeso molecular:354.53NS 383
CAS:<p>ASIC blocker with varying IC50: 0.12 μM in hASIC1a, and ineffective on hASIC2a/3; <5 μM on rASIC1a/2a/3; alleviates pain in inflamed/CCI rats.</p>Fórmula:C19H19N3O2Forma y color:SolidPeso molecular:321.37MSC-4381
CAS:<p>MSC-4381 (MCT4-IN-1) is an orally available and selectively modeled highly potent inhibitor of monocarboxylic acid transporter protein 4 (MCT4/SLC16A3) with potential anticancer and antitumor activity for the study of osteosarcoma.</p>Fórmula:C26H20ClN3O6SPureza:99.04%Forma y color:SolidPeso molecular:537.97Propanidid
CAS:<p>Propanidid (Sombrevin) is a gamma-aminobutyric acid type A receptor (GABAA) agonist and an intravenous anesthetic that lowers arterial blood pressure.</p>Fórmula:C18H27NO5Pureza:99.64%Forma y color:SolidPeso molecular:337.41BI-9627
CAS:<p>BI-9627 is an inhibitor of sodium-hydrogen exchanger isoform 1 (NHE1) (EC50: 31 nM).</p>Fórmula:C16H19F3N4O2Pureza:99.77%Forma y color:SolidPeso molecular:356.34GYKI 52466 dihydrochloride
CAS:<p>GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used to study neurological diseases.</p>Fórmula:C17H17Cl2N3O2Pureza:99.38%Forma y color:SolidPeso molecular:366.24(R)-3-Amino-4-hydroxybutanoic acid
CAS:<p>(R)-3-Amino-4-hydroxybutanoic acid,L-beta-Homoserine, is a full agonist at the human recombinant rho1 GABAC receptor, a modulator of GABAA and GABAB receptors.</p>Fórmula:C4H9NO3Pureza:99.92%Forma y color:SolidPeso molecular:119.12Cromakalim
CAS:<p>Cromakalim (BRL 34915) is an ATP-dependent K(+) channel opener, a smooth muscle relaxant with antiepileptic activity.</p>Fórmula:C16H18N2O3Pureza:99.39%Forma y color:SolidPeso molecular:286.33L-3373
CAS:<p>L-3373 is a competitive T3 (3,5,3'-triiodothyronine) antagonist with IC₅₀ values of 38 and 36 nM for alpha1-T3R and beta1-T3R, respectively.</p>Fórmula:C19H16I2O3Pureza:99.85%Forma y color:Off-White SolidPeso molecular:546.14Fanapanel hydrate
CAS:<p>Fanapanel hydrate selectively blocks AMPA/kainate over NMDA; Ki: 3.2 nM (quisqualate), 100 nM (kainate), 8.5 μM (NMDA).</p>Fórmula:C14H17F3N3O7PForma y color:SolidPeso molecular:427.27Piretanide
CAS:<p>Piretanide, an oral loop diuretic, effective and potassium-sparing, heart failure and hypertension with reduced electrolyte imbalance risk.</p>Fórmula:C17H18N2O5SForma y color:Pale Yellow PowderPeso molecular:362.4MDL 105519
CAS:<p>MDL 105519 is a selective, non-competitive antagonist of NMDA receptors. It inhibits cyclic GMP accumulation in brain slices, anxiolytic in rat models.</p>Fórmula:C18H11Cl2NO4Forma y color:SolidPeso molecular:376.19Naminidil
CAS:<p>Naminidil is an opener of cyanoguanidine KATP.</p>Fórmula:C15H19N5Pureza:98%Forma y color:SolidPeso molecular:269.34Furosemide-d5
CAS:<p>Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.</p>Fórmula:C12H11ClN2O5SForma y color:SolidPeso molecular:335.78Lesinurad sodium
CAS:<p>Lesinurad sodium (RDEA594 sodium) is a selective inhibitor of uric acid reabsorption and is used in the study of cardiovascular diseases.</p>Fórmula:C17H13BrN3NaO2SPureza:99.97%Forma y color:SolidPeso molecular:426.26Flecainide
CAS:<p>Flecainide is an orally administered antiarrhythmic agent acting as a sodium channel blocker and IKr inhibitor,PSVT.</p>Fórmula:C17H20F6N2O3Pureza:99.896%Forma y color:SolidPeso molecular:414.345-Hydroxydecanoic acid
CAS:<p>5-Hydroxydecanoic acid is a selective ATP-sensitive K+ (KATP) channel blocker (IC50 of ~30 μM). 5-Hydroxydecanoic acid is a substrate for mitochondrial outer membrane acyl-CoA synthetase and has antioxidant activity.</p>Fórmula:C10H20O3Pureza:99.24%Forma y color:SolidPeso molecular:188.26γ-DGG
CAS:<p>gamma-DGG is a competitive blocker of AMPA receptor.</p>Fórmula:C7H12N2O5Pureza:98%Forma y color:SolidPeso molecular:204.18Lansoprazole Sulfide D4
CAS:<p>Lansoprazole Sulfide D4 is a deuterium labeled Lansoprazole Sulfide. Lansoprazole Sulfide is an orally active anti-TB (Mycobacterium tuberculosis) agent with IC50 values of 0.59 μM intracellularly and 0.46 μM in broth.Lansoprazole Sulfide is an active metabolite of the proton pump inhibitor Lansoprazole.</p>Fórmula:C16H14F3N3OSPureza:98%Forma y color:SolidPeso molecular:357.39Padsevonil
CAS:<p>Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.</p>Fórmula:C14H14ClF5N4O2SPureza:99.63%Forma y color:SolidPeso molecular:432.80(S)-Lercanidipine D3 hydrochloride
CAS:<p>(S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.</p>Fórmula:C36H42ClN3O6Pureza:98%Forma y color:SolidPeso molecular:651.21Etifoxine
CAS:<p>Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.</p>Fórmula:C17H17ClN2OPureza:98%Forma y color:SolidPeso molecular:300.78Rapastinel
CAS:<p>Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.</p>Fórmula:C18H31N5O6Pureza:97.18%Forma y color:SolidPeso molecular:413.47PF-05198007
CAS:<p>PF-05198007 is a compound with a similar pharmacodynamic profile to PF-05089771. PF-05198007 is an effective and selective arylsulfonamide Nav1.7 inhibitor.</p>Fórmula:C19H12ClF4N5O3S2Pureza:98%Forma y color:SolidPeso molecular:533.91L-655708
CAS:<p>L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.</p>Fórmula:C18H19N3O4Pureza:98.41%Forma y color:PowderPeso molecular:341.36Naspm
CAS:<p>Naspm is a synthetic analogue of Joro spider toxin and is a antagonist iscalcium permeable AMPA (CP-AMPA) receptors.</p>Fórmula:C22H34N4OPureza:98%Forma y color:SolidPeso molecular:370.53KCNQ1 activator-1
CAS:<p>N-[4-(4-Methoxyphenyl)-2-thiazolyl]-2-piperidinecarboxamide is a potent KCNQ1 activator for LQTS research.</p>Fórmula:C22H23N3O4S2Pureza:99.71%Forma y color:SolidPeso molecular:457.57Ethacizine hydrochloride
CAS:<p>Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.</p>Fórmula:C22H28ClN3O3SPureza:98.08% - 98.08%Forma y color:SolidPeso molecular:449.99BTD
CAS:<p>BTD is a TRPC5 activator that activates heteromeric channel complexes composed of TRPC5 and its closest relatives TRPC1 or TRPC4.</p>Fórmula:C24H33N3O4SForma y color:SolidPeso molecular:459.6Ethyl tosylcarbamate
CAS:<p>Gliclazide blocks beta-cell ATP-sensitive K+ currents, IC50: 184 nM. Ethyl tosylcarbamate is a synthesis intermediate.</p>Fórmula:C10H13NO4SForma y color:SolidPeso molecular:243.28H-D-Allo-Ile-OH
CAS:<p>H-D-Allo-Ile-OH inhibits 3[H] gabapentin binding/voltage-dependent L-type calcium channels and can be used for studying neurological and psychiatric disorders.</p>Fórmula:C6H13NO2Pureza:99.92%Forma y color:SolidPeso molecular:131.17AM-2099
CAS:<p>AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.</p>Fórmula:C19H13F3N4O3S2Forma y color:SolidPeso molecular:466.46Vigabatrin Hydrochloride
CAS:<p>Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.</p>Fórmula:C6H11NO2·HClPureza:98%Forma y color:SolidPeso molecular:165.62CGP 36742
CAS:<p>CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).</p>Fórmula:C7H18NO2PForma y color:SolidPeso molecular:179.2MRK-016
CAS:<p>MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.</p>Fórmula:C17H20N8O2Pureza:99.76%Forma y color:SolidPeso molecular:368.39GYKI 53655 hydrochloride
CAS:<p>GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the study of neurological disorders.</p>Fórmula:C19H21ClN4O3Pureza:98.02%Forma y color:SolidPeso molecular:388.85β-Cyfluthrin
CAS:<p>β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.</p>Fórmula:C22H18Cl2FNO3Forma y color:SolidPeso molecular:434.29Lubiprostone hemiketal
CAS:<p>Lubiprostone (hemiketal) (RU-0211 (hemiketal)), a selective activator of the chloride channel 2 (CLCN2), facilitates the treatment of chronic idiopathic constipation and opioid-induced constipation. It functions by enhancing CLCN2 channel activity, which boosts chloride ion secretion in the intestines, subsequently increasing fluid secretion and improving intestinal peristalsis. Additionally, Lubiprostone (hemiketal) may be utilized in research related to chronic constipation and cancer.</p>Fórmula:C20H32F2O5Forma y color:SolidPeso molecular:390.46Neosolaniol
CAS:<p>Neosolaniol, a type A trichothecene mycotoxin produced by Fusarium species, strongly induces an anorectic (loss of appetite) response.</p>Fórmula:C19H26O8Pureza:98%Forma y color:SolidPeso molecular:382.4Crinecerfont hydrochloride
CAS:<p>SSR-125543, a potent CRF1 receptor non-peptide antagonist, effective in CAH research, taken orally.</p>Fórmula:C27H29Cl2FN2OSForma y color:SolidPeso molecular:519.5Flumazenil acid
CAS:<p>Flumazenil is an antagonist of GABAA receptor. Flumazenil acid is a metabolite of Flumazenil.</p>Fórmula:C13H10FN3O3Forma y color:SolidPeso molecular:275.24Mepivacaine
CAS:<p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>Fórmula:C15H22N2OPureza:99.35%Forma y color:SolidPeso molecular:246.35(R)-BPO-27
CAS:<p>(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.</p>Fórmula:C26H18BrN3O6Pureza:99.1%Forma y color:SolidPeso molecular:548.34(+)-SJ733
CAS:<p>(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.</p>Fórmula:C24H16F4N4O2Pureza:99.21%Forma y color:SolidPeso molecular:468.4Tetrabenazine-d6
CAS:<p>Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder.</p>Fórmula:C19H27NO3Pureza:98%Forma y color:SolidPeso molecular:323.46Valnoctamide
CAS:<p>Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.</p>Fórmula:C8H17NOPureza:98%Forma y color:SolidPeso molecular:143.23VU041
CAS:<p>VU041 inhibits mosquito Kir1 channels (IC50: An. gambiae 2.5μM, Ae. aegypti 1.7μM), less on mammalian Kir2.1 (12.7μM), and minimally on other Kir channels.</p>Fórmula:C19H20F3N3OPureza:98%Forma y color:SolidPeso molecular:363.38YM-244769 dihydrochloride
CAS:<p>YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.</p>Fórmula:C26H24Cl2FN3O3Pureza:98%Forma y color:SolidPeso molecular:516.39(R)-Tegoprazan
CAS:<p>(R)-Tegoprazan, a benzimidazole derivative, inhibits kidney H+/K+-ATPase (IC50: 98 nM). Potential in GI disease research.</p>Fórmula:C20H19F2N3O3Forma y color:SolidPeso molecular:387.38PF-04856264
CAS:<p>PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.</p>Fórmula:C20H15N5O3S2Pureza:97.43%Forma y color:SolidPeso molecular:437.5(R)-Lercanidipine-d3 hydrochloride
CAS:<p>(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.</p>Fórmula:C36H42ClN3O6Pureza:98%Forma y color:SolidPeso molecular:651.21Bamaquimast
CAS:<p>Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases.</p>Fórmula:C16H21N3O3Pureza:98.47%Forma y color:SolidPeso molecular:303.36Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Fórmula:C22H31ClN2OForma y color:SolidPeso molecular:374.95L-Palmitoylcarnitine
CAS:<p>L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.</p>Fórmula:C23H45NO4Pureza:97% - 99.81%Forma y color:SolidPeso molecular:399.61GI-530159
CAS:<p>TREK1/2 activator, selective over TRAAK/TASK3; hyperpolarizes neurons, depresses activity (EC50 = 0.76 μM).</p>Fórmula:C27H20F6N2O2Forma y color:White CrystalsPeso molecular:518.45(-)-α-Pinene
CAS:<p>(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,</p>Fórmula:C10H16Pureza:98.02% - 98.60%Forma y color:Colourless LiquidPeso molecular:136.23Clamikalant sodium
CAS:<p>Clamikalant sodium (HMR 1098) is an ATP-dependent potassium channel (KATP) cardiac-selective blocker, used in the study of arrhythmias.</p>Fórmula:C19H21ClN3NaO5S2Pureza:99.95%Forma y color:SolidPeso molecular:493.96MRS1845
CAS:<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Fórmula:C21H22N2O6Pureza:99.69%Forma y color:SolidPeso molecular:398.41Benzocaine hydrochloride
CAS:<p>Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and</p>Fórmula:C9H11NO2·HClPureza:98%Forma y color:SolidPeso molecular:201.65Triamterene D5
CAS:<p>Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.</p>Fórmula:C12H11N7Pureza:98%Forma y color:SolidPeso molecular:258.29QO-58
CAS:<p>QO-58 is a novel Kv7 activator (opener) that activates neuronal Kv7/KCNQ/M channels, danti-nociceptive effects on inflammatory pain</p>Fórmula:C18H8Cl2F4N4OPureza:99.17%Forma y color:SolidPeso molecular:443.18L-364,373
CAS:<p>KV7.1 (KCNQ1) channel activator</p>Fórmula:C25H20FN3OForma y color:SolidPeso molecular:397.44SDZ 220-581 hydrochloride
CAS:<p>SDZ 220-581 hydrochloride is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H18Cl2NO5PPureza:98%Forma y color:SolidPeso molecular:406.2Tetramethrin
CAS:<p>Tetramethrin is a type I pyrethroid insecticide that affects the inactivation process of sodium channels in insect neurons, prolonged sodium currents.</p>Fórmula:C19H25NO4Pureza:98.85%Forma y color:White Crystals Or PowderPeso molecular:331.41Poneratoxin acetate
<p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>Fórmula:C129H215N33O31S·xC2H4O2Forma y color:SolidPeso molecular:2756.35 (free base)BI-9627 hydrochloride
CAS:<p>BIX HCl is a sodium-hydrogen exchange type 1 inhibitor.</p>Fórmula:C16H20ClF3N4O2Forma y color:SolidPeso molecular:392.8HSK16149
CAS:<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Fórmula:C12H19NO2Forma y color:SolidPeso molecular:209.28SDZ 220-581 Ammonium salt
CAS:<p>SDZ 220-581 Ammonium salt is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H20ClN2O5PPureza:98%Forma y color:SolidPeso molecular:386.77Dibucaine hydrochloride
CAS:<p>Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.</p>Fórmula:C20H30ClN3O2Pureza:99.66%Forma y color:White PowderPeso molecular:379.92Lansoprazole-d4
CAS:<p>Lansoprazole D4 (AG-1749 D4) is a deuterium labeled Lansoprazole. Lansoprazole is an inhibitor of proton pump which prevents the stomach from producing acid.</p>Fórmula:C16H14F3N3O2SPureza:98%Forma y color:SolidPeso molecular:373.39(R)-Nicardipine
CAS:<p>(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Fórmula:C26H29N3O6Forma y color:SolidPeso molecular:479.53Luciferase, firefly
CAS:<p>Luciferase, firefly is a reporter gene in cellular imaging studies to quantify target gene expression levels and measure intracellular ATP content,</p>Pureza:98%Forma y color:SolidPeso molecular:N/ACabotegravir sodium
CAS:<p>Cabotegravir sodium inhibits HIV integrase (IC50: 2.5 nM), metabolized by UGT1A1, with minimal ARV interaction.</p>Fórmula:C19H16F2N3NaO5Forma y color:SolidPeso molecular:427.34SDZ 220-581
CAS:<p>SDZ 220-581 is a potent, orally active and competitive antagonist of NMDA receptor(pKi : 7.7).</p>Fórmula:C16H17ClNO5PPureza:98%Forma y color:SolidPeso molecular:369.74Nateglinide D5
CAS:<p>Nateglinide D5 is a deuterium labeled Nateglinide.</p>Fórmula:C19H27NO3Pureza:98%Forma y color:SolidPeso molecular:322.45TGN-073
CAS:<p>TGN-073 is an enhancer of aquaporin 4 (AQP4), a water channel in astrocytes. It shows an increase in lymphatic transport in the rat brain by up to 41%.</p>Fórmula:C18H16N2O3SForma y color:SolidPeso molecular:340.39617β-Estradiol sulfate sodium
CAS:<p>17β-Estradiol sulfate sodium (17β-Estradiol 3-sulfate sodium) is a neuroactive estrogen with vasoprotective properties that inhibits the growth of Neisseria brasiliensis and disrupts aquatic ecosystems.</p>Fórmula:C18H23NaO5SPureza:99%Forma y color:SolidPeso molecular:374.43SKA-121
CAS:<p>SKA-121 is a selective KCa3.1 activator (EC50s: 109 nM and 4.4 μM for KCa3.1 and KCa2.3, respectively).</p>Fórmula:C12H10N2OPureza:98%Forma y color:SolidPeso molecular:198.22Mexiletine-d6 hydrochloride
CAS:<p>Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.</p>Fórmula:C11H18ClNOPureza:98%Forma y color:SolidPeso molecular:221.76N-Methyl-DL-aspartic acid
CAS:<p>N-Methyl-DL-aspartic acid, a glutamate analogue and NMDA receptor agonist, is utilized in neurological disease research.</p>Fórmula:C5H9NO4Pureza:99.85%Forma y color:SolidPeso molecular:147.13UBP608
CAS:<p>UBP608 selectively inhibits NMDA GluN1/GluN2A receptors, 23x more than GluN1/GluN2D.</p>Fórmula:C10H5BrO4Forma y color:SolidPeso molecular:269.05YM-244769
CAS:<p>YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)</p>Fórmula:C26H22FN3O3Pureza:95.62%Forma y color:SolidPeso molecular:443.473,3-Diethylthiacarbocyanine iodide
CAS:<p>3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.</p>Fórmula:C21H21IN2S2Pureza:99.79%Forma y color:SolidPeso molecular:492.44Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Fórmula:C17H26ClNOPureza:99.80%Forma y color:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TastePeso molecular:295.85Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Fórmula:C18H12ClF4N5O2Pureza:98.6%Forma y color:SolidPeso molecular:441.77YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Fórmula:C20H22N2O3SPureza:98.78%Forma y color:SolidPeso molecular:370.47HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Fórmula:C18H21N5O3Pureza:99.69% - ≥95%Forma y color:SolidPeso molecular:355.39CCTA-1523
CAS:<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Fórmula:C16H15Cl2NO3Pureza:99.71%Forma y color:SolidPeso molecular:340.2VU0134992
CAS:<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Fórmula:C20H31BrN2O2Pureza:99.86%Forma y color:SolidPeso molecular:411.38Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Fórmula:C6H9NO4Pureza:99.77%Forma y color:SolidPeso molecular:159.14Omecamtiv mecarbil
CAS:<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Fórmula:C20H24FN5O3Pureza:98% - 99.23%Forma y color:SolidPeso molecular:401.43Dotinurad
CAS:<p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>Fórmula:C14H9Cl2NO4SPureza:97.43% - 98.04%Forma y color:SolidPeso molecular:358.2(S)-ATPO
CAS:<p>(S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.</p>Fórmula:C11H19N2O7PPureza:98.37% - 99.41%Forma y color:SolidPeso molecular:322.25Procyclidine hydrochloride
CAS:<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Fórmula:C19H30ClNOPureza:99.24% - 99.88%Forma y color:Crystals From Petroleum Ether White PowderPeso molecular:323.9DL-Menthol
CAS:<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Fórmula:C10H20OPureza:99.74%Forma y color:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecular:156.27γ-Acetylenic GABA
CAS:<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.143Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Fórmula:C10H12N2O3Pureza:99.38%Forma y color:White Crystalline PowderPeso molecular:208.21UBP551
CAS:<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Fórmula:C11H8O4Pureza:98.69%Forma y color:SolidPeso molecular:204.18DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Fórmula:C7H5FN2OPureza:97.84%Forma y color:SolidPeso molecular:152.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Fórmula:C34H60N14O12SPureza:96.79% - 99.65%Forma y color:White PowderPeso molecular:888.99OAC3
CAS:<p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>Fórmula:C15H11FN2OPureza:97.13%Forma y color:SolidPeso molecular:254.26Myomodulin acetate(110570-93-9 free base)
<p>Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.</p>Fórmula:C38H71N11O10S2Pureza:99.24%Forma y color:SolidPeso molecular:906.17Raxatrigine
CAS:<p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>Fórmula:C18H19FN2O2Pureza:98% - 99.43%Forma y color:SolidPeso molecular:314.35Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Fórmula:C38H52CaN2O8Pureza:98.97% - 99.96%Forma y color:White SolidPeso molecular:704.91HC067047 Hydrochloride(883031-03-6 free base)
CAS:<p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>Fórmula:C26H29ClF3N3O2Pureza:99.95%Forma y color:SolidPeso molecular:507.98Ivacaftor
CAS:<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Fórmula:C24H28N2O3Pureza:99% - 99.98%Forma y color:SolidPeso molecular:392.49NPPB
CAS:<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Fórmula:C16H16N2O4Pureza:99.95%Forma y color:Light Yellow To Yellow SolidPeso molecular:300.31NBQX
CAS:<p>NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.</p>Fórmula:C12H8N4O6SPureza:97.66% - 99.42%Forma y color:SolidPeso molecular:336.286-Methylflavone
CAS:<p>6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.</p>Fórmula:C16H12O2Pureza:99.69%Forma y color:SolidPeso molecular:236.27Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Fórmula:C15H14O4Pureza:98.06%Forma y color:SolidPeso molecular:258.27Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Fórmula:C17H16FN3O2SPureza:99.87% - 99.92%Forma y color:SolidPeso molecular:345.39TRPM8 antagonist WS-3
CAS:<p>TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).</p>Fórmula:C13H25NOPureza:97.64%Forma y color:DrypowderPeso molecular:211.34SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Fórmula:C10H12N2O3Pureza:99.84%Forma y color:SolidPeso molecular:208.21AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Fórmula:C34H31F2N3O3Pureza:99.61%Forma y color:SolidPeso molecular:567.62ICA-121431
CAS:<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Fórmula:C23H19N3O3S2Pureza:98.06%Forma y color:SolidPeso molecular:449.55SAR7334 hydrochloride
CAS:<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Fórmula:C21H24Cl3N3OPureza:98%Forma y color:SolidPeso molecular:440.79Selinexor (KPT-330)
CAS:<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Fórmula:C17H11F6N7OPureza:98% - 99.97%Forma y color:SolidPeso molecular:443.31Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2·C4H4O4Pureza:99.5% - 99.9%Forma y color:Off-White Crystalline PowderPeso molecular:420.39Homo-VK-II-36
CAS:<p>Homo-VK-II-36 (Homo-V-II-36) is a carvedilol analogue that acts by inhibiting store- overload-induced calcium release through the RyR2 channel.</p>Fórmula:C27H28N2O5Pureza:99.26%Forma y color:SolidPeso molecular:460.527-Chlorokynurenic acid sodium salt
CAS:<p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>Fórmula:C10H6ClNNaO3Forma y color:SolidPeso molecular:246.6α-Cyano-4-hydroxycinnamic acid
CAS:<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Fórmula:C10H7NO3Pureza:99.8% - 99.86%Forma y color:PowderPeso molecular:189.17Thonzonium Bromide
CAS:<p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>Fórmula:C32H55BrN4OPureza:98.48% - 99.94%Forma y color:SolidPeso molecular:591.71Linerixibat
CAS:<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Fórmula:C28H38N2O7SPureza:98.5% - 99.98%Forma y color:SolidPeso molecular:546.68ML365
CAS:<p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>Fórmula:C22H20N2O3Pureza:98.78%Forma y color:SolidPeso molecular:360.41Vanilloid receptor antagonist 1
CAS:<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Fórmula:C18H15N3O2Pureza:98.14%Forma y color:SolidPeso molecular:305.33Zoniporide hydrochloride hydrate
CAS:<p>Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.</p>Fórmula:C17H19ClN6O2Pureza:98%Forma y color:SolidPeso molecular:374.83SB-366791
CAS:<p>SB-366791 is a new and selective cinnamide TRPV1 antagonist.</p>Fórmula:C16H14ClNO2Pureza:99.51%Forma y color:SolidPeso molecular:287.74Optovin
CAS:<p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>Fórmula:C15H13N3OS2Pureza:99.47% - 99.67%Forma y color:SolidPeso molecular:315.41Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Fórmula:C24H32NO6ClPureza:99.9%Forma y color:SolidPeso molecular:465.97Vocacapsaicin
CAS:<p>Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.</p>Fórmula:C26H41N3O4Forma y color:SolidPeso molecular:459.631N-Me-aminopyrimidinone9
CAS:<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Fórmula:C16H21N3OSPureza:99.21%Forma y color:SolidPeso molecular:303.42SKA-31
CAS:<p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>Fórmula:C11H8N2SPureza:99.38%Forma y color:SolidPeso molecular:200.26Efonidipine hydrochloride
CAS:<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Fórmula:C34H39ClN3O7PForma y color:SolidPeso molecular:668.12Trofinetide
CAS:<p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>Fórmula:C13H21N3O6Pureza:98.70% - 99.50%Forma y color:SolidPeso molecular:315.32Nav1.8-IN-1
CAS:<p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>Fórmula:C20H15ClF3N3O2Pureza:97.59%Forma y color:SolidPeso molecular:421.86-(4-Methoxyphenyl)-3-pyridazinamine
CAS:<p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>Fórmula:C11H11N3OPureza:99.03%Forma y color:SolidPeso molecular:201.22Tulrampator
CAS:<p>Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.</p>Fórmula:C20H17FN4O3Pureza:99.77%Forma y color:SolidPeso molecular:380.37Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Fórmula:C17H24O4Pureza:98.22%Forma y color:SolidPeso molecular:292.37Vonoprazan fumarate
CAS:<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Fórmula:C17H16FN3O2S·C4H4O4Pureza:99.16% - 99.98%Forma y color:SolidPeso molecular:461.46(R)-baclofen
CAS:<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Fórmula:C10H12ClNO2Pureza:97.20% - 98.94%Forma y color:SolidPeso molecular:213.66CL 218872
CAS:<p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>Fórmula:C13H9F3N4Pureza:99.92%Forma y color:SolidPeso molecular:278.23Revaprazan
CAS:<p>Revaprazan: novel, K⁺-competitive acid blocker; reversibly halts gastric H⁺/K⁺-ATPase; rivals PPIs in acid reduction.</p>Fórmula:C22H23FN4Pureza:98%Forma y color:SolidPeso molecular:362.44TGN-020
CAS:<p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>Fórmula:C8H6N4OSPureza:99.54% - 99.99%Forma y color:SolidPeso molecular:206.22Ko 143
CAS:<p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>Fórmula:C26H35N3O5Pureza:99.01% - 99.89%Forma y color:SolidPeso molecular:469.57
