Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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Ataluren
CAS:<p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>Fórmula:C15H9FN2O3Pureza:99.16% - 99.84%Forma y color:SolidPeso molecular:284.24Raxatrigine hydrochloride
CAS:<p>Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.</p>Fórmula:C18H20ClFN2O2Pureza:98%Forma y color:SolidPeso molecular:350.82Rostafuroxin
CAS:<p>Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.</p>Fórmula:C23H34O4Pureza:99.08% - >99.99%Forma y color:SolidPeso molecular:374.51CX614
CAS:<p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>Fórmula:C13H13NO4Pureza:97.37%Forma y color:SolidPeso molecular:247.25Benzonatate
CAS:<p>Benzonatate is an antagonist of sodium channel protein.</p>Fórmula:C30H53NO11Pureza:99.92%Forma y color:Colorless To Faintly Yellow Oil LiquidPeso molecular:603.74Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Fórmula:C19H22O2Pureza:99.22% - 99.66%Forma y color:SolidPeso molecular:282.38Aptiganel hydrochloride
CAS:<p>Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>Fórmula:C20H22ClN3Pureza:99.89%Forma y color:SolidPeso molecular:339.86KPT276
CAS:<p>KPT276 (KPT 276) is an orally bioavailable selective inhibitor of nuclear export (SINE) that irreversibly bind to CRM1 and block the function of CRM1.</p>Fórmula:C16H10F8N4OPureza:99.89% - >99.99%Forma y color:SolidPeso molecular:426.26Tariquidar dihydrochloride
CAS:<p>Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).</p>Fórmula:C38H40Cl2N4O6Forma y color:SolidPeso molecular:719.65NBQX
CAS:<p>NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.</p>Fórmula:C12H8N4O6SPureza:97.66% - 99.42%Forma y color:SolidPeso molecular:336.28Etripamil
CAS:<p>Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.</p>Fórmula:C27H36N2O4Pureza:99.47% - 99.83%Forma y color:SolidPeso molecular:452.59Kv2-IN-A1
CAS:<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Fórmula:C20H17ClN4OSPureza:98.83%Forma y color:SolidPeso molecular:396.89Triclabendazole sulfoxide
CAS:<p>TCBZ-SO, a Triclabendazole metabolite, blocks ABCG2/BCRP and has anti-parasitic properties.</p>Fórmula:C14H9Cl3N2O2SPureza:98.02%Forma y color:SolidPeso molecular:375.66CFTR(inh)-172
CAS:<p>CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.</p>Fórmula:C18H10F3NO3S2Pureza:98% - 99.72%Forma y color:SolidPeso molecular:409.4Lansoprazole sulfone
CAS:<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Fórmula:C16H14F3N3O3SPureza:99.67%Forma y color:SolidPeso molecular:385.36Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Fórmula:C20H25NO2S2Pureza:99.25%Forma y color:White To Off-White Crystalline SolidPeso molecular:375.55Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Fórmula:C53H90O22Pureza:98.83% - 99.56%Forma y color:White PowderPeso molecular:1079.27Tirofiban hydrochloride monohydrate
CAS:<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Fórmula:C22H39ClN2O6SPureza:98.81% - >99.99%Forma y color:White SolidPeso molecular:495.07Phe-Met-Arg-Phe, amide acetate
<p>Phe-Met-Arg-Phe amide acetate (ED50=23 nM) triggers K+ current in caudodorsal neurons, co-localizes with neuropeptide Y in brain areas.</p>Fórmula:C31H46N8O6SPureza:99.4%Forma y color:SolidPeso molecular:658.82Levosimendan
CAS:<p>Levosimendan (OR1259) is a calcium sensitizer for acute heart failure, enhancing cardiac contractility without raising calcium levels.</p>Fórmula:C14H12N6OPureza:99.37% - 99.91%Forma y color:Yellow Crystalline PowderPeso molecular:280.28Chloroprocaine
CAS:<p>Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.</p>Fórmula:C13H19ClN2O2Forma y color:SolidPeso molecular:270.76AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Forma y color:SolidPeso molecular:354.38Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Fórmula:C17H11N5OPureza:99.81%Forma y color:SolidPeso molecular:301.3Esomeprazole
CAS:<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Fórmula:C17H19N3O3SPureza:97.3%Forma y color:SolidPeso molecular:345.42Esomeprazole potassium salt
CAS:<p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>Fórmula:C17H18KN3O3SForma y color:SolidPeso molecular:383.51SAR7334 hydrochloride
CAS:<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Fórmula:C21H24Cl3N3OPureza:98%Forma y color:SolidPeso molecular:440.79Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Fórmula:C18H12BrFN4OPureza:98.4%Forma y color:SolidPeso molecular:399.22Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Fórmula:C10H12N2O3Pureza:99.38%Forma y color:White Crystalline PowderPeso molecular:208.21Nisoxetine
CAS:<p>Nisoxetine is a selective NET (noradrenaline transporter) inhibitor (Kd=0.76 nM) capable of blocking voltage-gated sodium channels.</p>Fórmula:C17H21NO2Forma y color:SolidPeso molecular:271.35Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Fórmula:C22H25ClN2Pureza:99.46%Forma y color:SolidPeso molecular:352.9Flupirtine
CAS:<p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2Forma y color:SolidPeso molecular:304.32Icenticaftor
CAS:<p>Icenticaftor (QBW251) is an orally active potentiator of CFTR channel.</p>Fórmula:C12H13F6N3O3Pureza:99.76%Forma y color:SolidPeso molecular:361.24KCNQ2/3 activator-1
CAS:<p>KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.</p>Fórmula:C23H29FN2OPureza:99.16% - 99.47%Forma y color:SolidPeso molecular:368.49Rimtuzalcap
CAS:<p>Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and ET.</p>Fórmula:C18H24F2N6OPureza:99.64%Forma y color:SolidPeso molecular:378.42Raxatrigine
CAS:<p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>Fórmula:C18H19FN2O2Pureza:98% - 99.43%Forma y color:SolidPeso molecular:314.35Nateglinide
CAS:<p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>Fórmula:C19H27NO3Pureza:99.93% - 99.94%Forma y color:White Crystalline PowderPeso molecular:317.42Gabazine free base
CAS:<p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>Fórmula:C15H17N3O3Forma y color:SolidPeso molecular:287.31N-Me-aminopyrimidinone9
CAS:<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Fórmula:C16H21N3OSPureza:99.21%Forma y color:SolidPeso molecular:303.42GMQ hydrochloride
CAS:<p>GMQ hydrochloride, a potent ASIC modulator, activates ASIC3 at neutral pH and inhibits acid-induced peak current.</p>Fórmula:C10H12ClN5Pureza:99.64%Forma y color:SolidPeso molecular:237.692'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Forma y color:SolidPeso molecular:270.28Linerixibat
CAS:<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Fórmula:C28H38N2O7SPureza:98.5% - 99.98%Forma y color:SolidPeso molecular:546.68Benzamil
CAS:<p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>Fórmula:C13H14ClN7OPureza:99.79%Forma y color:SolidPeso molecular:319.75ML329
CAS:<p>ML329 is a small molecule inhibitor of MITF, inhibiting TRPM-1 promoter activity.</p>Fórmula:C16H12N2O4SPureza:98.96%Forma y color:SolidPeso molecular:328.34Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Fórmula:C17H24O4Pureza:98.22%Forma y color:SolidPeso molecular:292.37DQP 1105
CAS:<p>DQP 1105 is a NMDA receptor antagonist.</p>Fórmula:C29H24BrN3O4Pureza:98.6%Forma y color:SolidPeso molecular:558.42Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Forma y color:SolidPeso molecular:86.14UBP551
CAS:<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Fórmula:C11H8O4Pureza:98.69%Forma y color:SolidPeso molecular:204.18Omecamtiv mecarbil
CAS:<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Fórmula:C20H24FN5O3Pureza:98% - 99.23%Forma y color:SolidPeso molecular:401.43VU0134992
CAS:<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Fórmula:C20H31BrN2O2Pureza:99.86%Forma y color:SolidPeso molecular:411.38Disopyramide phosphate
CAS:<p>Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.</p>Fórmula:C21H32N3O5PForma y color:SolidPeso molecular:437.47Acamprosate calcium
CAS:<p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>Fórmula:C10H20CaN2O8S2Pureza:98% - 99.93%Forma y color:White Odorless Or Nearly Odorless PowderPeso molecular:400.48GSK369796 Dihydrochloride
CAS:<p>GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.</p>Fórmula:C20H24Cl3N3OPureza:>99.99%Forma y color:SolidPeso molecular:428.78Blebbistatin
CAS:<p>Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.</p>Fórmula:C18H16N2O2Pureza:99.88% - 99.97%Forma y color:Bright Yellow SolidPeso molecular:292.33TRPM8 antagonist WS-3
CAS:<p>TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).</p>Fórmula:C13H25NOPureza:97.64%Forma y color:DrypowderPeso molecular:211.34VU6036720 hydrochloride
<p>VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.</p>Fórmula:C20H23Cl2FN4O2SForma y color:SolidPeso molecular:473.39ML204
CAS:<p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>Fórmula:C15H18N2Pureza:98.1% - 99.72%Forma y color:SolidPeso molecular:226.32Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Fórmula:C16H14FN3OPureza:99.72%Forma y color:SolidPeso molecular:283.3α-Cyano-4-hydroxycinnamic acid
CAS:<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Fórmula:C10H7NO3Pureza:99.8% - 99.86%Forma y color:PowderPeso molecular:189.17BRITE-338733
CAS:<p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>Fórmula:C27H35N3O2Pureza:99.85%Forma y color:SolidPeso molecular:433.59Iptakalim Hydrochloride
CAS:<p>Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine</p>Fórmula:C9H22ClNPureza:98%Forma y color:SolidPeso molecular:179.731IDRA-21
CAS:<p>IDRA-21 is a positive AMPA receptor modulator.</p>Fórmula:C8H9ClN2O2SPureza:99.73%Forma y color:SolidPeso molecular:232.69Temgicoluril
CAS:<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Fórmula:C8H14N4O2Pureza:99.8%Forma y color:SolidPeso molecular:198.22DL-Menthol
CAS:<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Fórmula:C10H20OPureza:99.74%Forma y color:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecular:156.27AMG 517
CAS:<p>AMG 517 is an effective and specific TRPV1 antagonist, antagonizes proton (IC50: 0.76 nM), capsaicin (IC50: 0.62 nM) and heat activation (IC50: 1.3 nM) of TRPV1</p>Fórmula:C20H13F3N4O2SPureza:99.77% - 99.85%Forma y color:SolidPeso molecular:430.4SN 2
CAS:<p>SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.</p>Fórmula:C17H21NOPureza:99.86%Forma y color:SolidPeso molecular:255.35CCTA-1523
CAS:<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Fórmula:C16H15Cl2NO3Pureza:99.71%Forma y color:SolidPeso molecular:340.2YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Fórmula:C20H22N2O3SPureza:98.78%Forma y color:SolidPeso molecular:370.475,7-Dichlorokynurenic acid
CAS:<p>5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.</p>Fórmula:C10H5Cl2NO3Pureza:99.71%Forma y color:SolidPeso molecular:258.06Songorine
CAS:<p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>Fórmula:C22H31NO3Pureza:98% - 99.92%Forma y color:SolidPeso molecular:357.49Vanilloid receptor antagonist 1
CAS:<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Fórmula:C18H15N3O2Pureza:98.14%Forma y color:SolidPeso molecular:305.33Loreclezole
CAS:<p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>Fórmula:C10H6Cl3N3Pureza:99.78%Forma y color:SolidPeso molecular:274.53KM 91104
CAS:<p>KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.</p>Fórmula:C14H12N2O4Pureza:99.04%Forma y color:SolidPeso molecular:272.26Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Fórmula:C14H14O3Pureza:99.93% - ≥95%Forma y color:SolidPeso molecular:230.26AUT1
CAS:<p>AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).</p>Fórmula:C18H19N3O4Pureza:99.8% - 99.95%Forma y color:SolidPeso molecular:341.36Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Fórmula:C18H12ClF4N5O2Pureza:98.6%Forma y color:SolidPeso molecular:441.77Guanidinoethyl sulfonate
CAS:<p>Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist.</p>Fórmula:C3H9N3O3SPureza:99.43% - 99.47%Forma y color:SolidPeso molecular:167.19λ-Cyhalothrin
CAS:<p>λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.</p>Fórmula:C23H19ClF3NO3Pureza:99.76%Forma y color:SolidPeso molecular:449.85AM92016
CAS:<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Fórmula:C26H30Cl2N2O6SForma y color:SolidPeso molecular:569.49RN-1734
CAS:<p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>Fórmula:C14H22Cl2N2O2SPureza:99.1% - 99.3%Forma y color:SolidPeso molecular:353.31Esomeprazole magnesium salt
CAS:<p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>Fórmula:C17H21MgN3O3SForma y color:SolidPeso molecular:371.74Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Fórmula:C14H16ClN3O4S2Pureza:98.23% - 99.49%Forma y color:Crystals From Dilute Alcohol SolidPeso molecular:389.88Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Fórmula:C17H26ClNOPureza:99.80%Forma y color:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TastePeso molecular:295.85SKA-31
CAS:<p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>Fórmula:C11H8N2SPureza:99.38%Forma y color:SolidPeso molecular:200.26NBI-98782
CAS:<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Fórmula:C19H29NO3Pureza:99.29%Forma y color:SolidPeso molecular:319.44Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Fórmula:C19H17N4NaO2SPureza:99.06%Forma y color:SolidPeso molecular:388.42Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Fórmula:C6H9NO4Pureza:99.77%Forma y color:SolidPeso molecular:159.14Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Fórmula:C24H32NO6ClPureza:99.9%Forma y color:SolidPeso molecular:465.97XEN907
CAS:<p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>Fórmula:C21H21NO4Pureza:99.92%Forma y color:SolidPeso molecular:351.4Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Fórmula:C14H32N2O4Pureza:99.91% - 99.92%Forma y color:Viscous Liquid Liquid ViscousPeso molecular:292.41S107
CAS:<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Fórmula:C11H15NOSPureza:99.90%Forma y color:SolidPeso molecular:209.31RY785
CAS:<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Fórmula:C21H20N4O2SPureza:99.78%Forma y color:SolidPeso molecular:392.47Vanillyl butyl ether
CAS:<p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>Fórmula:C12H18O3Pureza:99.57%Forma y color:Yellowish Liquid LiquidPeso molecular:210.27Rbin-1
CAS:<p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>Fórmula:C13H12N4SPureza:99.83%Forma y color:SolidPeso molecular:256.33Epaminurad
CAS:<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Fórmula:C14H10Br2N2O3Forma y color:SolidPeso molecular:414.05Parimifasor
CAS:<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Fórmula:C18H11Cl2F4N5OPureza:96.77% - 98.97%Forma y color:SolidPeso molecular:460.21DL-Willardiine
CAS:<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Fórmula:C7H9N3O4Pureza:99.83%Forma y color:SolidPeso molecular:199.16A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Fórmula:C13H12ClNO3Pureza:98.54%Forma y color:SolidPeso molecular:265.69HC067047 Hydrochloride(883031-03-6 free base)
CAS:<p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>Fórmula:C26H29ClF3N3O2Pureza:99.95%Forma y color:SolidPeso molecular:507.98Dotinurad
CAS:<p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>Fórmula:C14H9Cl2NO4SPureza:97.43% - 98.04%Forma y color:SolidPeso molecular:358.2CTP disodium dihydrate
CAS:<p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>Fórmula:C9H18N3Na2O16P3Pureza:98.51%Forma y color:White Crystalline PowderPeso molecular:563.15PAP-1
CAS:<p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>Fórmula:C21H18O5Pureza:99.35% - 99.75%Forma y color:White SolidPeso molecular:350.36Levcromakalim
CAS:<p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>Fórmula:C16H18N2O3Pureza:99.74%Forma y color:SolidPeso molecular:286.33ML213
CAS:<p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>Fórmula:C17H23NOPureza:>99.99%Forma y color:SolidPeso molecular:257.37YHO-13351
CAS:<p>YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.</p>Fórmula:C27H37N3O7S2Pureza:97.88%Forma y color:SolidPeso molecular:579.73DL-AP5
CAS:<p>DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.</p>Fórmula:C5H12NO5PPureza:99.33%Forma y color:White Fine Crystalline PowderPeso molecular:197.13Pico145
CAS:<p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>Fórmula:C23H20ClF3N4O5Pureza:99.06%Forma y color:SolidPeso molecular:524.88rac-BHFF
CAS:<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Fórmula:C17H21F3O3Pureza:99.69% - >99.99%Forma y color:SolidPeso molecular:330.34Lomerizine
CAS:<p>Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.</p>Fórmula:C27H30F2N2O3Forma y color:SolidPeso molecular:468.54Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2·C4H4O4Pureza:99.5% - 99.9%Forma y color:Off-White Crystalline PowderPeso molecular:420.39Selinexor (KPT-330)
CAS:<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Fórmula:C17H11F6N7OPureza:98% - 99.97%Forma y color:SolidPeso molecular:443.31TRPM4-IN-1
CAS:<p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>Fórmula:C15H11Cl2NO4Pureza:97.22%Forma y color:SolidPeso molecular:340.16(S)-(-)-5-Fluorowillardiine hydrochloride
CAS:<p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>Fórmula:C7H9ClFN3O4Forma y color:SolidPeso molecular:253.62Unifiram
CAS:<p>Unifiram boosts cognition, enhances rat hippocampal signals (EC50=27 nM), and ups ACh in rat cortex.</p>Fórmula:C13H15FN2O3SPureza:99.9%Forma y color:SolidPeso molecular:298.33Tricaine methanesulfonate
CAS:<p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>Fórmula:C10H15NO5SPureza:99.259% - 99.86%Forma y color:White PowderPeso molecular:261.30Methyl homoveratrate
CAS:<p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>Fórmula:C11H14O4Pureza:99.48%Forma y color:SolidPeso molecular:210.23SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Fórmula:C18H21ClF3N3OPureza:99.03% - 99.95%Forma y color:SolidPeso molecular:387.83BzATP triethylammonium salt
CAS:<p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>Fórmula:C30H39N6O15P3Pureza:95% - 99.57%Forma y color:SolidPeso molecular:816.59MK6-83
CAS:<p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>Fórmula:C16H20N2O2S2Pureza:99.5%Forma y color:SolidPeso molecular:336.479-Phenanthrol
CAS:<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Fórmula:C14H10OPureza:98.48%Forma y color:SolidPeso molecular:194.23Amifampridine phosphate
CAS:<p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>Fórmula:C5H10N3O4PForma y color:SolidPeso molecular:207.12O4I1
CAS:<p>O4I1 is an effective Oct3/4 inducer.</p>Fórmula:C16H15NO2Pureza:96.25% - 99.47%Forma y color:SolidPeso molecular:253.3Sepimostat dimethanesulfonate
CAS:<p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>Fórmula:C23H27N5O8S2Forma y color:SolidPeso molecular:565.62Quinine hydrobromide
CAS:<p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>Fórmula:C20H25BrN2O2Forma y color:SolidPeso molecular:405.336ICA-121431
CAS:<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Fórmula:C23H19N3O3S2Pureza:98.06%Forma y color:SolidPeso molecular:449.55Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Fórmula:C17H16FN3O2SPureza:99.87% - 99.92%Forma y color:SolidPeso molecular:345.39Eniporide hydrochloride
CAS:<p>Eniporide hydrochloride (EMD-96785 hydrochloride) serves as a robust inhibitor of the sodium/hydrogen (Na+/H+) exchange process.</p>Fórmula:C14H17ClN4O3SForma y color:SolidPeso molecular:356.83Selamectin
CAS:<p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>Fórmula:C43H63NO11Pureza:99.84%Forma y color:SolidPeso molecular:769.96Esomeprazole hemistrontium
CAS:<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Fórmula:C34H36N6O6S2SrForma y color:SolidPeso molecular:776.44Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Fórmula:C15H14O4Pureza:98.06%Forma y color:SolidPeso molecular:258.27NPPB
CAS:<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Fórmula:C16H16N2O4Pureza:99.95%Forma y color:Light Yellow To Yellow SolidPeso molecular:300.31Flecainide acetate
CAS:<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Fórmula:C19H24F6N2O5Pureza:99.42%Forma y color:SolidPeso molecular:474.39Ivacaftor
CAS:<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Fórmula:C24H28N2O3Pureza:99% - 99.98%Forma y color:SolidPeso molecular:392.494-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Fórmula:C6H11NO3Pureza:98.51%Forma y color:SolidPeso molecular:145.16Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Fórmula:C13H8BrN4NaO3Forma y color:SolidPeso molecular:371.13Myomodulin acetate(110570-93-9 free base)
<p>Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.</p>Fórmula:C38H71N11O10S2Pureza:99.24%Forma y color:SolidPeso molecular:906.17NS6180
CAS:<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Fórmula:C16H12F3NOSPureza:99.83% - ≥95%Forma y color:SolidPeso molecular:323.33Azimilide Dihydrochloride
CAS:<p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>Fórmula:C23H30Cl3N5O3Pureza:97.59% - ≥95%Forma y color:SolidPeso molecular:530.88RQ-00203078
CAS:<p>RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.</p>Fórmula:C21H13ClF6N2O5SPureza:98% - 99.6%Forma y color:SolidPeso molecular:554.85Jujuboside A
CAS:<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Fórmula:C58H94O26Pureza:98% - >99.99%Forma y color:SolidPeso molecular:1207.35Amlodipine mesylate
CAS:<p>Amlodipine mesylate, an oral dihydropyridine Ca2+ blocker, treats angina, hypertension, and may be used in cancer research.</p>Fórmula:C21H29ClN2O8SForma y color:SolidPeso molecular:504.98DS-1971a
CAS:<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Fórmula:C20H21ClFN5O3SPureza:99.66%Forma y color:SolidPeso molecular:465.93Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Fórmula:C17H21ClF6N2O3Pureza:97.79%Forma y color:SolidPeso molecular:450.81Rufinamide
CAS:<p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>Fórmula:C10H8F2N4OPureza:99.77% - >99.99%Forma y color:White PowderPeso molecular:238.19Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Fórmula:(C20H36N2O3S)2·C4H4O4Pureza:99.68% - 99.74%Forma y color:SolidPeso molecular:885.23TRAM-34
CAS:<p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>Fórmula:C22H17ClN2Pureza:99.01% - 99.91%Forma y color:SolidPeso molecular:344.84Ko 143
CAS:<p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>Fórmula:C26H35N3O5Pureza:99.01% - 99.89%Forma y color:SolidPeso molecular:469.57Chloroprocaine hydrochloride
CAS:<p>Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.</p>Fórmula:C13H20Cl2N2O2Pureza:99.65%Forma y color:White Crystalline PowderPeso molecular:307.22BAY-8002
CAS:<p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>Fórmula:C20H14ClNO5SPureza:98.7% - 99.13%Forma y color:SolidPeso molecular:415.85Ropivacaine hydrochloride monohydrate
CAS:<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Fórmula:C17H29ClN2O2Pureza:99.94% - 99.95%Forma y color:White SolidPeso molecular:328.88Tetraethylammonium chloride
CAS:<p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>Fórmula:C8H20ClNPureza:≥95%Forma y color:White Solid Solid Particulate/PowderPeso molecular:165.7Ro 25-6981 Maleate
CAS:<p>Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders such as Parkinson's and epilepsy.</p>Fórmula:C26H33NO6Pureza:99.42%Forma y color:SolidPeso molecular:455.54JNJ-28583113
CAS:<p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>Fórmula:C19H21F3N2O2Pureza:98.57%Forma y color:SolidPeso molecular:366.38SRI-41315
CAS:<p>SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.</p>Fórmula:C22H19N3O2Pureza:99.87%Forma y color:SolidPeso molecular:357.41Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Forma y color:PowderPeso molecular:234.2Doxapram
CAS:<p>Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.</p>Fórmula:C24H30N2O2Pureza:99.42%Forma y color:SolidPeso molecular:378.51Darigabat
CAS:<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Fórmula:C22H21FN4O3SPureza:98.42% - 99.29%Forma y color:SolidPeso molecular:440.49Methionine
CAS:<p>Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor</p>Fórmula:C5H11NO2SPureza:99.13% - 99.62%Forma y color:SolidPeso molecular:149.21BL-1249
CAS:<p>BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).</p>Fórmula:C17H17N5Pureza:98% - 98.25%Forma y color:SolidPeso molecular:291.35VU590
CAS:<p>VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.</p>Fórmula:C24H32N4O7Pureza:98.06%Forma y color:SolidPeso molecular:488.53Bupivacaine
CAS:<p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>Fórmula:C18H28N2OPureza:99.83%Forma y color:SolidPeso molecular:288.43Dimiracetam
CAS:<p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>Fórmula:C6H8N2O2Pureza:>99.99% - >99.99%Forma y color:SolidPeso molecular:140.14ZT-1a
CAS:<p>ZT-1a is a SPAK inhibitor.ZT-1a inhibits SPAK.ZT-1a can be used for the prevention and treatment of neurodegenerative and neurocognitive disorders.</p>Fórmula:C22H15Cl3N2O2Pureza:99.77%Forma y color:SolidPeso molecular:445.73Safinamide
CAS:<p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>Fórmula:C17H19FN2O2Pureza:99.92%Forma y color:SolidPeso molecular:302.34Apinocaltamide
CAS:<p>Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.</p>Fórmula:C22H18F3N5OPureza:99.80%Forma y color:SolidPeso molecular:425.41Lanicemine dihydrochloride
CAS:<p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C13H16Cl2N2Pureza:98.37%Forma y color:SolidPeso molecular:271.19HUP30
CAS:<p>HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.</p>Fórmula:C14H15N3O3SPureza:99.96%Forma y color:SolidPeso molecular:305.35N-Methyl-L-leucin
CAS:<p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>Fórmula:C7H15NO2Pureza:99.87%Forma y color:SolidPeso molecular:145.2CX717
CAS:<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Fórmula:C11H11N3O3Pureza:99.81%Forma y color:SoildPeso molecular:233.23Mtb ATP synthase-IN-1
CAS:<p>Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.</p>Fórmula:C17H13N3O4Pureza:98.28%Forma y color:SolidPeso molecular:323.30VB124
CAS:<p>VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.</p>Fórmula:C23H23ClN2O4Pureza:99.21% - 99.57%Forma y color:SoildPeso molecular:426.89PF 03716556
CAS:<p>PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux</p>Fórmula:C22H26N4O3Pureza:99.79% - 99.85%Forma y color:SolidPeso molecular:394.47Propoxycaine hydrochloride
CAS:<p>Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.</p>Fórmula:C16H27ClN2O3Pureza:97.25%Forma y color:SolidPeso molecular:330.85Bupivacaine-d9
CAS:<p>Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.</p>Fórmula:C18H19D9N2OForma y color:SolidPeso molecular:297.48SAR7334
CAS:<p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Fórmula:C21H22ClN3OPureza:99.62% - 99.71%Forma y color:SolidPeso molecular:367.87Eleclazine
CAS:<p>Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).</p>Fórmula:C21H16F3N3O3Pureza:98.67%Forma y color:SolidPeso molecular:415.37MCT-IN-1
CAS:<p>MCT-IN-1 (compound 2) acts as a potent inhibitor of the monocarboxylate transporter (MCT), demonstrating IC50 values of 9 nM for MCT1 and 14 nM for MCT4.</p>Fórmula:C19H26N2O3Forma y color:SolidPeso molecular:330.42Eperisone
CAS:<p>Eperisone: a muscle relaxant for stiffness and pain, relaxes muscles, improves circulation, and mitigates pain by inhibiting reflexes and vasodilation.</p>Fórmula:C17H25NOForma y color:SolidPeso molecular:259.39Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46VGSC blocker-1
CAS:<p>VGSC blocker-1 inhibits 34.9% INa in nNav1.5 at 1 μM, reduces MDA-MB-231 invasion by 0.3%, non-toxic.</p>Fórmula:C24H32F2N2Forma y color:SolidPeso molecular:386.52FSC231
CAS:<p>FSC231 is a PICK1 inhibitor with analgesic activity, activating GSK-3β and ERK1/2.</p>Fórmula:C13H10Cl2N2O3Pureza:99.66%Forma y color:SolidPeso molecular:313.14Amlodipine besilate impurity G
CAS:<p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>Fórmula:C17H18ClNO4Pureza:98%Forma y color:SolidPeso molecular:335.78Cinepazide
CAS:<p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>Fórmula:C22H31N3O5Forma y color:White PowderPeso molecular:417.5Amlodipine hydrochloride
CAS:<p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>Fórmula:C20H26Cl2N2O5Forma y color:SolidPeso molecular:445.34PBFI-AM
CAS:<p>PBFI-AM is a useful tool to determine intracellular K + content [1] .</p>Fórmula:C58H62N2O24Forma y color:SolidPeso molecular:1171.11Methocarbamol D5
CAS:<p>Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.</p>Fórmula:C11H15NO5Pureza:98%Forma y color:SolidPeso molecular:246.27Topiramate D12
CAS:<p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>Fórmula:C12H21NO8SPureza:98%Forma y color:SolidPeso molecular:351.44Propafenone D7 hydrochloride
CAS:<p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>Fórmula:C21H28ClNO3Pureza:98%Forma y color:SolidPeso molecular:384.95Repaglinide D5
CAS:<p>Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.</p>Fórmula:C27H36N2O4Pureza:98%Forma y color:SolidPeso molecular:457.62Nifedipine-d6
CAS:<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Fórmula:C17H18N2O6Pureza:98%Forma y color:SolidPeso molecular:352.37BAY-390
CAS:<p>BAY-390, a selective TRPA1 inhibitor, crosses species, penetrates brains, with IC50s: 16-82 nM. Used in inflammation research.</p>Fórmula:C13H15F4NOForma y color:SolidPeso molecular:277.26Dofetilide D4
CAS:<p>Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.</p>Fórmula:C19H27N3O5S2Pureza:98%Forma y color:SolidPeso molecular:445.59Bumetanide-d5
CAS:<p>Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).</p>Fórmula:C17H20N2O5SPureza:98%Forma y color:SolidPeso molecular:369.45FFN 511 hydrochloride
CAS:<p>FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitter (FFNs) targeting VMA T2 that can be used to label baraminergic nerve endings.</p>Fórmula:C17H21ClN2O2Pureza:99.83%Forma y color:SoildPeso molecular:320.81ORM-10103
CAS:<p>ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nM</p>Fórmula:C20H16N2O4Pureza:99.9%Forma y color:SolidPeso molecular:348.35MNI-caged-NMDA
CAS:<p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>Fórmula:C14H17N3O6Pureza:98%Forma y color:SolidPeso molecular:323.30Tetradifon
CAS:<p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>Fórmula:C12H6Cl4O2SPureza:99.84%Forma y color:Yellowish Odorless OilPeso molecular:356.05A-317491 sodium salt hydrate
<p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>Fórmula:C33H29NNaO9Pureza:98%Forma y color:SolidPeso molecular:606.57Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Fórmula:C21H27NOForma y color:Needles From Petroleum Ether SolidPeso molecular:309.45DL-AP7
CAS:<p>DL-AP7: competitive NMDA antagonist, anticonvulsant, inhibits NMDA convulsions, impairs mice learning.</p>Fórmula:C7H16NO5PPureza:98%Forma y color:SolidPeso molecular:225.18LY 303511
CAS:<p>LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.</p>Fórmula:C19H18N2O2Pureza:98%Forma y color:SolidPeso molecular:306.36
