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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

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Se han encontrado 8626 productos de "Metabolismo"

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  • OMS-824

    CAS:
    <p>OMS-824 is a phosphodiesterase-10 inhibitor that slows or stops the hydrolysis of cAMP and cGMP.</p>
    Fórmula:C21H21BrN4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.32
  • 2-Iodoestradiol

    CAS:
    2-Iodoestradiol is an effective human sex hormone-binding globulin (SHBG) ligand.
    Fórmula:C18H23IO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:398.28
  • myomiR-IN-1

    CAS:
    <p>myomiR-IN-1 inhibits myoD translation in C2C12 cells, doesn't affect myoD mRNA, and reduces differentiation markers.</p>
    Fórmula:C33H27NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:533.57
  • α-RA-F

    CAS:
    <p>Alpha-RA-F increases collagen, lowers MMPs in human fibroblasts, non-toxic.</p>
    Fórmula:C16H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:300.31
  • ARI-3531

    CAS:
    <p>ARI-3531 is a selective prolyl endopeptidase inhibitor.</p>
    Fórmula:C15H22BN3O4
    Forma y color:Solid
    Peso molecular:319.16
  • Ipenoxazone

    CAS:
    <p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>
    Fórmula:C22H34N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:358.52
  • MLS000536924

    CAS:
    <p>MLS000536924 is a potent and selective competitive human epithelial 15-lipoxygenase-2 inhibitor.</p>
    Fórmula:C16H15N3S
    Forma y color:Solid
    Peso molecular:281.38
  • MMV-667492

    CAS:
    <p>MMV-667492 is an effective inhibitor of Ezrin.</p>
    Fórmula:C17H19N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:313.35
  • L-651392

    CAS:
    <p>L-651392 is an inhibitor of leukotriene.</p>
    Fórmula:C14H10BrNO3S
    Forma y color:Solid
    Peso molecular:352.2
  • L 30

    CAS:
    <p>L 30 is a blocker of the sodium channel.</p>
    Fórmula:C15H24N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:248.36
  • 4-Acetylsimvastatin

    CAS:
    <p>4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).</p>
    Fórmula:C27H40O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:460.6
  • PMPMEase-IN L-28

    CAS:
    <p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>
    Fórmula:C17H29FO2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:348.54
  • BFE-37

    CAS:
    <p>BFE-37 is a partial agonist of beta-adrenergic.</p>
    Fórmula:C16H23NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:277.36
  • Maxacalcitol

    CAS:
    <p>Maxacalcitol (22-Oxacalcitriol) is a ligand of VDR-like receptors and a non-serum calcium vitamin D3 analogue.</p>
    Fórmula:C26H42O4
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:418.61
  • 6-Hydroxyluteolin

    CAS:
    <p>6-Hydroxyluteolin, a flavonoid compound extracted from Salvia amarissima Ortega, inhibits aldose reductase (AR) and has antimicrobial activity.</p>
    Fórmula:C15H10O7
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:302.24
  • Senazodan hydrochloride

    CAS:
    <p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>
    Fórmula:C15H15ClN4O
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:302.76
  • IDO-IN-11

    CAS:
    <p>IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).</p>
    Fórmula:C19H23BrFN7O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:544.4
  • BKIDC-1553

    CAS:
    <p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>
    Fórmula:C22H23N5O2
    Forma y color:Solid
    Peso molecular:389.45
  • (E/Z)-Ensifentrine

    CAS:
    <p>RPL-554 (LS-193,855) is a dual PDE3/4 inhibitor with bronchodilator and anti-inflammatory properties, in trials for asthma and hay fever by Verona Pharma.</p>
    Fórmula:C26H31N5O4
    Forma y color:Solid
    Peso molecular:477.56
  • AMP-Deoxynojirimycin

    CAS:
    <p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>
    Fórmula:C22H39NO5
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:397.55
  • Epostane

    CAS:
    <p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>
    Fórmula:C22H31NO3
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:357.49
  • SHP2-IN-5

    CAS:
    <p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>
    Fórmula:C12H8O6
    Forma y color:Solid
    Peso molecular:248.19
  • JTP 103237

    CAS:
    <p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>
    Fórmula:C24H29F3N6O
    Forma y color:Solid
    Peso molecular:474.52
  • IDO-IN-12

    CAS:
    <p>IDO-IN-12 is an inhibitor of indoleamine 2,3-dioxygenase (IDO).</p>
    Fórmula:C13H11BrFN5O3S
    Pureza:99.727%
    Forma y color:Solid
    Peso molecular:416.23
  • α-Glucosidase-IN-6

    CAS:
    <p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>
    Fórmula:C24H17ClF3NO3S
    Forma y color:Solid
    Peso molecular:491.91
  • Endothelial lipase inhibitor-1

    CAS:
    <p>Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.</p>
    Fórmula:C22H22N4O4
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:406.43
  • Deltasonamide 2

    CAS:
    <p>Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>
    Fórmula:C30H39ClN6O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:647.25
  • THPP-4

    CAS:
    <p>THPP-4 inhibits phosphodiesterase 10A (PDE10A).</p>
    Fórmula:C20H21ClN6O2
    Forma y color:Solid
    Peso molecular:412.87
  • hCAI/II-IN-4

    CAS:
    <p>hCAI/II-IN-4 inhibits hCA I &amp; II (Ki: 16.95 &amp; 15.22 nM), hCA IX (Ki: 27.04 nM), has anti-hypoxia benefits and is low-toxic for AMS research.</p>
    Fórmula:C15H15N3O5S2
    Forma y color:Solid
    Peso molecular:381.43
  • CaV1.3 antagonist-1

    CAS:
    <p>CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.</p>
    Fórmula:C17H19ClN2O3
    Forma y color:Solid
    Peso molecular:334.8
  • STL1267

    CAS:
    <p>STL1267 is a REV-ERB agonist that crosses the blood-brain barrier and inhibits BMAL1 gene expression.</p>
    Fórmula:C17H11ClN4O
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:322.75
  • PF-04279405

    CAS:
    <p>PF-04279405 is a potent and selective glucokinase activator.</p>
    Fórmula:C25H25FN4O4
    Forma y color:Solid
    Peso molecular:464.49
  • AMPD2 inhibitor 1

    CAS:
    AMPD2 inhibitor 1 is an adenosine monophosphate deaminase 2 (AMPD2) inhibitor, useful for studying anorexia in the nervous system.
    Fórmula:C25H22N2O2
    Forma y color:Solid
    Peso molecular:382.45
  • Thialysine HCl

    CAS:
    <p>Thialysine HCl is a cytotoxic cysteine derivative that inhibits Escherichia coli, acting as a protein synthesis inhibitor and metabolite.</p>
    Fórmula:C5H13ClN2O2S
    Forma y color:Solid
    Peso molecular:200.69
  • BI-L 357

    CAS:
    <p>BI-L 357, a prodrug of BL-L 226, is a selective, orally active inhibitor of 5-lipoxygenase.</p>
    Fórmula:C18H18O4S
    Forma y color:Solid
    Peso molecular:330.4
  • TM6089

    CAS:
    <p>TM6089 is an inhibitor of Prolyl Hydroxylase that stimulates HIF activity without iron chelation, induces angiogenesis, and protects organ against ischemia.</p>
    Fórmula:C13H14N4O3S
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:306.34
  • SGK1-IN-1

    CAS:
    <p>SGK1-IN-1 (compound 14n) is a highly potent SGK1 (Serum/Glucocorticoid Regulated Kinase 1) inhibitor</p>
    Fórmula:C17H12ClFN6O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:418.83
  • SSI-4

    CAS:
    <p>SSI-4 is a Stearoyl CoA desaturase 1 (SCD1) inhibitor that can be labeled with carbon-11 (11C) for use as a ligand in small animal in vivo PET/CT imaging</p>
    Fórmula:C19H21ClN4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:388.85
  • Erythronic acid

    CAS:
    <p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>
    Fórmula:C4H8O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:136.1
  • hCA I-IN-2

    CAS:
    <p>hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).</p>
    Fórmula:C26H20BrN5O3S
    Forma y color:Solid
    Peso molecular:562.44
  • IACS-8968

    CAS:
    <p>IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Fórmula:C17H18F3N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.35
  • PGMI-004A

    CAS:
    <p>PGMI-004A is an effective inhibitor of phosphoglycerate mutase 1 (IC50: 13.1 μM).</p>
    Fórmula:C21H12F3NO6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:463.38
  • Kojibiose

    CAS:
    <p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>
    Fórmula:C12H22O11
    Pureza:99.933%
    Forma y color:Solid
    Peso molecular:342.3
  • IDO-IN-3

    CAS:
    <p>IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).</p>
    Fórmula:C11H12BrFN6O2
    Forma y color:Solid
    Peso molecular:359.15
  • Mufemilast

    CAS:
    <p>Mufemilast is an inhibitor of phosphodiesterase 4 (PDE4).</p>
    Fórmula:C20H22N2O7S2
    Forma y color:Solid
    Peso molecular:466.53
  • Dacisteine

    CAS:
    <p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>
    Fórmula:C7H11NO4S
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:205.23
  • (R)-Irsenontrine

    CAS:
    <p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>
    Fórmula:C22H22N4O3
    Forma y color:Solid
    Peso molecular:390.44
  • L-Xylulose

    CAS:
    <p>L-Xylulose: a rare sugar, key in metabolism, α-glucosidase inhibitor, lowers glucose, precursor to antiviral drug components.</p>
    Fórmula:C5H10O5
    Forma y color:Solid
    Peso molecular:150.13
  • IDO1/TDO-IN-2

    CAS:
    <p>IDO1/TDO-IN-2: IDO1/TDO inhibitor; IC50s: IDO1, 0.1μM; TDO, 0.07μM; potential for cancer research.</p>
    Fórmula:C16H9N3O2
    Forma y color:Solid
    Peso molecular:275.26
  • ML299

    CAS:
    <p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>
    Fórmula:C23H26BrFN4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:489.38
  • NCT-506

    CAS:
    <p>NCT-506 is an orally bioavailable inhibitors of aldehyde dehydrogenase 1A1 (ALDH1A1) (IC50 of 7 nM).</p>
    Fórmula:C25H23FN4O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:478.54
  • 2'-O-Methyladenosine

    CAS:
    <p>2'-O-Methyladenosine, a methylated adenine residue is found in the urine of normals and adenosine deaminase deficient patients.</p>
    Fórmula:C11H15N5O4
    Pureza:99.89%
    Forma y color:White Solid
    Peso molecular:281.27
  • Spiraprilat

    CAS:
    <p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>
    Fórmula:C20H26N2O5S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.56
  • ML218

    CAS:
    ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.
    Fórmula:C19H26Cl2N2O
    Pureza:99.2% - 99.45%
    Forma y color:Solid
    Peso molecular:369.33
  • MK-4409

    CAS:
    MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.
    Fórmula:C22H17ClFN3O2S
    Pureza:99.80% - 99.87%
    Forma y color:Solid
    Peso molecular:441.91
  • S07-2010

    CAS:
    <p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>
    Fórmula:C19H21N3O3S
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:371.45
  • Imazodan

    CAS:
    <p>Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.</p>
    Fórmula:C13H12N4O
    Pureza:98% - 98.31%
    Forma y color:Solid
    Peso molecular:240.26
  • Valibose

    CAS:
    <p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>
    Fórmula:C10H21NO6
    Forma y color:Solid
    Peso molecular:251.28
  • CAY10486

    CAS:
    <p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>
    Fórmula:C19H19NO4
    Forma y color:Solid
    Peso molecular:325.36
  • SCH-351591

    CAS:
    <p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>
    Fórmula:C17H10Cl2F3N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:432.18
  • ASP3662

    CAS:
    <p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>
    Fórmula:C19H16ClF3N4O2
    Forma y color:Solid
    Peso molecular:424.8
  • Trandolaprilate hydrate

    CAS:
    <p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>
    Fórmula:C22H32N2O6
    Forma y color:Solid
    Peso molecular:420.5
  • YCT529 free acid

    CAS:
    <p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>
    Fórmula:C29H25NO3
    Forma y color:Solid
    Peso molecular:435.51
  • SCD1 Inhibitor

    CAS:
    <p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>
    Fórmula:C21H20F3N3O3
    Forma y color:Solid
    Peso molecular:419.4
  • 14-dehydro Zymostenol

    CAS:
    <p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>
    Fórmula:C27H44O
    Forma y color:Solid
    Peso molecular:384.64
  • GlcN-6-P Synthase-IN-1

    CAS:
    <p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase &amp; CYP3A4. Has antimicrobial activity and CNS penetration.'</p>
    Fórmula:C20H21N7S
    Forma y color:Solid
    Peso molecular:391.49
  • DNJNAc

    CAS:
    <p>DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.</p>
    Fórmula:C8H16N2O4
    Pureza:98.65% - 99.37%
    Forma y color:Solid
    Peso molecular:204.22
  • 1-Methyluric acid

    CAS:
    <p>1-Methyluric acid (1-Methylurate) acts on the bladder mucosa and increases the levels of insulin, triglycerides, cholesterol, and blood glucose.</p>
    Fórmula:C6H6N4O3
    Pureza:98.05%
    Forma y color:Solid
    Peso molecular:182.14
  • MK-0952

    CAS:
    <p>MK-0952 treats memory loss and cognitive issues; it's a potent, selective PDE4 inhibitor with restricted blood activity.</p>
    Fórmula:C28H22FN3O4
    Forma y color:Solid
    Peso molecular:483.49
  • 3-Oxo-hop-22(29)-ene

    CAS:
    <p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>
    Fórmula:C30H48O
    Forma y color:Solid
    Peso molecular:424.7
  • LEO 39652

    CAS:
    <p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>
    Fórmula:C23H23N3O5
    Forma y color:Solid
    Peso molecular:421.45
  • Tyrphostin AG 1112

    CAS:
    <p>Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.</p>
    Fórmula:C15H10N6
    Forma y color:Solid
    Peso molecular:274.28
  • URB-694

    CAS:
    <p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Fórmula:C19H21NO3
    Forma y color:Solid
    Peso molecular:311.37
  • Nitrefazole

    CAS:
    <p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>
    Fórmula:C10H8N4O4
    Forma y color:Solid
    Peso molecular:248.19
  • DTP348

    CAS:
    <p>DTP348: Oral carbonic anhydrase IX inhibitor &amp; hypoxic cell radiosensitizer with sulfamide &amp; 5-nitroimidazole components.</p>
    Fórmula:C6H11N5O4S
    Forma y color:Solid
    Peso molecular:249.25
  • Oxythiamine diphosphate

    CAS:
    <p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>
    Fórmula:C12H17N3O8P2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:425.29
  • CM39

    CAS:
    <p>CM39 inhibits ALDH, linked to cancer stem-like cells &amp; chemoresistance.</p>
    Fórmula:C19H15FN4OS
    Forma y color:Solid
    Peso molecular:366.41
  • IDO1-IN-17

    CAS:
    <p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>
    Fórmula:C28H32BrClFN5O2
    Forma y color:Solid
    Peso molecular:604.94
  • Carbonic anhydrase inhibitor 13

    CAS:
    <p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>
    Fórmula:C17H15N5O3S2
    Forma y color:Solid
    Peso molecular:401.46
  • hCAIX-IN-6

    CAS:
    <p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>
    Fórmula:C18H12N2O4S
    Forma y color:Solid
    Peso molecular:352.36
  • UK-414,495

    CAS:
    <p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>
    Fórmula:C16H25N3O3S
    Forma y color:Solid
    Peso molecular:339.45
  • mIDH1-IN-1

    CAS:
    <p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>
    Fórmula:C25H27N3O5
    Forma y color:Solid
    Peso molecular:449.5
  • Enpp-1-IN-5

    CAS:
    <p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>
    Fórmula:C17H26N6O4S
    Forma y color:Solid
    Peso molecular:410.49
  • Oxagrelate

    CAS:
    <p>Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.</p>
    Fórmula:C14H16N2O4
    Forma y color:Solid
    Peso molecular:276.29
  • PDE5-IN-4

    CAS:
    <p>PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,</p>
    Fórmula:C21H27N5O5S
    Forma y color:Solid
    Peso molecular:461.53
  • Boc-Glu(OBzl)-OSu

    CAS:
    <p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>
    Fórmula:C21H26N2O8
    Forma y color:Solid
    Peso molecular:434.44
  • α-Amylase/α-Glucosidase-IN-2

    CAS:
    α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM
    Fórmula:C22H16ClN5
    Forma y color:Solid
    Peso molecular:385.85
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Fórmula:C20H21N3O
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:319.4
  • Spirapril

    CAS:
    <p>Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.</p>
    Fórmula:C22H30N2O5S2
    Forma y color:Solid
    Peso molecular:466.61
  • Enpp-1-IN-6

    CAS:
    <p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>
    Fórmula:C22H28N4O5S
    Forma y color:Solid
    Peso molecular:460.55
  • Teglarinad chloride

    CAS:
    <p>Teglarinad chloride (GMX-1777 chloride) is an inhibitor of NAMPT with antitumor activity that acts by interfering with DNA repair and inhibiting angiogenesis.</p>
    Fórmula:C30H43Cl2N5O8
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:672.6
  • mEH-IN-1

    CAS:
    <p>mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.</p>
    Fórmula:C16H17F6NOS
    Forma y color:Solid
    Peso molecular:385.37
  • SYN20028567

    CAS:
    <p>SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].</p>
    Fórmula:C20H29N3O3S
    Forma y color:Solid
    Peso molecular:391.53
  • Agn 190727

    CAS:
    <p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>
    Fórmula:C20H22O2
    Forma y color:Solid
    Peso molecular:294.39
  • α-Glycosidase-IN-1

    CAS:
    <p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>
    Fórmula:C21H19N9O6S2
    Forma y color:Solid
    Peso molecular:557.56
  • Glucosylceramide synthase-IN-1

    CAS:
    <p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>
    Fórmula:C24H20F4N2O3
    Forma y color:Solid
    Peso molecular:460.42
  • DHODH-IN-21

    CAS:
    <p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>
    Fórmula:C20H19ClF4N6O4
    Forma y color:Solid
    Peso molecular:518.85
  • SQ 28853

    CAS:
    <p>SQ 28853 is an inhibitor of ACE with diuretic properties.</p>
    Fórmula:C19H25ClN4NaO6S3
    Forma y color:Solid
    Peso molecular:560.05
  • Y-29794

    CAS:
    <p>Y-29794, a covalent POP inhibitor with a Ki of 0.95 nM, holds research potential for neurodegenerative diseases and cancer.</p>
    Fórmula:C22H32N2OS2
    Forma y color:Solid
    Peso molecular:404.63
  • Allopurinol riboside

    CAS:
    <p>Allopurinol riboside, an allopurinol metabolite, inhibits purine nucleoside phosphorylase in parasites with a Ki of 277 μM.</p>
    Fórmula:C10H12N4O5
    Pureza:99.46% - 99.73%
    Forma y color:Solid
    Peso molecular:268.23