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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8628 productos de "Metabolismo"

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  • Glyco-Obeticholic acid

    CAS:
    <p>Glyco-Obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is an agonist of the farnesoid X receptor (FXR).</p>
    Fórmula:C28H47NO5
    Pureza:99.77% - 99.95%
    Forma y color:Solid
    Peso molecular:477.68
  • Isomazole hydrochloride

    CAS:
    <p>Isomazole hydrochloride is a cardiotonic.</p>
    Fórmula:C14H14ClN3O2S
    Forma y color:Solid
    Peso molecular:323.8
  • Tryptophan, N-indol-3-ylacetyl- (6CI)

    CAS:
    <p>Tryptophan, N-indol-3-ylacetyl- (6CI) (Indole-3-acetyl-L-tryptophan) is involved in regulatory mechanisms for the control of auxin activity during physiological</p>
    Fórmula:C21H19N3O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:361.4
  • SR8278

    CAS:
    <p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>
    Fórmula:C18H19NO3S2
    Pureza:99.44% - 99.73%
    Forma y color:Solid
    Peso molecular:361.48
  • ASP-9521

    CAS:
    <p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>
    Fórmula:C19H26N2O3
    Pureza:95.11% - 96.96%
    Forma y color:Solid
    Peso molecular:330.42
  • Propiverine hydrochloride

    CAS:
    <p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>
    Fórmula:C23H30ClNO3
    Pureza:99.93%
    Forma y color:White Crystalling Power
    Peso molecular:403.94
  • CM10

    CAS:
    <p>CM10 is an aldehyde dehydrogenase 1A family(ALDH1A) inhibitor.</p>
    Fórmula:C20H23N3O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:321.42
  • Imidazole-5-propionic acid

    CAS:
    <p>Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination.</p>
    Fórmula:C6H8N2O2
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:140.14
  • Sacubitril hemicalcium salt

    CAS:
    <p>Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.</p>
    Fórmula:C48H56CaN2O10
    Pureza:99.86% - 99.93%
    Forma y color:Solid
    Peso molecular:861.06
  • Hydroxy Dimetridazole

    CAS:
    <p>Hydroxy Dimetridazole is a hydroxy metabolite of Dimetridazole which combats protozoan infections.</p>
    Fórmula:C5H7N3O3
    Pureza:99.83% - 99.85%
    Forma y color:Solid
    Peso molecular:157.13
  • Ziritaxestat

    CAS:
    <p>Ziritaxestat (GLPG1690), an autotaxin inhibitor, currently being evaluated in an exploratory phase 2 study in idiopathic pulmonary fibrosis patients.</p>
    Fórmula:C30H33FN8O2S
    Pureza:97% - 99.85%
    Forma y color:Solid
    Peso molecular:588.7
  • Captopril hydrochloride

    CAS:
    <p>Captopril hydrochloride: an oral ACE inhibitor (IC50: 0.025 μM), treats hypertension/heart failure, and blocks NDM-1 (IC50: 7.9 μM).</p>
    Fórmula:C9H16ClNO3S
    Forma y color:Solid
    Peso molecular:253.74
  • Dichlorphenamide

    CAS:
    <p>Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma.</p>
    Fórmula:C6H6Cl2N2O4S2
    Pureza:96.87% - 97.25%
    Forma y color:Needles From Dimethylsulfoxide + Water Solid
    Peso molecular:305.16
  • Cilostamide

    CAS:
    <p>Cilostamide (OPC3689) is a selective phosphodiesterase (PDE)3A and PDE3B inhibitor(IC50 values of 27 and 50 nM, respectively)</p>
    Fórmula:C20H26N2O3
    Pureza:98.87%
    Forma y color:White To Off-White Solid
    Peso molecular:342.43
  • Isradipine

    CAS:
    <p>Isradipine (PN 200-110), a dihydropyridine, is an antihypertensive calcium channel blocker that dilates arteries and reduces resistance.</p>
    Fórmula:C19H21N3O5
    Pureza:99.84% - 99.95%
    Forma y color:Yellow Solid
    Peso molecular:371.39
  • D-Pantothenic acid

    CAS:
    <p>D-Pantothenic acid (B5): water-soluble, antioxidant, in all living tissues, part of CoA &amp; B2 complex, needed for metabolism &amp; synthesizing cholesterol, etc.</p>
    Fórmula:C9H17NO5
    Pureza:99.85% - 99.92%
    Forma y color:Yellow Viscous Oil Solid
    Peso molecular:219.24
  • CP671305

    CAS:
    <p>CP671305 is an orally active, potent and selective inhibitor of phosphodiesterase-4-D.</p>
    Fórmula:C23H19FN2O7
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:454.4
  • (L)-Canavanine

    CAS:
    <p>(L)-Canavanine is antimutagenic activity.</p>
    Fórmula:C5H12N4O3
    Forma y color:Solid
    Peso molecular:176.17
  • β-Aminopropionitrile hydrochloride

    CAS:
    <p>β-Aminopropionitrile hydrochloride is a selective, oral, irreversible inhibitor of lysyl oxidase (LOX) that reduces metastatic seeding potential.</p>
    Fórmula:C3H7ClN2
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:106.55
  • Mibefradil dihydrochloride

    CAS:
    <p>Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type</p>
    Fórmula:C29H40Cl2FN3O3
    Pureza:99.45% - 99.72%
    Forma y color:Solid
    Peso molecular:568.55
  • 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine

    CAS:
    1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite that has been found in the aging mouse brain.
    Fórmula:C46H84NO8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:810.13
  • 1-Cyclohexyl-3-dodecyl urea

    CAS:
    1-Cyclohexyl-3-dodecyl urea (NCND) is a highly selective soluble epoxide hydrolase (sEH) inhibitor.
    Fórmula:C19H38N2O
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:310.52
  • 1,2-Dilauroyl-sn-glycerol

    CAS:
    <p>1,2-Dilauroyl-sn-glycerol ((S)-1,2-Dilaurin) is primarily composed of the interaction of 1,2-dilauroyl-sn-glycerol (1,2-DLG) with phosphatidylcholine (PC)</p>
    Fórmula:C27H52O5
    Pureza:99.93% - 99.95%
    Forma y color:Solid
    Peso molecular:456.7
  • 4-(benzyloxy)benzene-1-sulfonamide

    CAS:
    <p>4-(benzyloxy)benzene-1-sulfonamide is inhibitor of human recombinant CA-7.</p>
    Fórmula:C13H13NO3S
    Pureza:97.54%
    Forma y color:Solid
    Peso molecular:263.31
  • S29434

    CAS:
    <p>S29434 (NMDPEF) is a potent, competitiveinhibitor of quinone reductase 2 (QR2;IC50:5-16nM).</p>
    Fórmula:C21H18N4O3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:374.39
  • KY-226

    CAS:
    <p>KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,)</p>
    Fórmula:C27H31NO3S2
    Pureza:99.4%
    Forma y color:Solid
    Peso molecular:481.67
  • ABT-639

    CAS:
    <p>ABT-639 is a potent and selective T-type calcium channel blocker.</p>
    Fórmula:C20H20ClF2N3O3S
    Pureza:99.12% - 99.77%
    Forma y color:Solid
    Peso molecular:455.91
  • WWL70

    CAS:
    <p>WWL70 is a selective alpha/beta hydrolase domain 6 inhibitors (IC50: 70 nM).</p>
    Fórmula:C27H23N3O3
    Pureza:98.38% - 98.53%
    Forma y color:Solid
    Peso molecular:437.49
  • YM-58483

    CAS:
    <p>YM-58483 (BTP2) is a specific and effective inhibitor of CRAC channels and subsequent Ca2+ signals.</p>
    Fórmula:C15H9F6N5OS
    Pureza:99.33% - 99.64%
    Forma y color:Solid
    Peso molecular:421.32
  • Tuna AI acetate


    <p>Tuna AI acetate is an inhibitor of angiotensin-converting enzyme (ACE) in non-competitive manner derived from tuna muscle.</p>
    Fórmula:C46H68N12O14
    Pureza:98.49%
    Forma y color:Solid
    Peso molecular:1013.1
  • VAS2870

    CAS:
    VAS2870 is an inhibitor of NADPH oxidase (NOX).
    Fórmula:C18H12N6OS
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:360.39
  • Oroxylin A

    CAS:
    <p>Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion and enhances leukemia treatment.</p>
    Fórmula:C16H12O5
    Pureza:98.72% - 99.55%
    Forma y color:Solid
    Peso molecular:284.26
  • Biocytin

    CAS:
    <p>Biocytin, a D-biotin and L-lysine conjugate, maps brain connections via a secondary amide bond.</p>
    Fórmula:C16H28N4O4S
    Pureza:97.23%
    Forma y color:White Solid
    Peso molecular:372.48
  • Panaxadiol

    CAS:
    <p>Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng.</p>
    Fórmula:C30H52O3
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:460.73
  • Mitochondrial fusion promoter M1

    CAS:
    Mitochondrial fusion promoter M1, a modulator of mitochondrial dynamics, enhances mitochondrial function and cellular respiration, and has shown efficacy in
    Fórmula:C14H10Cl4N2O
    Pureza:99.54% - 99.54%
    Forma y color:Solid
    Peso molecular:364.05
  • Darexaban

    CAS:
    <p>Darexaban (YM-150) selectively inhibits Factor Xa, reducing clotting and risk of heart/stroke events.</p>
    Fórmula:C27H30N4O4
    Pureza:98.33%
    Forma y color:Solid
    Peso molecular:474.55
  • Carbobenzoxyphenylalanine

    CAS:
    <p>Carbobenzoxyphenylalanine (NSC-402059) is a thermolysin inhibitor.</p>
    Fórmula:C17H17NO4
    Pureza:99.71%
    Forma y color:White Amorphous Powder
    Peso molecular:299.32
  • Azumolene

    CAS:
    Azumolene (EU4093 free base)
    Fórmula:C13H9BrN4O3
    Pureza:98.1% - 98.35%
    Forma y color:Solid
    Peso molecular:349.14
  • BIM-46187 4HCl

    CAS:
    <p>BIM-46187 4HCl (PH-064 4HCl) is a heterotrimeric G-protein complex inhibitor.</p>
    Fórmula:C44H62Cl4N8O2S2
    Pureza:99.26% - 99.63%
    Forma y color:Solid
    Peso molecular:940.95
  • Gcase activator 1

    CAS:
    <p>Gcase activator 1 (LTI-291) is a glucocerebrosidase (Gcase) activator.</p>
    Fórmula:C20H30N4O2
    Pureza:99.25% - 99.31%
    Forma y color:Solid
    Peso molecular:358.48
  • Ponalrestat

    CAS:
    <p>Ponalrestat is an aldose reductase inhibitor.</p>
    Fórmula:C17H12BrFN2O3
    Pureza:97.34% - 99.86%
    Forma y color:Solid
    Peso molecular:391.19
  • Dimethyl DL-Glutamate (hydrochloride)

    CAS:
    <p>Dimethyl DL-glutamate boosts insulin release in response to glucose.</p>
    Fórmula:C7H14ClNO4
    Pureza:≥95%
    Forma y color:Solid
    Peso molecular:211.64
  • Milacemide

    CAS:
    <p>Milacemide is a glycine prodrug and MAO-B inhibitor.</p>
    Fórmula:C7H16N2O
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:144.21
  • Enoxaparin sodium

    CAS:
    <p>Enoxaparin, a low-weight heparin approved by FDA for STEMI, enhances antithrombin and prevents clotting by inhibiting factors XIa, IXa, Xa, IIa.</p>
    Fórmula:C42H59N3Na4O35S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1322
  • EAAT2 activator 1

    CAS:
    <p>EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein</p>
    Fórmula:C16H11ClFN3S
    Pureza:98.86%
    Forma y color:Solid
    Peso molecular:331.8
  • ML-095 hydrochloride

    CAS:
    ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.
    Fórmula:C13H15ClN2O3
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:282.72
  • PF-9601N

    CAS:
    <p>PF-9601N: potent, selective MAO-BI with neuroprotection in PD models.</p>
    Fórmula:C19H18N2O
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:290.36
  • ML351

    CAS:
    <p>ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).</p>
    Fórmula:C15H11N3O
    Pureza:97.67%
    Forma y color:Solid
    Peso molecular:249.27
  • trifarotene

    CAS:
    <p>Trifarotene (CD5789) is a RARγ agonist, 65x more selective than RARα and 16x than RARβ, with EC50 of 7.7 nM.</p>
    Fórmula:C29H33NO4
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:459.58
  • TH5427

    CAS:
    <p>TH5427 is a lead NUDT5 inhibitor(MG assay IC50 = 29 nM).</p>
    Fórmula:C20H20Cl2N8O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:491.33
  • Mirogabalin

    CAS:
    <p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>
    Fórmula:C12H19NO2
    Pureza:98.57%
    Forma y color:Solid
    Peso molecular:209.28
  • ISX-9

    CAS:
    <p>ISX-9 (Isoxazole 9) is necessary to activate neuron-specific genes as neurogenesis inducer.</p>
    Fórmula:C11H10N2O2S
    Pureza:97.81% - ≥95%
    Forma y color:Solid
    Peso molecular:234.27
  • Furafylline

    CAS:
    <p>Furafylline is a selective inhibitor of human cytochrome P450 (CYP)1A2 (IC50 : 0.07 μM),</p>
    Fórmula:C12H12N4O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:260.25
  • Pentamidine dimesylate

    CAS:
    <p>Pentamidine dimesylate blocks (Ca)S100B-p53, aiding p53 activity against melanoma.</p>
    Fórmula:C20H28N4O5S
    Forma y color:Solid
    Peso molecular:436.53
  • THPP-1

    CAS:
    THPP-1 is a potent and orally bioavailable inhibitor of PDE10A(Ki of 1 nM and 1.3 nM for human and rat PDE10A, respectively).
    Fórmula:C23H21ClN6O3
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:464.9
  • L-Leucyl-L-Leucine methyl ester hydrochloride

    CAS:
    <p>L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.</p>
    Fórmula:C13H27ClN2O3
    Pureza:98.41% - 99.63%
    Forma y color:Solid
    Peso molecular:294.81
  • Osoresnontrine

    CAS:
    <p>Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.</p>
    Fórmula:C16H17N5O2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:311.34
  • BMS-309403

    CAS:
    BMS309403 is a potent and selective inhibitor of adipocyte fatty acid binding protein aFABP.Cost-effective and quality-assured.
    Fórmula:C31H26N2O3
    Pureza:99.52% - 99.76%
    Forma y color:Solid
    Peso molecular:474.55
  • ABX-1431

    CAS:
    <p>ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).</p>
    Fórmula:C20H22F9N3O2
    Pureza:99.8% - 99.96%
    Forma y color:Solid
    Peso molecular:507.39
  • (E/Z)-Teriflunomide

    CAS:
    <p>(E/Z)-Teriflunomide (Aubagio), a orally-available Pyrimidine Synthesis Inhibitor, is used to treat relapsing multiple sclerosis.</p>
    Fórmula:C12H9F3N2O2
    Pureza:99.49% - 99.76%
    Forma y color:White Solid
    Peso molecular:270.21
  • HA130

    CAS:
    <p>HA130 is a selective ATX (autotaxin) inhibitor.</p>
    Fórmula:C24H19BFNO5S
    Pureza:98.26% - ≥95%
    Forma y color:Solid
    Peso molecular:463.29
  • Mephenytoin

    CAS:
    <p>Mephenytoin (Phenantoin) is an anticonvulsant and a substrate of CYP2C19 and CYP2B6.</p>
    Fórmula:C12H14N2O2
    Pureza:99.67% - 99.91%
    Forma y color:Crystals Solid
    Peso molecular:218.25
  • Edoxaban hydrochloride

    CAS:
    <p>Edoxaban (DU-176b) HCl: Oral, selective Factor Xa inhibitor, Ki 0.561 nM; prevents thromboembolic disease.</p>
    Fórmula:C24H31Cl2N7O4S
    Forma y color:Solid
    Peso molecular:584.52
  • Nepicastat hydrochloride

    CAS:
    <p>Nepicastat hydrochloride (RS-25560-197 hydrochloride) is a selective, orally active, dopamine-beta-hydroxylase inhibitor that crosses the blood-brain barrier.</p>
    Fórmula:C14H15F2N3S·HCl
    Pureza:98.35% - 99.74%
    Forma y color:Solid
    Peso molecular:331.81
  • TB5

    CAS:
    TB5 is a potent, selective and reversible inhibitor of hMAO-B.
    Fórmula:C15H14BrNOS
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:336.25
  • N-(p-amylcinnamoyl) Anthranilic Acid

    CAS:
    N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.
    Fórmula:C21H23NO3
    Pureza:99.35% - 99.67%
    Forma y color:Solid
    Peso molecular:337.41
  • PDM2

    CAS:
    <p>PDM 2 is a potent and selective aryl hydrocarbon receptor (AhR) antagonist.</p>
    Fórmula:C14H9Cl3
    Pureza:99.44%
    Forma y color:Solid
    Peso molecular:283.58
  • (R)-3-Hydroxy-4,4-dimethyldihydrofuran-2(3H)-one

    CAS:
    <p>Pantolactone belongs to the class of organic compounds known as gamma-butyrolactones. gamma-Butyrolactones are compounds containing a gamma-butyrolactone moiety, which consists of an aliphatic five-member ring with four carbon atoms, one oxygen atom, and </p>
    Fórmula:C6H10O3
    Pureza:99.41%
    Forma y color:White Crystalline Powder Or Crystals
    Peso molecular:130.14
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:354.38
  • NFAT Inhibitor-2

    CAS:
    <p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>
    Fórmula:C22H20F2N2O4S
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:446.47
  • ML355

    CAS:
    <p>ML355, a specific, effective 12-Lipoxygenase(12-LOX) inhibitors(IC50=0.34 μM), possess favorable ADME properties.</p>
    Fórmula:C21H19N3O4S2
    Pureza:98.02% - 98.2%
    Forma y color:Solid
    Peso molecular:441.52
  • Fomepizole

    CAS:
    <p>Fomepizole (4-Methylpyrazole), a competitive inhibitor of alcohol dehydrogenase, is used as an antidote in methanol or ethylene glycol poisoning.</p>
    Fórmula:C4H6N2
    Pureza:98.1% - 99.94%
    Forma y color:Yellow <13°C Solid >13°C Liquid
    Peso molecular:82.1
  • MPO-IN-28

    CAS:
    <p>MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.</p>
    Fórmula:C11H13N5O
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:231.25
  • Barnidipine hydrochloride

    CAS:
    <p>Barnidipine HCl is a potent dihydropyridine Ca²⁺ blocker with 0.35 nM IC50 in pig coronary artery.</p>
    Fórmula:C27H30ClN3O6
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:528
  • Tienilic Acid

    CAS:
    <p>Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity</p>
    Fórmula:C13H8Cl2O4S
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:331.17
  • Inosine

    CAS:
    Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!
    Fórmula:C10H12N4O5
    Pureza:99.51% - 99.89%
    Forma y color:Solid
    Peso molecular:268.23
  • LY195448 HCl

    CAS:
    <p>LY195448 HCl is a phenethanolamine shown anti-tumour activity. It blocks cells at metaphase.</p>
    Fórmula:C20H27ClN2O2
    Forma y color:Solid
    Peso molecular:362.89
  • BPTES

    CAS:
    <p>BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.</p>
    Fórmula:C24H24N6O2S3
    Pureza:95.83% - 99.64%
    Forma y color:Solid
    Peso molecular:524.68
  • TEPP-46

    CAS:
    <p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C17H16N4O2S2
    Pureza:98.21% - 98.77%
    Forma y color:Solid
    Peso molecular:372.46
  • 3-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one

    CAS:
    <p>DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 nM, respectively)</p>
    Fórmula:C18H13NO
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:259.3
  • Tarenflurbil

    CAS:
    <p>Tarenflurbil, the R-enantiomer of flurbiprofen, lacks COX inhibition and was tested for Alzheimer's treatment.</p>
    Fórmula:C15H13FO2
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:244.26
  • RS-25344

    CAS:
    <p>RS-25344: a strong PDE4 blocker, curbs eosinophil movement, boosts sperm motility in vitro.</p>
    Fórmula:C19H13N5O4
    Pureza:98.98%
    Forma y color:Solid
    Peso molecular:375.34
  • CP-640186

    CAS:
    <p>CP-640186 is an isozyme-nonselective ACCase inhibitor. The IC50s of CP-640186 is 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively.</p>
    Fórmula:C30H35N3O3
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:485.62
  • Bepridil hydrochloride

    CAS:
    <p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>
    Fórmula:C24H35ClN2O
    Pureza:99.45% - 99.68%
    Forma y color:Solid
    Peso molecular:403
  • R162

    CAS:
    <p>R162 is an effective glutamate dehydrogenase 1 (GDH1) inhibitor.</p>
    Fórmula:C17H12O3
    Pureza:96.21% - 98.15%
    Forma y color:Solid
    Peso molecular:264.28
  • 2′-Deoxyadenosine 5′-monophosphate disodium

    CAS:
    <p>2′-Deoxyadenosine 5′-monophosphate disodium, a nucleic acid AMP derivative, is a deoxyribonucleotide present in DNA.</p>
    Fórmula:C10H14N5Na2O6P
    Pureza:98.96%
    Forma y color:Solid
    Peso molecular:377.2
  • p-Fluoro-L-phenylalanine

    CAS:
    <p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>
    Fórmula:C9H10FNO2
    Pureza:99.63%
    Forma y color:White To Off-White Powder
    Peso molecular:183.18
  • THP104c

    CAS:
    <p>THP104c is an inhibitor of mitochondrial fission.</p>
    Fórmula:C20H16N4O2S
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:376.43
  • N-Boc-O-tosyl hydroxylamine

    CAS:
    <p>N-Boc-O-tosyl hydroxylamine is nitrogen source for the N-amination of aryl and alkyl amines.</p>
    Fórmula:C12H17NO5S
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:287.33
  • Tropifexor

    CAS:
    <p>Tropifexor (LJN452) is a novel and highly potent agonist of FXR with an EC50 of 0.2 nM.</p>
    Fórmula:C29H25F4N3O5S
    Pureza:99.3% - 99.85%
    Forma y color:Solid
    Peso molecular:603.58
  • Dalcetrapib

    CAS:
    <p>Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol.</p>
    Fórmula:C23H35NO2S
    Pureza:97.98% - >99.99%
    Forma y color:Solid
    Peso molecular:389.59
  • WIN 18446

    CAS:
    <p>inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)</p>
    Fórmula:C12H20Cl4N2O2
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:366.11
  • AZ876

    CAS:
    <p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>
    Fórmula:C24H29N3O3S
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:439.57
  • Indoximod

    CAS:
    <p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>
    Fórmula:C12H14N2O2
    Pureza:97.82% - 99.55%
    Forma y color:Solid
    Peso molecular:218.25
  • 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

    CAS:
    <p>4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-</p>
    Fórmula:C7H8F3N3O4S2
    Pureza:98.58%
    Forma y color:Solid
    Peso molecular:319.28
  • UK-5099

    CAS:
    <p>UK-5099 (PF-1005023) is a potent MPC inhibitor with an IC50 of 50 nM in rat heart mitochondria.</p>
    Fórmula:C18H12N2O2
    Pureza:97.39% - >99.99%
    Forma y color:Solid
    Peso molecular:288.3
  • SR3335

    CAS:
    <p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>
    Fórmula:C13H9F6NO3S2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:405.34
  • HSL-IN-3

    CAS:
    <p>HSL-IN-3 (HSL inhibitor 3) is a boronic acid derivative that is an inhibitor of hormone-sensitive lipase(HSL).</p>
    Fórmula:C14H19BO4
    Pureza:99.402%
    Forma y color:Solid
    Peso molecular:262.11
  • Des(benzylpyridyl) Atazanavi

    CAS:
    <p>The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.</p>
    Fórmula:C26H43N5O7
    Pureza:98% - 99.75%
    Forma y color:Solid
    Peso molecular:537.65
  • BAY-218

    CAS:
    <p>Bindarit (AF2838) is an aryl hydrocarbon receptor (AHR) antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C20H17ClFN3O3
    Pureza:99.46% - 99.85%
    Forma y color:Solid
    Peso molecular:401.82
  • Tuftsin 3TFA

    CAS:
    <p>Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.</p>
    Fórmula:C27H43F9N8O12
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:842.66
  • YM-750

    CAS:
    <p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>
    Fórmula:C31H36N2O
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:452.63
  • Bifemelane hydrochloride

    CAS:
    <p>Bifemelane hydrochloride is a MAO inhibitor</p>
    Fórmula:C18H23NO·HCl
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:305.84
  • SC-57461A

    CAS:
    <p>SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor.</p>
    Fórmula:C20H26ClNO3
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:363.9
  • PHGDH-inactive

    CAS:
    <p>PHGDH inactive is inactive against PHGDH and serves as a negative control for NCT-502 and NCT-503 [1].</p>
    Fórmula:C17H21N5S
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:327.45
  • L-Homocystine

    CAS:
    <p>Homocystine briefly forms before turning into cystathionine via vitamin B6; linked to schizophrenia and neural tube defects; folic acid lowers risk.</p>
    Fórmula:C8H16N2O4S2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:268.35
  • Cytidine 5'-diphosphate disodium

    CAS:
    Cytidine 5'-diphosphate disodium (CDP sodium salt) produces CTP to support DNA and RNA biosynthesis and ribonucleotide reductase to produce dCMP.
    Fórmula:C9H13N3Na2O11P2
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:447.14
  • 4-Nonylphenylboronic acid

    CAS:
    <p>4-Nonylphenylboronic acid is a inhibitor of FAAH.</p>
    Fórmula:C15H25BO2
    Pureza:97.63%
    Forma y color:Solid
    Peso molecular:248.17
  • YM976

    CAS:
    YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)
    Fórmula:C17H16ClN3O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:313.78
  • LXR-623

    CAS:
    <p>LXR-623 (WAY 252623) is an orally bioavailable and highly specifical synthetic modulator of LXR.</p>
    Fórmula:C21H12ClF5N2
    Pureza:97.91% - 99.24%
    Forma y color:Solid
    Peso molecular:422.78
  • CD437

    CAS:
    <p>CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.</p>
    Fórmula:C27H26O3
    Pureza:98.92% - 99.63%
    Forma y color:Solid
    Peso molecular:398.49
  • Neomangiferin

    CAS:
    Neomangiferin combats fatty liver in rats and inhibits an enzyme linked to bone loss.
    Fórmula:C25H28O16
    Pureza:99.41% - 99.83%
    Forma y color:Solid
    Peso molecular:584.48
  • RHC 80267

    CAS:
    <p>RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)</p>
    Fórmula:C20H34N4O4
    Pureza:99.54%
    Forma y color:White Solid
    Peso molecular:394.51
  • BMS-779788

    CAS:
    <p>BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).</p>
    Fórmula:C28H29ClN2O3S
    Pureza:98.65% - 99.24%
    Forma y color:Solid
    Peso molecular:509.06
  • Enoximone

    CAS:
    <p>Enoximone is a selective inhibitor of phosphodiesterase III (PDE3), with treatment of congestive heart failure.</p>
    Fórmula:C12H12N2O2S
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:248.3
  • Ensifentrine

    CAS:
    <p>Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3(IC50: 0.4 nM) is 3,440 times higher than that for PDE4(IC50: 1479 nM), that</p>
    Fórmula:C26H31N5O4
    Pureza:99.76% - 99.94%
    Forma y color:Solid
    Peso molecular:477.56
  • Clinofibrate

    CAS:
    <p>Clinofibrate lowers lipids, blocks HMGCR (IC50: 0.47 mM), and controls cholesterol/triacylglycerides.</p>
    Fórmula:C28H36O6
    Pureza:>99.99%
    Forma y color:White Crystalline Powder
    Peso molecular:468.58
  • Adamantanine

    CAS:
    <p>Adamantanine (NSC-145160) is an amino acid transport inhibitor.</p>
    Fórmula:C11H17NO2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:195.26
  • GW3965 hydrochloride

    CAS:
    <p>GW3965 hydrochloride (GW3965 HCl) is an effective and specific LXR agonist for hLXRα/β (EC50: 190/30 nM).</p>
    Fórmula:C33H31ClF3NO3·HCl
    Pureza:98.9% - 99.51%
    Forma y color:Solid
    Peso molecular:618.51
  • A 922500

    CAS:
    <p>A 922500 (DGAT-1 Inhibitor 4a) is an inhibitor for human and mouse DGAT-1, good selectivity over related acyltransferases, hERG, and a panel of anti-targets.</p>
    Fórmula:C26H24N2O4
    Pureza:97.34% - 97.66%
    Forma y color:Solid
    Peso molecular:428.48
  • Torcetrapib

    CAS:
    <p>Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.</p>
    Fórmula:C26H25F9N2O4
    Pureza:98% - 99.59%
    Forma y color:Lipid
    Peso molecular:600.47
  • trans-4-Hydroxycyclohexanecarboxylic Acid

    CAS:
    <p>trans-4-Hydroxycyclohexanecarboxylic Acid is an organic intermediate.</p>
    Fórmula:C7H12O3
    Pureza:96.24%
    Forma y color:Solid
    Peso molecular:144.17
  • Verdiperstat

    CAS:
    Verdiperstat (AZD 3241) is a selective, irreversible, orally active myeloperoxidase inhibitor for neurodegenerative brain diseases.
    Fórmula:C11H15N3O2S
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:253.32
  • Eprobemide

    CAS:
    <p>Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).</p>
    Fórmula:C14H19ClN2O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:282.77
  • 8-Azaadenosine

    CAS:
    <p>8-Azaadenosine inhibits ADAR1, blocks RNA editing, and reduces thyroid cancer cell proliferation and spread.</p>
    Fórmula:C9H12N6O4
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:268.23
  • Nifurtimox

    CAS:
    <p>Nifurtimox (BAY-A-2502) is an antiprotozoal agent (IC50s = 9.91, 12.28, and 10.44 μM against Taluahuén, LQ, and Brener strains of T.</p>
    Fórmula:C10H13N3O5S
    Pureza:99.87% - 99.89%
    Forma y color:Solid
    Peso molecular:287.29
  • A939572

    CAS:
    <p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of &lt;4 nM for mSCD1 and 37 nM for hSCD1.</p>
    Fórmula:C20H22ClN3O3
    Pureza:99.96% - ≥95%
    Forma y color:Solid
    Peso molecular:387.86
  • Glycylsarcosine

    CAS:
    <p>Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosine</p>
    Fórmula:C5H10N2O3
    Pureza:98.47%
    Forma y color:Solid
    Peso molecular:146.14
  • CK2-IN-1

    CAS:
    <p>CK2 inhibitor</p>
    Fórmula:C14H9NO3
    Pureza:97.28%
    Forma y color:Solid
    Peso molecular:239.23
  • VY-3-135

    CAS:
    <p>VY-3-135 is an orally active, stable and specific acetyl-CoA synthetase 2 (ACSS2) inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C26H27N3O3
    Pureza:99.25% - 99.79%
    Forma y color:Solid
    Peso molecular:429.51
  • S-(2-Carboxypropyl)cysteine

    CAS:
    <p>S-(2-Carboxypropyl)cysteine is a urinary metabolite of S-(2-Carboxypropyl)glutathione.</p>
    Fórmula:C7H13NO4S
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:207.25
  • Phenidone

    CAS:
    Phenidone inhibits COX/LOX, reducing rat autoimmune paralysis and lowering blood pressure in hypertensive rats.
    Fórmula:C9H10N2O
    Pureza:97.24%
    Forma y color:White Solid Solid Crystalline
    Peso molecular:162.19
  • Betrixaban hydrochloride(330942-05-7(free base))


    <p>Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5</p>
    Fórmula:C23H23Cl2N5O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:488.36
  • Navoximod

    CAS:
    <p>Navoximod (GDC-0919) (NLG- 919, GDC-0919) is a potent indoleamine-(2,3)-dioxygenase (IDO) pathway inhibitor (Ki/EC50: 7 nM/75 nM).</p>
    Fórmula:C18H21FN2O2
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:316.37
  • PF-3845

    CAS:
    <p>PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.</p>
    Fórmula:C24H23F3N4O2
    Pureza:99.54% - 99.58%
    Forma y color:Solid
    Peso molecular:456.46
  • FPL64176

    CAS:
    <p>FPL64176 is a L-type calcium channels activator.</p>
    Fórmula:C22H21NO3
    Pureza:98.68%
    Forma y color:Solid
    Peso molecular:347.41
  • Pyridaben

    CAS:
    <p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>
    Fórmula:C19H25ClN2OS
    Pureza:97.11% - 99.75%
    Forma y color:Solid
    Peso molecular:364.93
  • Tipifarnib (S enantiomer)

    CAS:
    <p>Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).</p>
    Fórmula:C27H22Cl2N4O
    Pureza:99.05%
    Forma y color:Solid
    Peso molecular:489.4
  • AM-2394

    CAS:
    <p>AM-2394 is an effective and specific Glucokinase agonist (GKA, EC50: 60 nM), which catalyzes the phosphorylation of glucose to glucose-6-phosphate.</p>
    Fórmula:C22H25N5O4
    Pureza:99.01% - 99.62%
    Forma y color:Solid
    Peso molecular:423.46
  • 1,2-Didecanoyl-sn-glycero-3-phosphocholi

    CAS:
    <p>1,2-Didecanoyl PC: synthetic phospholipid aiding peptide drug and insulin absorption.</p>
    Fórmula:C28H56NO8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:565.72
  • Fantofarone

    CAS:
    <p>Fantofarone (SR 33557) is a highly potent antagonist of Calcium Channel.</p>
    Fórmula:C31H38N2O5S
    Pureza:96.13% - 99.19%
    Forma y color:Solid
    Peso molecular:550.71
  • AMG-3969

    CAS:
    <p>AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).</p>
    Fórmula:C21H20F6N4O3S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:522.46
  • Telotristat Etiprate

    CAS:
    <p>Telotristat Etiprate (LX 1606 Hippurate) is an orally bioavailable, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.</p>
    Fórmula:C27H26ClF3N6O3·C9H9NO3
    Pureza:99.21% - 99.83%
    Forma y color:White Solid
    Peso molecular:754.15
  • Acebilustat

    CAS:
    <p>Acebilustat (CTX-4430) (ZK322) is an effective and specific leukotriene B4 hydrolase inhibitor.</p>
    Fórmula:C29H27N3O4
    Pureza:99.59% - 99.88%
    Forma y color:Solid
    Peso molecular:481.54
  • Fabomotizole hydrochloride

    CAS:
    <p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>
    Fórmula:C15H22ClN3O2S
    Pureza:99.54% - >99.99%
    Forma y color:Solid
    Peso molecular:343.87
  • SEP-0372814

    CAS:
    SEP-0372814 is a potent inhibitor of PDE10.
    Fórmula:C21H19N7
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:369.42
  • MLCK inhibitor peptide 18 acetate


    MLCK inhibitor peptide 18 acetate: Selective (IC50=50nM), 4000x more than CaM kinase II. Does not block PKA. Cell-permeable.
    Fórmula:C62H109N23O13
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:1384.67
  • PHD-1-IN-1

    CAS:
    PHD-1-IN-1 is a potent inhibitor of hypoxia-inducible factor prolylhydroxylase domain-1 (PHD-1) enzyme(IC50 = 0.034 μM).
    Fórmula:C13H8N4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:220.23
  • DG051

    CAS:
    <p>DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).</p>
    Fórmula:C21H25Cl2NO4
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:426.33
  • Fenretinide

    CAS:
    <p>Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.</p>
    Fórmula:C26H33NO2
    Pureza:98% - 99.68%
    Forma y color:Yellow Powder
    Peso molecular:391.55
  • Bay K 8644

    CAS:
    <p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>
    Fórmula:C16H15F3N2O4
    Pureza:99.41%
    Forma y color:Yellow Powder
    Peso molecular:356.3
  • Fraxinellone

    CAS:
    <p>1.</p>
    Fórmula:C14H16O3
    Pureza:99.35% - 99.92%
    Forma y color:Solid
    Peso molecular:232.27
  • N-Acetyl-β-Asp-Glu

    CAS:
    <p>N-Acetyl-β-Asp-Glu is a peptide neurotransmitter, the third most common neurotransmitter in the mammalian nervous system.</p>
    Fórmula:C11H16N2O8
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:304.25
  • TM5275 sodium

    CAS:
    TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).
    Fórmula:C28H27ClN3NaO5
    Pureza:98.8% - 99.74%
    Forma y color:Solid
    Peso molecular:543.98
  • Sevelamer hydrochloride

    CAS:
    <p>Sevelamer hydrochloride (Sevelamer HCl) is a phosphate binding drug used to treat hyperphosphatemia via binding to dietary phosphate and prevents its absorption</p>
    Fórmula:(C3H7N·C3H5ClO·HCl)x
    Pureza:98%
    Forma y color:Solid
    Peso molecular:186.08
  • Izilendustat hydrochloride

    CAS:
    <p>Izilendustat hydrochloride inhibits prolyl hydroxylase, stabilizing HIF-1α/HIF-2, with potential to treat various HIF-1α diseases.</p>
    Fórmula:C22H29Cl2N3O4
    Forma y color:Solid
    Peso molecular:470.39
  • Hydramethylnon

    CAS:
    <p>Hydramethylnon (AC217300) is an insecticide primarily. Hydramethylnon is used for fire ants.</p>
    Fórmula:C25H24F6N4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:494.48
  • GOT1 inhibitor-1

    CAS:
    <p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>
    Fórmula:C19H19ClN4O
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:354.83
  • Vardenafil hydrochloride trihydrate

    CAS:
    <p>Vardenafil hydrochloride trihydrate (BAY38-9456) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.</p>
    Fórmula:C23H32N6O4S·HCl·3H2O
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:579.11
  • URB602

    CAS:
    URB602 is a specific monoacylglycerol lipase (MGL) inhibitor, which inhibits rat brain MGL (IC50: 28±4 μM) through a noncompetitive mechanism.
    Fórmula:C19H21NO2
    Pureza:99.64% - 99.9%
    Forma y color:Off-White Solid
    Peso molecular:295.38
  • Uridine 5′-triphosphate tris salt

    CAS:
    <p>Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) is an agonist to the P2Y receptor and has been used to study concentrations of intracellular</p>
    Fórmula:C21H48N5O24P3
    Pureza:99.04% - 99.94%
    Forma y color:Solid
    Peso molecular:847.55
  • Bestatin trifluoroacetate

    CAS:
    <p>Bestatin trifluoroacetate inhibits CD13/APN and leukotriene A4 hydrolase, used in cancer research.</p>
    Fórmula:C18H25F3N2O6
    Forma y color:Solid
    Peso molecular:422.401
  • Ziconotide Acetate (107452-89-1 free base)

    CAS:
    <p>Ziconotide Acetate (Prialt, 107452-89-1) is an analgesic for neuropathic pain, acting on N-type calcium channels to block pain signals.</p>
    Fórmula:C102H172N36O32S7
    Pureza:99.52% - 99.87%
    Forma y color:Solid
    Peso molecular:2639.2
  • 3-Amino-2-oxazolidinone

    CAS:
    <p>3-Amino-2-oxazolidinone (AOZ) is the metabolite of Furazolidone. It is always be detected as a indicator of furazolidone residues in vivo.</p>
    Fórmula:C3H6N2O2
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:102.09
  • Tempol

    CAS:
    <p>Tempol (Tanol) is a superoxide scavenger. It has anti-inflammatory, neuroprotective and analgesic effects.</p>
    Fórmula:C9H18NO2
    Pureza:97% - 99.74%
    Forma y color:4-Hydroxy-Tempo Appears As Orange Flakes Solid Flakes
    Peso molecular:172.25
  • Tebufenpyrad

    CAS:
    <p>Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant</p>
    Fórmula:C18H24ClN3O
    Pureza:98.63% - 99.16%
    Forma y color:Solid
    Peso molecular:333.86
  • GSK0660

    CAS:
    <p>GSK0660 is an antagonist and inverse agonist of PPARβ/δ.</p>
    Fórmula:C19H18N2O5S2
    Pureza:99.26% - ≥95%
    Forma y color:Solid
    Peso molecular:418.49
  • Zofenopril

    CAS:
    <p>Zofenopril is an angiotensin-converting enzyme (ACE) inhibitor (IC50: 81 μM).</p>
    Fórmula:C22H23NO4S2
    Forma y color:Solid
    Peso molecular:429.55
  • Dorzolamide hydrochloride

    CAS:
    <p>Dorzolamide hydrochloride (MK507 hydrochloride) is the hydrochloride salt form of dorzolamide, an inhibitor of carbonic anhydrase, a zinc-containing enzyme that</p>
    Fórmula:C10H17ClN2O4S3
    Pureza:99.48% - 99.67%
    Forma y color:White Off-White Crystalline Powder
    Peso molecular:360.9
  • Raphin1 acetate

    CAS:
    <p>Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor.</p>
    Fórmula:C10H12Cl2N4O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:291.13
  • IBMX

    CAS:
    <p>IBMX (Methylisobutylxanthine) is a broad-spectrum phosphodiesterase (PDE) inhibitor with inhibitory activity against PDE3, PDE4, and PDE5 (IC50=6.5/26.3/31.7 μM</p>
    Fórmula:C10H14N4O2
    Pureza:98% - >99.99%
    Forma y color:Off-White
    Peso molecular:222.24
  • Quilseconazole

    CAS:
    <p>Quilseconazole is an effective, orally active fungal Cyp51 inhibitor. it also binds tightly to cryptococcal CYP51 but weakly inhibits humans CYP450 enzymes.</p>
    Fórmula:C22H14F7N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:513.37
  • amflutizole

    CAS:
    <p>Amflutizole used for the treatment of gout, and is a Xanthine oxidase inhibitor</p>
    Fórmula:C11H7F3N2O2S
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:288.246
  • ATP

    CAS:
    <p>ATP (Adenosine triphosphate) provides cellular energy, participates in overall energy balance, and maintains intracellular homeostasis.</p>
    Fórmula:C10H16N5O13P3
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:507.18
  • ICI 63197

    CAS:
    ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.
    Fórmula:C9H13N5O
    Pureza:99.70%
    Forma y color:White Solid
    Peso molecular:207.23
  • CDD3506

    CAS:
    <p>CDD3506 (1-TRITYL-1H-IMIDAZOL-4-AMINE) increases high-density lipoprotein cholesterol by targeting hepatic CYP3A.</p>
    Fórmula:C22H19N3
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:325.41
  • Alfacalcidol

    CAS:
    <p>Alfacalcidol (Etalpha) (1-hydroxycholecalciferol; Alpha D3; 1.alpha.-Hydroxyvitamin D3) is a non-selective VDR activator medication.</p>
    Fórmula:C27H44O2
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:400.64
  • Lomerizine dihydrochloride

    CAS:
    <p>Lomerizine dihydrochloride (KB-2796) is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.</p>
    Fórmula:C27H30F2N2O3·2HCl
    Pureza:99.26% - 99.80%
    Forma y color:Colourless Crystalline Solid
    Peso molecular:541.46
  • DL-AP3

    CAS:
    <p>DL-AP3 is a competitive group I metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase.</p>
    Fórmula:C3H8NO5P
    Pureza:98.18% - ≥98%
    Forma y color:White Powder
    Peso molecular:169.07
  • Nequinate

    CAS:
    <p>Nequinate is an anticoccidial agent, preventing coccidiosis .</p>
    Fórmula:C22H23NO4
    Pureza:96.43%
    Forma y color:Light Yellow Odorless Powder
    Peso molecular:365.42
  • CDN1163

    CAS:
    <p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>
    Fórmula:C20H20N2O2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:320.39
  • Levamlodipine besylate

    CAS:
    <p>Levamlodipine besylate, or S-amlodipine (CAS 103129-82-4), is the active enantiomer of amlodipine, used to treat hypertension and angina.</p>
    Fórmula:C26H31ClN2O8S
    Pureza:99.78% - 99.79%
    Forma y color:Solid
    Peso molecular:567.05
  • Ethyl 3,4-dihydroxybenzoate

    CAS:
    <p>Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.</p>
    Fórmula:C9H10O4
    Pureza:99.88%
    Forma y color:White Crystal Or Powder
    Peso molecular:182.17
  • LHW090-A7

    CAS:
    <p>LHW090-A7 is an neutral endopeptidase (NEP) inhibitor, and an enzyme responsible for the metabolic inactivation of enkephalins.</p>
    Fórmula:C20H22ClNO4
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:375.85
  • (E,E)-RAMB4

    CAS:
    <p>PTP1B-IN-8 is a potent and selective inhibitor of protein tyrosine phosphatase-1B (PTP1B).</p>
    Fórmula:C19H13Cl4NO
    Pureza:96.03%
    Forma y color:Solid
    Peso molecular:413.12
  • AA26-9

    CAS:
    <p>AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.</p>
    Fórmula:C7H10N4O
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:166.18
  • JNJ-42165279

    CAS:
    <p>JNJ-42165279 selectively inactivates FAAH without notably affecting other enzymes, ion channels, receptors, or CYPs/hERG at 10 μM.</p>
    Fórmula:C18H17ClF2N4O3
    Pureza:99.67% - 99.88%
    Forma y color:Solid
    Peso molecular:410.8
  • Indisulam

    CAS:
    <p>Indisulam (E 7070) is a dual-action anticancer drug, blocking G1/S cell cycle transition by degrading cyclin E and activating p53/p21.</p>
    Fórmula:C14H12ClN3O4S2
    Pureza:98.68% - 99.77%
    Forma y color:Solid
    Peso molecular:385.85
  • AKR1C3-IN-1

    CAS:
    <p>AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3(IC50 of 13 nM).</p>
    Fórmula:C16H15NO4S
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:317.36
  • Ethyl potassium malonate

    CAS:
    <p>Ethyl potassium malonate, a competitive inhibitor of the enzyme succinate dehydrogenase, acts as a precursor to produce (trimethylsilyl)ethyl malonate, which is</p>
    Fórmula:C5H7KO4
    Pureza:99.71%
    Forma y color:White Crystals Or Powder
    Peso molecular:170.21
  • Sacubitril sodium

    CAS:
    <p>Sacubitril sodium (AHU-377) is potent NEP inhibitor with an IC50=5 nM for the treatment of heart failure or in combination with antihypertensive agents.</p>
    Fórmula:C24H28NNaO5
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:433.47
  • LJ570

    CAS:
    <p>LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, respectively[)</p>
    Fórmula:C27H22O3
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:394.46
  • AGI-5198

    CAS:
    <p>AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).</p>
    Fórmula:C27H31FN4O2
    Pureza:97.37% - 99.23%
    Forma y color:Solid
    Peso molecular:462.56
  • H2S Donor 5a

    CAS:
    <p>H2S Donor 5a is a H2S donor that could mimic the slow and continuous H(2)S generation process.</p>
    Fórmula:C14H11NO2S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:257.31
  • Trandolapril

    CAS:
    <p>Trandolapril is an orally administered angiotensin converting enzyme (ACE) inhibitor that is hydrolysed to the active diacid trandolaprilat.</p>
    Fórmula:C24H34N2O5
    Pureza:99.70% - 99.83%
    Forma y color:White Powder
    Peso molecular:430.54
  • N6022

    CAS:
    <p>N6022(IC50 of 8 nM) is an effective, reversible, and selective S-Nitrosoglutathione reductase(GSNOR) inhibitor.</p>
    Fórmula:C24H22N4O3
    Pureza:98.24% - 98.32%
    Forma y color:Solid
    Peso molecular:414.46
  • Clorgyline

    CAS:
    <p>Clorgyline,M&amp;B 9302, an irreversible and selective MAO-A inhibitor with the advantages of oral activity and blood-brain barrier permeability, antidepressant.</p>
    Fórmula:C13H15Cl2NO
    Pureza:98.39%
    Forma y color:Solid
    Peso molecular:272.17
  • Amino Tadalafil

    CAS:
    <p>Amino tadalafil is a potent phosphodiesterase 5 (PDE5) inhibitor.</p>
    Fórmula:C21H18N4O4
    Pureza:99.85%
    Forma y color:White Powder
    Peso molecular:390.39
  • LDHA-IN-4

    CAS:
    <p>LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.</p>
    Fórmula:C25H27N3O6S
    Pureza:98.17% - 99.68%
    Forma y color:Solid
    Peso molecular:497.56
  • Balipodect

    CAS:
    <p>Balipodect (TAK063) is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is &gt;15000-fold over other PDEs.</p>
    Fórmula:C23H17FN6O2
    Pureza:98% - 99.79%
    Forma y color:Solid
    Peso molecular:428.42