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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

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Se han encontrado 8626 productos de "Metabolismo"

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  • 1,2-Dipalmitoyl-sn-glycerol 3-phosphate

    CAS:
    <p>1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.</p>
    Fórmula:C35H69O8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:648.89
  • ARN-6039

    CAS:
    <p>ARN-6039 is an oral RORγ inverse agonist for Autoimmune Neuroinflammation, active in HEK 293 cells and CD4+T cells.</p>
    Fórmula:C21H21F3N2O3
    Forma y color:Solid
    Peso molecular:406.40
  • Flurtamone

    CAS:
    <p>Flurtamone is an agricultural chemical. Flurtamone mainly used as an herbicide.</p>
    Fórmula:C18H14F3NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:333.30
  • RPR132595A

    CAS:
    RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).
    Fórmula:C28H30N4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:518.56
  • DC-6-14

    CAS:
    <p>DC-6-14 is a cationic lipid known for its gene transfection activity, commonly utilized in the synthesis of liposomes.</p>
    Fórmula:C37H73ClN2O5
    Forma y color:Solid
    Peso molecular:661.44
  • sEH inhibitor-17

    CAS:
    <p>sEH inhibitor-17 (compound 4f) is an orally active soluble epoxide hydrolase (sEH) inhibitor with an IC50 value of 2.94 nM. This compound exhibits anti-inflammatory properties.</p>
    Fórmula:C18H21F3N2O4S
    Forma y color:Solid
    Peso molecular:418.43
  • Prothioconazole

    CAS:
    <p>Prothioconazole (Proline 480 SC Fungicide) is a chiral triazole fungicide in plant pathogen control.</p>
    Fórmula:C14H15Cl2N3OS
    Pureza:99.77%
    Forma y color:Un3077 9/Pg 3
    Peso molecular:344.26
  • PAT-494

    CAS:
    <p>PAT-494 is an inhibitor of type II Autotaxin.</p>
    Fórmula:C20H16FN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:349.36
  • SHP2-IN-29

    CAS:
    <p>SHP2-IN-29 (Compound 3), a potent inhibitor of SHP2, exhibits an IC 50 of 0.18 μM. Additionally, this compound demonstrates inhibitory activity against PTP1B and TCPTP, with IC 50 values of 4.27 μM and 4.74 μM, respectively.</p>
    Fórmula:C16H20O4
    Forma y color:Solid
    Peso molecular:276.33
  • MDI-2268

    CAS:
    <p>MDI-2268, an inhibitor of plasma kallikrein inhibitor 1 (PAI-1), exhibits strong antithrombotic properties. It plays a role in regulating blood coagulation by promoting fibrinolysis and is applicable in research related to deep vein thrombosis.</p>
    Fórmula:C10H10F3N3O3
    Forma y color:Solid
    Peso molecular:277.20
  • Transketolase-IN-3

    CAS:
    <p>Transketolase-IN-3: potent TK inhibitor with herbicidal effects on DS and AR, useful for herbicide research.</p>
    Fórmula:C20H9ClF3NO3
    Forma y color:Solid
    Peso molecular:403.74
  • Acetaminophen mercapturate

    CAS:
    <p>Paracetamol Mercapturate is a metabolite of Acetaminophen. It can also be used in the biological study of urinary antihypertensive drugs.</p>
    Fórmula:C13H16N2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:312.34
  • Leucylarginine

    CAS:
    <p>Leucylarginine hinders antinociception induced by L-arginine.</p>
    Fórmula:C12H25N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:287.36
  • Desmethylnortriptyline

    CAS:
    <p>Desmethylnortriptyline, a tricyclic antidepressant metabolite of nortriptyline and amitriptyline, treats depression.</p>
    Fórmula:C18H19N
    Pureza:98%
    Forma y color:Solid
    Peso molecular:249.35
  • PPM1A-IN-1

    CAS:
    <p>PPM1A-IN-1 (Compound IV-4) is an inhibitor of the PP2C Ser/Thr protein phosphatase Mg2+/Mn2+-dependent 1A. It exhibits antibacterial activity against Mycobacterium tuberculosis.</p>
    Fórmula:C16H15BrFNO2
    Forma y color:Solid
    Peso molecular:352.2
  • FAAH-IN-8

    CAS:
    <p>FAAH-IN-8 (compound 11) is a competitive inhibitor of FAAH with an IC50 of 6.7 nM and a Ki of 5 nM. It exhibits high blood-brain permeability and a significant antioxidant profile without neurotoxicity [1].</p>
    Fórmula:C18H14N4O
    Forma y color:Solid
    Peso molecular:302.33
  • Trimosulfa

    CAS:
    <p>Trimosulfa is a combination of trimethoprim and sulfamethoxazole, an antibiotic combination. Sulfamethoxazole inhibits dihydropteroate synthase, while trimethoprim inhibits dihydrofolate reductase (dihydrofolate reductase), making it effective for mild to moderate bacterial infections against many Gram-negative and Gram-positive bacteria.</p>
    Fórmula:C24H29N7O6S
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:543.6
  • 1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine

    CAS:
    1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.
    Fórmula:C44H84NO8P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:786.11
  • Descarbamoyl cefuroxime

    CAS:
    Descarbamoyl cefuroxime is also an intermediate in the synthesis of cephalosporin antibiotics. Decarbamyl cefuroxime is a degradation product of cefuroxime.
    Fórmula:C15H15N3O7S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.36
  • HSL-IN-5

    CAS:
    <p>HSL-IN-5 (Example 21) is a hormone-sensitive lipase (HSL) inhibitor with an IC₅₀ value of 0.2 μM, suitable for diabetes research.</p>
    Fórmula:C18H23F3N2O4
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:388.38
  • Roflumilast Impurity E

    CAS:
    <p>Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast acts as a selective and long-acting the enzyme PDE-4 inhibitor(IC50 value of 0.8 nM).</p>
    Fórmula:C13H8Cl2F2N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:349.12
  • LAPAO

    CAS:
    <p>Lauramide propyl amine oxide is an amphoteric surfactant</p>
    Fórmula:C17H36N2O2
    Forma y color:Solid
    Peso molecular:300.48
  • Dihydro Dutasteride

    CAS:
    <p>Dihydro Dutasteride is a metabolite of Dutasteride. Dutasteride is an effective inhibitor of five α-reductase isozymes.</p>
    Fórmula:C27H32F6N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:530.55
  • H-Arg-Lys-OH

    CAS:
    <p>H-Arg-Lys-OH is a dipeptide formed from L-lysine residues and L-arginyl.</p>
    Fórmula:C12H26N6O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.37
  • Sodium lauroyl glutamate

    CAS:
    <p>Sodium lauroyl glutamate (Acylglutamate LS-11) is an amino acid detergent and increases the solubility of long-chain alkyl gallates such as alkyl gallates.</p>
    Fórmula:C17H30NNaO5
    Pureza:97.13%
    Forma y color:Solid
    Peso molecular:351.41
  • AKU-005

    CAS:
    <p>AKU-005 is a dual inhibitor of FAAH and MAGL, exhibiting IC50 values of 63 nM and 389 nM against rat and human FAAH, respectively. This compound has potential for researching trigeminal nociceptive hypersensitivity.</p>
    Fórmula:C20H21N5O
    Forma y color:Solid
    Peso molecular:347.41
  • Atorvastatin acetonide

    CAS:
    <p>Atorvastatin acetonide, an impurity in Atorvastatin, lowers blood lipids; from patent WO2011131605A1.</p>
    Fórmula:C36H39FN2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:598.7
  • Proadifen

    CAS:
    <p>Proadifen is a non-selective cytochrome P450 enzymes inhibitor, preventing some types of drug metabolism.</p>
    Fórmula:C23H31NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:353.5
  • ent-Tadalafil

    CAS:
    ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS).
    Fórmula:C22H19N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:389.4
  • Prasugrel chloride impurity

    CAS:
    <p>Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.</p>
    Fórmula:C20H21ClFNO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:409.9
  • 1-Decanesulfonic acid

    CAS:
    <p>1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.</p>
    Fórmula:C10H22O3S
    Forma y color:Solid
    Peso molecular:222.35
  • Tolrestat

    CAS:
    <p>Tolrestat (AY-27773) is a potent inhibitor of aldose reductase (IC50 = 35 nM).</p>
    Fórmula:C16H14F3NO3S
    Pureza:98.89% - >99.99%
    Forma y color:Solid
    Peso molecular:357.35
  • PF-05175157

    CAS:
    <p>PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,</p>
    Fórmula:C23H27N5O2
    Pureza:98% - 99.92%
    Forma y color:Solid
    Peso molecular:405.49
  • 4-POBN

    CAS:
    <p>4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).</p>
    Fórmula:C7H9N3O
    Pureza:99.60%
    Forma y color:White Crystalline Powder
    Peso molecular:151.17
  • Calcipotriol monohydrate

    CAS:
    <p>Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.</p>
    Fórmula:C27H42O4
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:430.62
  • Tesaglitazar

    CAS:
    <p>Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα</p>
    Fórmula:C20H24O7S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:408.47
  • PCI-27483

    CAS:
    <p>PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.</p>
    Fórmula:C26H24N6O9S
    Pureza:98.55%
    Forma y color:Solid
    Peso molecular:596.57
  • BIBB 515

    CAS:
    <p>BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.</p>
    Fórmula:C22H21ClN2O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:380.87
  • E3330

    CAS:
    <p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>
    Fórmula:C21H30O6
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:378.46
  • 3-Phenylbutyric acid

    CAS:
    <p>3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.</p>
    Fórmula:C10H12O2
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:164.2
  • L-m-Tyrosine

    CAS:
    <p>L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.</p>
    Fórmula:C9H11NO3
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:181.19
  • UK-414,495

    CAS:
    <p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>
    Fórmula:C16H25N3O3S
    Forma y color:Solid
    Peso molecular:339.45
  • Darexaban glucuronide

    CAS:
    <p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>
    Fórmula:C33H38N4O10
    Forma y color:Solid
    Peso molecular:650.68
  • Sterculic acid

    CAS:
    <p>Sterculic acid inhibits SCD1 with IC50 of 0.9μM, affecting Δ9D desaturase activity.</p>
    Fórmula:C19H34O2
    Forma y color:Solid
    Peso molecular:294.47
  • hCAIX-IN-11

    CAS:
    <p>hCAIX-IN-11 inhibits carbonic anhydrases IX &amp; XII with Ki of 32.7 nM &amp; 623.5 nM, respectively.</p>
    Fórmula:C21H15ClN4O3
    Forma y color:Solid
    Peso molecular:406.82
  • hCAI/II-IN-5

    CAS:
    <p>hCAI/II-IN-5 inhibits human carbonic anhydrase I &amp; II, α-Glycosidase, and AChE, for diabetes, heart failure, Alzheimer's, ulcers, epilepsy research.</p>
    Fórmula:C21H18Cl2N8O4S2
    Forma y color:Solid
    Peso molecular:581.45
  • LY 56110

    CAS:
    <p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>
    Fórmula:C17H12Cl2N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:315.2
  • (R)-Bromoenol lactone

    CAS:
    <p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>
    Fórmula:C16H13BrO2
    Forma y color:Solid
    Peso molecular:317.18
  • LB42908

    CAS:
    <p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>
    Fórmula:C32H31N5O3
    Forma y color:Solid
    Peso molecular:533.62
  • N-Oleoyl Leucine

    CAS:
    <p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>
    Fórmula:C24H45NO3
    Pureza:98.25%
    Forma y color:Solid
    Peso molecular:395.62
  • Loxoprofenol-SRS

    CAS:
    <p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>
    Fórmula:C15H20O3
    Forma y color:Solid
    Peso molecular:248.32
  • TPN729MA

    CAS:
    <p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>
    Fórmula:C29H40N6O8S
    Forma y color:Solid
    Peso molecular:632.73
  • 14-dehydro Zymostenol

    CAS:
    <p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>
    Fórmula:C27H44O
    Forma y color:Solid
    Peso molecular:384.64
  • 103D5R

    CAS:
    <p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>
    Fórmula:C20H21N3O2
    Forma y color:Solid
    Peso molecular:335.4
  • JBP485

    CAS:
    <p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>
    Fórmula:C8H12N2O4
    Forma y color:Solid
    Peso molecular:200.19
  • Anserinone B

    CAS:
    <p>Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).</p>
    Fórmula:C11H14O4
    Forma y color:Solid
    Peso molecular:210.23
  • EDP-305

    CAS:
    <p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>
    Fórmula:C36H58N2O5S
    Forma y color:Solid
    Peso molecular:630.92
  • CAY10486

    CAS:
    <p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>
    Fórmula:C19H19NO4
    Forma y color:Solid
    Peso molecular:325.36
  • Valibose

    CAS:
    <p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>
    Fórmula:C10H21NO6
    Forma y color:Solid
    Peso molecular:251.28
  • (R)-Irsenontrine

    CAS:
    <p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>
    Fórmula:C22H22N4O3
    Forma y color:Solid
    Peso molecular:390.44
  • URB532

    CAS:
    <p>URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Fórmula:C18H21NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:299.36
  • Fluindione

    CAS:
    <p>Fluindione is a hematologic drug.</p>
    Fórmula:C15H9FO2
    Forma y color:Solid
    Peso molecular:240.23
  • Glyoxalase I inhibitor 2

    CAS:
    <p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>
    Fórmula:C24H23N3O4S
    Forma y color:Solid
    Peso molecular:449.52
  • DMPAC-Chol

    CAS:
    <p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>
    Fórmula:C33H58N2O2
    Forma y color:Solid
    Peso molecular:514.83
  • hCAIX-IN-7

    CAS:
    <p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: &gt;10000 nM).</p>
    Fórmula:C18H12FNO3
    Forma y color:Solid
    Peso molecular:309.29
  • GNE-3500

    CAS:
    <p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>
    Fórmula:C24H30FN3O3S
    Forma y color:Solid
    Peso molecular:459.58
  • YM-75466

    CAS:
    <p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>
    Fórmula:C28H35N5O8S2
    Forma y color:Solid
    Peso molecular:633.74
  • BMS 740808

    CAS:
    <p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>
    Fórmula:C31H27F3N6O3
    Forma y color:Solid
    Peso molecular:588.58
  • TMCB

    CAS:
    <p>CK2 and ERK8 inhibitor</p>
    Fórmula:C11H9Br4N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:534.82
  • DHODH-IN-21

    CAS:
    <p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>
    Fórmula:C20H19ClF4N6O4
    Forma y color:Solid
    Peso molecular:518.85
  • HIF-PHD-IN-2

    CAS:
    <p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>
    Fórmula:C17H15N5O3S
    Forma y color:Solid
    Peso molecular:369.4
  • α-Amylase-IN-2

    CAS:
    α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =
    Fórmula:C39H52BrNO4
    Forma y color:Solid
    Peso molecular:678.74
  • HIF-1α-IN-3

    CAS:
    <p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>
    Fórmula:C19H17N5O2
    Forma y color:Solid
    Peso molecular:347.37
  • MDK-4823

    CAS:
    <p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>
    Fórmula:C28H36N4O
    Forma y color:Solid
    Peso molecular:444.61
  • Enpp-1-IN-8

    CAS:
    <p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>
    Fórmula:C19H26N6O4S
    Forma y color:Solid
    Peso molecular:434.51
  • FAAH-IN-7


    <p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>
    Fórmula:C26H29N3O4
    Forma y color:Solid
    Peso molecular:447.53
  • hCAIX-IN-3

    CAS:
    <p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>
    Fórmula:C21H21BrN6O4S
    Forma y color:Solid
    Peso molecular:533.4
  • α-Glucosidase-IN-21

    CAS:
    <p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>
    Fórmula:C24H23NO2S
    Forma y color:Solid
    Peso molecular:389.51
  • 3,3-Dimethyl-1-butanol

    CAS:
    <p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>
    Fórmula:C6H14O
    Forma y color:Solid
    Peso molecular:102.17
  • IDO1-IN-15

    CAS:
    <p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>
    Fórmula:C13H14BrFN6O3
    Forma y color:Solid
    Peso molecular:401.19
  • hCAXII-IN-1

    CAS:
    <p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>
    Fórmula:C20H17NO5
    Forma y color:Solid
    Peso molecular:351.35
  • DP00477

    CAS:
    <p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>
    Fórmula:C17H11ClF3N3OS
    Forma y color:Solid
    Peso molecular:397.8
  • D-threo-PPMP hydrochloride

    CAS:
    <p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>
    Fórmula:C29H51ClN2O3
    Forma y color:Solid
    Peso molecular:511.19
  • Lp-PLA2-IN-3

    CAS:
    <p>Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.</p>
    Fórmula:C20H13ClF3N3O3S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:467.85
  • Hydroxychlorodenafil

    CAS:
    <p>Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>
    Fórmula:C19H23ClN4O3
    Forma y color:Solid
    Peso molecular:390.86
  • HS79

    CAS:
    <p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>
    Fórmula:C19H22N4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.47
  • Andolast

    CAS:
    <p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>
    Fórmula:C15H11N9O
    Forma y color:Solid
    Peso molecular:333.31
  • sEH inhibitor-14

    CAS:
    <p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>
    Fórmula:C16H12F3N3O4
    Forma y color:Soild
    Peso molecular:367.28
  • Enpp-1-IN-5

    CAS:
    <p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>
    Fórmula:C17H26N6O4S
    Forma y color:Solid
    Peso molecular:410.49
  • mIDH1-IN-1

    CAS:
    <p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>
    Fórmula:C25H27N3O5
    Forma y color:Solid
    Peso molecular:449.5
  • Glucokinase activator 3

    CAS:
    <p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>
    Fórmula:C26H33N2O9PS2
    Forma y color:Solid
    Peso molecular:612.65
  • IDO-IN-14

    CAS:
    <p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>
    Fórmula:C23H23ClN4O2
    Forma y color:Solid
    Peso molecular:422.91
  • FXR agonist 4


    <p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>
    Fórmula:C21H28ClN3O
    Forma y color:Solid
    Peso molecular:373.92
  • CYP1B1-IN-3

    CAS:
    <p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>
    Fórmula:C20H16FN3O2S2
    Forma y color:Solid
    Peso molecular:413.49
  • DTP348

    CAS:
    <p>DTP348: Oral carbonic anhydrase IX inhibitor &amp; hypoxic cell radiosensitizer with sulfamide &amp; 5-nitroimidazole components.</p>
    Fórmula:C6H11N5O4S
    Forma y color:Solid
    Peso molecular:249.25
  • Nitrefazole

    CAS:
    <p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>
    Fórmula:C10H8N4O4
    Forma y color:Solid
    Peso molecular:248.19
  • URB-694

    CAS:
    <p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Fórmula:C19H21NO3
    Forma y color:Solid
    Peso molecular:311.37
  • DGAT1-IN-3

    CAS:
    <p>DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.</p>
    Fórmula:C20H19F3N4O3
    Forma y color:Solid
    Peso molecular:420.39
  • Nampt-IN-7

    CAS:
    <p>Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).</p>
    Fórmula:C20H21N5O3
    Forma y color:Solid
    Peso molecular:379.41
  • FASN-IN-4

    CAS:
    <p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>
    Fórmula:C26H27N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:477.58
  • AMPD2 inhibitor 2


    <p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>
    Fórmula:C26H27F2N3O3
    Forma y color:Solid
    Peso molecular:467.51
  • ME-143

    CAS:
    <p>ME-143, a 2nd-gen NADH oxidase inhibitor, blocks WNT/β-catenin pathway, active against various cancers in vitro/vivo.</p>
    Fórmula:C21H18O4
    Forma y color:Solid
    Peso molecular:334.37
  • MDPD

    CAS:
    <p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>
    Fórmula:C21H19N3O3
    Forma y color:Solid
    Peso molecular:361.39
  • Antiproliferative agent-10


    <p>Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.</p>
    Fórmula:C35H36Cl2N7PRu
    Forma y color:Solid
    Peso molecular:757.66
  • LY 113174

    CAS:
    <p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>
    Fórmula:C17H10Cl2N2
    Forma y color:Solid
    Peso molecular:313.18
  • FC11409B

    CAS:
    <p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>
    Fórmula:C29H23BF4N2O3S
    Forma y color:Solid
    Peso molecular:566.38
  • Lp-PLA2-IN-4

    CAS:
    <p>Lp-PLA2-IN-4, a potent inhibitor of Lp-PLA2/PAF-AH, may target Alzheimer's, atherosclerosis. (WO2021228159A1, Compound 38)</p>
    Fórmula:C23H18F5N3O4
    Forma y color:Solid
    Peso molecular:495.4
  • Flutolanil

    CAS:
    <p>Flutolanil: a fungicide targeting R. solani in rice, toxic to zebrafish.</p>
    Fórmula:C17H16F3NO2
    Forma y color:Solid
    Peso molecular:323.31
  • JZP-MA-13


    <p>JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.</p>
    Fórmula:C14H15FN4O3S
    Forma y color:Solid
    Peso molecular:338.36
  • BRD9500

    CAS:
    <p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>
    Fórmula:C15H18FN3O2
    Forma y color:Solid
    Peso molecular:291.32
  • Glyoxalase I inhibitor 4

    CAS:
    <p>Glyoxalase I inhibitor 4 is a potent inhibitor of glyoxalase I (GLO1) (Ki: 10 nM).</p>
    Fórmula:C17H21IN4O8S
    Forma y color:Solid
    Peso molecular:568.34
  • BMP-22

    CAS:
    <p>BMP-22 selectively inhibits autotaxin (IC50=170 nM), blocks LPA production and MM1 cell invasion, and reduces lung metastases in mice at 0.5 mg/kg/day.</p>
    Fórmula:C22H39O3P
    Forma y color:Solid
    Peso molecular:382.52
  • SAHO

    CAS:
    <p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>
    Fórmula:C14H20N6O6S
    Forma y color:Solid
    Peso molecular:400.41
  • SHP2-IN-5

    CAS:
    <p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>
    Fórmula:C12H8O6
    Forma y color:Solid
    Peso molecular:248.19
  • Tebuconazole-d9

    CAS:
    <p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>
    Fórmula:C16H13ClD9N3O
    Forma y color:Solid
    Peso molecular:316.87
  • CD 1530

    CAS:
    <p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>
    Fórmula:C27H26O3
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:398.49
  • JMS-053

    CAS:
    <p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>
    Fórmula:C13H8N2O2S
    Pureza:≥98.0%
    Forma y color:Solid
    Peso molecular:256.28
  • Glycogen phosphorylase-IN-1

    CAS:
    <p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>
    Fórmula:C17H15ClF2N4O4
    Pureza:97.98% - 98.15%
    Forma y color:Solid
    Peso molecular:412.78
  • AQX-MN115

    CAS:
    <p>AQX-MN115 is an SH2- containing inositol 5- phosphatase modulator.</p>
    Fórmula:C21H30O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:314.46
  • Bamethan sulfate

    CAS:
    <p>Bamethan sulfate is a Vasodilator.</p>
    Fórmula:C24H40N2O8S
    Forma y color:Solid
    Peso molecular:516.65
  • Ethylene thiourea

    CAS:
    <p>Ethylene thiourea (NCIC03372) is a pesticide used in fruit and vegetable production.</p>
    Fórmula:C3H6N2S
    Pureza:≥98%
    Forma y color:Needles Prisms From Alcohol Or Amyl Alcohol
    Peso molecular:102.16
  • Pteropterin

    CAS:
    <p>Pteropterin is an antineoplastic agent.</p>
    Fórmula:C29H33N9O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:699.63
  • Alitame

    CAS:
    <p>Alitame is a high-intensity sweetener and sugar substitute widely used in biochemical experiments and drug synthesis research.</p>
    Fórmula:C14H25N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:331.43
  • DCYM21

    CAS:
    <p>DCYM21: Menin-MLL inhibitor, halts leukemia cell growth with MLL changes, causing arrest and differentiation.</p>
    Fórmula:C26H33ClN2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:409.01
  • Sermetacin

    CAS:
    <p>Sermetacin is an anti-inflammatory agent.</p>
    Fórmula:C22H21ClN2O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:444.86
  • AZD-3289

    CAS:
    <p>AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>
    Fórmula:C24H14F5N5
    Forma y color:Solid
    Peso molecular:467.39
  • tHGA

    CAS:
    <p>tHGA is a potent inhibitor of lipoxygenase.</p>
    Fórmula:C18H24O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:304.38
  • GW648495

    CAS:
    <p>GW648495 is a PfDHODH inhibitor that shows greater than 4,000-fold selectivity for the malarial enzyme.</p>
    Fórmula:C16H13N5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:275.31
  • ts-SA

    CAS:
    <p>ts-SA is a metalloenzyme carbonic anhydrase (CA) inhibitor. It is active against 7 out of 10 human CA isoforms.</p>
    Fórmula:C14H15N3O5S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:369.42
  • Fexaramate

    CAS:
    <p>Fexaramate is a potent, selective agonist of farnesoid X receptor.</p>
    Fórmula:C31H37NO5
    Forma y color:Solid
    Peso molecular:503.63
  • Oncrasin-72

    CAS:
    Oncrasin-72 is an analog of oncrasin-1. It has antitumor activity mediated by JNK activation and STAT3 inhibition.
    Fórmula:C16H14ClNO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:271.74
  • iGP-5

    CAS:
    <p>iGP-5 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>
    Fórmula:C21H17N3O3
    Forma y color:Solid
    Peso molecular:359.38
  • α-RA-F

    CAS:
    <p>Alpha-RA-F increases collagen, lowers MMPs in human fibroblasts, non-toxic.</p>
    Fórmula:C16H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:300.31
  • myomiR-IN-1

    CAS:
    <p>myomiR-IN-1 inhibits myoD translation in C2C12 cells, doesn't affect myoD mRNA, and reduces differentiation markers.</p>
    Fórmula:C33H27NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:533.57
  • 2-Iodoestradiol

    CAS:
    2-Iodoestradiol is an effective human sex hormone-binding globulin (SHBG) ligand.
    Fórmula:C18H23IO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:398.28
  • OMS-824

    CAS:
    <p>OMS-824 is a phosphodiesterase-10 inhibitor that slows or stops the hydrolysis of cAMP and cGMP.</p>
    Fórmula:C21H21BrN4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.32
  • PF-05387252

    CAS:
    PF-05387252 is an effective and selective inhibitor of the IRAK4.
    Fórmula:C25H27N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:429.51
  • AF267

    CAS:
    <p>AF267 is a M1 muscarinic agonist that works by restoring cognitive impairments.</p>
    Fórmula:C10H18N2OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:214.33
  • Clinolamide

    CAS:
    <p>Clinolamide is an antilipidemic agent.</p>
    Fórmula:C24H43NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:361.6
  • Dehydro-ZINC39395747

    CAS:
    Dehydro-ZINC39395747 enhances NO in cells and inhibits cytochrome b5 reductase 3 (IC50: 9.14μM, Kd: 1.11μM).
    Fórmula:C12H9N3O2S2
    Forma y color:Solid
    Peso molecular:291.35
  • Bucricaine

    CAS:
    <p>Bucricaine is an anesthetic drug.</p>
    Fórmula:C17H22N2
    Forma y color:Solid
    Peso molecular:254.37
  • Nafenopin

    CAS:
    <p>Nafenopin is a peroxisome proliferator, it is used to promote liver tumors and has been used as an antihyperlipoproteinemic agent.</p>
    Fórmula:C20H22O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:310.39
  • CM026

    CAS:
    <p>CM026 inhibits ALDH1A1 selectively, binds to its aldehyde pocket uncompetitively.</p>
    Fórmula:C22H30N6O4
    Forma y color:Solid
    Peso molecular:442.51
  • ABT-418

    CAS:
    <p>ABT-418, a nicotinic acetylcholine receptor (nAchR) agonist, is used potentially for the treatment of attention deficit disorder.</p>
    Fórmula:C9H14N2O
    Forma y color:Solid
    Peso molecular:166.22
  • Safrazine Hydrochloride

    CAS:
    <p>Safrazine Hydrochloride is a monoamine oxidase inhibitor (MOI) that is irreversible.</p>
    Fórmula:C11H17ClN2O2
    Forma y color:Solid
    Peso molecular:244.718
  • MDK-0738

    CAS:
    <p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>
    Fórmula:C15H16O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:244.29
  • 4&prime;-Deoxyphlorizin

    CAS:
    <p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>
    Fórmula:C21H24O9
    Forma y color:Solid
    Peso molecular:420.41
  • CP-319340(free base)

    CAS:
    <p>CP-319340 free base is a inhibitor of microsomal triglyceride transfer protein (MTP) .</p>
    Fórmula:C27H23F3N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:476.49
  • MP-10 succinate

    CAS:
    <p>MP-10 succinate is a potent and specific inhibitor of PDE10A.</p>
    Fórmula:C29H26N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:510.54
  • LYPLAL1-IN-1

    CAS:
    LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.
    Fórmula:C29H29N7O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:539.59
  • Brocresine

    CAS:
    <p>Brocresine is an aromatic L-amino acid decarboxylase inhibitor. It has both a peripheral and central action.</p>
    Fórmula:C7H8BrNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:218.05
  • NE21650

    CAS:
    <p>NE21650, a bisphosphonate, inhibits isopentenyl diphosphate isomerase and farnesyl diphosphate synthase.</p>
    Fórmula:C8H13NO7P2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:297.14
  • Zofenoprilat arginine

    CAS:
    <p>Zofenoprilat arginine is an antihypertensive.</p>
    Fórmula:C21H33N5O5S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:499.65
  • ABL127

    CAS:
    ABL127 inhibits PME-1 with IC50s of 6.4 nM in HEK293T cells and 4.2 nM in MDA-MB-231 cells.
    Fórmula:C17H20N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:332.35
  • Butaperazine maleate

    CAS:
    <p>Butaperazine maleate, a phenothiazine derivative, is an antipsychotic.</p>
    Fórmula:C32H39N3O9S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:641.73
  • Albifylline

    CAS:
    <p>Albifylline: a xanthine derivative, anti-asthmatic, reduces leukocyte adhesion, enhances liver microcirculation post-hemorrhagic shock.</p>
    Fórmula:C13H20N4O3
    Forma y color:Solid
    Peso molecular:280.32
  • AHR-activator-1023

    CAS:
    <p>AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.</p>
    Fórmula:C14H8Cl2N2O
    Forma y color:Solid
    Peso molecular:291.13
  • LY 79771

    CAS:
    <p>LY-79771, a phenethanolamine antiobesity agent, can be effective in preventing fat regain following energy deprivation.</p>
    Fórmula:C18H24ClNO2
    Forma y color:Solid
    Peso molecular:321.84
  • ML350

    CAS:
    <p>ML350 (CYM-50202) is a potent KOR antagonist (IC50: 12.6 nM), selective over DOR/MOR, with high solubility and CNS penetration, lacking long-term effects.</p>
    Fórmula:C18H26BrN3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:412.32
  • 2-Methyldecanenitrile

    CAS:
    <p>2-Methyldecanenitrile, intense peach scent with lactone notes, stable in all pH, effective at low concentration.</p>
    Fórmula:C11H21N
    Pureza:98%
    Forma y color:Colourless Liquid Liquid
    Peso molecular:167.29
  • GA11

    CAS:
    <p>GA11is an inhibitor of ALDH1. It also displays anti-GBM effects in vitro and in vivo.</p>
    Fórmula:C19H14N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:270.33
  • Chlorambucyl-proline

    CAS:
    <p>Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.</p>
    Fórmula:C19H26Cl2N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:401.33
  • Otamixaban

    CAS:
    Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.
    Fórmula:C25H26N4O4
    Pureza:98.08%
    Forma y color:Solid
    Peso molecular:446.5
  • FASN-IN-5

    CAS:
    <p>FASN-IN-5 is a FASN inhibitor, useful for studying cancer and metabolic diseases.</p>
    Fórmula:C29H26N4O2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:462.54
  • A 85 4777

    CAS:
    <p>A 85 4777, a homoperazine derivative, is an anti-inflammatory agent with nonclassical immunosuppressive properties.</p>
    Fórmula:C20H32N2O2
    Forma y color:Solid
    Peso molecular:332.48
  • Ciraparantag TFA

    CAS:
    <p>Ciraparantag TFA reverses anticoagulants by inhibiting thrombin and factor Xa.</p>
    Fórmula:C26H50F6N12O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:740.74
  • NP603

    CAS:
    <p>NP603 is a cell-permeable inhibitor of FGFR1, PDGFRβ, and VEGFR2 that binds to the ATP pocket. It also is a very weak EGFR inhibitor.</p>
    Fórmula:C26H26N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.49
  • MRL-871

    CAS:
    <p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>
    Fórmula:C22H12ClF3N2O3
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:444.79
  • Transketolase-IN-4

    CAS:
    <p>Transketolase-IN-4: IC50 3.9 μM; targets M. tuberculosis DXS (IC50 114.1 μM) &amp; hinders SW620, LS174T, MIA PaCa-2 tumor cell growth.</p>
    Fórmula:C19H14ClN3O
    Pureza:99.07%
    Forma y color:Solid
    Peso molecular:335.79
  • 7ETMC

    CAS:
    <p>7ETMC inhibits Human Cytochrome P450s 1A1/1A2 with IC50: 0.46/0.50 μM; not effective on P450s 2A6/2B1 even at 50 μM.</p>
    Fórmula:C14H12O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:212.24
  • PDE5-IN-6c

    CAS:
    <p>PDE5-IN-6c is a potent and selective inhibitor of PDE5A1.</p>
    Fórmula:C23H21ClN4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.89
  • SQ-24,798

    CAS:
    <p>SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).</p>
    Fórmula:C7H15N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:205.28
  • CG-707

    CAS:
    <p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>
    Fórmula:C20H17NO3S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:383.48
  • (R)-DNMDP

    CAS:
    <p>(R)-DNMDP is a potent and selective cancer cytotoxic agent that directly binds PDE3A and has an EC50 500-fold lower than that of (S)-DNMDP against HeLa.</p>
    Fórmula:C15H20N4O3
    Forma y color:Solid
    Peso molecular:304.34
  • MK-4409

    CAS:
    MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.
    Fórmula:C22H17ClFN3O2S
    Pureza:99.80% - 99.87%
    Forma y color:Solid
    Peso molecular:441.91
  • RV01

    CAS:
    <p>RV01, a resveratrol-like quinoline, inhibits DNA damage, ALDH2 expression, and has antioxidant and anti-inflammatory properties.</p>
    Fórmula:C17H13NO2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:263.29
  • FTX-6746

    CAS:
    <p>FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.</p>
    Fórmula:C16H7ClF2N2O
    Pureza:98.68%
    Forma y color:Solid
    Peso molecular:316.69
  • Tilivapram

    CAS:
    <p>Tilivapram is a PDE4 (phosphodiesterase IV) inhibitor that can be used in the study of mental illness.</p>
    Fórmula:C16H15Cl2N3O4
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:384.21
  • Tritoqualine

    CAS:
    <p>Tritoqualine is used as an inhibitor of histidine decarboxylase.</p>
    Fórmula:C26H32N2O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:500.54
  • Pparδ agonist 2

    CAS:
    <p>Pparδ agonist 2 is an agonist of PPARδ.</p>
    Fórmula:C20H18F3N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:437.44
  • Enazadrem

    CAS:
    <p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>
    Fórmula:C18H25N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:299.41
  • CaV1.3 antagonist-1

    CAS:
    <p>CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.</p>
    Fórmula:C17H19ClN2O3
    Forma y color:Solid
    Peso molecular:334.8
  • STL1267

    CAS:
    <p>STL1267 is a REV-ERB agonist that crosses the blood-brain barrier and inhibits BMAL1 gene expression.</p>
    Fórmula:C17H11ClN4O
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:322.75
  • IACS-8968 S-enantiomer

    CAS:
    <p>IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Fórmula:C17H18F3N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.35
  • Angiogenesis agent 1

    CAS:
    <p>Compound C-31, a salidroside-based glycoside, activates HIF-1α and may aid in diabetic limb ischemia studies.</p>
    Fórmula:C20H24O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:376.4
  • Erythronic acid

    CAS:
    <p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>
    Fórmula:C4H8O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:136.1
  • LZWL02003

    CAS:
    <p>LZWL02003, an anti-neuroinflammatory agent, demonstrates a protective effect on MPP+-induced neuronal damage and reduces ROS expression.</p>
    Fórmula:C18H18N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:294.35
  • WAY127093B racemate

    CAS:
    <p>WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.</p>
    Fórmula:C23H28N4O4
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:424.49
  • IDO inhibitor 1

    CAS:
    <p>IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 &lt;100 nM).with potential immunomodulating and antineoplastic activities.</p>
    Fórmula:C11H13BrFN7O4S
    Pureza:99.805%
    Forma y color:Solid
    Peso molecular:438.23
  • SQ-31765

    CAS:
    <p>SQ-31765 is a blocker of benzazepine calcium channel.</p>
    Fórmula:C24H27F3N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:464.48
  • Imazodan

    CAS:
    <p>Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.</p>
    Fórmula:C13H12N4O
    Pureza:98% - 98.31%
    Forma y color:Solid
    Peso molecular:240.26
  • CYP11B2-IN-1

    CAS:
    <p>CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。</p>
    Fórmula:C18H18FN3O
    Pureza:99.79% - 99.89%
    Forma y color:Solid
    Peso molecular:311.35
  • CDC25B-IN-1

    CAS:
    <p>CDC25B-IN-1 is an inhibitor of CDC25B with a Ki of 8.5 μM. CDC25B-IN-1 increases the G2/M phase by inhibiting cell proliferation and colony formation.</p>
    Fórmula:C20H19NO3
    Pureza:97.05%
    Forma y color:Solid
    Peso molecular:321.37
  • AZD8329

    CAS:
    <p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>
    Fórmula:C25H31N3O3
    Pureza:99.31%
    Forma y color:Solid
    Peso molecular:421.53
  • 2-Hydroxy atorvastatin calcium salt

    CAS:
    <p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>
    Fórmula:C33H34FN2O60·5Ca
    Pureza:97.06%
    Forma y color:Solid
    Peso molecular:593.68
  • α-Glucosidase-IN-4

    CAS:
    α-Glucosidase-IN-4 is a potent α-glucosidase inhibitor with antihypertensive and hypoglycemic activity.
    Fórmula:C19H14O4
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:306.31
  • SRPKIN-1

    CAS:
    SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
    Fórmula:C27H21FN2O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.53
  • SK-216

    CAS:
    <p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>
    Fórmula:C29H29NNa2O6
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:533.52
  • VU0155056

    CAS:
    <p>VU0155056 is a dual PLD1/2 inhibitor with IC50 &lt; 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>
    Fórmula:C25H26N4O2
    Pureza:98.6% - 99.15%
    Forma y color:Solid
    Peso molecular:414.5
  • AGI-14100

    CAS:
    <p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>
    Fórmula:C29H22ClF4N5O3
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:599.96