
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(271 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(98 productos)
- Lípido(58 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8626 productos de "Metabolismo"
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1,2-Dipalmitoyl-sn-glycerol 3-phosphate
CAS:<p>1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.</p>Fórmula:C35H69O8PPureza:98%Forma y color:SolidPeso molecular:648.89ARN-6039
CAS:<p>ARN-6039 is an oral RORγ inverse agonist for Autoimmune Neuroinflammation, active in HEK 293 cells and CD4+T cells.</p>Fórmula:C21H21F3N2O3Forma y color:SolidPeso molecular:406.40Flurtamone
CAS:<p>Flurtamone is an agricultural chemical. Flurtamone mainly used as an herbicide.</p>Fórmula:C18H14F3NO2Pureza:98%Forma y color:SolidPeso molecular:333.30RPR132595A
CAS:RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).Fórmula:C28H30N4O6Pureza:98%Forma y color:SolidPeso molecular:518.56DC-6-14
CAS:<p>DC-6-14 is a cationic lipid known for its gene transfection activity, commonly utilized in the synthesis of liposomes.</p>Fórmula:C37H73ClN2O5Forma y color:SolidPeso molecular:661.44sEH inhibitor-17
CAS:<p>sEH inhibitor-17 (compound 4f) is an orally active soluble epoxide hydrolase (sEH) inhibitor with an IC50 value of 2.94 nM. This compound exhibits anti-inflammatory properties.</p>Fórmula:C18H21F3N2O4SForma y color:SolidPeso molecular:418.43Prothioconazole
CAS:<p>Prothioconazole (Proline 480 SC Fungicide) is a chiral triazole fungicide in plant pathogen control.</p>Fórmula:C14H15Cl2N3OSPureza:99.77%Forma y color:Un3077 9/Pg 3Peso molecular:344.26PAT-494
CAS:<p>PAT-494 is an inhibitor of type II Autotaxin.</p>Fórmula:C20H16FN3O2Pureza:98%Forma y color:SolidPeso molecular:349.36SHP2-IN-29
CAS:<p>SHP2-IN-29 (Compound 3), a potent inhibitor of SHP2, exhibits an IC 50 of 0.18 μM. Additionally, this compound demonstrates inhibitory activity against PTP1B and TCPTP, with IC 50 values of 4.27 μM and 4.74 μM, respectively.</p>Fórmula:C16H20O4Forma y color:SolidPeso molecular:276.33MDI-2268
CAS:<p>MDI-2268, an inhibitor of plasma kallikrein inhibitor 1 (PAI-1), exhibits strong antithrombotic properties. It plays a role in regulating blood coagulation by promoting fibrinolysis and is applicable in research related to deep vein thrombosis.</p>Fórmula:C10H10F3N3O3Forma y color:SolidPeso molecular:277.20Transketolase-IN-3
CAS:<p>Transketolase-IN-3: potent TK inhibitor with herbicidal effects on DS and AR, useful for herbicide research.</p>Fórmula:C20H9ClF3NO3Forma y color:SolidPeso molecular:403.74Acetaminophen mercapturate
CAS:<p>Paracetamol Mercapturate is a metabolite of Acetaminophen. It can also be used in the biological study of urinary antihypertensive drugs.</p>Fórmula:C13H16N2O5SPureza:98%Forma y color:SolidPeso molecular:312.34Leucylarginine
CAS:<p>Leucylarginine hinders antinociception induced by L-arginine.</p>Fórmula:C12H25N5O3Pureza:98%Forma y color:SolidPeso molecular:287.36Desmethylnortriptyline
CAS:<p>Desmethylnortriptyline, a tricyclic antidepressant metabolite of nortriptyline and amitriptyline, treats depression.</p>Fórmula:C18H19NPureza:98%Forma y color:SolidPeso molecular:249.35PPM1A-IN-1
CAS:<p>PPM1A-IN-1 (Compound IV-4) is an inhibitor of the PP2C Ser/Thr protein phosphatase Mg2+/Mn2+-dependent 1A. It exhibits antibacterial activity against Mycobacterium tuberculosis.</p>Fórmula:C16H15BrFNO2Forma y color:SolidPeso molecular:352.2FAAH-IN-8
CAS:<p>FAAH-IN-8 (compound 11) is a competitive inhibitor of FAAH with an IC50 of 6.7 nM and a Ki of 5 nM. It exhibits high blood-brain permeability and a significant antioxidant profile without neurotoxicity [1].</p>Fórmula:C18H14N4OForma y color:SolidPeso molecular:302.33Trimosulfa
CAS:<p>Trimosulfa is a combination of trimethoprim and sulfamethoxazole, an antibiotic combination. Sulfamethoxazole inhibits dihydropteroate synthase, while trimethoprim inhibits dihydrofolate reductase (dihydrofolate reductase), making it effective for mild to moderate bacterial infections against many Gram-negative and Gram-positive bacteria.</p>Fórmula:C24H29N7O6SPureza:99.93%Forma y color:SolidPeso molecular:543.61-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine
CAS:1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.Fórmula:C44H84NO8PPureza:98%Forma y color:SolidPeso molecular:786.11Descarbamoyl cefuroxime
CAS:Descarbamoyl cefuroxime is also an intermediate in the synthesis of cephalosporin antibiotics. Decarbamyl cefuroxime is a degradation product of cefuroxime.Fórmula:C15H15N3O7SPureza:98%Forma y color:SolidPeso molecular:381.36HSL-IN-5
CAS:<p>HSL-IN-5 (Example 21) is a hormone-sensitive lipase (HSL) inhibitor with an IC₅₀ value of 0.2 μM, suitable for diabetes research.</p>Fórmula:C18H23F3N2O4Pureza:99.96%Forma y color:SolidPeso molecular:388.38Roflumilast Impurity E
CAS:<p>Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast acts as a selective and long-acting the enzyme PDE-4 inhibitor(IC50 value of 0.8 nM).</p>Fórmula:C13H8Cl2F2N2O3Pureza:98%Forma y color:SolidPeso molecular:349.12LAPAO
CAS:<p>Lauramide propyl amine oxide is an amphoteric surfactant</p>Fórmula:C17H36N2O2Forma y color:SolidPeso molecular:300.48Dihydro Dutasteride
CAS:<p>Dihydro Dutasteride is a metabolite of Dutasteride. Dutasteride is an effective inhibitor of five α-reductase isozymes.</p>Fórmula:C27H32F6N2O2Pureza:98%Forma y color:SolidPeso molecular:530.55H-Arg-Lys-OH
CAS:<p>H-Arg-Lys-OH is a dipeptide formed from L-lysine residues and L-arginyl.</p>Fórmula:C12H26N6O3Pureza:98%Forma y color:SolidPeso molecular:302.37Sodium lauroyl glutamate
CAS:<p>Sodium lauroyl glutamate (Acylglutamate LS-11) is an amino acid detergent and increases the solubility of long-chain alkyl gallates such as alkyl gallates.</p>Fórmula:C17H30NNaO5Pureza:97.13%Forma y color:SolidPeso molecular:351.41AKU-005
CAS:<p>AKU-005 is a dual inhibitor of FAAH and MAGL, exhibiting IC50 values of 63 nM and 389 nM against rat and human FAAH, respectively. This compound has potential for researching trigeminal nociceptive hypersensitivity.</p>Fórmula:C20H21N5OForma y color:SolidPeso molecular:347.41Atorvastatin acetonide
CAS:<p>Atorvastatin acetonide, an impurity in Atorvastatin, lowers blood lipids; from patent WO2011131605A1.</p>Fórmula:C36H39FN2O5Pureza:98%Forma y color:SolidPeso molecular:598.7Proadifen
CAS:<p>Proadifen is a non-selective cytochrome P450 enzymes inhibitor, preventing some types of drug metabolism.</p>Fórmula:C23H31NO2Pureza:98%Forma y color:SolidPeso molecular:353.5ent-Tadalafil
CAS:ent-Tadalafil (ent-IC-351), compound (6S,12aS), is a inactive cis-enantiomer of compound (6R,12aS).Fórmula:C22H19N3O4Pureza:98%Forma y color:SolidPeso molecular:389.4Prasugrel chloride impurity
CAS:<p>Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.</p>Fórmula:C20H21ClFNO3SPureza:98%Forma y color:SolidPeso molecular:409.91-Decanesulfonic acid
CAS:<p>1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.</p>Fórmula:C10H22O3SForma y color:SolidPeso molecular:222.35Tolrestat
CAS:<p>Tolrestat (AY-27773) is a potent inhibitor of aldose reductase (IC50 = 35 nM).</p>Fórmula:C16H14F3NO3SPureza:98.89% - >99.99%Forma y color:SolidPeso molecular:357.35PF-05175157
CAS:<p>PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,</p>Fórmula:C23H27N5O2Pureza:98% - 99.92%Forma y color:SolidPeso molecular:405.494-POBN
CAS:<p>4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).</p>Fórmula:C7H9N3OPureza:99.60%Forma y color:White Crystalline PowderPeso molecular:151.17Calcipotriol monohydrate
CAS:<p>Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.</p>Fórmula:C27H42O4Pureza:99.95%Forma y color:SolidPeso molecular:430.62Tesaglitazar
CAS:<p>Tesaglitazar is a potent and selective peroxide PPARα / γ receptor dual agonist with a more potent affinity for PPARγ than PPARα, The EC50 values for rat PPARα</p>Fórmula:C20H24O7SPureza:99.95%Forma y color:SolidPeso molecular:408.47PCI-27483
CAS:<p>PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.</p>Fórmula:C26H24N6O9SPureza:98.55%Forma y color:SolidPeso molecular:596.57BIBB 515
CAS:<p>BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.</p>Fórmula:C22H21ClN2O2Pureza:99.68%Forma y color:SolidPeso molecular:380.87E3330
CAS:<p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>Fórmula:C21H30O6Pureza:99.52%Forma y color:SolidPeso molecular:378.463-Phenylbutyric acid
CAS:<p>3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.</p>Fórmula:C10H12O2Pureza:98.26%Forma y color:SolidPeso molecular:164.2L-m-Tyrosine
CAS:<p>L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.</p>Fórmula:C9H11NO3Pureza:99.8%Forma y color:SolidPeso molecular:181.19UK-414,495
CAS:<p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>Fórmula:C16H25N3O3SForma y color:SolidPeso molecular:339.45Darexaban glucuronide
CAS:<p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>Fórmula:C33H38N4O10Forma y color:SolidPeso molecular:650.68Sterculic acid
CAS:<p>Sterculic acid inhibits SCD1 with IC50 of 0.9μM, affecting Δ9D desaturase activity.</p>Fórmula:C19H34O2Forma y color:SolidPeso molecular:294.47hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Fórmula:C21H15ClN4O3Forma y color:SolidPeso molecular:406.82hCAI/II-IN-5
CAS:<p>hCAI/II-IN-5 inhibits human carbonic anhydrase I & II, α-Glycosidase, and AChE, for diabetes, heart failure, Alzheimer's, ulcers, epilepsy research.</p>Fórmula:C21H18Cl2N8O4S2Forma y color:SolidPeso molecular:581.45LY 56110
CAS:<p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>Fórmula:C17H12Cl2N2Pureza:98%Forma y color:SolidPeso molecular:315.2(R)-Bromoenol lactone
CAS:<p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>Fórmula:C16H13BrO2Forma y color:SolidPeso molecular:317.18LB42908
CAS:<p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>Fórmula:C32H31N5O3Forma y color:SolidPeso molecular:533.62N-Oleoyl Leucine
CAS:<p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>Fórmula:C24H45NO3Pureza:98.25%Forma y color:SolidPeso molecular:395.62Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Fórmula:C15H20O3Forma y color:SolidPeso molecular:248.32TPN729MA
CAS:<p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>Fórmula:C29H40N6O8SForma y color:SolidPeso molecular:632.7314-dehydro Zymostenol
CAS:<p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>Fórmula:C27H44OForma y color:SolidPeso molecular:384.64103D5R
CAS:<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Fórmula:C20H21N3O2Forma y color:SolidPeso molecular:335.4JBP485
CAS:<p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>Fórmula:C8H12N2O4Forma y color:SolidPeso molecular:200.19Anserinone B
CAS:<p>Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).</p>Fórmula:C11H14O4Forma y color:SolidPeso molecular:210.23EDP-305
CAS:<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92CAY10486
CAS:<p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>Fórmula:C19H19NO4Forma y color:SolidPeso molecular:325.36Valibose
CAS:<p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>Fórmula:C10H21NO6Forma y color:SolidPeso molecular:251.28(R)-Irsenontrine
CAS:<p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>Fórmula:C22H22N4O3Forma y color:SolidPeso molecular:390.44URB532
CAS:<p>URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.</p>Fórmula:C18H21NO3Pureza:98%Forma y color:SolidPeso molecular:299.36Fluindione
CAS:<p>Fluindione is a hematologic drug.</p>Fórmula:C15H9FO2Forma y color:SolidPeso molecular:240.23Glyoxalase I inhibitor 2
CAS:<p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>Fórmula:C24H23N3O4SForma y color:SolidPeso molecular:449.52DMPAC-Chol
CAS:<p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>Fórmula:C33H58N2O2Forma y color:SolidPeso molecular:514.83hCAIX-IN-7
CAS:<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Fórmula:C18H12FNO3Forma y color:SolidPeso molecular:309.29GNE-3500
CAS:<p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>Fórmula:C24H30FN3O3SForma y color:SolidPeso molecular:459.58YM-75466
CAS:<p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>Fórmula:C28H35N5O8S2Forma y color:SolidPeso molecular:633.74BMS 740808
CAS:<p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>Fórmula:C31H27F3N6O3Forma y color:SolidPeso molecular:588.58TMCB
CAS:<p>CK2 and ERK8 inhibitor</p>Fórmula:C11H9Br4N3O2Pureza:98%Forma y color:SolidPeso molecular:534.82DHODH-IN-21
CAS:<p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>Fórmula:C20H19ClF4N6O4Forma y color:SolidPeso molecular:518.85HIF-PHD-IN-2
CAS:<p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>Fórmula:C17H15N5O3SForma y color:SolidPeso molecular:369.4α-Amylase-IN-2
CAS:α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =Fórmula:C39H52BrNO4Forma y color:SolidPeso molecular:678.74HIF-1α-IN-3
CAS:<p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>Fórmula:C19H17N5O2Forma y color:SolidPeso molecular:347.37MDK-4823
CAS:<p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>Fórmula:C28H36N4OForma y color:SolidPeso molecular:444.61Enpp-1-IN-8
CAS:<p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>Fórmula:C19H26N6O4SForma y color:SolidPeso molecular:434.51FAAH-IN-7
<p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>Fórmula:C26H29N3O4Forma y color:SolidPeso molecular:447.53hCAIX-IN-3
CAS:<p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>Fórmula:C21H21BrN6O4SForma y color:SolidPeso molecular:533.4α-Glucosidase-IN-21
CAS:<p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>Fórmula:C24H23NO2SForma y color:SolidPeso molecular:389.513,3-Dimethyl-1-butanol
CAS:<p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>Fórmula:C6H14OForma y color:SolidPeso molecular:102.17IDO1-IN-15
CAS:<p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>Fórmula:C13H14BrFN6O3Forma y color:SolidPeso molecular:401.19hCAXII-IN-1
CAS:<p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>Fórmula:C20H17NO5Forma y color:SolidPeso molecular:351.35DP00477
CAS:<p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>Fórmula:C17H11ClF3N3OSForma y color:SolidPeso molecular:397.8D-threo-PPMP hydrochloride
CAS:<p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>Fórmula:C29H51ClN2O3Forma y color:SolidPeso molecular:511.19Lp-PLA2-IN-3
CAS:<p>Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.</p>Fórmula:C20H13ClF3N3O3SPureza:99.65%Forma y color:SolidPeso molecular:467.85Hydroxychlorodenafil
CAS:<p>Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>Fórmula:C19H23ClN4O3Forma y color:SolidPeso molecular:390.86HS79
CAS:<p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>Fórmula:C19H22N4SPureza:98%Forma y color:SolidPeso molecular:338.47Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Fórmula:C15H11N9OForma y color:SolidPeso molecular:333.31sEH inhibitor-14
CAS:<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Fórmula:C16H12F3N3O4Forma y color:SoildPeso molecular:367.28Enpp-1-IN-5
CAS:<p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>Fórmula:C17H26N6O4SForma y color:SolidPeso molecular:410.49mIDH1-IN-1
CAS:<p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>Fórmula:C25H27N3O5Forma y color:SolidPeso molecular:449.5Glucokinase activator 3
CAS:<p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>Fórmula:C26H33N2O9PS2Forma y color:SolidPeso molecular:612.65IDO-IN-14
CAS:<p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>Fórmula:C23H23ClN4O2Forma y color:SolidPeso molecular:422.91FXR agonist 4
<p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>Fórmula:C21H28ClN3OForma y color:SolidPeso molecular:373.92CYP1B1-IN-3
CAS:<p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>Fórmula:C20H16FN3O2S2Forma y color:SolidPeso molecular:413.49DTP348
CAS:<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Fórmula:C6H11N5O4SForma y color:SolidPeso molecular:249.25Nitrefazole
CAS:<p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>Fórmula:C10H8N4O4Forma y color:SolidPeso molecular:248.19URB-694
CAS:<p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>Fórmula:C19H21NO3Forma y color:SolidPeso molecular:311.37DGAT1-IN-3
CAS:<p>DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.</p>Fórmula:C20H19F3N4O3Forma y color:SolidPeso molecular:420.39Nampt-IN-7
CAS:<p>Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).</p>Fórmula:C20H21N5O3Forma y color:SolidPeso molecular:379.41FASN-IN-4
CAS:<p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>Fórmula:C26H27N3O4SPureza:98%Forma y color:SolidPeso molecular:477.58AMPD2 inhibitor 2
<p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>Fórmula:C26H27F2N3O3Forma y color:SolidPeso molecular:467.51ME-143
CAS:<p>ME-143, a 2nd-gen NADH oxidase inhibitor, blocks WNT/β-catenin pathway, active against various cancers in vitro/vivo.</p>Fórmula:C21H18O4Forma y color:SolidPeso molecular:334.37MDPD
CAS:<p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>Fórmula:C21H19N3O3Forma y color:SolidPeso molecular:361.39Antiproliferative agent-10
<p>Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.</p>Fórmula:C35H36Cl2N7PRuForma y color:SolidPeso molecular:757.66LY 113174
CAS:<p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>Fórmula:C17H10Cl2N2Forma y color:SolidPeso molecular:313.18FC11409B
CAS:<p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>Fórmula:C29H23BF4N2O3SForma y color:SolidPeso molecular:566.38Lp-PLA2-IN-4
CAS:<p>Lp-PLA2-IN-4, a potent inhibitor of Lp-PLA2/PAF-AH, may target Alzheimer's, atherosclerosis. (WO2021228159A1, Compound 38)</p>Fórmula:C23H18F5N3O4Forma y color:SolidPeso molecular:495.4Flutolanil
CAS:<p>Flutolanil: a fungicide targeting R. solani in rice, toxic to zebrafish.</p>Fórmula:C17H16F3NO2Forma y color:SolidPeso molecular:323.31JZP-MA-13
<p>JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.</p>Fórmula:C14H15FN4O3SForma y color:SolidPeso molecular:338.36BRD9500
CAS:<p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>Fórmula:C15H18FN3O2Forma y color:SolidPeso molecular:291.32Glyoxalase I inhibitor 4
CAS:<p>Glyoxalase I inhibitor 4 is a potent inhibitor of glyoxalase I (GLO1) (Ki: 10 nM).</p>Fórmula:C17H21IN4O8SForma y color:SolidPeso molecular:568.34BMP-22
CAS:<p>BMP-22 selectively inhibits autotaxin (IC50=170 nM), blocks LPA production and MM1 cell invasion, and reduces lung metastases in mice at 0.5 mg/kg/day.</p>Fórmula:C22H39O3PForma y color:SolidPeso molecular:382.52SAHO
CAS:<p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>Fórmula:C14H20N6O6SForma y color:SolidPeso molecular:400.41SHP2-IN-5
CAS:<p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>Fórmula:C12H8O6Forma y color:SolidPeso molecular:248.19Tebuconazole-d9
CAS:<p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>Fórmula:C16H13ClD9N3OForma y color:SolidPeso molecular:316.87CD 1530
CAS:<p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>Fórmula:C27H26O3Pureza:98.13%Forma y color:SolidPeso molecular:398.49JMS-053
CAS:<p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>Fórmula:C13H8N2O2SPureza:≥98.0%Forma y color:SolidPeso molecular:256.28Glycogen phosphorylase-IN-1
CAS:<p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>Fórmula:C17H15ClF2N4O4Pureza:97.98% - 98.15%Forma y color:SolidPeso molecular:412.78AQX-MN115
CAS:<p>AQX-MN115 is an SH2- containing inositol 5- phosphatase modulator.</p>Fórmula:C21H30O2Pureza:98%Forma y color:SolidPeso molecular:314.46Bamethan sulfate
CAS:<p>Bamethan sulfate is a Vasodilator.</p>Fórmula:C24H40N2O8SForma y color:SolidPeso molecular:516.65Ethylene thiourea
CAS:<p>Ethylene thiourea (NCIC03372) is a pesticide used in fruit and vegetable production.</p>Fórmula:C3H6N2SPureza:≥98%Forma y color:Needles Prisms From Alcohol Or Amyl AlcoholPeso molecular:102.16Pteropterin
CAS:<p>Pteropterin is an antineoplastic agent.</p>Fórmula:C29H33N9O12Pureza:98%Forma y color:SolidPeso molecular:699.63Alitame
CAS:<p>Alitame is a high-intensity sweetener and sugar substitute widely used in biochemical experiments and drug synthesis research.</p>Fórmula:C14H25N3O4SPureza:98%Forma y color:SolidPeso molecular:331.43DCYM21
CAS:<p>DCYM21: Menin-MLL inhibitor, halts leukemia cell growth with MLL changes, causing arrest and differentiation.</p>Fórmula:C26H33ClN2Pureza:98%Forma y color:SolidPeso molecular:409.01Sermetacin
CAS:<p>Sermetacin is an anti-inflammatory agent.</p>Fórmula:C22H21ClN2O6Pureza:98%Forma y color:SolidPeso molecular:444.86AZD-3289
CAS:<p>AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>Fórmula:C24H14F5N5Forma y color:SolidPeso molecular:467.39tHGA
CAS:<p>tHGA is a potent inhibitor of lipoxygenase.</p>Fórmula:C18H24O4Pureza:98%Forma y color:SolidPeso molecular:304.38GW648495
CAS:<p>GW648495 is a PfDHODH inhibitor that shows greater than 4,000-fold selectivity for the malarial enzyme.</p>Fórmula:C16H13N5Pureza:98%Forma y color:SolidPeso molecular:275.31ts-SA
CAS:<p>ts-SA is a metalloenzyme carbonic anhydrase (CA) inhibitor. It is active against 7 out of 10 human CA isoforms.</p>Fórmula:C14H15N3O5S2Pureza:98%Forma y color:SolidPeso molecular:369.42Fexaramate
CAS:<p>Fexaramate is a potent, selective agonist of farnesoid X receptor.</p>Fórmula:C31H37NO5Forma y color:SolidPeso molecular:503.63Oncrasin-72
CAS:Oncrasin-72 is an analog of oncrasin-1. It has antitumor activity mediated by JNK activation and STAT3 inhibition.Fórmula:C16H14ClNOPureza:98%Forma y color:SolidPeso molecular:271.74iGP-5
CAS:<p>iGP-5 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>Fórmula:C21H17N3O3Forma y color:SolidPeso molecular:359.38α-RA-F
CAS:<p>Alpha-RA-F increases collagen, lowers MMPs in human fibroblasts, non-toxic.</p>Fórmula:C16H16N2O4Pureza:98%Forma y color:SolidPeso molecular:300.31myomiR-IN-1
CAS:<p>myomiR-IN-1 inhibits myoD translation in C2C12 cells, doesn't affect myoD mRNA, and reduces differentiation markers.</p>Fórmula:C33H27NO6Pureza:98%Forma y color:SolidPeso molecular:533.572-Iodoestradiol
CAS:2-Iodoestradiol is an effective human sex hormone-binding globulin (SHBG) ligand.Fórmula:C18H23IO2Pureza:98%Forma y color:SolidPeso molecular:398.28OMS-824
CAS:<p>OMS-824 is a phosphodiesterase-10 inhibitor that slows or stops the hydrolysis of cAMP and cGMP.</p>Fórmula:C21H21BrN4O4Pureza:98%Forma y color:SolidPeso molecular:473.32PF-05387252
CAS:PF-05387252 is an effective and selective inhibitor of the IRAK4.Fórmula:C25H27N5O2Pureza:98%Forma y color:SolidPeso molecular:429.51AF267
CAS:<p>AF267 is a M1 muscarinic agonist that works by restoring cognitive impairments.</p>Fórmula:C10H18N2OSPureza:98%Forma y color:SolidPeso molecular:214.33Clinolamide
CAS:<p>Clinolamide is an antilipidemic agent.</p>Fórmula:C24H43NOPureza:98%Forma y color:SolidPeso molecular:361.6Dehydro-ZINC39395747
CAS:Dehydro-ZINC39395747 enhances NO in cells and inhibits cytochrome b5 reductase 3 (IC50: 9.14μM, Kd: 1.11μM).Fórmula:C12H9N3O2S2Forma y color:SolidPeso molecular:291.35Bucricaine
CAS:<p>Bucricaine is an anesthetic drug.</p>Fórmula:C17H22N2Forma y color:SolidPeso molecular:254.37Nafenopin
CAS:<p>Nafenopin is a peroxisome proliferator, it is used to promote liver tumors and has been used as an antihyperlipoproteinemic agent.</p>Fórmula:C20H22O3Pureza:98%Forma y color:SolidPeso molecular:310.39CM026
CAS:<p>CM026 inhibits ALDH1A1 selectively, binds to its aldehyde pocket uncompetitively.</p>Fórmula:C22H30N6O4Forma y color:SolidPeso molecular:442.51ABT-418
CAS:<p>ABT-418, a nicotinic acetylcholine receptor (nAchR) agonist, is used potentially for the treatment of attention deficit disorder.</p>Fórmula:C9H14N2OForma y color:SolidPeso molecular:166.22Safrazine Hydrochloride
CAS:<p>Safrazine Hydrochloride is a monoamine oxidase inhibitor (MOI) that is irreversible.</p>Fórmula:C11H17ClN2O2Forma y color:SolidPeso molecular:244.718MDK-0738
CAS:<p>MDK-0738 is a potent and selective aldo-keto reductase 1C3 inhibitor.</p>Fórmula:C15H16O3Pureza:98%Forma y color:SolidPeso molecular:244.294′-Deoxyphlorizin
CAS:<p>4'-Deoxyphlorizin inhibits glucose transport; Km 0.59 nM, Ki 0.33 nM for phlorizin hydrolase.</p>Fórmula:C21H24O9Forma y color:SolidPeso molecular:420.41CP-319340(free base)
CAS:<p>CP-319340 free base is a inhibitor of microsomal triglyceride transfer protein (MTP) .</p>Fórmula:C27H23F3N4OPureza:98%Forma y color:SolidPeso molecular:476.49MP-10 succinate
CAS:<p>MP-10 succinate is a potent and specific inhibitor of PDE10A.</p>Fórmula:C29H26N4O5Pureza:98%Forma y color:SolidPeso molecular:510.54LYPLAL1-IN-1
CAS:LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.Fórmula:C29H29N7O4Pureza:98%Forma y color:SolidPeso molecular:539.59Brocresine
CAS:<p>Brocresine is an aromatic L-amino acid decarboxylase inhibitor. It has both a peripheral and central action.</p>Fórmula:C7H8BrNO2Pureza:98%Forma y color:SolidPeso molecular:218.05NE21650
CAS:<p>NE21650, a bisphosphonate, inhibits isopentenyl diphosphate isomerase and farnesyl diphosphate synthase.</p>Fórmula:C8H13NO7P2Pureza:98%Forma y color:SolidPeso molecular:297.14Zofenoprilat arginine
CAS:<p>Zofenoprilat arginine is an antihypertensive.</p>Fórmula:C21H33N5O5S2Pureza:98%Forma y color:SolidPeso molecular:499.65ABL127
CAS:ABL127 inhibits PME-1 with IC50s of 6.4 nM in HEK293T cells and 4.2 nM in MDA-MB-231 cells.Fórmula:C17H20N2O5Pureza:98%Forma y color:SolidPeso molecular:332.35Butaperazine maleate
CAS:<p>Butaperazine maleate, a phenothiazine derivative, is an antipsychotic.</p>Fórmula:C32H39N3O9SPureza:98%Forma y color:SolidPeso molecular:641.73Albifylline
CAS:<p>Albifylline: a xanthine derivative, anti-asthmatic, reduces leukocyte adhesion, enhances liver microcirculation post-hemorrhagic shock.</p>Fórmula:C13H20N4O3Forma y color:SolidPeso molecular:280.32AHR-activator-1023
CAS:<p>AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.</p>Fórmula:C14H8Cl2N2OForma y color:SolidPeso molecular:291.13LY 79771
CAS:<p>LY-79771, a phenethanolamine antiobesity agent, can be effective in preventing fat regain following energy deprivation.</p>Fórmula:C18H24ClNO2Forma y color:SolidPeso molecular:321.84ML350
CAS:<p>ML350 (CYM-50202) is a potent KOR antagonist (IC50: 12.6 nM), selective over DOR/MOR, with high solubility and CNS penetration, lacking long-term effects.</p>Fórmula:C18H26BrN3O3Pureza:98%Forma y color:SolidPeso molecular:412.322-Methyldecanenitrile
CAS:<p>2-Methyldecanenitrile, intense peach scent with lactone notes, stable in all pH, effective at low concentration.</p>Fórmula:C11H21NPureza:98%Forma y color:Colourless Liquid LiquidPeso molecular:167.29GA11
CAS:<p>GA11is an inhibitor of ALDH1. It also displays anti-GBM effects in vitro and in vivo.</p>Fórmula:C19H14N2Pureza:98%Forma y color:SolidPeso molecular:270.33Chlorambucyl-proline
CAS:<p>Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.</p>Fórmula:C19H26Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:401.33Otamixaban
CAS:Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.Fórmula:C25H26N4O4Pureza:98.08%Forma y color:SolidPeso molecular:446.5FASN-IN-5
CAS:<p>FASN-IN-5 is a FASN inhibitor, useful for studying cancer and metabolic diseases.</p>Fórmula:C29H26N4O2Pureza:99.88%Forma y color:SolidPeso molecular:462.54A 85 4777
CAS:<p>A 85 4777, a homoperazine derivative, is an anti-inflammatory agent with nonclassical immunosuppressive properties.</p>Fórmula:C20H32N2O2Forma y color:SolidPeso molecular:332.48Ciraparantag TFA
CAS:<p>Ciraparantag TFA reverses anticoagulants by inhibiting thrombin and factor Xa.</p>Fórmula:C26H50F6N12O6Pureza:98%Forma y color:SolidPeso molecular:740.74NP603
CAS:<p>NP603 is a cell-permeable inhibitor of FGFR1, PDGFRβ, and VEGFR2 that binds to the ATP pocket. It also is a very weak EGFR inhibitor.</p>Fórmula:C26H26N2O5Pureza:98%Forma y color:SolidPeso molecular:446.49MRL-871
CAS:<p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>Fórmula:C22H12ClF3N2O3Pureza:99.66%Forma y color:SolidPeso molecular:444.79Transketolase-IN-4
CAS:<p>Transketolase-IN-4: IC50 3.9 μM; targets M. tuberculosis DXS (IC50 114.1 μM) & hinders SW620, LS174T, MIA PaCa-2 tumor cell growth.</p>Fórmula:C19H14ClN3OPureza:99.07%Forma y color:SolidPeso molecular:335.797ETMC
CAS:<p>7ETMC inhibits Human Cytochrome P450s 1A1/1A2 with IC50: 0.46/0.50 μM; not effective on P450s 2A6/2B1 even at 50 μM.</p>Fórmula:C14H12O2Pureza:98%Forma y color:SolidPeso molecular:212.24PDE5-IN-6c
CAS:<p>PDE5-IN-6c is a potent and selective inhibitor of PDE5A1.</p>Fórmula:C23H21ClN4O2Pureza:98%Forma y color:SolidPeso molecular:420.89SQ-24,798
CAS:<p>SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).</p>Fórmula:C7H15N3O2SPureza:98%Forma y color:SolidPeso molecular:205.28CG-707
CAS:<p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>Fórmula:C20H17NO3S2Pureza:98%Forma y color:SolidPeso molecular:383.48(R)-DNMDP
CAS:<p>(R)-DNMDP is a potent and selective cancer cytotoxic agent that directly binds PDE3A and has an EC50 500-fold lower than that of (S)-DNMDP against HeLa.</p>Fórmula:C15H20N4O3Forma y color:SolidPeso molecular:304.34MK-4409
CAS:MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.Fórmula:C22H17ClFN3O2SPureza:99.80% - 99.87%Forma y color:SolidPeso molecular:441.91RV01
CAS:<p>RV01, a resveratrol-like quinoline, inhibits DNA damage, ALDH2 expression, and has antioxidant and anti-inflammatory properties.</p>Fórmula:C17H13NO2Pureza:99.93%Forma y color:SolidPeso molecular:263.29FTX-6746
CAS:<p>FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.</p>Fórmula:C16H7ClF2N2OPureza:98.68%Forma y color:SolidPeso molecular:316.69Tilivapram
CAS:<p>Tilivapram is a PDE4 (phosphodiesterase IV) inhibitor that can be used in the study of mental illness.</p>Fórmula:C16H15Cl2N3O4Pureza:99.87%Forma y color:SolidPeso molecular:384.21Tritoqualine
CAS:<p>Tritoqualine is used as an inhibitor of histidine decarboxylase.</p>Fórmula:C26H32N2O8Pureza:98%Forma y color:SolidPeso molecular:500.54Pparδ agonist 2
CAS:<p>Pparδ agonist 2 is an agonist of PPARδ.</p>Fórmula:C20H18F3N3O3SPureza:98%Forma y color:SolidPeso molecular:437.44Enazadrem
CAS:<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Fórmula:C18H25N3OPureza:98%Forma y color:SolidPeso molecular:299.41CaV1.3 antagonist-1
CAS:<p>CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.</p>Fórmula:C17H19ClN2O3Forma y color:SolidPeso molecular:334.8STL1267
CAS:<p>STL1267 is a REV-ERB agonist that crosses the blood-brain barrier and inhibits BMAL1 gene expression.</p>Fórmula:C17H11ClN4OPureza:99.19%Forma y color:SolidPeso molecular:322.75IACS-8968 S-enantiomer
CAS:<p>IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Fórmula:C17H18F3N5O2Pureza:98%Forma y color:SolidPeso molecular:381.35Angiogenesis agent 1
CAS:<p>Compound C-31, a salidroside-based glycoside, activates HIF-1α and may aid in diabetic limb ischemia studies.</p>Fórmula:C20H24O7Pureza:98%Forma y color:SolidPeso molecular:376.4Erythronic acid
CAS:<p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>Fórmula:C4H8O5Pureza:98%Forma y color:SolidPeso molecular:136.1LZWL02003
CAS:<p>LZWL02003, an anti-neuroinflammatory agent, demonstrates a protective effect on MPP+-induced neuronal damage and reduces ROS expression.</p>Fórmula:C18H18N2O2Pureza:98%Forma y color:SolidPeso molecular:294.35WAY127093B racemate
CAS:<p>WAY127093B racemate is the racemate of WAY127093B. WAY127093B is a phosphodiesterase IV inhibitor with oral activity in rats and guinea pigs.</p>Fórmula:C23H28N4O4Pureza:99.67%Forma y color:SolidPeso molecular:424.49IDO inhibitor 1
CAS:<p>IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 <100 nM).with potential immunomodulating and antineoplastic activities.</p>Fórmula:C11H13BrFN7O4SPureza:99.805%Forma y color:SolidPeso molecular:438.23SQ-31765
CAS:<p>SQ-31765 is a blocker of benzazepine calcium channel.</p>Fórmula:C24H27F3N2O4Pureza:98%Forma y color:SolidPeso molecular:464.48Imazodan
CAS:<p>Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.</p>Fórmula:C13H12N4OPureza:98% - 98.31%Forma y color:SolidPeso molecular:240.26CYP11B2-IN-1
CAS:<p>CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。</p>Fórmula:C18H18FN3OPureza:99.79% - 99.89%Forma y color:SolidPeso molecular:311.35CDC25B-IN-1
CAS:<p>CDC25B-IN-1 is an inhibitor of CDC25B with a Ki of 8.5 μM. CDC25B-IN-1 increases the G2/M phase by inhibiting cell proliferation and colony formation.</p>Fórmula:C20H19NO3Pureza:97.05%Forma y color:SolidPeso molecular:321.37AZD8329
CAS:<p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>Fórmula:C25H31N3O3Pureza:99.31%Forma y color:SolidPeso molecular:421.532-Hydroxy atorvastatin calcium salt
CAS:<p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>Fórmula:C33H34FN2O60·5CaPureza:97.06%Forma y color:SolidPeso molecular:593.68α-Glucosidase-IN-4
CAS:α-Glucosidase-IN-4 is a potent α-glucosidase inhibitor with antihypertensive and hypoglycemic activity.Fórmula:C19H14O4Pureza:99.69%Forma y color:SolidPeso molecular:306.31SRPKIN-1
CAS:SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).Fórmula:C27H21FN2O3SPureza:98%Forma y color:SolidPeso molecular:472.53SK-216
CAS:<p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>Fórmula:C29H29NNa2O6Pureza:98.29%Forma y color:SolidPeso molecular:533.52VU0155056
CAS:<p>VU0155056 is a dual PLD1/2 inhibitor with IC50 < 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>Fórmula:C25H26N4O2Pureza:98.6% - 99.15%Forma y color:SolidPeso molecular:414.5AGI-14100
CAS:<p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>Fórmula:C29H22ClF4N5O3Pureza:99.91%Forma y color:SolidPeso molecular:599.96

