GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.024 productos)
- Receptor de adenosina(249 productos)
- Receptor adrenérgico(3.030 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(159 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(217 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(443 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(22 productos)
- Receptor de glucagón(196 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(42 productos)
- Receptor de opioides(326 productos)
- PAFR(14 productos)
- PKA(54 productos)
- Receptor S1P(17 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5981 productos de "GPCR / proteína G"
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CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Fórmula:C15H18Cl2N4OPureza:99.5%Forma y color:SolidPeso molecular:341.24Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Fórmula:C18H18ClNS·HClPureza:99.76%Forma y color:White PowderPeso molecular:352.32Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Fórmula:C26H35NO7Pureza:98.53% - 99.43%Forma y color:CoaPeso molecular:473.57Amiselimod hydrochloride
CAS:Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Fórmula:C19H31ClF3NO3Pureza:99.55%Forma y color:SolidPeso molecular:413.9Ref: TM-T10305
1mg38,00€2mg49,00€5mg80,00€10mg120,00€25mg215,00€50mg354,00€100mg512,00€200mg738,00€1mL*10mM (DMSO)88,00€Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Fórmula:C19H21NSPureza:99.93%Forma y color:SolidPeso molecular:295.44Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Forma y color:White Or Almost White Crystalline PowderPeso molecular:463.79CYM 50769
CAS:CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).Fórmula:C24H17ClN2O3Pureza:98% - 99.08%Forma y color:SolidPeso molecular:416.86Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Forma y color:White Crystalline PowderPeso molecular:313.86Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Forma y color:SolidPeso molecular:307.39ML-180
CAS:ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .Fórmula:C20H25ClN4O2Pureza:99.74%Forma y color:SolidPeso molecular:388.89Ref: TM-T12075
1mg35,00€2mg52,00€5mg77,00€10mg114,00€25mg207,00€50mg363,00€100mg550,00€1mL*10mM (DMSO)86,00€hGPR91 antagonist 1
CAS:hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).Fórmula:C31H23F4N3OPureza:98.89%Forma y color:SolidPeso molecular:529.53Ref: TM-T11560
1mg90,00€5mg192,00€10mg281,00€25mg480,00€50mg655,00€100mg888,00€1mL*10mM (DMSO)212,00€Alfuzosin hydrochloride
CAS:Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).Fórmula:C19H27N5O4·HClPureza:99.78%Forma y color:White To Off-White SolidPeso molecular:425.91KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Fórmula:C26H40N4O8Pureza:98.46%Forma y color:SolidPeso molecular:536.62Ref: TM-T15656
1mg109,00€2mg158,00€5mg260,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€1mL*10mM (DMSO)305,00€Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Forma y color:SolidPeso molecular:449.4Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:98.55%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Forma y color:Colorless To Pink SolidPeso molecular:495.53Ref: TM-T1504
5mg35,00€10mg52,00€25mg78,00€50mg96,00€100mg104,00€200mg133,00€1500mg267,00€1mL*10mM (DMSO)38,00€Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Forma y color:White Or Kind Of White PowderPeso molecular:287.36Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Forma y color:White To Off-White Crystalline PowderPeso molecular:383.51Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Fórmula:C19H26ClNO2Pureza:99.35%Forma y color:SolidPeso molecular:335.87Noradrenaline bitartrate
CAS:Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.Fórmula:C12H19NO10Pureza:99.53% - >99.99%Forma y color:SolidPeso molecular:337.28Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H11ClFNO2Pureza:99.98%Forma y color:SoildPeso molecular:231.65Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:99.99% - >99.99%Forma y color:SolidPeso molecular:367.87Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Forma y color:White Crystalline PowderPeso molecular:341.43Salmeterol
CAS:Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.Fórmula:C25H37NO4Pureza:99.2% - 99.9%Forma y color:SolidPeso molecular:415.57Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Forma y color:PowderPeso molecular:522.55Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFórmula:C17H19N3·HClPureza:98% - 99.53%Forma y color:White Or Almost White Crystalline PowderPeso molecular:301.82Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Fórmula:C13H16N4Pureza:98.34% - 99.73%Forma y color:SolidPeso molecular:228.29Senktide acetate
Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.Fórmula:C42H59N7O13SPureza:98.26%Forma y color:SolidPeso molecular:902.02Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Forma y color:Colourless Flake Crystalline SolidPeso molecular:448.39Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Forma y color:SolidPeso molecular:461.81(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H10FNO2Pureza:97.82%Forma y color:SoildPeso molecular:195.19Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Fórmula:C17H22Cl2N4Pureza:99.79%Forma y color:SolidPeso molecular:353.29AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Fórmula:C17H14O5Pureza:97.59%Forma y color:SolidPeso molecular:298.29Ref: TM-T14148
1mg35,00€5mg66,00€10mg96,00€25mg168,00€50mg264,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)71,00€Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFórmula:C10H13NO4Pureza:98.95% - 99.86%Forma y color:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Forma y color:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:99.08%Forma y color:SolidPeso molecular:631.59Ref: TM-T11174
5mg52,00€10mg80,00€25mg144,00€50mg205,00€100mg324,00€200mg477,00€1mL*10mM (DMSO)73,00€Olinciguat
CAS:Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.Fórmula:C21H16F5N7O3Pureza:99.33% - 99.71%Forma y color:SolidPeso molecular:509.39Ref: TM-T16383
1mg178,00€5mg454,00€10mg655,00€25mg1.026,00€50mg1.406,00€100mg1.863,00€1mL*10mM (DMSO)502,00€Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Fórmula:C9H15ClNO5PPureza:99.84%Forma y color:SolidPeso molecular:283.65MP-A08
CAS:MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.Fórmula:C27H25N3O4S2Pureza:97.44%Forma y color:SolidPeso molecular:519.64Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Fórmula:C16H26ClNO3Pureza:99.94% - ≥95%Forma y color:SolidPeso molecular:315.84YNT-185
CAS:YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,Fórmula:C33H37N5O5SPureza:99.67%Forma y color:SolidPeso molecular:615.74Phenothiazine
CAS:Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.Fórmula:C12H9NSPureza:99.95%Forma y color:Yellow Solid PelletsPeso molecular:199.27NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Fórmula:C20H24ClN3OPureza:99.56%Forma y color:SolidPeso molecular:357.88Ref: TM-T12207
1mg74,00€5mg140,00€10mg215,00€25mg373,00€50mg522,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)156,00€Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Forma y color:SolidPeso molecular:266.55Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Forma y color:SolidPeso molecular:395.43Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Forma y color:SolidPeso molecular:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Fórmula:C21H24ClNOPureza:99.77% - >99.99%Forma y color:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Forma y color:SolidPeso molecular:384.9Ezlopitant
CAS:Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.Fórmula:C31H38N2OPureza:97.49%Forma y color:SolidPeso molecular:454.65
