
GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(249 productos)
- Receptor adrenérgico(3.018 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(158 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(217 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(23 productos)
- Receptor de glucagón(194 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(327 productos)
- PAFR(14 productos)
- PKA(60 productos)
- Receptor S1P(18 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5983 productos de "GPCR / proteína G"
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Phenoxybenzamine hydrochloride
CAS:Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.Fórmula:C18H23Cl2NOPureza:98.04% - >99.99%Forma y color:Antihypertensive DrugPeso molecular:340.3Ornidazole
CAS:Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.Fórmula:C7H10ClN3O3Pureza:99.47%Forma y color:Crystalline SolidPeso molecular:219.63Iobenguane sulfate
CAS:Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.Fórmula:C8H10IN3H2O4SPureza:99.04%Forma y color:SolidPeso molecular:324.12Ref: TM-T15588
5mg66,00€10mg96,00€25mg197,00€50mg354,00€100mg530,00€500mg1.153,00€1mL*10mM (DMSO)73,00€Relamorelin
CAS:Relamorelin(BIM28131, RM131) is a selective and potent ghrelin/growth hormone secretagogue receptor (GHSR) agonist.Cost-effective and quality-assured.Fórmula:C43H50N8O5SPureza:99.26% - >99.99%Forma y color:SolidPeso molecular:790.97Clozapine
CAS:Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Fórmula:C18H19ClN4Pureza:99.91% - 99.93%Forma y color:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecular:326.82Ref: TM-T0455
1g425,00€10mg34,00€25mg49,00€50mg66,00€100mg90,00€200mg161,00€500mg286,00€1mL*10mM (DMSO)44,00€Strontium ranelate
CAS:Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.Fórmula:C12H6N2O8S·2SrPureza:98.97%Forma y color:Crystalline SolidPeso molecular:513.49Isoprenaline hydrochloride
CAS:Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.Fórmula:C11H18ClNO3Pureza:98% - 99.65%Forma y color:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Peso molecular:247.719Ozagrel
CAS:Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of
Fórmula:C13H12N2O2Pureza:97.90% - 99.38%Forma y color:White PowderPeso molecular:228.25Molindone hydrochloride
CAS:Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.
Fórmula:C16H24N2O2·HClPureza:99% - 99.99%Forma y color:SolidPeso molecular:312.84Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Fórmula:C84H107ClN18O18Pureza:98.66%Forma y color:SolidPeso molecular:1692.34Paliperidone
CAS:Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Fórmula:C23H27FN4O3Pureza:95% - 99.08%Forma y color:Off White To Light Orange Coloured SolidPeso molecular:426.48Roluperidone
CAS:Roluperidone (CYR-101) is a novel cyclic amide derivative.Fórmula:C22H23FN2O2Pureza:96.08% - 97.77%Forma y color:SolidPeso molecular:366.43ML-109
CAS:ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
Fórmula:C31H29N3O5Pureza:98.63%Forma y color:SolidPeso molecular:523.58Tolamolol
CAS:Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in theFórmula:C19H24N2O4Pureza:98.59%Forma y color:SolidPeso molecular:344.4Tenilapine
CAS:Tenilapine is a neuroleptic compound that can be used to study atypical antipsychotics.Fórmula:C17H16N4S2Pureza:99.58% - >99.99%Forma y color:SoildPeso molecular:340.47(±) Clopidogrel hydrogen sulfate
CAS:(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clotsFórmula:C16H16ClNO2S·H2SO4Pureza:98.67% - 99.04%Forma y color:Colorless To Light Yellow LiquidPeso molecular:419.9Triprolidine hydrochloride monohydrate
CAS:Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Fórmula:C19H25ClN2OPureza:99.68% - 99.81%Forma y color:White Crystalline PowderPeso molecular:332.87Tegaserod maleate
CAS:Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.Fórmula:C20H27N5O5Pureza:98% - 99.06%Forma y color:White PowderPeso molecular:417.46Ref: TM-T1551
10mg44,00€25mg74,00€50mg113,00€100mg188,00€200mg285,00€500mg482,00€1mL*10mM (DMSO)48,00€GANT 58
CAS:GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).Fórmula:C24H16N4SPureza:99.53%Forma y color:SolidPeso molecular:392.48GTS-21 dihydrochloride
CAS:GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.Fórmula:C19H20N2O2·2HClPureza:98.54% - >99.99%Forma y color:SolidPeso molecular:381.3Ref: TM-T2663
5mg51,00€10mg85,00€25mg115,00€50mg144,00€100mg216,00€200mg325,00€500mg545,00€1mL*10mM (DMSO)57,00€
