GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(249 productos)
- Receptor adrenérgico(3.022 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(158 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(217 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(23 productos)
- Receptor de glucagón(194 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(327 productos)
- PAFR(14 productos)
- PKA(60 productos)
- Receptor S1P(18 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5983 productos de "GPCR / proteína G"
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6-Iodopravadoline
CAS:6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.Fórmula:C23H25IN2O3Pureza:99.29%Forma y color:Off-White SolidPeso molecular:504.36Ref: TM-T14204
1mg38,00€2mg52,00€5mg70,00€10mg90,00€25mg198,00€50mg326,00€100mg520,00€1mL*10mM (DMSO)99,00€Clopidogrel hydrogen sulfate
CAS:Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.Fórmula:C16H16ClNO2S·H2SO4Pureza:99.57% - 99.79%Forma y color:SolidPeso molecular:419.9Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Fórmula:C24H29ClF3N5O5SPureza:97.91%Forma y color:SoildPeso molecular:592.03Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Fórmula:C72H95ClN14O14Pureza:>99.99%Forma y color:SolidPeso molecular:1416.06AM-8123
CAS:AM-8123: oral APJ agonist, potent, inhibits cAMP, activates Gα, key for cardiovascular research.Fórmula:C27H33N7O5SPureza:99.59% - 99.76%Forma y color:SolidPeso molecular:567.66Rebamipide
CAS:Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.Fórmula:C19H15ClN2O4Pureza:99.48% - 99.61%Forma y color:White PowderPeso molecular:370.79Midodrine hydrochloride
CAS:Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.
Fórmula:C12H19ClN2O4Pureza:99.79% - >99.99%Forma y color:Crystalline SolidPeso molecular:290.74Paroxetine hydrochloride
CAS:Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.Fórmula:C19H21ClFNO3Pureza:98% - 99.99%Forma y color:White Crystalline PowderPeso molecular:365.826Sertraline hydrochloride
CAS:Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.Fórmula:C17H18Cl3NPureza:99.12% - 99.99%Forma y color:Solid PowderPeso molecular:342.69Ref: TM-T0482
5mg49,00€10mg59,00€25mg98,00€50mg170,00€100mg222,00€200mg289,00€500mg487,00€1mL*10mM (DMSO)54,00€Iobenguane sulfate
CAS:Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.Fórmula:C8H10IN3H2O4SPureza:99.04%Forma y color:SolidPeso molecular:324.12Ref: TM-T15588
5mg66,00€10mg96,00€25mg197,00€50mg354,00€100mg530,00€500mg1.153,00€1mL*10mM (DMSO)73,00€Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Fórmula:C21H27N3O5Pureza:99.51% - 99.7%Forma y color:White Crystalline PowderPeso molecular:401.47Aripiprazole Lauroxil
CAS:Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Fórmula:C36H51Cl2N3O4Pureza:99.64%Forma y color:SolidPeso molecular:660.71Ref: TM-T14319
10mg46,00€25mg69,00€50mg90,00€100mg123,00€200mg178,00€500mg300,00€1mL*10mM (DMSO)50,00€p-MPPI hydrochloride
CAS:p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Fórmula:C25H28ClIN4O2Pureza:99.95%Forma y color:SolidPeso molecular:578.87Ref: TM-T16421
2mg38,00€5mg56,00€10mg88,00€25mg138,00€50mg222,00€100mg351,00€200mg522,00€1mL*10mM (DMSO)94,00€Efloxate
CAS:Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.Fórmula:C19H16O5Pureza:99.66%Forma y color:SolidPeso molecular:324.33Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Fórmula:C21H26NO10PPureza:97.04%Forma y color:SoildPeso molecular:483.41(R)-Terazosin
CAS:R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).Fórmula:C19H25N5O4Pureza:98.96% - 99.79%Forma y color:SolidPeso molecular:387.43Ref: TM-T12643
1mg44,00€2mg60,00€5mg90,00€10mg138,00€25mg227,00€50mg334,00€100mg469,00€500mgA consultar1mL*10mM (DMSO)100,00€Carebastine
CAS:Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.Fórmula:C32H37NO4Pureza:99.16%Forma y color:Off-White SolidPeso molecular:499.64Cinnarizine
CAS:Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Fórmula:C26H28N2Pureza:99.94%Forma y color:SolidPeso molecular:368.51Tetrabenazine
CAS:Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Fórmula:C19H27NO3Pureza:98% - 99.91%Forma y color:White To Off-White White To Off-White SolidPeso molecular:317.42Mianserin hydrochloride
CAS:Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Fórmula:C18H21ClN2Pureza:99.63% - 99.82%Forma y color:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedPeso molecular:300.83
