GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(251 productos)
- Receptor adrenérgico(3.028 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(158 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(218 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(36 productos)
- GRK(33 productos)
- GTPasa(23 productos)
- Receptor de glucagón(195 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(42 productos)
- Receptor de opioides(327 productos)
- PAFR(14 productos)
- PKA(61 productos)
- Receptor S1P(18 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
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Se han encontrado 6012 productos de "GPCR / proteína G"
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Gemeprost
CAS:Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.Fórmula:C23H38O5Pureza:98%Forma y color:SolidPeso molecular:394.54PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFórmula:C123H215N39O28SPureza:98%Forma y color:SolidPeso molecular:2720.33A 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Fórmula:C22H22ClNForma y color:SolidPeso molecular:335.87Ethoxyquin Dimer
CAS:Ethoxyquin dimer is an antioxidant, metabolite of ethoxyquin, that protects fish meal/oil fats but can cause liver damage in mice.Fórmula:C28H36N2O2Forma y color:SolidPeso molecular:432.608Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2
CAS:Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2 is a biologically active peptide functioning as a selective agonist for Protease Activated Receptor 1 (PAR-1), a subtypeFórmula:C42H63FN12O8Forma y color:SolidPeso molecular:883.02(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.Fórmula:C54H76N14O11Forma y color:SolidPeso molecular:1097.27Cannabigerorcinic Acid
CAS:Cannabigerorcinic acid, structurally akin to recognized phytocannabinoids, serves as an analytical reference standard designed for research and forensic purposes.Fórmula:C18H24O4Forma y color:SolidPeso molecular:304.386PAMP-12(human, porcine)
CAS:Potent endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 57.2 nM). Corresponds to amino acids 9 to 20 of proadrenomedullin.Fórmula:C77H119N25O14Pureza:98%Forma y color:SolidPeso molecular:1618.95W140 HBr
CAS:[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.Fórmula:C16H28BrN2O4PPureza:99.85%Forma y color:SoildPeso molecular:423.28Ref: TM-T60204
1mg115,00€2mg172,00€5mg255,00€1mL*10mM (DMSO)284,00€10mg375,00€25mg562,00€50mg787,00€100mg1.074,00€GEP44
GEP44 is a peptide-biased triple agonist targeting the glucagon-like peptide-1 receptor (GLP-1R), neuropeptide Y1 receptor (Y1-R), and neuropeptide Y2 receptor (Y2-R). It induces GLP-1R-dependent insulin secretion in rat and human islets by offsetting the actions of Y1-R and GLP-1R agonism, controlled by Y1-R antagonists. Additionally, GEP44 enhances glucose uptake in muscle tissue through Y1-R mediation independent of insulin and significantly reduces food intake and body weight in diet-induced obese rat models. GEP44 is utilized in studies related to obesity and type 2 diabetes.Forma y color:Odour Solid3-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Fórmula:C19H19ClN2OForma y color:SolidPeso molecular:326.82Nesiritide acetate
CAS:Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.Fórmula:C143H244N50O42S4C2H4O2Forma y color:SolidPeso molecular:3524.1meta-Fluoxetine (hydrochloride)
CAS:meta-Fluoxetine (hydrochloride) can be used in related research in the field of life sciences. Its product number is T37474 and CAS number is 79088-29-2.Fórmula:C17H19ClF3NOForma y color:SolidPeso molecular:345.79Prostaglandin F2α 1,11-lactone
CAS:Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.Fórmula:C20H32O4Pureza:98%Forma y color:SolidPeso molecular:336.47GRP (porcine)
CAS:GRP: agonist for GRPR, stimulates amygdala GABA release reducing fear in mice, aids mitogenesis, GI function, and appetite control.Fórmula:C126H198N38O31S2Pureza:98%Forma y color:SolidPeso molecular:2805.315-HT5AR/5-HT6R ligand-1
5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.Fórmula:C25H30N4O2SForma y color:SolidPeso molecular:450.6Kisspeptin 13
CAS:Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Fórmula:C78H107N21O18Forma y color:SolidPeso molecular:1626.8111β-Prostaglandin E2
CAS:11β-PGE2 is the C-11 epimer of PGE2.Fórmula:C20H32O5Forma y color:SolidPeso molecular:352.47BNP (1-21), Pro (Human)
CAS:BNP (1-21), Pro (Human) is a 21-amino acid peptide and a form of B-Type Natriuretic Peptide (BNP), a cardiac natriuretic hormone.Fórmula:C89H144N28O35Peso molecular:2166.26β-MSH, human
CAS:beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).Fórmula:C118H174N34O35SPureza:98%Forma y color:SolidPeso molecular:2660.92
