GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(248 productos)
- Receptor adrenérgico(3.031 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(154 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(216 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(22 productos)
- Receptor de glucagón(191 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(325 productos)
- PAFR(14 productos)
- PKA(59 productos)
- Receptor S1P(17 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5963 productos de "GPCR / proteína G"
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AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Fórmula:C17H14O5Pureza:97.59%Forma y color:SolidPeso molecular:298.29Ref: TM-T14148
1mg35,00€5mg66,00€10mg96,00€25mg168,00€50mg264,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)71,00€Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Forma y color:White Or Kind Of White PowderPeso molecular:287.36(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:99.08%Forma y color:SolidPeso molecular:631.59Ref: TM-T11174
5mg50,00€10mg75,00€25mg137,00€50mg195,00€100mg306,00€200mg452,00€1mL*10mM (DMSO)70,00€Quetiapine
CAS:Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Forma y color:White To Off-White Crystalline PowderPeso molecular:383.51Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Fórmula:C16H26ClNO3Pureza:99.94% - ≥95%Forma y color:SolidPeso molecular:315.84Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Fórmula:C19H23NO·HClPureza:98.72%Forma y color:SolidPeso molecular:317.85Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Noradrenaline bitartrate
CAS:Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.Fórmula:C12H19NO10Pureza:99.53% - >99.99%Forma y color:SolidPeso molecular:337.28Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:99.99% - >99.99%Forma y color:SolidPeso molecular:367.87Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:98.55%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFórmula:C10H13NO4Pureza:98.95% - 99.86%Forma y color:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Fórmula:C26H27N5O2Pureza:99.61%Forma y color:Light Yellow SolidPeso molecular:441.52Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Forma y color:White Or Almost White Crystalline PowderPeso molecular:463.79Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Forma y color:SolidPeso molecular:266.55Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Forma y color:Colorless To Pink SolidPeso molecular:495.53Ref: TM-T1504
5mg34,00€10mg50,00€25mg73,00€50mg92,00€100mg99,00€200mg126,00€1500mg267,00€1mL*10mM (DMSO)35,00€KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Fórmula:C26H40N4O8Pureza:98.46%Forma y color:SolidPeso molecular:536.62Ref: TM-T15656
1mg109,00€2mg158,00€5mg260,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€1mL*10mM (DMSO)305,00€Cisapride
CAS:Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.Fórmula:C23H29ClFN3O4Pureza:99.77%Forma y color:White To Slightly Biege Powder SolidPeso molecular:465.95Ref: TM-T1291
5mg47,00€10mg59,00€25mg77,00€50mg99,00€100mg135,00€200mg235,00€500mg394,00€1mL*10mM (DMSO)55,00€Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Forma y color:White Crystalline PowderPeso molecular:313.86Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Forma y color:SolidPeso molecular:307.39DPTN dihydrochloride
CAS:DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Fórmula:C22H20Cl2N4OSPureza:99.95%Forma y color:SoildPeso molecular:459.39
