GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.043 productos)
- Receptor de adenosina(214 productos)
- Receptor adrenérgico(3.182 productos)
- Receptor de bombesina(37 productos)
- Receptor de bradicinina(63 productos)
- CXCR(167 productos)
- CaSR(31 productos)
- Receptor de cannabinoides(223 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(85 productos)
- Receptor GNRH(89 productos)
- GPCR19(38 productos)
- GRK(41 productos)
- GTPasa(24 productos)
- Receptor de glucagón(203 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(389 productos)
- Receptor LPA(22 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(54 productos)
- Receptor de opioides(332 productos)
- PAFR(12 productos)
- PKA(57 productos)
- Receptor S1P(21 productos)
- SGLT(32 productos)
- Receptor sigma(48 productos)
Mostrar 19 subcategorías más
Se han encontrado 5952 productos para "GPCR / proteína G".
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Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H11ClFNO2Pureza:99.98%Forma y color:SolidPeso molecular:231.65Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:99.99% - >99.99%Forma y color:White SolidPeso molecular:367.87Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Fórmula:C22H23N3O2Pureza:99.29% - 99.97%Forma y color:White SolidPeso molecular:361.44Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Forma y color:SolidPeso molecular:266.55Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Forma y color:White SolidPeso molecular:448.39(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFórmula:C10H10FNO2Pureza:97.82%Forma y color:SolidPeso molecular:195.19AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Fórmula:C17H14O5Pureza:97.59%Forma y color:SolidPeso molecular:298.29Ref: TM-T14148
1mg34,00€5mg63,00€1mL*10mM (DMSO)67,00€10mg92,00€25mg165,00€50mg250,00€100mg401,00€200mg580,00€Phenothiazine
CAS:Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.Fórmula:C12H9NSPureza:99.95%Forma y color:SolidPeso molecular:199.27Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Forma y color:White SolidPeso molecular:260.3Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Forma y color:SolidPeso molecular:384.99-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFórmula:C10H13N5Pureza:99.98%Forma y color:White SolidPeso molecular:203.24Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Forma y color:White SolidPeso molecular:287.36PF429242 dihydrochloride
CAS:PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).Fórmula:C25H37Cl2N3O2Pureza:99.68%Forma y color:White ViscousPeso molecular:482.49KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Fórmula:C26H40N4O8Pureza:98.46%Forma y color:SolidPeso molecular:536.62Ref: TM-T15656
1mg109,00€2mg158,00€5mg260,00€1mL*10mM (DMSO)305,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€Olinciguat
CAS:Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.Fórmula:C21H16F5N7O3Pureza:99.33% - 99.97%Forma y color:SolidPeso molecular:509.39Ref: TM-T16383
1mg170,00€5mg430,00€1mL*10mM (DMSO)475,00€10mg620,00€25mg973,00€50mg1.333,00€100mg1.765,00€Succinate/succinate receptor antagonist 1
CAS:Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.Fórmula:C17H15N3OPureza:99.53%Forma y color:SolidPeso molecular:277.32Ref: TM-T67915
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg86,00€25mg161,00€50mg245,00€100mg363,00€200mg515,00€MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Fórmula:C24H26F3N3O4Pureza:99.98%Forma y color:SolidPeso molecular:477.48Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Fórmula:C24H28N2O3Pureza:99.60% - 99.96%Forma y color:SolidPeso molecular:392.49Fluoxetine
CAS:Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.Fórmula:C17H18F3NOPureza:99.07% - 99.28%Forma y color:Transparent LiquidPeso molecular:309.33Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Fórmula:C17H20N4SPureza:99.86% - ≥95%Forma y color:SolidPeso molecular:312.43
