GPCR / proteína G
Los inhibidores de GPCR/proteínas G son compuestos que se dirigen a los receptores acoplados a proteínas G (GPCR) y a las proteínas G asociadas, que desempeñan roles cruciales en la transmisión de señales desde el exterior hacia el interior de las células. Estos inhibidores son esenciales para estudiar las vías de señalización mediadas por los GPCR, que están involucradas en numerosos procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la neurotransmisión. Los inhibidores de GPCR también son importantes en el desarrollo de fármacos, ya que muchos agentes terapéuticos tienen como objetivo estos receptores. En CymitQuimica, ofrecemos una amplia gama de inhibidores de GPCR/proteínas G de alta calidad para apoyar su investigación en farmacología, biología celular y campos relacionados.
Subcategorías de "GPCR / proteína G"
- Receptor 5-HT(1.025 productos)
- Receptor de adenosina(248 productos)
- Receptor adrenérgico(2.994 productos)
- Receptor de bombesina(35 productos)
- Receptor de bradicinina(61 productos)
- CXCR(154 productos)
- CaSR(34 productos)
- Receptor de cannabinoides(216 productos)
- Colecistoquinina(1 productos)
- Receptor de dopamina(445 productos)
- Receptor de endotelina(86 productos)
- Receptor GNRH(84 productos)
- GPCR19(33 productos)
- GRK(33 productos)
- GTPasa(23 productos)
- Receptor de glucagón(191 productos)
- Hedgehog / Smoothened(49 productos)
- Receptor de histamina(385 productos)
- Receptor LPA(21 productos)
- Receptor de melatonina(26 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(325 productos)
- PAFR(14 productos)
- PKA(59 productos)
- Receptor S1P(17 productos)
- SGLT(31 productos)
- Receptor sigma(46 productos)
Mostrar 19 subcategorías más
Se han encontrado 5964 productos de "GPCR / proteína G"
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Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Fórmula:C19H21NSPureza:99.93%Forma y color:SolidPeso molecular:295.44Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Forma y color:Colorless To Pink SolidPeso molecular:495.53Ref: TM-T1504
5mg34,00€10mg50,00€25mg73,00€50mg92,00€100mg99,00€200mg126,00€1500mg267,00€1mL*10mM (DMSO)35,00€Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Forma y color:White Or Almost White Crystalline PowderPeso molecular:463.79Acetophenazine dimaleate
CAS:Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Forma y color:SolidPeso molecular:643.71hGPR91 antagonist 1
CAS:hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).Fórmula:C31H23F4N3OPureza:98.89%Forma y color:SolidPeso molecular:529.53Ref: TM-T11560
1mg90,00€5mg192,00€10mg281,00€25mg480,00€50mg655,00€100mg888,00€1mL*10mM (DMSO)212,00€Alfuzosin hydrochloride
CAS:Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).Fórmula:C19H27N5O4·HClPureza:99.78%Forma y color:White To Off-White SolidPeso molecular:425.91Urapidil hydrochloride
CAS:Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Fórmula:C20H29N5O3·HClPureza:99.58%Forma y color:White Or Off-White Crystalline PowderPeso molecular:423.94Cefaclor monohydrate
CAS:Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.Fórmula:C15H16ClN3O5SPureza:97.36% - 99.9%Forma y color:White Crystaling PowderPeso molecular:385.82JNJ-18038683
CAS:JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Fórmula:C26H28ClN3O7Pureza:97.29%Forma y color:SolidPeso molecular:529.97Ref: TM-T11720
2mg35,00€5mg50,00€10mg90,00€25mg170,00€50mg259,00€100mg383,00€200mg545,00€1mL*10mM (DMSO)55,00€PF429242 dihydrochloride
CAS:PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Fórmula:C25H37Cl2N3O2Pureza:99.68%Forma y color:SolidPeso molecular:482.49Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFórmula:C10H13NO4Pureza:98.95% - 99.86%Forma y color:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Fórmula:C19H26ClNO2Pureza:99.35%Forma y color:SolidPeso molecular:335.87Granisetron hydrochloride
CAS:Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFórmula:C18H25ClN4OPureza:99.88% - 99.93%Forma y color:White To Off-White Crystalline SolidPeso molecular:348.87Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Forma y color:White Crystalline PowderPeso molecular:434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Fórmula:C22H29N3O4SPureza:98.55%Forma y color:Yellowish White Crystalline PowderPeso molecular:431.55Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:99.99% - >99.99%Forma y color:SolidPeso molecular:367.87Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Forma y color:White Crystalline PowderPeso molecular:313.86TSHR antagonist S37
CAS:TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).Fórmula:C25H20N2O3S2Pureza:98.35%Forma y color:SolidPeso molecular:460.57Ref: TM-T13216
1mg64,00€2mg92,00€5mg130,00€10mg200,00€25mg371,00€50mg553,00€100mg788,00€500mg1.603,00€1mL*10mM (DMSO)172,00€Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Forma y color:SolidPeso molecular:307.39Cericlamine
CAS:Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Fórmula:C12H17Cl2NOPureza:99.06%Forma y color:SolidPeso molecular:262.18
