Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(9 produits)
- BCL(1 produits)
- Caspase(154 produits)
- FOXO1(2 produits)
- IAP(67 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(135 produits)
- PDK(9 produits)
- PERK(23 produits)
- Sérine/thréonine kinase(17 produits)
- Survivant(14 produits)
- TNF(93 produits)
- c-RET(61 produits)
- p53(63 produits)
Affichez 6 plus de sous-catégories
6225 produits trouvés pour "Apoptose"
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Malachite green oxalate
CAS :Malachite green oxalate is a triphenylmethane dye which can be used to detect the release of phosphate in enzymatic reactions.Formule :C23H25N2·C2HO4C2H2O4Couleur et forme :Dark Green Crystals With A Metallic LusterMasse moléculaire :463.51RX-3117
CAS :RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog.Formule :C10H12FN3O4Degré de pureté :97.46%Couleur et forme :SolidMasse moléculaire :257.22Ref: TM-T16813
1mg148,00€2mg200,00€5mg294,00€1mL*10mM (DMSO)303,00€10mg420,00€25mg690,00€50mg964,00€100mg1.305,00€3-Dehydrotrametenolic acid
CAS :3-Dehydrotrametenolic acid is a potential anticancer agent against H-ras transformed tumor and a promising candidate for a new type of insulin-sensitizing drug.Formule :C30H46O3Degré de pureté :98.5% - 99.25%Couleur et forme :SolidMasse moléculaire :454.68Ref: TM-T5S0620
1mg46,00€5mg92,00€1mL*10mM (DMSO)108,00€10mg147,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€Cabozantinib hydrochloride
CAS :Cabozantinib hydrochloride (XL184) is a potent pan-tyrosine kinases inhibitor that inhibits VEGFR2, c-Met, Kit, Axl, and Flt4 (IC50s: 0.035, 1.3, 4.6, 7 and 6Formule :C28H25ClFN3O5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :537.96Ref: TM-T5164
1mg42,00€2mg52,00€5mg65,00€10mg92,00€25mg160,00€50mg235,00€100mg330,00€200mg538,00€500mg860,00€Enzastaurin 2HCl
CAS :Enzastaurin (DB-102/LY317615) is a macrocyclic bisindolemaleimide inhibiting protein kinase C beta to reduce tumor blood supply.Formule :C32H31Cl2N5O2Couleur et forme :SolidMasse moléculaire :588.53Polydatin
CAS :Polydatin, a resveratrol glycoside from Polygonum cuspidatum, inhibits platelet aggregation, alters lipid ratios, and modulates cell functions.Formule :C20H22O8Degré de pureté :97.2% - 98.94%Couleur et forme :White Fine PowderMasse moléculaire :390.38SC-43
CAS :SC-43 is a potent and orally active agonist of SHP-1 (PTPN6).Formule :C21H13ClF3N3O2Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :431.8Cidofovir sodium
CAS :Cidofovir sodium, an injectable antiviral for AIDS-related CMV retinitis, is a DNA polymerase inhibitor.Formule :C8H12N3Na2O6PCouleur et forme :SolidMasse moléculaire :323.1523ONO-4059 analog
CAS :ONO-4059 analog (ONO-WG-307)ue is an analogue of ONO-4059, which is a highly potent and selective oral BTK inhibitor with IC50 of 23.9 nM. Phase 1.Formule :C25H24N6O3Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :456.5Ref: TM-T6921
1mg43,00€2mg56,00€1mL*10mM (DMSO)90,00€5mg93,00€10mg137,00€25mg264,00€50mg439,00€100mg627,00€MK-8745
CAS :MK-8745 is a potent and selective Aurora A inhibitor.Formule :C20H19ClFN5OSDegré de pureté :99.09% - 99.79%Couleur et forme :SolidMasse moléculaire :431.91HS-1793
CAS :HS-1793, resveratrol-like, reduces HIF-1, VEGF in hypoxia, and curbs human breast cancer growth in mouse model.Formule :C16H12O3Degré de pureté :98.16% - 99.82%Couleur et forme :SolidMasse moléculaire :252.26Galanthamine
CAS :Galanthamine (Galantamine) is an acetylcholinesterase (AChE)inhibitor(IC50 : 500 nM), can reduce brain damage induced by hypoxia-ischemia.Formule :C17H21NO3Degré de pureté :98.03% - 99.87%Couleur et forme :Off-White SolidMasse moléculaire :287.35Cidofovir
CAS :Cidofovir ((S)-HPMPC) 通过特异性抑制病毒 DNA 合成来抑制病毒复制。Formule :C8H14N3O6PDegré de pureté :99.24% - 99.76%Couleur et forme :Fluffy White PowderMasse moléculaire :279.19STM2457
CAS :View and buy STM2457 from TargetMol.STM2457 is a first-in-class, highly potent, selective and orally active inhibitor of METTL3.Cited in 2 publications.Formule :C25H28N6O2Degré de pureté :97.44% - 98.90%Couleur et forme :SolidMasse moléculaire :444.53Cucurbitacin B
CAS :Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.Formule :C32H46O8Degré de pureté :97.1% - 99.93%Couleur et forme :SolidMasse moléculaire :558.70Citric acid
CAS :Citric acid (Citro) is a weak organic tricarboxylic acid found in citrus fruits, a food additive and a natural preservative. High-Quality, Low-Cost!Formule :C6H8O7Degré de pureté :98.88%Couleur et forme :White Solid CrystallineMasse moléculaire :192.12KRAS inhibitor-9
CAS :KRAS inhibitor-9 (DUN09716) hinders GTP-KRAS formation, with a Kd of 92 μM, causes G2/M arrest, and induces apoptosis in mutated NSC-LC cells.Formule :C13H9ClN2S2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :292.81Ref: TM-T8756
1mg57,00€2mg81,00€5mg113,00€1mL*10mM (DMSO)136,00€10mg178,00€25mg334,00€50mg485,00€100mg622,00€GSK2656157
CAS :GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay.Formule :C23H21FN6ODegré de pureté :98.59% - >99.99%Couleur et forme :SolidMasse moléculaire :416.45Ref: TM-T2654
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg77,00€25mg135,00€50mg245,00€100mg442,00€200mg598,00€PRIMA-1
CAS :PRIMA-1 (NSC-281668) is a mutant p53 reactivator. It induces apoptosis and inhibits growth of human tumors with mutant p53.Formule :C9H15NO3Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :185.22Ref: TM-T6954
5mg49,00€1mL*10mM (DMSO)54,00€10mg70,00€25mg133,00€50mg195,00€100mg349,00€200mg518,00€500mg830,00€Kinsenoside
CAS :Kinsenoside ((+)-Kinsenoside) shows significant antihepatotoxic, and anti-inflammatory activities.Formule :C10H16O8Degré de pureté :99.2% - 99.92%Couleur et forme :SolidMasse moléculaire :264.23Prexasertib dihydrochloride
CAS :Prexasertib dihydrochloride (LY2606368) inhibits CHK1 (Ki: 0.9 nM); IC50: CHK2 8 nM, RSK 9 nM.Formule :C18H21Cl2N7O2Degré de pureté :98.46% - 99.82%Couleur et forme :SolidMasse moléculaire :438.31Ref: TM-T4327
1mg43,00€2mg56,00€5mg93,00€1mL*10mM (DMSO)96,00€10mg137,00€25mg259,00€50mg405,00€100mg597,00€500mg1.251,00€5-Geranoxy-7-methoxycoumarin
CAS :5-Geranoxy-7-methoxycoumarin shows antifungal activity.Formule :C20H24O4Degré de pureté :98.94% - 99.99%Couleur et forme :SolidMasse moléculaire :328.4Ref: TM-TN3110
1mg99,00€5mg231,00€1mL*10mM (DMSO)244,00€10mg343,00€25mg575,00€50mg802,00€100mg1.108,00€GSK2983559 active metabolite
CAS :GSK2983559 active metabolite (RIPK2-IN-1) is a potent, selective receptor-interacting protein-2 (RIP2) kinase inhibitor.Formule :C21H22N4O4S2Degré de pureté :97.07% - 99.57%Couleur et forme :SolidMasse moléculaire :458.55Parthenolide
CAS :Parthenolide ((-)-Parthenolide) is a natural sesquiterpene lactone that is an NF-κB and HDAC1 inhibitor with anti-inflammatory effect. Cost-effective and quality-assured.Formule :C15H20O3Degré de pureté :98.19% - 99.46%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :248.32Fraxetin
CAS :Fraxetin (7,8-dihydroxy-6-methoxy coumarin) has dual-antioxidative ,hepatoprotective and antihyperglycemic functions, it shows potent protective effects againstFormule :C10H8O5Degré de pureté :98% - 99.84%Couleur et forme :Light Yellow Crystalline FlakesMasse moléculaire :208.17PP1
CAS :PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is 5 nM/ 6 nM, respectively.Formule :C16H19N5Degré de pureté :99% - 99.88%Couleur et forme :Off-White To Grey SolidMasse moléculaire :281.36Ref: TM-T6196
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)89,00€10mg112,00€25mg190,00€50mg268,00€100mg421,00€500mg945,00€Nystatin
CAS :Nystatin (Fungicidin) is a topical and oral antifungal agent with activity against many species of yeast and candida albicans, which is used largely to treatFormule :C47H79NO19Degré de pureté :69.55% - 99.86%Couleur et forme :Yellow SuspensionMasse moléculaire :962.137Amifostine sodium
CAS :Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formule :C5H15N2NaO3PSCouleur et forme :SolidMasse moléculaire :237.21SKLB4771
CAS :SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.Formule :C25H27N7O3S2Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :537.66Ref: TM-T2051
1mg63,00€2mg93,00€5mg124,00€1mL*10mM (DMSO)148,00€10mg177,00€25mg371,00€50mg557,00€100mg792,00€500mg1.611,00€TASIN-1 Hydrochloride
CAS :TASIN-1 Hydrochloride (TASIN-1 HCl) is a selective inhibitor of truncated APC that acts by selectively killing colorectal cancer cells that express truncatedFormule :C18H29ClN2O3SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :388.95Ref: TM-T24855
1mg73,00€5mg136,00€1mL*10mM (DMSO)142,00€10mg187,00€25mg318,00€50mg452,00€100mg627,00€200mg845,00€TPCK
CAS :TPCK is an irreversible inhibitor of chymotrypsin-like proteases that affect cell proliferation, apoptosis, and tumorigenesisFormule :C17H18ClNO3SDegré de pureté :97.33%Couleur et forme :PowderMasse moléculaire :351.85Aurintricarboxylic acid
CAS :Aurintricarboxylic acid (NSC-4056) blocks nucleases and topoisomerases, stopping nucleic acid binding.Formule :C22H14O9Degré de pureté :97.1%Couleur et forme :Deep Red Coarse Crystalline PowderMasse moléculaire :422.34PX-12
CAS :PX-12, a Trx-1 inhibitor, promotes apoptosis, reduces HIF-1α/VEGF, and inhibits tumor growth, suggesting use in advanced cancer therapy.Formule :C7H12N2S2Degré de pureté :98% - 99.21%Couleur et forme :SolidMasse moléculaire :188.31L524-0366
CAS :L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.
Formule :C13H13ClN4OSDegré de pureté :98.6% - 99.13%Couleur et forme :SolidMasse moléculaire :308.79Glycochenodeoxycholic Acid
CAS :Glycochenodeoxycholic Acid (Lithocholylglycine) is a glycine conjugate of lithocholic acid, a bile acid.Formule :C26H43NO5Degré de pureté :97% - 99.97%Couleur et forme :SolidMasse moléculaire :449.62Ref: TM-T4588
5mg34,00€10mg49,00€1mL*10mM (DMSO)54,00€25mg79,00€50mg104,00€100mg154,00€200mg220,00€500mg374,00€SRT 2183
CAS :SRT 2183 is a selective activator of Sirtuin-1 (SIRT1, EC1.5 : 0.36 μM).Formule :C27H24N4O2SDegré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :468.57Ref: TM-T16932
1mg50,00€2mg72,00€5mg107,00€1mL*10mM (DMSO)111,00€10mg165,00€25mg283,00€50mg430,00€100mg622,00€Baohuoside I
CAS :Baohuoside I (Icariside-II) is a component of Epimedium koreanum, exhibits anti-inflammatory activity and anti-osteoporosis activities.Formule :C27H30O10Degré de pureté :97.64% - 98.14%Couleur et forme :SolidMasse moléculaire :514.52Ref: TM-T3396
2mg43,00€5mg63,00€10mg92,00€1mL*10mM (DMSO)123,00€25mg170,00€50mg268,00€100mg447,00€200mg623,00€Shepherdin 79-87 acetate
Shepherdin 79-87 acetate is a peptidomimetic antagonist of the complex between Hsp90 and survivin, another key regulator of tumor cell viability.Formule :C43H68N12O14SDegré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :1009.14Tenilsetam
CAS :Tenilsetam: an endonuclease, nootropic, AGE inhibitor potential for Alzheimer's.Formule :C8H10N2OSDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :182.24Ref: TM-T8583
1mg58,00€1mL*10mM (DMSO)96,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Benzarone
CAS :Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum.Formule :C17H14O3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :266.29Afatinib
CAS :Afatinib (BIBW 2992) is an irreversible and orally EGFR family inhibitor that inhibits EGFR and HER2. Afatinib has antitumor activity. Cost effective and quality assured.Formule :C24H25ClFN5O3Degré de pureté :98.56% - 99.9%Couleur et forme :Off-White SolidMasse moléculaire :485.94Ref: TM-T21312
5mg34,00€10mg49,00€1mL*10mM (DMSO)50,00€25mg81,00€50mg109,00€100mg137,00€200mg168,00€500mg284,00€Melatonin
CAS :Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formule :C13H16N2O2Degré de pureté :98% - 99.89%Couleur et forme :Pale Yellow Leaflets From Benzene SolidMasse moléculaire :232.283-hydroxy-3-phenylpentanamide
CAS :Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.
Formule :C11H15NO2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :193.24Stavudine sodium
CAS :Stavudine sodium, an oral HIV-1/2 inhibitor, also hinders mtDNA replication, NLRP3 inflammasome, and Amyloid-β autophagy, prompting apoptosis.Formule :C10H11N2NaO4Couleur et forme :SolidMasse moléculaire :246.198GW 441756
CAS :GW 441756 is a specific Tropomyosin-related kinase A (TrkA) inhibitor with an IC50 value of 2 nM.Formule :C17H13N3ODegré de pureté :97.73% - 99.8%Couleur et forme :SolidMasse moléculaire :275.3Dapivirine
CAS :Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.Formule :C20H19N5Degré de pureté :98% - 99.77%Couleur et forme :SolidMasse moléculaire :329.4Hypericin
CAS :Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. Cost-effective and quality-assured.Formule :C30H16O8Degré de pureté :98.90% - ≥98%Couleur et forme :Red-Coloured Anthraquinone-DerivativeMasse moléculaire :504.44Ref: TM-T6S0923
1mg54,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg172,00€25mg341,00€50mg504,00€100mg705,00€500mg1.431,00€AZD1208 hydrochloride
CAS :AZD1208 hydrochloride is a highly selective, potent and orally active PIM inhibitor.Formule :C21H22ClN3O2SCouleur et forme :SolidMasse moléculaire :415.94Dubermatinib
CAS :Dubermatinib (TP0903) is a potent and selective Axl kinase inhibitor.Formule :C24H30ClN7O2SDegré de pureté :98.65% - 99.58%Couleur et forme :SolidMasse moléculaire :516.06NSC 3852
CAS :NSC 3852 is a potent inhibitor of histone deacetylase.Formule :C9H6N2O2Degré de pureté :99.64%Couleur et forme :Slightly Yellow To Yellow-Green PowderMasse moléculaire :174.16Hexamethylene bisacetamide
CAS :Hexamethylene bisacetamide inhibits BET Bromodomain Proteins.Formule :C10H20N2O2Degré de pureté :99.94%Couleur et forme :White FlakesMasse moléculaire :200.284-Nitroquinoline 1-oxide
CAS :4-Nitroquinoline 1-oxide (4-NQO) is a chemical carcinogen that induces mutations in bacteria, fungi, and animals through the formation of large amounts ofFormule :C9H6N2O3Degré de pureté :97.4% - 99.94%Couleur et forme :Yellow Needles Or Plates From Acetone Physical Description Yellowish-Brown Plates Or Needles Or Yellow Solid (Ntp 1992)Masse moléculaire :190.16PDL-1 cpd 10
CAS :PDL-1 cpd 10 is a novel small molecule PD-L1 inhititor.Formule :C21H23N5O2Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :377.44PD184161
CAS :PD184161 is a novel, orally-active MEK inhibitor. PD184161 inhibited MEK activity (IC50 = 10-100 nM) in a time- and concentration-dependent manner[1].Formule :C17H13BrClF2IN2O2Degré de pureté :99.40%Couleur et forme :SolidMasse moléculaire :557.56Ref: TM-T21635
1mg35,00€2mg49,00€5mg74,00€10mg119,00€25mg259,00€50mg430,00€100mg620,00€200mg888,00€500mg1.333,00€Perillyl alcohol
CAS :Perillyl Alcohol, a monoterpene with antitumor properties, inhibits protein activation blocking cancer cell growth.Formule :C10H16ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :152.23Z-DEVD-FMK
CAS :Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,Formule :C30H41FN4O12Degré de pureté :96.19% - 99.69%Couleur et forme :SolidMasse moléculaire :668.66Ibuprofen sodium
CAS :Ibuprofen sodium is a selective COX-1 inhibitor, anti-inflammatory, and NO donor, used in pain, swelling, and cancer research.Formule :C13H17NaO2Couleur et forme :SolidMasse moléculaire :228.267Pectolinarin
CAS :Pectolinarin is a Cirsium isolate with anti-inflammatory activity.Formule :C29H34O15Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :622.57Tomivosertib HCl
CAS :Tomivosertib (eFT508) is a MNK1/2 inhibitor that blocks eIF4E phosphorylation, hindering tumor growth and immune signaling.Formule :C17H21ClN6O2Couleur et forme :SolidMasse moléculaire :376.845ZM 336372
CAS :ZM 336372 is a potent and selective c-Raf inhibitor.Formule :C23H23N3O3Degré de pureté :97.24% - 97.51%Couleur et forme :SolidMasse moléculaire :389.45Buparlisib
CAS :Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM for p110α, p110β, and p110δ).Formule :C18H21F3N6O2Degré de pureté :95.32% - 98.45%Couleur et forme :SolidMasse moléculaire :410.39Ref: TM-T1827
5mg59,00€1mL*10mM (DMSO)65,00€10mg80,00€25mg88,00€50mg109,00€100mg137,00€200mg222,00€500mg403,00€Pifithrin-β hydrobromide
CAS :Pifithrin-β hydrobromide (Cyclic PFT-α) is an inhibitor of p53; reversibly blocks p53-dependent transcriptional activation and apoptosis.Formule :C16H17BrN2SDegré de pureté :99.24% - 99.74%Couleur et forme :SolidMasse moléculaire :349.29Tangeretin
CAS :Tangeretin (NSC-618905), a flavonoid from citrus fruit peels, has been proven to play an important role in anti-inflammatory responses and neuroprotectiveFormule :C20H20O7Degré de pureté :98.83% - 98.97%Couleur et forme :Yellow CrystallineMasse moléculaire :372.37Amsilarotene
CAS :Amsilarotene (TAC101) blocks RB phosphorylation, boosts 2 CDK inhibitors, halts cell cycle, and reduces thymidylate synthase and cyclin A levels.Formule :C20H27NO3Si2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :385.6Ref: TM-T21314
1mg40,00€2mg54,00€1mL*10mM (DMSO)90,00€5mg92,00€10mg133,00€25mg259,00€50mg371,00€100mg530,00€200mg717,00€Oxaprozin potassium
CAS :Oxaprozin potassium is an oral COX inhibitor (IC50: 2.2 μM for COX-1, 36 μM for COX-2), induces apoptosis, and blocks NF-κB activation.Formule :C18H14KNO3Couleur et forme :SolidMasse moléculaire :331.412Rigosertib sodium
CAS :Rigosertib sodium (ON-01910), a non-ATP-competitive inhibitor of PLK1(IC50=9 nM), exhibits 30-fold higher specificity activity over Plk2 and no effect on Plk3.Formule :C21H24NNaO8SDegré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :473.47Epibrassinolide
CAS :Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator withFormule :C28H48O6Degré de pureté :97.57% - 98.11%Couleur et forme :SolidMasse moléculaire :480.68Amifostine trihydrate
CAS :Amifostine trihydrate (WR2721) is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.Formule :C5H15N2O3PS·3H2ODegré de pureté :99.71% - 99.80%Couleur et forme :SolidMasse moléculaire :268.27Rosiglitazone potassium
CAS :Rosiglitazone (BRL 49653) is an oral PPARγ agonist (EC50: 60 nM), TRPC5 activator (EC50: 30 μM), and TRPM3 inhibitor, used in obesity and diabetes research.Formule :C18H18KN3O3SCouleur et forme :SolidMasse moléculaire :395.52Dantrolene
CAS :Dantrolene is a postsynaptic muscle relaxant by inhibiting Ca2+ ions release from sarcoplasmic reticulum stores by antagonizing ryanodine receptors.Formule :C14H10N4O5Degré de pureté :99.97%Couleur et forme :Crystals From Aq DimethylformamideMasse moléculaire :314.25Ref: TM-T8452
5mg52,00€1mL*10mM (DMSO)59,00€10mg77,00€25mg92,00€50mg160,00€100mg200,00€200mg295,00€500mg497,00€Alemtuzumab
CAS :Alemtuzumab is a humanized monoclonal antibody against CD52 an antigen found on the surface of normal and malignant lymphocytes.
Degré de pureté :97.2% (SDS-PAGE); 96.7% (SEC-HPLC) - 98.00%Couleur et forme :LiquidMasse moléculaire :146.04 kDaRottlerin
CAS :Rottlerin (NSC-56346), a Mallotus Philippinensis extract, inhibits PKC (3-100 μM IC50); triggers apoptosis by activating caspase 3.Formule :C30H28O8Degré de pureté :97.41% - 99.44%Couleur et forme :Orange To Brown PowderMasse moléculaire :516.54Ferrostatin-1
CAS :Ferrostatin-1 (Fer-1) is a potent and selective inhibitor of iron death, potently inhibits Erastin-induced iron death in HT-1080 cells. High-Quality, Low-Cost!Formule :C15H22N2O2Degré de pureté :96.1% - 99.68%Couleur et forme :SolidMasse moléculaire :262.35RO8994
CAS :RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).Formule :C31H31Cl2FN4O4Degré de pureté :99.31% - 99.44%Couleur et forme :SolidMasse moléculaire :613.51Ref: TM-T3517
1mg38,00€2mg50,00€5mg82,00€1mL*10mM (DMSO)100,00€10mg120,00€25mg219,00€50mg344,00€100mg512,00€Oxysophoridine
CAS :Oxysophoridine protects against brain ischemia and heart damage through antioxidant, anti-apoptotic, and anti-inflammatory effects.Formule :C15H24N2O2Degré de pureté :98.15% - >99.99%Couleur et forme :SolidMasse moléculaire :264.36ABT-737
CAS :ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.Formule :C42H45ClN6O5S2Degré de pureté :98.15% - >99.99%Couleur et forme :SolidMasse moléculaire :813.43Ref: TM-T2099
2mgÀ demander5mg66,00€1mL*10mM (DMSO)73,00€10mg80,00€25mg130,00€50mg222,00€100mg389,00€BMS-8
CAS :BMS-8 is a novel inhibitor of the PD-1/PD-L1 interaction (IC50: 7.2 μM) by binding directly to PD-L1 and inducing the formation of PD-L1 homodimers.Formule :C27H28BrNO3Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :494.42Ref: TM-T26859
1mg37,00€5mg79,00€1mL*10mM (DMSO)86,00€10mg124,00€25mg222,00€50mg340,00€100mg505,00€200mg705,00€Voreloxin hydrochloride
CAS :Voreloxin hydrochloride (SNS-595 hydrochloride) is a potent inhibitor of Topoisomerase II with broad-spectrum anti-tumor activity.Formule :C18H20ClN5O4SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :437.9LASSBio-1135
CAS :LASSBio-1135 is an orally effective antagonist of TRPV1 and inhibitor of TNF-α production.Formule :C18H14N4Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :286.33Eprenetapopt
CAS :Eprenetapopt (PRIMA-1Met) restores wild-type conformation and function to mutant p53, and triggers apoptosis in tumor cells.Formule :C10H17NO3Degré de pureté :98.75% - 99.57%Couleur et forme :SolidMasse moléculaire :199.25Ref: TM-T4414
5mg70,00€1mL*10mM (DMSO)77,00€10mg100,00€25mg195,00€50mg349,00€100mg618,00€500mg1.251,00€Flavokawain B
CAS :Flavokawain B inhibits NO and PGE2, causes oxidative stress, and induces apoptosis, with potential for treating prostate cancer.Formule :C17H16O4Degré de pureté :99.94% - >99.99%Couleur et forme :SolidMasse moléculaire :284.31Capmatinib 2HCl.H2O
CAS :Capmatinib 2HCl.H2O (NVP-INC280 2HCl.H2O) is an orally bioavailable inhibitor of the proto-oncogene c-Met (HGFR)with potential antineoplastic activity.Formule :C23H21Cl2FN6O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :503.36Ref: TM-T8825
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg63,00€25mg84,00€50mg92,00€100mg126,00€500mg250,00€Navtemadlin
CAS :Navtemadlin (AMG232) is a potent, selective and orally available inhibitor of p53-MDM2 interaction (IC50: 0.6 nM).Cost-effective and quality-assured.Formule :C28H35Cl2NO5SDegré de pureté :95.55% - 99.08%Couleur et forme :SolidMasse moléculaire :568.55DMU-212
CAS :DMU-212, a Resveratrol derivative, has antimitotic, antiproliferative, antioxidant properties; induces apoptosis via ERK1/2.Formule :C18H20O4Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :300.35Ref: TM-T36674
2mg34,00€5mg50,00€1mL*10mM (DMSO)56,00€10mg84,00€25mg152,00€50mg259,00€100mg385,00€500mg873,00€Cannabigerol
CAS :Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormule :C21H32O2Degré de pureté :99.59% - 99.92%Couleur et forme :SolidMasse moléculaire :316.48Ref: TM-TN1465
1mg138,00€2mg203,00€5mg298,00€1mL*10mM (DMSO)306,00€10mg449,00€25mg765,00€50mg1.054,00€100mg1.423,00€Orantinib
CAS :Orantinib (NSC 702827) , a excellent effective against PDGFR autophosphorylation with Ki of 8 nM, also highly inhibits Flk-1 and FGFR1 trans-phosphorylation.Formule :C18H18N2O3Degré de pureté :98.92% - 99.52%Couleur et forme :SolidMasse moléculaire :310.35Carfilzomib
CAS :Carfilzomib (PR-171) is a proteasome inhibitor that irreversibly binds to the chymotrypsin of the 20S proteasome.Formule :C40H57N5O7Degré de pureté :99.6% - 99.84%Couleur et forme :SolidMasse moléculaire :719.91PUMA BH3 Free base
PUMA BH3 acetate (PUMA BH3 Free base) is a p53 positive regulator of apoptosis (PUMA) BH3 domain polypeptide that acts as a direct activator of Bak with a Kd ofFormule :C130H206N42O45SDegré de pureté :96.64%Couleur et forme :SolidMasse moléculaire :3109.35Brassinolide
CAS :Brassinolide (Brassin lactone) is a plant hormone isolated from rapeseed (Brassica napus) promoting stem elongation and cell division.Formule :C28H48O6Degré de pureté :98% - 99.189%Couleur et forme :Off-White SolidMasse moléculaire :480.68L-Buthionine-(S,R)-sulfoximine hydrochloride
L-Buthionine-(S,R)-sulfoximine hydrochloride is a fast, irreversible γ-GCS inhibitor that depletes glutathione. IC50: 1.9-29 μM in various tumors.Formule :C8H19ClN2O3SCouleur et forme :SolidMasse moléculaire :258.77DD1
CAS :DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.Formule :C16H14N2O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :282.29Ref: TM-T8978
1mg71,00€5mg131,00€1mL*10mM (DMSO)138,00€10mg215,00€25mg338,00€50mg465,00€100mg630,00€200mg850,00€SRS11-92
CAS :SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.47Ref: TM-T8922
1mg46,00€5mg80,00€1mL*10mM (DMSO)105,00€10mg116,00€25mg227,00€50mg359,00€100mg550,00€500mg1.159,00€Pyrogallol
CAS :Pyrogallol (Piral) is a white crystalline powder and a powerful reducing agent prepared by heating gallic acid.Formule :C6H6O3Degré de pureté :99.88% - 99.91%Couleur et forme :SoildMasse moléculaire :126.11JG-98
CAS :JG-98 is an allosteric Hsp70 inhibitor, displays high active against the breast cancer cell lines MDA-MB-231 and MCF-7 (EC50s: 0.4/0.7 μM).Formule :C24H21Cl2N3OS3Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :534.53DC260126
CAS :DC260126 is a small-molecule antagonist of FFA1 (GPR40)Formule :C16H18FNO2SDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :307.38Rimiducid
CAS :Rimiducid, a tacrolimus analogue, dimerizes FKBP domains to activate Caspase 9 and induce apoptosis; binds FKBP12 weakly.Formule :C78H98N4O20Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :1411.63Ref: TM-T14298
1mg129,00€2mg177,00€5mg285,00€10mg420,00€25mg692,00€50mg973,00€100mg1.305,00€500mg2.602,00€MK-2206 dihydrochloride
CAS :MK-2206 dihydrochloride (MK-2206 2HCl) is a variant Akt inhibitor that inhibits Akt1, Akt2, and Akt3 (IC50=8/12/65 nM) with orally active, highly potent andFormule :C25H23Cl2N5ODegré de pureté :99.228% - 99.94%Couleur et forme :SolidMasse moléculaire :480.39Ref: TM-T1952
2mg34,00€5mg49,00€1mL*10mM (DMSO)52,00€10mg66,00€25mg90,00€50mg137,00€100mg205,00€200mg334,00€500mg552,00€NSC 15364
CAS :NSC 15364 (1,3-Bis(4-aminophenyl)urea) can be used for screening of ALR inhibitors by detection of hydrogen peroxide production Measured in Biochemical System.Formule :C13H14N4ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :242.28Mirodenafil dihydrochloride
CAS :Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.Formule :C26H39Cl2N5O5SDegré de pureté :99.64% - 99.78%Couleur et forme :SolidMasse moléculaire :604.59AZ5576 racemate
CAS :AZ5576 racemate, potent Cdk9 inhibitor, oral, IC50 <5nM; disrupts RNAPII, aids AML treatment, kills MV411 cells.Formule :C21H24FN3O3Couleur et forme :SolidMasse moléculaire :385.43
