
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5593 produits trouvés pour "Apoptose"
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CP-31398 dihydrochloride
CAS :<p>CP-31398 dihydrochloride is a p53 stabilizer which stabilizes the active conformation of p53 and promotes p53 activity in cancer cell lines.</p>Formule :C22H28Cl2N4ODegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :435.4Suberoyl bis-hydroxamic acid
CAS :<p>SBHA is an HDAC inhibitor, an enzyme key to transcription, cell cycle, and development.</p>Formule :C8H16N2O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :204.22PF-4989216
CAS :<p>PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.</p>Formule :C18H13FN6OSDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :380.4WT-161
CAS :<p>WT161 is a potent and selective inhibitor of HDAC6 (IC50:0.40 nM).</p>Formule :C27H30N4O3Degré de pureté :95.98% - 98.34%Couleur et forme :SolidMasse moléculaire :458.55Pexidartinib
CAS :<p>Pexidartinib (PLX-3397) is a capsule formulation containing a small-molecule receptor tyrosine kinase (RTK) inhibitor of KIT, CSF1R and FLT3 with potential</p>Formule :C20H15ClF3N5Degré de pureté :98.34% - 99.45%Couleur et forme :SolidMasse moléculaire :417.81G-749
CAS :<p>G-749, a new-type FLT3 inhibitor, exhibits effective and sustained inhibition of the FLT3 wild type and mutants.</p>Formule :C25H25BrN6O2Degré de pureté :98.32% - 99.60%Couleur et forme :SolidMasse moléculaire :521.41Obacunone
CAS :<p>Obacunone: cytotoxic to prostate cells, anti-S. Typhimurium, may inhibit breast cancer and aromatase, trigger apoptosis.</p>Formule :C26H30O7Degré de pureté :98% - ≥95%Couleur et forme :White PowderMasse moléculaire :454.51NVP-HSP990
CAS :<p>NVP-HSP990 (HSP990) is an effective and specific HSP90α/β inhibitor (IC50: 0.6 /0.8 nM).</p>Formule :C20H18FN5O2Degré de pureté :98.03% - 99.32%Couleur et forme :SolidMasse moléculaire :379.39PF-3758309 hydrochloride
CAS :<p>PF-3758309 hydrochloride (PF-03758309 hydrochloride) , is a PAK4 inhibitor, is also a n orally bioavailable small-molecule inhibitor of p21-activated kinase 4 (</p>Formule :C25H31ClN8OSDegré de pureté :98.83% - >99.99%Couleur et forme :SolidMasse moléculaire :527.08Panobinostat
CAS :<p>Panobinostat (NVP-LBH589) is a broad-spectrum HDAC inhibitor (IC50=5 nM) with oral activity and non-selectivity.</p>Formule :C21H23N3O2Degré de pureté :97.2% - 99.81%Couleur et forme :Yellow SolidMasse moléculaire :349.43PHA-767491 hydrochloride
CAS :<p>PHA-767491 (CAY-10572) is a potent Cdc7/CDK9 inhibitor (IC50: 10/34 nM), selective against GSK3-β, CDK1/2, CDK5, MK2, CHK2, PLK1.</p>Formule :C12H12ClN3ODegré de pureté :99.56% - 99.92%Couleur et forme :SolidMasse moléculaire :249.69Capmatinib 2HCl
CAS :<p>Capmatinib 2HCl (INC-280 2HCl), a c-MET inhibitor, is potent (IC50 = 0.13 nM), highly specific, and induces apoptosis in tumor cells.</p>Formule :C23H19Cl2FN6ODegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :485.34Phenazine methylsulfate
CAS :<p>Phenazine methylsulfate is anti-bacterial agents.</p>Formule :C14H14N2O4SDegré de pureté :97.67% - >99.99%Couleur et forme :Yellow CrystallineMasse moléculaire :306.34α-Thujone
CAS :<p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>Formule :C10H16ODegré de pureté :97.02% - 98.41%Couleur et forme :Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Masse moléculaire :152.23COTI-2
CAS :<p>COTI-2, an orally available thiosemicarbazone, is an activator of mutant forms of the p53 protein with potential antineoplastic activity.</p>Formule :C19H22N6SDegré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :366.48C-DIM12
CAS :<p>C-DIM12 boosts Nurr1 gene expression, heightens Nurr1 protein in neurons, and improves survival against 6-OHDA.</p>Formule :C23H17ClN2Degré de pureté :97.72% - ≥95%Couleur et forme :SolidMasse moléculaire :356.85SJ-172550
CAS :<p>SJ-172550 is a small molecule inhibitor of MDMX (EC50: 5 μM).</p>Formule :C22H21ClN2O5Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :428.87Kahweol
CAS :<p>Kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the LPS-induced activation of NF-kappaB by preventing IkappaB</p>Formule :C20H26O3Degré de pureté :99.26% - 99.86%Couleur et forme :Off-White To Yellow SolidMasse moléculaire :314.42Oleic acid
CAS :<p>Oleic acid, a common unsaturated fat, is used in oleates, lotions, and as a pharma solvent.</p>Formule :C18H34O2Degré de pureté :97.14% - 99.91%Couleur et forme :Colorless Or Nearly Colorless Liq (Above 5-7 Deg C) Oleic Acid Is A Colorless To Pale Yellow Liquid With A Mild Odor Floats On Water (Uscg 1999)Masse moléculaire :282.46RA-9
CAS :<p>RA-9 is a potent and selective proteasome-associated inhibitor of deubiquitinating enzymes (DUBs), with favorable toxicity profile and anticancer activity.</p>Formule :C19H15N3O5Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :365.34AVN-944
CAS :<p>AVN-944 (VX-944)(VX-944) is a selective, noncompetitive inhibitor of human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.</p>Formule :C25H27N5O5Degré de pureté :99.07% - ≥95%Couleur et forme :SolidMasse moléculaire :477.51GW 441756
CAS :<p>GW 441756 is a specific Tropomyosin-related kinase A (TrkA) inhibitor with an IC50 value of 2 nM.</p>Formule :C17H13N3ODegré de pureté :97.73% - 99.8%Couleur et forme :SolidMasse moléculaire :275.3R406
CAS :<p>R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.</p>Formule :C22H23FN6O5·C6H6O3SDegré de pureté :97.67% - 98.82%Couleur et forme :SolidMasse moléculaire :628.63R406 free base
CAS :<p>R406 free base (R406 (free base)) is a potent Syk inhibitor.</p>Formule :C22H23FN6O5Degré de pureté :97.64% - 99.11%Couleur et forme :SolidMasse moléculaire :470.45Rosiglitazone
CAS :<p>Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity.</p>Formule :C18H19N3O3SDegré de pureté :98.61% - 99.87%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :357.433-Dehydrotrametenolic acid
CAS :<p>3-Dehydrotrametenolic acid is a potential anticancer agent against H-ras transformed tumor and a promising candidate for a new type of insulin-sensitizing drug.</p>Formule :C30H46O3Degré de pureté :98.5% - 99.25%Couleur et forme :SolidMasse moléculaire :454.68Adalimumab
CAS :<p>Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.</p>Degré de pureté :95% - 99.50%Couleur et forme :LiquidMasse moléculaire :145.4 kDaSolasodine
CAS :<p>Solasodine, a toxic alkaloid from Solanaceae, kills HeLa cervical cancer and U937 leukemia cells.</p>Formule :C27H43NO2Degré de pureté :99.64% - 99.94%Couleur et forme :SolidMasse moléculaire :413.64BIBR 1532
CAS :<p>BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).</p>Formule :C21H17NO3Degré de pureté :98.49% - 98.90%Couleur et forme :SolidMasse moléculaire :331.36(Rac)-Benpyrine
CAS :<p>(Rac)-Benpyrine is a potent and orally active inhibitor of TNF-α.</p>Formule :C16H16N6ODegré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :308.34Leachianone A
CAS :<p>Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced cytotoxicity.</p>Formule :C26H30O6Degré de pureté :98.53% - 99.79%Couleur et forme :SolidMasse moléculaire :438.51L-Glutamic acid monosodium salt
CAS :<p>L-Glutamic acid monosodium salt (MSG) (Monosodium glutamate) is an activator of mGlu1 receptor.</p>Formule :C5H8NO4·NaDegré de pureté :99.93%Couleur et forme :White Solid CrystallineMasse moléculaire :169.11Citric acid
CAS :<p>Citric acid (Citro) is a weak organic tricarboxylic acid found in citrus fruits, a food additive and a natural preservative. High-Quality, Low-Cost!</p>Formule :C6H8O7Degré de pureté :98.88%Couleur et forme :White Solid CrystallineMasse moléculaire :192.12ONO-4059 analog
CAS :<p>ONO-4059 analog (ONO-WG-307)ue is an analogue of ONO-4059, which is a highly potent and selective oral BTK inhibitor with IC50 of 23.9 nM. Phase 1.</p>Formule :C25H24N6O3Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :456.5Galgravin
CAS :<p>Galgravin combats inflammation, safeguards neurons, promotes neurite growth, and resists Abeta25-35 and MPP+ toxicity.</p>Formule :C22H28O5Degré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :372.45Sanguinarine
CAS :<p>Sanguinarine (Pseudochelerythrine) is a specific inhibitor of Rac1b with anti-microbial, anti-oxidant and anti-inflammatory properties.</p>Formule :C20H14NO4Degré de pureté :99.04% - 99.76%Couleur et forme :SolidMasse moléculaire :332.33Polydatin
CAS :<p>Polydatin, a resveratrol glycoside from Polygonum cuspidatum, inhibits platelet aggregation, alters lipid ratios, and modulates cell functions.</p>Formule :C20H22O8Degré de pureté :97.2% - 98.94%Couleur et forme :White Fine PowderMasse moléculaire :390.38Quercetin Dihydrate
CAS :<p>Quercetin Dihydrate (Sophoretin) is a flavonoid natural product that activates or inhibits the activity of many proteins. It activates SIRT1 and inhibits PI3K.</p>Formule :C15H10O7·2H2ODegré de pureté :97.77%Couleur et forme :Yellow SolidMasse moléculaire :338.27Atractylenolide II
CAS :<p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>Formule :C15H20O2Degré de pureté :99.89% - 99.93%Couleur et forme :SolidMasse moléculaire :232.32API-1
CAS :<p>API-1 (NSC-177223) is a potent inhibitor of Akt. It induces GSK3-dependent, β-TrCP- and FBXW7-mediated Mcl-1 degradation, resulting in induction of apoptosis .</p>Formule :C13H15N5O6Degré de pureté :97.15%Couleur et forme :SolidMasse moléculaire :337.29L-Glutamic acid
CAS :<p>L-Glutamic acid is an agonist of glutamate receptors, including metabotropic glutamate receptors (mGluR), AMPA, NMDA, and KA. High-Quality, Low-Cost!</p>Formule :C5H9NO4Degré de pureté :99.14% - 99.55%Couleur et forme :White Solid CrystallineMasse moléculaire :147.13PND-1186
CAS :<p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>Formule :C25H26F3N5O3Degré de pureté :99.14% - 99.75%Couleur et forme :SolidMasse moléculaire :501.5Bafetinib
CAS :<p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>Formule :C30H31F3N8ODegré de pureté :94.16% - 99.68%Couleur et forme :SolidMasse moléculaire :576.62PHT-427
CAS :<p>PHT-427 (CS-0223) is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity binding for the PH domains of Akt and PDPK1).</p>Formule :C20H31N3O2S2Degré de pureté :97.54% - >99.99%Couleur et forme :SolidMasse moléculaire :409.61Brazilin
CAS :<p>1.</p>Formule :C16H14O5Degré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :286.28Onvansertib
CAS :<p>Onvansertib (NMS-1286937) is a PLK1 inhibitor with high selectivity and oral activity. Onvansertib has antitumor activity. Cost-effective and quality-assured.</p>Formule :C24H27F3N8O3Degré de pureté :98.3% - 99.88%Couleur et forme :SolidMasse moléculaire :532.52SBI-0640756
CAS :<p>SBI-0640756 (SBI-756) (SBI-756) is a first-in-class inhibitor that targets eIF4G1 and disrupts the eIF4F complex.</p>Formule :C23H14ClFN2O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :404.82D-Pantothenic acid sodium
CAS :<p>D-Pantothenic acid sodium, a sodium salt of D-pantothenate, is a vital B5 derivative, aiding fat, carb, and amino acid oxidation.</p>Formule :C9H16NNaO5Degré de pureté :97.98%Couleur et forme :White PowderMasse moléculaire :241.22Darapladib
CAS :<p>Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.</p>Formule :C36H38F4N4O2SDegré de pureté :99.82% - >99.99%Couleur et forme :SolidMasse moléculaire :666.77Hematoporphyrin dihydrochloride
CAS :<p>Hematoporphyrin dihydrochloride (Hematoporphyrin IX dihydrochloride) is a substrate for affinity chromatography of heme-binding proteins.</p>Formule :C34H40Cl2N4O6Degré de pureté :90.11%Couleur et forme :SolidMasse moléculaire :671.61PluriSIn 1
CAS :<p>PluriSIn 1 (NSC 14613) blocks SCD1, key in oleic acid creation, showing lipid metabolism's role in hPSCs.</p>Formule :C12H11N3ODegré de pureté :99.19% - 99.63%Couleur et forme :SolidMasse moléculaire :213.24BTSA1
CAS :<p>BTSA1: High-affinity BAX activator inducing conformational changes for apoptosis.</p>Formule :C21H14N6OS2Degré de pureté :99.60% - 99.71%Couleur et forme :SolidMasse moléculaire :430.51Cambinol
CAS :<p>Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.</p>Formule :C21H16N2O2SDegré de pureté :98.02% - 99.83%Couleur et forme :SolidMasse moléculaire :360.43Azadirachtin
CAS :<p>Azadirachtin has antifungal activity, used as an insecticide.</p>Formule :C35H44O16Degré de pureté :98.11% - 99.713%Couleur et forme :SolidMasse moléculaire :720.71Lumichrome
CAS :<p>Lumichrome, a riboflavin metabolite, influences plant growth, ascidian metamorphosis, bacterial communication, and blocks riboflavin uptake.</p>Formule :C12H10N4O2Degré de pureté :99.69% - 99.93%Couleur et forme :SolidMasse moléculaire :242.23Jaceosidin
CAS :<p>Jaceosidin: anti-oxidant, anti-inflammatory, anti-cancer, immunosuppressive; affects CYP1A2/UGT1A1/UGT1A7 metabolism.</p>Formule :C17H14O7Degré de pureté :98.23% - 99.28%Couleur et forme :SolidMasse moléculaire :330.29Ruxolitinib
CAS :<p>Ruxolitinib (INCB018424) is a JAK1/2 inhibitor (IC50=3.3/2.8 nM) that is potent and selective.</p>Formule :C17H18N6Degré de pureté :99.4% - >99.99%Couleur et forme :SolidMasse moléculaire :306.36Eribulin mesylate
CAS :<p>Eribulin mesylate (E7389), a microtubule inhibitor, treats metastatic breast cancer by halting cell division.</p>Formule :C41H63NO14SDegré de pureté :97.02% - >99.99%Couleur et forme :SolidMasse moléculaire :826XI-006
CAS :<p>NSC-207895 (XI-006) suppresses MDMX with IC50 of 2.5 μM, leading to enhanced p53 stabilization/activation and DNA damage, and regulates MDM2, an E3 ligase.</p>Formule :C11H13N5O4Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :279.25Cabozantinib
CAS :<p>Cabozantinib (XL184) is a multi-targeted tyrosine kinase receptor inhibitor that inhibits VEGFR2, c-Met, Kit, Axl, and Flt3 (IC50=0.035/1.3/4.6/7/11.3 nM).</p>Formule :C28H24FN3O5Degré de pureté :99.68% - 99.88%Couleur et forme :SolidMasse moléculaire :501.513,4-Dicaffeoylquinic acid
CAS :<p>3,4-Dicaffeoylquinic acid (Isochlorogenic acid B) has antioxidant activity.</p>Formule :C25H24O12Degré de pureté :96.33% - 98.82%Couleur et forme :SolidMasse moléculaire :516.45PRIMA-1
CAS :<p>PRIMA-1 (NSC-281668) is a mutant p53 reactivator. It induces apoptosis and inhibits growth of human tumors with mutant p53.</p>Formule :C9H15NO3Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :185.22GSK2656157
CAS :<p>GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay.</p>Formule :C23H21FN6ODegré de pureté :98.59% - >99.99%Couleur et forme :SolidMasse moléculaire :416.45KRAS inhibitor-9
CAS :<p>KRAS inhibitor-9 (DUN09716) hinders GTP-KRAS formation, with a Kd of 92 μM, causes G2/M arrest, and induces apoptosis in mutated NSC-LC cells.</p>Formule :C13H9ClN2S2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :292.81BAI1
CAS :<p>BAI1 (Bax channel blocker) is a potent inhibitor of Bax-mediated mitochondrial cytochrome C release (IC50: 0.52 μM).</p>Formule :C19H21Br2N3ODegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :467.2LQZ-7I
CAS :<p>LQZ-7I is an inhibitor of surviving-targeting. It orally effectively inhibits xenograft tumor growth and induces survivin loss in tumors</p>Formule :C20H14F2N4Degré de pureté :99.81% - 99.87%Couleur et forme :SolidMasse moléculaire :348.356-Thioguanine
CAS :<p>6-Thioguanine (2-Amino-6-purinethiol) is an antineoplastic compound which also has antimetabolite action. The drug is used in the therapy of acute leukemia.</p>Formule :C5H5N5SDegré de pureté :98.34% - >99.99%Couleur et forme :Odorless Or Almost Odorless Pale Yellow Crystalline PowderMasse moléculaire :167.19Adaphostin
CAS :<p>Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.</p>Formule :C24H27NO4Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :393.48Karanjin
CAS :<p>Karanjin, a flavonoid from karanja seeds, boosts GLUT4, AMPK in muscles, and triggers cancer cell apoptosis.</p>Formule :C18H12O4Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :292.29Mivebresib
CAS :<p>Mivebresib (ABBV-075) is a potent BET inhibitor with antitumor effects, disrupting gene expression and MYC, TMPRSS2-ETS proteins.</p>Formule :C22H19F2N3O4SDegré de pureté :98.74% - 99.32%Couleur et forme :SolidMasse moléculaire :459.47Madecassoside
CAS :<p>Madecassoside (Asiaticoside A) is a pentacyclic triterpene extracted from Centella asitica (L.) with anti-inflammatory, anti-oxidative and anti-aging activities</p>Formule :C48H78O20Degré de pureté :99.46% - 99.85%Couleur et forme :White PowderMasse moléculaire :975.12Z-FA-FMK
CAS :<p>Z-FA-FMK can irreversibly inhibit cysteine protease and also inhibit effector caspases.</p>Formule :C21H23FN2O4Degré de pureté :98.84% - 99.68%Couleur et forme :SolidMasse moléculaire :386.42PI-1840
CAS :<p>PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.</p>Formule :C22H26N4O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :394.47Soyasapogenol B
CAS :<p>Soyasapogenol B has anti-cancer, hypocholesterolemic, anticomplementary, hepatoprotective effects, it inhibits proliferation of cultured Hep-G2.</p>Formule :C30H50O3Degré de pureté :99.51% - 99.81%Couleur et forme :SolidMasse moléculaire :458.72Pantoprazole
CAS :<p>Pantoprazole (BY1023) is a proton pump inhibitor used for short-term treatment of erosion and ulceration of the esophagus caused by gastroesophageal reflux</p>Formule :C16H15F2N3O4SDegré de pureté :99.28% - 99.63%Couleur et forme :Almost White SolidMasse moléculaire :383.37ATH686
CAS :<p>ATH686 is an potent and selective Inhibitor of FLT3.</p>Formule :C25H28F3N7O2Degré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :515.53Embelin
CAS :<p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>Formule :C17H26O4Degré de pureté :97.07% - 99.88%Couleur et forme :SolidMasse moléculaire :294.39VER-50589
CAS :<p>VER-50589 is a potent HSP90 inhibitor.</p>Formule :C19H17ClN2O5Degré de pureté :99.96% - >99.99%Couleur et forme :SolidMasse moléculaire :388.8Calycosin
CAS :<p>Calycosin modulates estrogen receptors, induces apoptosis in cancers, and shows skin-lightening by inhibiting tyrosinase (IC50: 38.4µM).</p>Formule :C16H12O5Degré de pureté :99.91% - >99.99%Couleur et forme :White PowderMasse moléculaire :284.26FIN56
CAS :<p>FIN56 is a specific inducer of ferroptosis.</p>Formule :C25H31N3O5S2Degré de pureté :99.72% - 99.78%Couleur et forme :SolidMasse moléculaire :517.66Volasertib
CAS :<p>Volasertib (BI 6727) (BI-6727) is a potent inhibitor of PLK1 (IC50: 0.87 nM), inducing mitotic arrest and apoptosis.</p>Formule :C34H50N8O3Degré de pureté :98% - 99.72%Couleur et forme :SolidMasse moléculaire :618.81Triptolide
CAS :<p>Triptolide (PG490) belongs to the tricyclic diterpenoid group of natural products and is an inhibitor of NF-κB activation.</p>Formule :C20H24O6Degré de pureté :97.19% - 99.97%Couleur et forme :White To Off-White SolidMasse moléculaire :360.4RO8994
CAS :<p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>Formule :C31H31Cl2FN4O4Degré de pureté :99.31% - 99.44%Couleur et forme :SolidMasse moléculaire :613.51Epibrassinolide
CAS :<p>Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator with</p>Formule :C28H48O6Degré de pureté :97.57% - 98.11%Couleur et forme :SolidMasse moléculaire :480.68Hypericin
CAS :<p>Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. Cost-effective and quality-assured.</p>Formule :C30H16O8Degré de pureté :99.05% - ≥98%Couleur et forme :Red-Coloured Anthraquinone-DerivativeMasse moléculaire :504.44Afatinib
CAS :<p>Afatinib (BIBW 2992) is an irreversible and orally EGFR family inhibitor that inhibits EGFR and HER2. Afatinib has antitumor activity. Cost effective and quality assured.</p>Formule :C24H25ClFN5O3Degré de pureté :98.56% - 99.9%Couleur et forme :Off-White SolidMasse moléculaire :485.94Glycochenodeoxycholic Acid
CAS :<p>Glycochenodeoxycholic Acid (Lithocholylglycine) is a glycine conjugate of lithocholic acid, a bile acid.</p>Formule :C26H43NO5Degré de pureté :97% - 99.97%Couleur et forme :SolidMasse moléculaire :449.62Telekin
CAS :<p>Telekin, a sesquiterpene lactone from Carpesium divaricatum, strongly inhibits cancer cell growth.</p>Formule :C15H20O3Degré de pureté :99.86% - 99.97%Couleur et forme :SolidMasse moléculaire :248.32AT7519
CAS :<p>AT7519 is a CDK1/2/4/6/9 inhibitor (IC50: 10-210 nM). It is less effective to CDK3 and little active to CDK7.</p>Formule :C16H17Cl2N5O2Degré de pureté :98.88% - 99.65%Couleur et forme :SolidMasse moléculaire :382.24Malabaricone B
CAS :<p>Malabaricone B is a Spice-derived phenolic, it induces mitochondrial damage in lung cancer cells via a p53-independent pathway.</p>Formule :C21H26O4Degré de pureté :99.84% - 99.91%Couleur et forme :SolidMasse moléculaire :342.43(E/Z)-TG003
CAS :<p>(E/Z)-TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor.</p>Formule :C13H15NO2SDegré de pureté :98% - 99.04%Couleur et forme :SolidMasse moléculaire :249.33BI-3802
CAS :<p>BI-3802, a highly potent BCL6 degrader, targets and inhibits the Bric-à-brac (BTB) domain of BCL6, exhibiting an IC50 value of ≤3 nM.</p>Formule :C24H29ClN6O3Degré de pureté :97.93% - 98.58%Couleur et forme :SolidMasse moléculaire :484.98JG-98
CAS :<p>JG-98 is an allosteric Hsp70 inhibitor, displays high active against the breast cancer cell lines MDA-MB-231 and MCF-7 (EC50s: 0.4/0.7 μM).</p>Formule :C24H21Cl2N3OS3Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :534.53TD52
CAS :<p>TD52, an Erlotinib derivative, is an oral CIP2A cancer inhibitor that disrupts Elk1's attachment to the CIP2A promoter.</p>Formule :C24H16N4Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :360.41Rilmenidine hemifumarate
CAS :<p>Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.</p>Formule :C10H16N2OC4H4O4Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :238.28TREM2-IN-1
CAS :<p>TREM2-IN-1 (OPA) is a platinum-based TREM2 inhibitor with anti-cancer and anti-tumor activity, inhibiting the immune-regulatory activity of TREM2 on macrophages</p>Formule :C46H68N2O20PtDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :1164.12Pitavastatin sodium
CAS :<p>Pitavastatin sodium inhibits HMG-CoA reductase, enhances LDL-C receptors, and has various protective effects.</p>Formule :C25H23FNNaO4Couleur et forme :SolidMasse moléculaire :443.45WHI-P154
CAS :<p>WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.</p>Formule :C16H14BrN3O3Degré de pureté :98% - 99.67%Couleur et forme :SolidMasse moléculaire :376.2S63845
CAS :<p>S63845 is a selective myeloid leukemia 1(MCL1) inhibitor that binds to human MCL1 with a Kd of 0.19 nM.Cost-effective and quality-assured.</p>Formule :C39H37ClF4N6O6SDegré de pureté :97.7% - ≥98%Couleur et forme :SolidMasse moléculaire :829.26Mdivi-1
CAS :<p>Mdivi-1 (Mitochondrial division inhibitor 1) is a mitochondrial division inhibitor that inhibits DRP1 and Dynamin I (IC50=1-10 μM).</p>Formule :C15H10Cl2N2O2SDegré de pureté :96.57% - 99.23%Couleur et forme :SolidMasse moléculaire :353.22Quinidine
CAS :<p>Quinidine is a stereoisomer of the antimalarial agent quinine and a class Ia antiarrhythmic agent. for the treatment of abnormal heart rhythms and also malaria.</p>Formule :C20H24N2O2Degré de pureté :97.03% - 99.99%Couleur et forme :Crystals With 2 5 Mol Water Of Crystallization; Crystals From Dilute Alcohol Physical Description Crystals Or White Powder (Ntp 1992)Masse moléculaire :324.42PYR-41
CAS :<p>PYR-41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2.</p>Formule :C17H13N3O7Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :371.3Lupeol
CAS :<p>Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.</p>Formule :C30H50ODegré de pureté :98% - 99.96%Couleur et forme :Needles From Alcohol Acetone White PowderMasse moléculaire :426.72Purvalanol A
CAS :<p>Purvalanol A (NG-60) is an effective and cell-permeable CDK inhibitor with IC50 of 70/4/35/850 nM for cdk2-cyclin A/B/E, and cdk4-cyclin D1, respectively.</p>Formule :C19H25ClN6ODegré de pureté :98.13% - 99.68%Couleur et forme :PowderMasse moléculaire :388.89Meisoindigo
CAS :<p>Meisoindigo (Natura-α) is a derivative of indigo natural, might induces apoptosis and myeloid differentiation of acute myeloid leukemia (AML).</p>Formule :C17H12N2O2Degré de pureté :98.03% - 98.19%Couleur et forme :SolidMasse moléculaire :276.29Pinosylvin
CAS :<p>Pinosylvin (5-Styrylresorcinol) induces autophagy via AMPK activation. Pinosylvin is likely to act as a pro-angiogenic factor.</p>Formule :C14H12O2Degré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :212.24M50054
CAS :<p>Apoptosis Inhibitor was a novel inhibitor of programmed cell death associate with caspase-3 inhibition.</p>Formule :C13H16O4Degré de pureté :97.8%Couleur et forme :SolidMasse moléculaire :236.26BI-847325
CAS :<p>BI-847325 is a selective dual inhibitor of MEK and aurora kinases (AK) with IC50 values of 4 and 15 nM for human MEK2 and AK-C, respectively.</p>Formule :C29H28N4O2Degré de pureté :97.13% - 97.54%Couleur et forme :SolidMasse moléculaire :464.56BI 2536
CAS :<p>BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM). It has 4- and 11-fold greater selectivity than Plk2 and Plk3.</p>Formule :C28H39N7O3Degré de pureté :98% - 99.88%Couleur et forme :SolidMasse moléculaire :521.65Copanlisib
CAS :<p>Copanlisib (BAY 80-6946), a PI3K inhibitor, may block tumor growth and improve cancer treatment efficacy.</p>Formule :C23H28N8O4Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :480.52Avicularin
CAS :<p>Avicularin reduces inflammation via ERK pathway in RAW 264.7 cells and hinders lipid buildup in adipocytes by limiting glucose uptake and fatty acid synthesis.</p>Formule :C20H18O11Degré de pureté :97.02% - 99.94%Couleur et forme :White PowderMasse moléculaire :434.35PD146176
CAS :<p>PD146176 (NSC-168807) is an inhibitor of 15-Lipoxygenase (15-LO) , it inhibits rabbit reticulocyte 15-LO with Ki of 197 nM and IC50 of 0.54 μM.</p>Formule :C15H11NSDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :237.32Terrestrosin D
CAS :<p>Terrestrosin D triggers apoptosis, halts cell cycles, and blocks angiogenesis in tumor cells, displaying anti-cancer effects.</p>Formule :C50H80O23Degré de pureté :99.92% - 99.96%Couleur et forme :SolidMasse moléculaire :1049.16Ganetespib
CAS :<p>Ganetespib (STA-9090) is a synthetic small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity.</p>Formule :C20H20N4O3Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :364.4Aminopurvalanol A
CAS :<p>Aminopurvalanol A is a competitive, selective and cell-permeable inhibitor of cyclin-dependent kinase (CDK) that potently inhibits Cyclin A/cdk2, Cyclin B/cdk1</p>Formule :C19H26ClN7ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :403.91Apomine
CAS :<p>Apomine (SR-9223i) 是一种 HMG-CoA-还原酶抑制剂,可在体外促进骨髓瘤细胞的凋亡,并与体内骨髓瘤的调节有关。 Apomine 加速 3-羟基-3-甲基戊二酰-CoA 还原酶的降解并刺激低密度脂蛋白受体活性。 Apomine 通过下调 3-羟基-3-甲基戊二酰-CoA 还原酶来增强洛伐他汀对骨髓瘤细胞的抗肿瘤作用。</p>Formule :C28H52O7P2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :562.66TBHQ
CAS :<p>TBHQ (tert-Butylhydroquinone) is an antioxidant that induces an antioxidant response through the redox-sensitive transcription factor Nrf2.</p>Formule :C10H14O2Degré de pureté :99.17% - 99.53%Couleur et forme :White Solid PowderMasse moléculaire :166.22Ginsenoside Rh2
CAS :<p>Ginsenoside Rh2 (20(S)-Ginsenoside Rh2), an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug.</p>Formule :C36H62O8Degré de pureté :99.20% - 99.76%Couleur et forme :White PowderMasse moléculaire :622.87Ginsenoside F2
CAS :<p>Ginsenoside F2 halts breast CSCs growth, induces apoptosis via intrinsic pathway and impairs mitochondria.</p>Formule :C42H72O13Degré de pureté :99.04% - 99.3%Couleur et forme :SolidMasse moléculaire :785.01HA14-1
CAS :<p>HA14-1, a Bcl-2/Bcl-XL antagonist, is a non-peptidic ligand of a Bcl-2 surface pocket (IC50: ~9 μM).</p>Formule :C17H17BrN2O5Degré de pureté :95.07% - 98%Couleur et forme :SolidMasse moléculaire :409.23LCL161
CAS :<p>LCL161 is a SMAC mimetic, an IAP antagonist with oral activity that inhibits XIAP and cIAP1. LCL161 has potential antitumor activity. Cost-effective and quality-assured.</p>Formule :C26H33FN4O3SDegré de pureté :99.13% - 99.87%Couleur et forme :SolidMasse moléculaire :500.63Mocetinostat
CAS :<p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>Formule :C23H20N6ODegré de pureté :99% - 99.21%Couleur et forme :SolidMasse moléculaire :396.44AG1024
CAS :<p>AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).</p>Formule :C14H13BrN2ODegré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :305.17Sertaconazole
CAS :<p>Sertaconazole is a broad-spectrum antifungal.</p>Formule :C20H15Cl3N2OSDegré de pureté :99.483%Couleur et forme :SolidMasse moléculaire :437.77Rigosertib
CAS :<p>Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by disrupting PI3K/Akt.</p>Formule :C21H25NO8SDegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :451.49PI-103
CAS :<p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>Formule :C19H16N4O3Degré de pureté :97.79% - 99.3%Couleur et forme :SolidMasse moléculaire :348.36ML311
CAS :<p>ML311 is a selective inhibitor of the Mcl-1/Bim interaction.</p>Formule :C23H24F3N3ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :415.45Asiaticoside
CAS :<p>Asiaticoside, in Centella asiatica, may treat wounds/burns.</p>Formule :C48H78O19Degré de pureté :98% - 99.96%Couleur et forme :PowderMasse moléculaire :959.12SC66
CAS :<p>SC66 is a AKT inhibitor in HepG2, HA22T/VGH, and PLC/PRF/5 cells (IC50: about 0.75 μg/ml, at 72 h).</p>Formule :C18H16N2ODegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :276.33Rhosin hydrochloride
CAS :<p>Rhosin hydrochloride is a specific inhibitor of the RhoA subfamily Rho GTPases.Cost-effective and quality-assured.</p>Formule :C20H20Cl2N6ODegré de pureté :97.33% - 98.92%Couleur et forme :SolidMasse moléculaire :431.318NADPH tetracyclohexanamine
CAS :<p>NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.</p>Formule :C45H82N11O17P3Degré de pureté :98.73% - 99.05%Couleur et forme :SolidMasse moléculaire :1142.12Idasanutlin
CAS :<p>Idasanutlin (Ro 5503781) (RG-7388) is an effective and specific p53-MDM2 inhibitor (IC50: 6 nM).</p>Formule :C31H29Cl2F2N3O4Degré de pureté :99.13% - 99.88%Couleur et forme :SolidMasse moléculaire :616.48CPTH2
CAS :<p>CPTH2 is a histone acetyltransferase inhibitor modulating Gcn5 network.</p>Formule :C14H14ClN3SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :291.8ZMC1
CAS :<p>NSC-319726 (ZMC1), a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).</p>Formule :C11H14N4SDegré de pureté :98.97% - 99.76%Couleur et forme :SolidMasse moléculaire :234.32RAD51 Inhibitor B02
CAS :<p>RAD51 Inhibitor B02 (B02) (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM.</p>Formule :C22H17N3ODegré de pureté :99.72% - 99.89%Couleur et forme :SolidMasse moléculaire :339.39Bendamustine
CAS :<p>Bendamustine (SDX105) for the treatment of Non-Hodgkin Lymphomas and Chronic Lymphocytic Leukemia</p>Formule :C16H21Cl2N3O2Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :358.26Sertaconazole nitrate
CAS :<p>Sertaconazole nitrate, a broad-spectrum topical antifungal, treats skin and mucosal infections.</p>Formule :C20H15Cl3N2OS·HNO3Degré de pureté :98.66% - 99.65%Couleur et forme :SolidMasse moléculaire :500.78Almorexant
CAS :<p>Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for OX1 and 0.17 nM for OX2.</p>Formule :C29H31F3N2O3Degré de pureté :97.75% - 98.02%Couleur et forme :SolidMasse moléculaire :512.56Grape Seed Extract
CAS :<p>Grape Seed Extract (Grape Seed P.E.) is exudate from seeds of the grape plant Vitis vinifera, composed of oils and secondary plant metabolites.</p>Formule :C32H30O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :590.581CVT-11127
CAS :<p>CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.</p>Formule :C25H23Cl2N5O3Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :512.39N-Ethylmaleimide
CAS :<p>N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor. Cost-effective and quality-assured.</p>Formule :C6H7NO2Degré de pureté :99.50%Couleur et forme :White SolidMasse moléculaire :125.13Cucurbitacin IIA
CAS :<p>1.</p>Formule :C32H50O8Degré de pureté :98.62% - 99.87%Couleur et forme :SolidMasse moléculaire :562.73OSI-930
CAS :<p>OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.</p>Formule :C22H16F3N3O2SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :443.44Tanespimycin
CAS :<p>Tanespimycin (KOS 953) is an Hsp90 inhibitor (IC50=5 nM) and is selective. Tanespimycin depletes intracellular STK38/NDR1. High-Quality, Low-Cost!</p>Formule :C31H43N3O8Degré de pureté :99.07% - 99.83%Couleur et forme :Dark Purple SolidMasse moléculaire :585.692-tert-Butyl-1,4-benzoquinone
CAS :<p>TBQ, a BHA metabolite, activates Nrf2 and S-arylates Keap1 in RAW264.7 cells.</p>Formule :C10H12O2Degré de pureté :97.19%Couleur et forme :SolidMasse moléculaire :164.2Quizartinib
CAS :<p>Quizartinib (AC220) is an inhibitor of FLT3 (Kd: 1.6 nM) and demonstrates high selectivity for FLT3 when tested against a panel of 227 additional kinases.</p>Formule :C29H32N6O4SDegré de pureté :98% - 99.42%Couleur et forme :SolidMasse moléculaire :560.67Caudatin
CAS :<p>Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.</p>Formule :C28H42O7Degré de pureté :98.83% - 99.9%Couleur et forme :SolidMasse moléculaire :490.63Taurochenodeoxycholic acid sodium
CAS :<p>Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).</p>Formule :C26H44NNaO6SDegré de pureté :98.23% - 99.45%Couleur et forme :White To Off-White PowderMasse moléculaire :521.68GSK-J4
CAS :<p>GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.</p>Formule :C24H27N5O2Degré de pureté :98.24% - 99.98%Couleur et forme :SolidMasse moléculaire :417.5Angelicin
CAS :<p>Angelicin (Isopsoralen), is a furanocoumarin with anti-Y, antiviral, anti-inflammatory activity.</p>Formule :C11H6O3Degré de pureté :99.86% - 99.89%Couleur et forme :White SolidMasse moléculaire :186.16Fimasartan
CAS :<p>Fimasartan (BR-A-657), an ARB, treats hypertension and heart failure; safe with hydrochlorothiazide.</p>Formule :C27H31N7OSDegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :501.65Lenalidomide hemihydrate
CAS :<p>Lenalidomide hemihydrate inhibits TNF-α (IC50=13nM) and binds CRBN/DDB1 complexes.</p>Formule :C13H13N3O3H2ODegré de pureté :96.22%Couleur et forme :SolidMasse moléculaire :268.28ASTX660
CAS :<p>Tolinapant (ASTX660) is an orally bioavailable cIAP1/2 and XIAP antagonist.Cost-effective and quality-assured.</p>Formule :C30H42FN5O3Degré de pureté :98.33% - 99.85%Couleur et forme :SolidMasse moléculaire :539.68Palomid 529
CAS :<p>Palomid 529 (SG 00529) has been used in trials studying the treatment of Age-Related Macular Degeneration.</p>Formule :C24H22O6Degré de pureté :98.40% - 98.59%Couleur et forme :SolidMasse moléculaire :406.43BI-6C9
CAS :<p>BI-6C9 is an inhibitor of tBid (Kd = 20 μM).BI-6c9 prevented MOMP and mitochondrial fission, and protected the cells from cell death.</p>Formule :C23H25N3O4S2Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :471.59Alogliptin
CAS :<p>Alogliptin (SYR-322)(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of <10 nM, exhibits greater than 10, 000-fold selectivity over DPP-8 and DPP-9</p>Formule :C18H21N5O2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :339.39Takinib
CAS :<p>Takinib (EDHS-206) is a specific and effective TAK1 inhibitor(IC50= 9.5 nM).</p>Formule :C18H18N4O2Degré de pureté :98.29% - 99.35%Couleur et forme :SolidMasse moléculaire :322.36ML-210
CAS :<p>ML-210 (CID 49766530) is a glutathione peroxidase 4 (GPX4) inhibitor. ML-210 has antitumor activity and induces ferroptosis. Cost-effective and quality-assured.</p>Formule :C22H20Cl2N4O4Degré de pureté :97% - 99.03%Couleur et forme :SolidMasse moléculaire :475.32UMI-77
CAS :<p>UMI-77 is a selective Mcl-1 inhibitor. UMI-77 binds to the BH3-binding groove of Mcl-1.Cost-effective and quality-assured.</p>Formule :C18H14BrNO5S2Degré de pureté :96% - 99.57%Couleur et forme :SolidMasse moléculaire :468.34ACBI1
CAS :<p>ACBI1 is a potent PROTAC degrader of BAF ATPase subunits SMARCA2 and SMARCA4, also degrades the polybromo-associated BAF (PBAF) complex member PBRM1, with DC50s</p>Formule :C49H58FN9O7SDegré de pureté :97.54% - 98.15%Couleur et forme :SolidMasse moléculaire :936.1[8]-Shogaol
CAS :<p>[8]-Shogaol is a component of ginger and maintains anti-inflammatory activity as a cyclooxygenase-2 inhibitor.</p>Formule :C19H28O3Degré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :304.42R-7050
CAS :<p>R-7050 (TNF-α Antagonist III), a tumor necrosis factor receptor (TNFR) antagonist, exhibits heightened selectivity for TNFα.</p>Formule :C16H8ClF3N4SDegré de pureté :98.64% - 99.8%Couleur et forme :SolidMasse moléculaire :380.77(+)-Nortrachelogenin
CAS :<p>(+)-Nortrachelogenin is a lignan isolated from Wikstroemia indica C.A. Meyer (Thymelaeaceae). (+)-Nortrachelogenin possesses antileukemic activity.</p>Formule :C20H22O7Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :374.38Cidofovir dihydrate
CAS :<p>Cidofovir dihydrate: Injectable anti-CMV; suppresses CMV by inhibiting viral DNA polymerase; treats CMV retinitis in AIDS.</p>Formule :C8H18N3O8PDegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :315.22Erdafitinib
CAS :<p>Erdafitinib (JNJ-42756493) is a quinoxaline derivative compound, acts on FGFR1/2/3/4.</p>Formule :C25H30N6O2Degré de pureté :97.00% - 99.07%Couleur et forme :SolidMasse moléculaire :446.54ASK1-IN-1
CAS :<p>ASK1-IN-1 inhibits apoptosis kinase 1, crucial in cell stress responses, with 21 nM IC50.</p>Formule :C19H19N9O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :405.41Taurochenodeoxycholic Acid
CAS :<p>Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.</p>Formule :C26H45NO6SDegré de pureté :99.53% - 99.86%Couleur et forme :SolidMasse moléculaire :499.7MGH-CP1
CAS :<p>MGH-CP1 inhibits TEAD2/4 auto-palmitoylation with IC50 of 710 and 672 nM, respectively.</p>Formule :C20H24N4OSDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :368.5BAY 61-3606 dihydrochloride
CAS :<p>BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).</p>Formule :C20H18N6O3·2HClDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :463.32Lycorine
CAS :<p>Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.</p>Formule :C16H17NO4Degré de pureté :98.60% - 99.95%Couleur et forme :SolidMasse moléculaire :287.312BAct
CAS :<p>2BAct is a novel eif2b activator, preventing neurological defects caused by a chronic integrated stress response</p>Formule :C19H16ClF3N4O3Degré de pureté :97.97% - 99.04%Couleur et forme :SolidMasse moléculaire :440.8Irigenin
CAS :<p>Irigenin mediates its antimetastatic effect by specifically and selectively blocking the α9β1 and α4β1 integrin binding sites on the C-C loop of the Extra</p>Formule :C18H16O8Degré de pureté :99.50% - 99.85%Couleur et forme :SolidMasse moléculaire :360.31ML141
CAS :<p>ML141 (CID-2950007) is an effective, specific and reversible non-competitive inhibitor of Rho family GTPase cdc42 (IC50: 200 nM).</p>Formule :C22H21N3O3SDegré de pureté :99.36% - 99.56%Couleur et forme :SolidMasse moléculaire :407.49SW106065
CAS :<p>SW106065 is a novel pharmacologic inducer of apoptosis in MPNST (malignant peripheral nerve sheath tumors). SW106065 inhibits ATP consumption of sMPNST.</p>Formule :C10H8N2OSDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :204.25(S)-(+)-Rolipram
CAS :<p>(S)-(+)-Rolipram ((+)-Rolipram) inhibits human monocyte cyclic AMP-specific PDE4 with IC50 of 0.75 μM, has anti-inflammatory and anti-depressant activity in the</p>Formule :C16H21NO3Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :275.34Nur77 modulator 1
CAS :<p>Nur77 modulator 1: binds at 3.58 μM, boosts expression, alters location, triggers ER stress/autophagy, induces apoptosis, and fights hepatoma.</p>Formule :C28H25N5O2SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :495.6KRIBB11
CAS :<p>KRIBB11 is an inhibitor of Heat shock factor (HSF) inhibitor.</p>Formule :C13H12N6O2Degré de pureté :97.25% - 99.91%Couleur et forme :SolidMasse moléculaire :284.27Asperosaponin VI
CAS :<p>Asperosaponin VI, from Dipsacus asper rhizome, treats back pain, hematoma, and fractures.</p>Formule :C47H76O18Degré de pureté :97.15% - 99.79%Couleur et forme :SolidMasse moléculaire :929.1Ginsenoside Rg6
CAS :<p>Ginsenoside Rg6 inhibits the proliferation and induces apoptosis of human lymphoma JK cells</p>Formule :C42H70O12Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :767GSK2334470
CAS :<p>GSK2334470 is a novel PDK1 inhibitor (IC50: ~10 nM, in a cell-free assay), with no inhibitory at other close related AGC-kinases.</p>Formule :C25H34N8ODegré de pureté :99.57% - 99.87%Couleur et forme :SolidMasse moléculaire :462.59Dictamine
CAS :<p>Dictamine (Dectamine) shows anticholinesterase, anti-inflammatory, mutagenic, and has antimicrobial activity against bacteria and fungi.</p>Formule :C12H9NO2Degré de pureté :99.72% - 99.889%Couleur et forme :SolidMasse moléculaire :199.21Masitinib
CAS :<p>Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in animals, specifically dogs.</p>Formule :C28H30N6OSDegré de pureté :97.56% - >99.99%Couleur et forme :SolidMasse moléculaire :498.64RSL3
CAS :<p>View and buy RSL3 from TargetMol.RSL3 is a VDAC-independent ferroptosis activator.Cited in 10 publications.</p>Formule :C23H21ClN2O5Degré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :440.88Schisandrin C
CAS :<p>Schisandrin C (Wuweizisu-C) is a phytochemical lignan isolated from Schizandra chinensis Baill; shows anticancer-effects in human leukemia U937 cells.</p>Formule :C22H24O6Degré de pureté :99.44% - 99.56%Couleur et forme :SolidMasse moléculaire :384.42WM-3835
CAS :<p>WM-3835, a specific KAT7 inhibitor, potently halts OS cell growth, migration, and induces apoptosis.</p>Formule :C20H17FN2O4SDegré de pureté :97.78% - 99.36%Couleur et forme :SolidMasse moléculaire :400.42Venetoclax
CAS :<p>Venetoclax (ABT-199) is a selective inhibitor of Bcl-2 (Ki < 0.010 nM), binding over 3 orders of magnitude less avidly to Bcl-xL, and Bcl-W (Kis = 48/245 nM).</p>Formule :C45H50ClN7O7SDegré de pureté :98.00% - 99.97%Couleur et forme :SolidMasse moléculaire :868.44Monomethyl auristatin E
CAS :<p>Monomethyl auristatin E (MMAE) (MMAE), an antimitotic agent, inhibits cell division by blocking the polymerization of tubulin and also has inhibition of</p>Formule :C39H67N5O7Degré de pureté :98.47% - 99.9%Couleur et forme :SolidMasse moléculaire :717.98Limonin
CAS :<p>Limonin (Citrolimonin) is a triterpenoid enriched in citrus fruits, which has antivirus and antitumor ability.</p>Formule :C26H30O8Degré de pureté :99.65% - 99.66%Couleur et forme :White To Slightly Off White PowderMasse moléculaire :470.51(-)-Huperzine A
CAS :<p>(-)-Huperzine A: Lycopodium alkaloid, AChE inhibitor, treats Alzheimer's in China.</p>Formule :C15H18N2ODegré de pureté :99.19% - >99.99%Couleur et forme :White To Slight White Crystaline PowderMasse moléculaire :242.32Zoledronic Acid
CAS :<p>Zoledronic Acid (ZOL 446) 是一种含氮二磷酸盐,能抑制破骨细胞的分化和凋亡,具有高效的抗骨质再吸收活性,也有抗癌作用。</p>Formule :C5H10N2O7P2Degré de pureté :98% - 99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :272.09Troglitazone
CAS :<p>Troglitazone (Romglizone) is a PPARγ agonist with anti-inflammatory and anti-tumor activity.</p>Formule :C24H27NO5SDegré de pureté :98% - 99.8%Couleur et forme :Yellow SolidMasse moléculaire :441.54KYP-2047
CAS :<p>KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor.</p>Formule :C20H25N3O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :339.43Artemisitene
CAS :<p>Artemisitene, an oxidized antimalarial derivative of Artemisinin, stems from precursors like Artemisinin B and Artemisinic acid.</p>Formule :C15H20O5Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :280.32BAM7
CAS :<p>BAM 7 is a direct and specific activator of proapoptotic Bax (EC50: 3.3 μM).</p>Formule :C21H19N5O2SDegré de pureté :98.51% - 98.68%Couleur et forme :SolidMasse moléculaire :405.47Glyphosate
CAS :<p>Glyphosate (Atila) is an herbicide. It also is a possible carcinogen to humans.</p>Formule :C3H8NO5PDegré de pureté :99.12% - 99.91%Couleur et forme :White Crystals (Darkens) Ph (1% Solution In Water) 2 5 (Ntp 1992)Masse moléculaire :169.07GSK621
CAS :<p>GSK621 is a specific and potent AMPK activator.</p>Formule :C26H20ClN3O5Degré de pureté :97.02% - 97.05%Couleur et forme :SolidMasse moléculaire :489.91Sodium Oxamate
CAS :<p>Sodium Oxamate (Oxamic acid sodium salt) is an LDH inhibitor that specifically inhibits LDHA.</p>Formule :C2H2NNaO3Degré de pureté :99.23% - ≥98%Couleur et forme :White Crystalline PowderMasse moléculaire :111.03SC99
CAS :SC99 inhibits JAK2-STAT3, reducing STAT3 genes, platelet activity, and has anti-myeloma, anti-thrombotic effects.Formule :C15H8Cl2FN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :336.15Cichoric Acid
CAS :<p>Cichoric Acid (Dicaffeoyltartaric acid) is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues.</p>Formule :C22H18O12Degré de pureté :97.87% - 98.77%Couleur et forme :SolidMasse moléculaire :474.37BML-210
CAS :<p>BML-210 (CAY10433) is a new-type HDAC inhibitor.</p>Formule :C20H25N3O2Degré de pureté :96.37% - 98.12%Couleur et forme :SolidMasse moléculaire :339.43
