Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(196 produits)
- Caséine Kinase(138 produits)
- DHFR(32 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(85 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(134 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(86 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(22 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(45 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9182 produits trouvés pour "Métabolisme"
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CP-609754
CAS :CP-609754 shows selective inhibition of farnesyltransferase.Formule :C29H22ClN3O2Degré de pureté :99.86% - 99.87%Couleur et forme :SolidMasse moléculaire :479.96Ref: TM-T38050
1mg55,00€5mg116,00€10mg187,00€25mg319,00€50mg449,00€100mg638,00€200mg840,00€1mL*10mM (DMSO)134,00€CS 722
CAS :CS 722 is a centrally acting muscle relaxant. CS-722 exerts its muscle relaxant action by affecting both the supraspinal structure and the spinal cord.Formule :C16H20Cl2N2O4Couleur et forme :SolidMasse moléculaire :375.25Olprinone
CAS :Olprinone (Loprinone)(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor.Olprinone has been reported to improve microcirculation and attenuateFormule :C14H10N4ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :250.26Sacubitril
CAS :Sacubitril (AHU-377) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril is a component of the heart failure medicine LCZ696.
Formule :C24H29NO5Degré de pureté :97.72% - 97.91%Couleur et forme :SolidMasse moléculaire :411.49Voglibose
CAS :Voglibose (Glustat), an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemiaFormule :C10H21NO7Degré de pureté :98% - 99.90%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :267.28Firibastat
CAS :Firibastat (RB150) is a glutamyl aminopeptidase antagonist and an orally active brain penetrating prodrug of EC33.
Formule :C8H20N2O6S4Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :368.51Sephin1 Hydrochloride
CAS :Sephin1 HCl selectively inhibits PPP1R15A, enhancing eIF2α phosphorylation to protect cells from proteostatic flaws.Formule :C8H10Cl2N4Couleur et forme :SolidMasse moléculaire :233.1Kresoxim-Methyl
CAS :Kresoxim-methyl is a strobilurin fungicide,inhibits conidial germination of V. inaequalis isolates from apple orchards .Formule :C18H19NO4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :313.35MASM7
CAS :MASM7: mitochondrial fusion activator, a cyclopenta[b]thiophene derivative used in molecular structures.Formule :C22H23N5O2S2Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :453.58Ref: TM-T50093
1mg69,00€5mg147,00€10mg224,00€25mg358,00€50mg512,00€100mg707,00€200mg982,00€1mL*10mM (DMSO)164,00€IDO-IN-1
CAS :IDO-IN-1: potent IDO inhibitor, IC50 of 59 nM (enzyme), 12 nM (HeLa cells).Formule :C9H7BrFN5O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :316.09Ref: TM-T7181
1mg49,00€5mg96,00€10mg155,00€25mg269,00€50mg404,00€100mg567,00€200mg763,00€1mL*10mM (DMSO)110,00€Cyclo(his-pro)
CAS :Cyclo(his-pro) is a cyclic dipeptide that shields against oxidative damage by activating Nrf2.Formule :C11H14N4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :234.25MSDC 0160
CAS :MSDC 0160 (CAY10415) is a prototype mTOT-modulating insulin sensitizer being used in trials studying the treatment of Type 2 Diabetes and Alzheimer's Disease.Formule :C19H18N2O4SDegré de pureté :98.11% - 99.53%Couleur et forme :SolidMasse moléculaire :370.42Ref: TM-T2607
1mg35,00€2mg50,00€5mg77,00€10mg99,00€25mg154,00€50mg197,00€100mg350,00€1mL*10mM (DMSO)82,00€Acipimox sodium
CAS :Acipimox sodium is an antilipolytic, enhancing leptin, curbing lipolysis and FFAs, and boosting insulin sensitivity.Formule :C6H5N2NaO3Couleur et forme :SolidMasse moléculaire :176.11Tetrahydropapaverine hydrochloride
CAS :Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.Formule :C20H26ClNO4Degré de pureté :99.08%Couleur et forme :White Crystal PowderMasse moléculaire :379.8786-Aminocaproic acid hydrochloride
CAS :6-Aminocaproic acid HCl: Potent oral antifibrinolytic; blocks plasminogen binding; used for bleeding disorder research.Formule :C6H14ClNO2Couleur et forme :SolidMasse moléculaire :167.634Pyributicarb
CAS :Pyributicarb (TSH-888) is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).Formule :C18H22N2O2SDegré de pureté :99.702% - ≥95%Couleur et forme :SolidMasse moléculaire :330.44PCC0208009
CAS :PCC0208009 (IDO-IN-2) is an IDO inhibitor.Formule :C29H35N7ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :497.63Ref: TM-T4142
1mg44,00€2mg56,00€5mg93,00€10mg142,00€25mg258,00€50mg439,00€100mg605,00€1mL*10mM (DMSO)92,00€Phenprocoumon
CAS :Phenprocoumon is an antagonist of vitamin K(IC50:1 μM).Formule :C18H16O3Degré de pureté :95.79% - 97.98%Couleur et forme :Fine White Crystalline Powder SolidMasse moléculaire :280.32Ro 20-1724
CAS :Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) is a widely used inhibitor of cyclic nucleotide phosphodiesterase with IC50 of 2.0 μM and Ki of 3.1Formule :C15H22N2O3Degré de pureté :98.82% - 99.79%Couleur et forme :SolidMasse moléculaire :278.35Udenafil
CAS :Udenafil is an inhibitor of PDE5 .Formule :C25H36N6O4SDegré de pureté :99.90%Couleur et forme :Off-White SolidMasse moléculaire :516.66Ref: TM-T17199
5mg50,00€10mg80,00€25mg140,00€50mg219,00€100mg319,00€200mg457,00€1mL*10mM (DMSO)52,00€Icerguastat
CAS :Icerguastat (IFB-088) is a selective inhibitor of holophosphatase. Icerguastat selectively inhibited a regulatory subunit of protein phosphatase 1 in vivo.Formule :C8H9ClN4Degré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :196.64Amifostine sodium
CAS :Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formule :C5H15N2NaO3PSCouleur et forme :SolidMasse moléculaire :237.21Mutant IDH1-IN-1
CAS :Mutant IDH1-IN-1 is a potent mutant IDH1 R132 h inhibitor with IC50 < 0.1 uM.Formule :C30H31FN4O2Degré de pureté :99.49% - >99.99%Couleur et forme :SolidMasse moléculaire :498.59Ref: TM-T2043
2mg44,00€5mg67,00€10mg94,00€25mg173,00€50mg249,00€100mg363,00€200mg490,00€1mL*10mM (DMSO)71,00€AS-252424
CAS :AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; >10 fold selectivity for PI3Kγ versus PI3Kα.Formule :C14H8FNO4SDegré de pureté :99.06% - 99.09%Couleur et forme :SolidMasse moléculaire :305.28Ref: TM-T6208
1mg37,00€2mg52,00€5mg77,00€10mg128,00€25mg205,00€50mg309,00€100mg447,00€500mg973,00€1mL*10mM (DMSO)84,00€ML348
CAS :ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Formule :C18H17ClF3N3O3Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :415.79Ref: TM-T3439
2mg44,00€5mg65,00€10mg92,00€25mg215,00€50mg334,00€100mg537,00€200mg750,00€500mg1.134,00€2-Oxobutanoic acid
CAS :2-Oxobutanoic acid, from cystathionine lysis and threonine degradation, becomes propionyl-CoA for the citric acid cycle.Formule :C4H6O3Degré de pureté :97% - 99.47%Couleur et forme :SolidMasse moléculaire :102.09B2
CAS :B2 (Linazolamide intermediate B impurity 2) promotes inclusion formation in cellular models of Huntington's disease and Parkinson's diseaseFormule :C20H17ClN4O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :396.83Deserpidine hydrochloride
CAS :Deserpidine hydrochloride is an antihypertensive, ACE-inhibiting drug derived from Rauwolfia, reducing blood pressure and aldosterone secretion.Formule :C32H39ClN2O8Couleur et forme :SolidMasse moléculaire :615.12TP0463518
CAS :TP-0463518 is a highly potent HIF prolyl hydroxylase (PHD) inhibitor (IC50s: 13 nM and 18 nM for human and rat PHD2, respectively).Formule :C20H18ClN3O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :431.83Ibiglustat hydrochloride
CAS :Ibiglustat hydrochloride is a potent and selective Glucosylceramide synthase inhibitor and ceramide glucosyltransferase inhibitor.Formule :C20H25ClFN3O2SCouleur et forme :SolidMasse moléculaire :425.95JNJ-1661010
CAS :JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.Formule :C19H19N5OSDegré de pureté :99.79% - 99.97%Couleur et forme :SolidMasse moléculaire :365.45CP-91149
CAS :CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM in the presence of glucose, 5- to 10-fold less potent in the absence ofFormule :C21H22ClN3O3Degré de pureté :99.66% - 99.81%Couleur et forme :SolidMasse moléculaire :399.87Ref: TM-T6455
2mg35,00€5mg51,00€10mg84,00€25mg137,00€50mg197,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)57,00€Potassium 2-hydroxy-2-methylsuccinate
CAS :Potassium 2-hydroxy-2-methylsuccinate ((±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt) is a type of endogenous metabolite.Formule :C5H6K2O5Degré de pureté :99.96% - ≥98%Couleur et forme :SolidMasse moléculaire :224.29Nitecapone
CAS :Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Formule :C12H11NO6Degré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :265.226-Phosphogluconic acid
CAS :6-Phosphogluconic acid competitively inhibits PGI with Ki: 0.048 mM for glucose 6-P, 0.042 mM for fructose 6-P.Formule :C6H13O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :276.14Tebuconazole
CAS :Tebuconazole: azole fungicide, inhibits CYP51 with IC50s 0.9 μM (C. albicans) and 1.3 μM (human).Formule :C16H22ClN3ODegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :307.82L-Gulose
CAS :L-Gulose: unnatural L-hexose, sweet syrup, vitamin C biosynthesis intermediate.Formule :C6H12O6Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :180.16Oxytetracycline Dihydrate
CAS :Oxytetracycline Dihydrate (Terramycin Dihydrate) is a prescription antibiotic, interfering with the ability of bacteria to produce essential proteins.Formule :C22H24N2O9·2H2ODegré de pureté :99.80%Couleur et forme :CrystallineMasse moléculaire :496.46RPI-1
CAS :RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.
Formule :C17H15NO4Degré de pureté :98.91% - ≥95%Couleur et forme :SolidMasse moléculaire :297.31Alagebrium chloride
CAS :Alagebrium chloride (ALT711) inhibits AGEs, lowers systolic blood pressure, and benefits diastolic patients.Formule :C13H14ClNOSDegré de pureté :99.65% - 99.77%Couleur et forme :SolidMasse moléculaire :267.77RHC 80267
CAS :RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Formule :C20H34N4O4Degré de pureté :99.54%Couleur et forme :White SolidMasse moléculaire :394.51Uridine 5′-triphosphate tris salt
CAS :Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) is an agonist to the P2Y receptor and has been used to study concentrations of intracellularFormule :C21H48N5O24P3Degré de pureté :99.04% - 99.94%Couleur et forme :SolidMasse moléculaire :847.55L-Leucyl-L-Leucine methyl ester hydrochloride
CAS :L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) is a dipeptide condensation product of L-leucine methyl ester. Cost-effective and quality-assured.Formule :C13H27ClN2O3Degré de pureté :98.41% - 99.63%Couleur et forme :SolidMasse moléculaire :294.81CM10
CAS :CM10 is an aldehyde dehydrogenase 1A family(ALDH1A) inhibitor.Formule :C20H23N3ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :321.42Aranidipine
CAS :Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.Formule :C19H20N2O7Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :388.37Enecadin HCl
CAS :Enecadin HCl is a voltage-dependent sodium and calcium channel blocker.Formule :C21H29ClFN3OCouleur et forme :SolidMasse moléculaire :393.93Lazabemide hydrochloride
CAS :Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki：7.9nM).Formule :C8H11Cl2N3ODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :236.098Liquiritin
CAS :Liquiritin (Liquiritigenin-4'-O-glucoside) (LIQ) is a main component among the licorice flavonoids, and possesses anti-inflammatory and anti-cancer abilities.Formule :C21H22O9Degré de pureté :98.16% - 98.66%Couleur et forme :SolidMasse moléculaire :418.39AGI-6780
CAS :AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.Formule :C21H18F3N3O3S2Degré de pureté :98.19% - 99.7%Couleur et forme :SolidMasse moléculaire :481.51Ref: TM-T1809
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg220,00€50mg393,00€100mg587,00€500mg1.264,00€1mL*10mM (DMSO)85,00€Tienilic Acid
CAS :Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
Formule :C13H8Cl2O4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :331.17PFK-015
CAS :PFK-015 (PFK15) is an effective inhibitor of PFKFB3 (IC50: 110 nM) and inhibits PFKFB3 activity in Y cells (IC50: 20 nM).Formule :C17H12N2ODegré de pureté :99.7% - 99.85%Couleur et forme :SolidMasse moléculaire :260.29Ref: TM-T2455
2mg40,00€5mg57,00€10mg88,00€25mg159,00€50mg250,00€100mg376,00€200mg550,00€1mL*10mM (DMSO)57,00€7-Hydroxy-3,4-dihydro-2(1H)-quinolinone
CAS :7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .Formule :C9H9NO2Degré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :163.17Oseltamivir acid
CAS :Oseltamivir acid (GS4071) is a potent influenza virus neuraminidase inhibitor and the prodrug of GS4071.Formule :C14H24N2O4Degré de pureté :97.66% - 98.88%Couleur et forme :SolidMasse moléculaire :284.35Ref: TM-T5186
1mg34,00€5mg70,00€10mg103,00€25mg187,00€50mg286,00€100mg409,00€200mg590,00€1mL*10mM (DMSO)75,00€IMR-1A
CAS :IMR-1A is the metabolite of IMR-1 which is a novel class of Notch inhibitors targeting the transcriptional activation with IC50 of 6 μMol/L.Formule :C13H11NO5S2Degré de pureté :97.1% - 99.76%Couleur et forme :SolidMasse moléculaire :325.36Ref: TM-T3540
1mg47,00€5mg92,00€10mg145,00€25mg295,00€50mg477,00€100mg715,00€200mg964,00€1mL*10mM (DMSO)99,00€NCC007
CAS :NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.Formule :C22H28F3N7Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :447.5Rolipram
CAS :Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Formule :C16H21NO3Degré de pureté :99.22% - >99.99%Couleur et forme :SolidMasse moléculaire :275.34Nampt-IN-1
CAS :Nampt-IN-1 (LSN3154567) (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM.Formule :C20H25N3O5SDegré de pureté :99.28% - 99.4%Couleur et forme :SolidMasse moléculaire :419.49Ref: TM-T4376
1mg37,00€2mg49,00€5mg79,00€10mg130,00€25mg245,00€50mg409,00€100mg605,00€1mL*10mM (DMSO)87,00€Y-29794 Tosylate
CAS :Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.Formule :C30H42N2O4S3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :590.86PQ-10
CAS :PQ-10 (A-844337) is a PDE-10 inhibitor. PQ-10 induces brain glucose metabolism patterns, which may be a potential translational biomarker.
Formule :C22H21N5O3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :403.43SR1001
CAS :SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).Formule :C15H13F6N3O4S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :477.4CP-640186 hydrochloride
CAS :CP-640186 hydrochloride (CP 640186 HCl) is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor, including rat liver ACC1 (IC50: 53 nM) and rat
Formule :C30H36ClN3O3Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :522.08Edoxaban Tosylate Monohydrate
CAS :Edoxaban(DU-176) is an oral factor Xa (FXa) inhibitor in clinical development for stroke prevention.Formule :C31H40ClN7O8S2Degré de pureté :99.86% - 99.91%Couleur et forme :SolidMasse moléculaire :738.27Fondaparinux sodium
CAS :Fondaparinux sodium (SR-90107A) is an antithrombin-dependent factor Xa inhibitor with antithrombotic activity.Formule :C31H43N3Na10O49S8Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :1728.08HNHA
CAS :HNHA is an inhibitor of HDAC.Formule :C17H21NO2SDegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :303.42Ref: TM-T21806
1mg44,00€5mg84,00€10mg135,00€25mg279,00€50mg445,00€100mg640,00€200mg879,00€1mL*10mM (DMSO)90,00€FOY 251
CAS :FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.Formule :C17H19N3O7SDegré de pureté :97.11% - 99.33%Couleur et forme :SolidMasse moléculaire :409.41Ref: TM-T8676
1mg51,00€5mg110,00€10mg177,00€25mg300,00€50mg424,00€100mg605,00€500mg1.198,00€1mL*10mM (DMSO)126,00€Dimethylfraxetin
CAS :Dimethylfraxetin (6,7,8-Trimethoxycoumarin) is a Carbonic anhydrase inhibitor(Ki：0.0097 μM)Formule :C12H12O5Degré de pureté :99.96% - ≥95%Couleur et forme :SolidMasse moléculaire :236.22EMD638683
CAS :EMD638683,a novel SGK inhibitor with antihypertensive potency(with an IC50 of 3 μM).Formule :C18H18F2N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.34Ref: TM-T6635
1mg74,00€2mg92,00€5mg150,00€10mg233,00€25mg358,00€50mg517,00€100mg737,00€200mg982,00€1mL*10mM (DMSO)120,00€Rosiptor
CAS :Rosiptor (AQX-1125) (AQX-1125) is an orally-active and specific phosphatase SHIP1 activator with anti-inflammatory effects.Formule :C20H35NO2Degré de pureté :99.53% - 99.73%Couleur et forme :SolidMasse moléculaire :321.5HA 155
CAS :HA 155 (Autotaxin Inhibitor IV) is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.Formule :C24H19BFNO5SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :463.29Roflumilast N-oxide
CAS :Roflumilast N-oxide is an inhibitor of PDE type 4.Formule :C17H14Cl2F2N2O4Degré de pureté :98.19% - 99.69%Couleur et forme :SolidMasse moléculaire :419.21Ref: TM-T4462
1mg35,00€2mg52,00€5mg74,00€10mg99,00€25mg170,00€50mg274,00€100mg350,00€500mg840,00€1mL*10mM (DMSO)69,00€Melilotic acid
CAS :3-(2-Hydroxyphenyl)propanoic acid, aka melilotic acid, found in cytoplasm, in foods like herbs, beetroot, cinnamon.Formule :C9H10O3Degré de pureté :99.65% - 99.83%Couleur et forme :SolidMasse moléculaire :166.17PD 128042
CAS :PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formule :C23H39NO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.56KML29
CAS :KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.Formule :C24H21F6NO7Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :549.42K-Ras-PDEδ-IN-1
CAS :K-Ras-PDEδ-IN-1 is a potent inhibitor of competitive K-Ras-PDEδ.It binds to the farnesyl binding pocket of PDEδ(Kd of 8 nM).
Formule :C25H26FN5O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :447.5Cilomilast
CAS :Cilomilast (SB-207499) is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.Formule :C20H25NO4Degré de pureté :97.37% - 99.52%Couleur et forme :White SolidMasse moléculaire :343.42BI-0115
CAS :BI-0115 inhibits LOX-1, preventing oxLDL uptake by triggering receptor inhibition and dimer formation.Formule :C15H14ClN3ODegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :287.74UCPH-101
CAS :UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Formule :C27H22N2O3Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :422.48Ref: TM-T4138
1mg50,00€2mg75,00€5mg130,00€10mg203,00€25mg409,00€50mg655,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)142,00€AGI-5198
CAS :AGI-5198 (IDH-C35) is a highly effective and specific inhibitor of IDH1 R132H/R132C mutants (IC50: 0.07/0.16 μM).Formule :C27H31FN4O2Degré de pureté :97.37% - 99.23%Couleur et forme :SolidMasse moléculaire :462.56LHW090-A7
CAS :LHW090-A7 is an neutral endopeptidase (NEP) inhibitor, and an enzyme responsible for the metabolic inactivation of enkephalins.Formule :C20H22ClNO4Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :375.85ML-030
CAS :ML-030 is a potent PDE4 inhibitor, selective for subtypes (A1, B1, B2, C1, D2) with IC50 ranging from 6.7 to 452 nM.Formule :C20H20N4O4SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :412.46ICI 63197
CAS :ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.Formule :C9H13N5ODegré de pureté :99.70%Couleur et forme :White SolidMasse moléculaire :207.23Raphin1 acetate
CAS :Raphin1 acetate is a selective and orally bioavailable regulatory phosphatase PPP1R15B (R15B) inhibitor.Formule :C10H12Cl2N4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :291.13Orthanilamide
CAS :Orthanilamide (Orthanilamide) is a molecule containing the sulfonamide functional group attached to an aniline.Formule :C6H8N2O2SDegré de pureté :99.72% - 99.96%Couleur et forme :White To Pale Cream Crystalline Powder Or CrystalsMasse moléculaire :172.2Sevelamer hydrochloride
CAS :Sevelamer hydrochloride (Sevelamer HCl) is a phosphate binding drug used to treat hyperphosphatemia via binding to dietary phosphate and prevents its absorption
Formule :(C3H7N·C3H5ClO·HCl)xDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :186.08Fraxinellone
CAS :1.Formule :C14H16O3Degré de pureté :99.35% - 99.92%Couleur et forme :SolidMasse moléculaire :232.27Ref: TM-T6S0071
2mg34,00€5mg50,00€10mg84,00€25mg152,00€50mg222,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)81,00€DG051
CAS :DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).Formule :C21H25Cl2NO4Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :426.33Ref: TM-TQ0047
2mg37,00€5mg74,00€10mg116,00€25mg239,00€50mg380,00€100mg610,00€200mg815,00€1mL*10mM (DMSO)84,00€Tebufenpyrad
CAS :Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicantFormule :C18H24ClN3ODegré de pureté :98.63% - 99.16%Couleur et forme :SolidMasse moléculaire :333.86SC-57461A
CAS :SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor.Formule :C20H26ClNO3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :363.94-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
CAS :4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) is a carbonic anhydrase inhibitor, used as a potential anti-Formule :C7H8F3N3O4S2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :319.28Tuftsin 3TFA
CAS :Tuftsin 3TFA is a tetrapeptide. It is a macrophage/microglial activator.Formule :C27H43F9N8O12Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :842.66ABX-1431
CAS :ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).Formule :C20H22F9N3O2Degré de pureté :99.8% - 99.96%Couleur et forme :SolidMasse moléculaire :507.39ISX-9
CAS :ISX-9 (Isoxazole 9) is necessary to activate neuron-specific genes as neurogenesis inducer.Formule :C11H10N2O2SDegré de pureté :97.81% - ≥95%Couleur et forme :SolidMasse moléculaire :234.27Ref: TM-T2003
2mg48,00€5mg72,00€10mg97,00€25mg155,00€50mg210,00€100mg378,00€500mg889,00€1mL*10mM (DMSO)79,00€trifarotene
CAS :Trifarotene (CD5789) is a RARγ agonist, 65x more selective than RARα and 16x than RARβ, with EC50 of 7.7 nM.
Formule :C29H33NO4Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :459.58Furafylline
CAS :Furafylline is a selective inhibitor of human cytochrome P450 (CYP)1A2 (IC50 : 0.07 μM),Formule :C12H12N4O3Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :260.25Ref: TM-T7410
1mg119,00€5mg235,00€10mg349,00€25mg593,00€50mg832,00€100mg1.159,00€200mg1.568,00€1mL*10mM (DMSO)268,00€ML351
CAS :ML351 is a potent and selective inhibitor of human 15-lipoxygenase-1 (15 LOX)(IC50: 200 nM).Formule :C15H11N3ODegré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :249.27Ref: TM-T21902
1mg50,00€5mg105,00€10mg167,00€25mg334,00€50mg505,00€100mg713,00€1mL*10mM (DMSO)117,00€Osoresnontrine
CAS :Osoresnontrine is a potent and selective inhibitor of PDE9A (IC50 of 52 nM),and can be used in the research of memory.Formule :C16H17N5O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :311.34Ref: TM-T8515
1mg38,00€2mg50,00€5mg81,00€10mg119,00€25mg188,00€50mg350,00€100mg522,00€200mg748,00€1mL*10mM (DMSO)89,00€VAS2870
CAS :VAS2870 is an inhibitor of NADPH oxidase (NOX).Formule :C18H12N6OSDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :360.39BMS-309403
CAS :BMS309403 is a potent and selective inhibitor of adipocyte fatty acid binding protein aFABP.Cost-effective and quality-assured.Formule :C31H26N2O3Degré de pureté :99.52% - 99.98%Couleur et forme :SolidMasse moléculaire :474.55Imidazole-5-propionic acid
CAS :Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination.Formule :C6H8N2O2Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :140.14Sacubitril hemicalcium salt
CAS :Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM.Formule :C48H56CaN2O10Degré de pureté :99.86% - 99.93%Couleur et forme :SolidMasse moléculaire :861.06Ref: TM-T4200
2mg39,00€5mg52,00€10mg64,00€25mg94,00€50mg106,00€100mg155,00€200mg207,00€1mL*10mM (DMSO)64,00€
