Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(197 produits)
- Caséine Kinase(139 produits)
- DHFR(30 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(63 produits)
- Facteur Xa(87 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(233 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(56 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(36 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(62 produits)
- Lipoxygénase(134 produits)
- MAO(84 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(84 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(17 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(43 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9198 produits trouvés pour "Métabolisme"
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Prasugrel chloride impurity
CAS :Prasugrel chloride impurity is an orally active antagonist of P2Y12 receptor, and inhibits ADP-induced platelet aggregation.Formule :C20H21ClFNO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :409.9PD 113413
CAS :PD 113413 is a metabolite of quinapril, an angiotensin-converting enzyme inhibitor for the treatment of hypertension and congestive heart failure.Formule :C23H24N2O4Couleur et forme :SolidMasse moléculaire :392.45Desmethylnortriptyline
CAS :Desmethylnortriptyline, a tricyclic antidepressant metabolite of nortriptyline and amitriptyline, treats depression.Formule :C18H19NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.35(+)-Xylariamide A
CAS :(+)-Xylariamide A is a probe used for mycobacterial and fungal carbonic anhydrase.Formule :C14H14ClNO6Couleur et forme :SolidMasse moléculaire :327.72Leucylarginine
CAS :Leucylarginine hinders antinociception induced by L-arginine.Formule :C12H25N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.36Z-Arg(Z)2-OH
CAS :Z-Arg(Z)2-OH can be used in the assay to screen proteolytic activities in mite homogenates.Formule :C30H32N4O8Degré de pureté :99.1400%Couleur et forme :SolidMasse moléculaire :576.6Roflumilast Impurity E
CAS :Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast acts as a selective and long-acting the enzyme PDE-4 inhibitor(IC50 value of 0.8 nM).Formule :C13H8Cl2F2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.12Bitertanol
CAS :Bitertanol (KWG 0599) is a triazole fungicide. Bitertanol inhibits demethylation, disrupts membrane function, and prevents sterol synthesis.Formule :C20H23N3O2Degré de pureté :99.88%Couleur et forme :Clear Browm Clear LiquidMasse moléculaire :337.428-Azaadenine
CAS :8-Azaadenine (NSC-32797) is an inhibitor of xanthine oxidase with IC50 of 0.54 μM and Ki of 0.66 μM.Formule :C4H4N6Degré de pureté :99.68%Couleur et forme :White PowderMasse moléculaire :136.11Descarbamoyl cefuroxime
CAS :Descarbamoyl cefuroxime is also an intermediate in the synthesis of cephalosporin antibiotics. Decarbamyl cefuroxime is a degradation product of cefuroxime.Formule :C15H15N3O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.36BAY-721973
CAS :BAY-721973 is a bio-active chemical.Formule :C21H16ClF3N4O4Couleur et forme :SolidMasse moléculaire :480.821,2-Dibehenoyl-sn-glycero-3-phosphocholine
CAS :1,2-Dibehenoyl-sn-glycero-3-phosphocholine (DBPC), a phospholipid integral to cell membranes, facilitates the formation of micelles, liposomes, and various artificial membranes [1].Formule :C48H80NO8PCouleur et forme :SolidMasse moléculaire :830.141ARN-6039
CAS :ARN-6039 is an oral RORγ inverse agonist for Autoimmune Neuroinflammation, active in HEK 293 cells and CD4+T cells.Formule :C21H21F3N2O3Couleur et forme :SolidMasse moléculaire :406.40H-Arg-Lys-OH
CAS :H-Arg-Lys-OH is a dipeptide formed from L-lysine residues and L-arginyl.Formule :C12H26N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.37PAT-494
CAS :PAT-494 is an inhibitor of type II Autotaxin.Formule :C20H16FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.36JZP-MA-11
CAS :"JZP-MA-11 is a PET ligand that selectively targets ABHD6, inhibits with 126 nM IC50, and crosses the BBB for preclinical brain studies."Formule :C15H17FN4O2SCouleur et forme :SolidMasse moléculaire :336.38Trimosulfa
CAS :Trimosulfa is a combination of trimethoprim and sulfamethoxazole, an antibiotic combination. Sulfamethoxazole inhibits dihydropteroate synthase, while trimethoprim inhibits dihydrofolate reductase (dihydrofolate reductase), making it effective for mild to moderate bacterial infections against many Gram-negative and Gram-positive bacteria.Formule :C24H29N7O6SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :543.61-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine
CAS :1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.Formule :C44H84NO8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :786.11Sodium lauroyl glutamate
CAS :Sodium lauroyl glutamate (Acylglutamate LS-11) is an amino acid detergent and increases the solubility of long-chain alkyl gallates such as alkyl gallates.Formule :C17H30NNaO5Degré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :351.41Tetrachlorvinphos
CAS :Tetrachlorvinphos, an organophosphate cholinesterase inhibitor, is used as an insecticide. It has low toxicity to mammals.Formule :C10H9Cl4O4PDegré de pureté :98%Couleur et forme :Less Crystals Or White Powder Colorless Crystals Or White PowderMasse moléculaire :365.965-Hydroxy-L-tryptophan-4,6,7-d3
CAS :5-Hydroxy-L-tryptophan-4,6,7-d3 is a 2H labeled L-5-Hydroxytryptophan. L-5-Hydroxytryptophan (L-5-HTP) is a dietary supplement.Formule :C11H9D3N2O3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :223.241,2-Dipalmitoyl-sn-glycerol 3-phosphate
CAS :1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.Formule :C35H69O8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.89Nitrophenide
CAS :Nitrophenide, a 3,3'-Dinitrodiphenyl disulfide, blocks M1PDH in the mannitol cycle, serving as an anticoccidial.Formule :C12H8N2O4S2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :308.333-O-Methyltolcapone
CAS :3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Formule :C15H13NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.27DC-6-14
CAS :DC-6-14 is a cationic lipid known for its gene transfection activity, commonly utilized in the synthesis of liposomes.Formule :C37H73ClN2O5Couleur et forme :SolidMasse moléculaire :661.44RPR132595A
CAS :RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).Formule :C28H30N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.56Flurtamone
CAS :Flurtamone is an agricultural chemical. Flurtamone mainly used as an herbicide.Formule :C18H14F3NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.303-Phenylbutyric acid
CAS :3-Phenylbutyric acid, from compost soil, metabolizes via benzene and side-chain oxidation.
Formule :C10H12O2Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :164.2PCI-27483
CAS :PCI-27483 is an activated coagulation factor VIIa inhibitor with antithrombotic effects in a baboon model of arterial thrombosis.Formule :C26H24N6O9SDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :596.57BIBB 515
CAS :BIBB 515 inhibits OSC, reducing cholesterol in hamsters by up to 25% with specific dosing.Formule :C22H21ClN2O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :380.87Calcipotriol monohydrate
CAS :Calcipotriol monohydrate, a Vitamin D3 analog, binds well to the vitamin D receptor, used in psoriasis research.Formule :C27H42O4Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :430.62PF-05175157
CAS :PF 05175157 is an inhibitor of acetyl-CoA carboxylase 1 (ACC1) and ACC2 (IC50s = 27, 33, 23.5, and 50.4 nM for human ACC1, human ACC2, rat ACC1, and rat ACC2,Formule :C23H27N5O2Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :405.49Ref: TM-T7163
1mg34,00€2mg44,00€5mg63,00€1mL*10mM (DMSO)70,00€10mg90,00€25mg173,00€50mg295,00€100mg477,00€200mg677,00€E3330
CAS :E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.Formule :C21H30O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :378.461-Decanesulfonic acid
CAS :1-Decanesulfonic acid (Decane-1-sulfonic acid) is a potential amyloid beta peptide (Aβ40) inhibitor, useful for studying cardiovascular diseases.Formule :C10H22O3SCouleur et forme :SolidMasse moléculaire :222.354-POBN
CAS :4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM).Formule :C7H9N3ODegré de pureté :99.60%Couleur et forme :White Crystalline PowderMasse moléculaire :151.17L-m-Tyrosine
CAS :L-m-Tyrosine (3-Hydroxy-L-Phenylalanine) is a non-natural amino acid.Formule :C9H11NO3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :181.1911β-HSD1-IN-9
CAS :11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.Formule :C13H9F3N2OCouleur et forme :SolidMasse moléculaire :266.22Thialysine HCl
CAS :Thialysine HCl is a cytotoxic cysteine derivative that inhibits Escherichia coli, acting as a protein synthesis inhibitor and metabolite.Formule :C5H13ClN2O2SCouleur et forme :SolidMasse moléculaire :200.69CL 242817
CAS :CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).Formule :C18H21NO5SCouleur et forme :SolidMasse moléculaire :363.43Nampt-IN-7
CAS :Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).Formule :C20H21N5O3Couleur et forme :SolidMasse moléculaire :379.41DGAT1-IN-3
CAS :DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.Formule :C20H19F3N4O3Couleur et forme :SolidMasse moléculaire :420.39Ro-15-2041
CAS :Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.Formule :C12H12BrN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.15SGK1-IN-1
CAS :SGK1-IN-1 (compound 14n) is a highly potent SGK1 (Serum/Glucocorticoid Regulated Kinase 1) inhibitorFormule :C17H12ClFN6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :418.83RYL-552
CAS :RYL-552 is a potent inhibitor of PfNDH2.Formule :C24H17F4NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.39GKA-71
CAS :GKA-71 is an effective glucokinase activator (GKA).Formule :C21H23N3O6S2Couleur et forme :SolidMasse moléculaire :477.55JNJ-61803534
CAS :JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.Formule :C23H23Cl2F6N3O4SCouleur et forme :SolidMasse moléculaire :622.41Umbralisib tosylate
CAS :Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.Formule :C38H32F3N5O6SCouleur et forme :SolidMasse moléculaire :743.75Lith-O-Asp
CAS :Lith-O-Asp is a sialytransferase (ST) inhibitor,(IC50s:12-37 μM).Formule :C28H45NO6Couleur et forme :SolidMasse moléculaire :491.66SSI-4
CAS :SSI-4 is a Stearoyl CoA desaturase 1 (SCD1) inhibitor that can be labeled with carbon-11 (11C) for use as a ligand in small animal in vivo PET/CT imagingFormule :C19H21ClN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.85IDO1-IN-21
CAS :IDO1-IN-21 (compound 10m), with an IC50 of 0.64 μM, acts as an IDO1 inhibitor and has demonstrated efficacy in suppressing tumor growth in murine models [1].Formule :C21H19F2N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.45Antitumor agent-87
CAS :Antitumor agent-87: potent, high CYP1A1 affinity (Ki 0.23µM), antiproliferative, arrests G2/M cell cycle.
Formule :C22H28N2O6SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :448.53SYN20028567
CAS :SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].Formule :C20H29N3O3SCouleur et forme :SolidMasse moléculaire :391.53mEH-IN-1
CAS :mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.Formule :C16H17F6NOSCouleur et forme :SolidMasse moléculaire :385.37N-Phenylthiourea
CAS :N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.Formule :C7H8N2SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :152.2217β-HSD10-IN-2
CAS :17β-HSD10-IN-2 (compound 11), a benzothiazolylurea-based inhibitor, specifically targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), avoidingFormule :C15H10ClN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :363.7814R(15S)-EET
CAS :14R(15S)-EET, an oxylipin and a metabolite of arachidonic acid, is produced through the oxidation of arachidonic acid by the cytochrome P450 (CYP) isoforms CYP2C8 and CYP2C9. At a concentration of 10 µM, 14R(15S)-EET causes relaxation in precontracted isolated bovine coronary arteries.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47PDE5-IN-6c
CAS :PDE5-IN-6c is a potent and selective inhibitor of PDE5A1.Formule :C23H21ClN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.89CYP1B1-IN-3
CAS :CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.Formule :C20H16FN3O2S2Couleur et forme :SolidMasse moléculaire :413.49ZM223
CAS :ZM223 is an inhibitor of NEDD8 activating enzyme (NAE).Formule :C23H17F3N4O2S2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :502.53Ref: TM-T13412
1mg109,00€2mg163,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€PKM2 activator 4
CAS :PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.Formule :C16H16N2O4SCouleur et forme :SolidMasse moléculaire :332.37FXR agonist 4
FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.Formule :C21H28ClN3OCouleur et forme :SolidMasse moléculaire :373.92hCA IX-IN-2
hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferativeFormule :C23H24N2O4STeCouleur et forme :SolidMasse moléculaire :552.11TDP1 Inhibitor-1
CAS :TDP1 Inhibitor-1 is a potent inhibitor of Tyrosyl-DNA Phosphodiesterase 1 (TDP1) (IC50 of 7 μM).Formule :C26H26N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :446.49OMDM-3
CAS :OMDM-3 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 16.6 μM).Formule :C29H43NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.66HIF-1/2α-IN-2
CAS :HIF-1/2α-IN-2 is a potent inhibitor of HIF-1/2α, which effectively reduces the levels of HIF-1/2α.Formule :C16H11FN4O2SCouleur et forme :SolidMasse moléculaire :342.35P-3FAX-Neu5Ac
CAS :P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.Formule :C22H30FNO14Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :551.47MY33-3 hydrochloride
CAS :MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.Formule :C16H14ClF6NS2Couleur et forme :SolidMasse moléculaire :433.867β,27-dihydroxy Cholesterol
CAS :7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt.Formule :C27H46O3Couleur et forme :SolidMasse moléculaire :418.65ACC1/2-IN-1
CAS :ACC1/2-IN-1 is a potent inhibitor of ACC1/2 and acts on ACC1 (IC50: 98.06 nM) and ACC2 (IC50: 29.43 nM). ACC1/2-IN-1 can be used in cancer research.Formule :C34H32N4O4Couleur et forme :SolidMasse moléculaire :560.64α-Glucosidase-IN-10
CAS :α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.Formule :C21H15BrN4O2SCouleur et forme :SolidMasse moléculaire :467.34TUPS
CAS :TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.Formule :C14H18F3N3O4SCouleur et forme :SolidMasse moléculaire :381.37AX 048
CAS :Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.Formule :C22H41NO4Couleur et forme :SolidMasse moléculaire :383.57ATX inhibitor 11
CAS :ATX inhibitor 11 blocks autotaxin (IC50: 2.7 nM), reduces fibrosis and α-SMA in mice. Useful for lung fibrosis studies.Formule :C32H35N5O6Couleur et forme :SolidMasse moléculaire :585.65CAY10485
CAS :CAY10485 blocks human ACAT-1 & ACAT-2 (IC50: 95 & 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.Formule :C27H27NO7Couleur et forme :SolidMasse moléculaire :477.51SGK1 inhibitor
CAS :SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.Formule :C17H12Cl2N6O2SCouleur et forme :SolidMasse moléculaire :435.29hCAIX-IN-8
CAS :hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.Formule :C19H16N4O6Couleur et forme :SolidMasse moléculaire :396.35JTP-4819
CAS :JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.Formule :C19H25N3O4Couleur et forme :SolidMasse moléculaire :359.42AMG-221
CAS :AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.Formule :C14H22N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :266.4Boc-Glu(OBzl)-OSu
CAS :Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.Formule :C21H26N2O8Couleur et forme :SolidMasse moléculaire :434.44α-Amylase/α-Glucosidase-IN-2
CAS :α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μMFormule :C22H16ClN5Couleur et forme :SolidMasse moléculaire :385.857ETMC
CAS :7ETMC inhibits Human Cytochrome P450s 1A1/1A2 with IC50: 0.46/0.50 μM; not effective on P450s 2A6/2B1 even at 50 μM.Formule :C14H12O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :212.24IDO inhibitor 1
CAS :IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 <100 nM).with potential immunomodulating and antineoplastic activities.Formule :C11H13BrFN7O4SDegré de pureté :99.805%Couleur et forme :SolidMasse moléculaire :438.23Ref: TM-T7660
1mg94,00€2mg138,00€5mg192,00€1mL*10mM (DMSO)220,00€10mg294,00€25mg427,00€50mg625,00€100mg889,00€500mg1.783,00€NPP1-IN-1
CAS :NPP1-IN-1 is a highly potent inhibitor of NPP enzymes, effectively inhibiting NPP1 with an IC 50 value of 0.15 μM and NPP3 with an IC 50 value of 40 μM [1].Formule :C27H21NO2Couleur et forme :SolidMasse moléculaire :391.46Ornithine-α-ketoglutarate
CAS :Ornithine-α-ketoglutarate (L-Ornithine-α-ketoglutarate) is a salt formed of 2 molecules of ornithine and 1 alpha-ketoglutarate.Formule :C10H18N2O7Degré de pureté :≥98%Couleur et forme :White PowderMasse moléculaire :278.26Xylamidine tosylate
CAS :Xylamidine tosylate is a Serotonin inhibitor with reproductive effectsFormule :C26H32N2O5SCouleur et forme :SolidMasse moléculaire :484.61Moschamine
CAS :Moschamine is an inhibitor of mitochondrial superoxide overproduction.Formule :C20H20N2O4Couleur et forme :SolidMasse moléculaire :352.38PDE7-IN-2
CAS :PDE7-IN-2 is an inhibitor of phosphodiesterase 7 (IC50 = 2.1 µM) and can be used in Parkinson's disease studies.Formule :C14H11ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.77Letimide HCl
CAS :Letimide HCl is an analgesic agent.Formule :C14H19ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.771-Methyluric acid
CAS :1-Methyluric acid (1-Methylurate) acts on the bladder mucosa and increases the levels of insulin, triglycerides, cholesterol, and blood glucose.Formule :C6H6N4O3Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :182.14NP603
CAS :NP603 is a cell-permeable inhibitor of FGFR1, PDGFRβ, and VEGFR2 that binds to the ATP pocket. It also is a very weak EGFR inhibitor.Formule :C26H26N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :446.49U-0521
CAS :U-0521, an inhibitor of catechol-O-methyltransferase (COMT), enhances the availability and utilization of levodopa in the brain.Formule :C10H12O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :180.2(Z)-10-Hydroxynortriptyline
CAS :(Z)-10-Hydroxynortriptyline ((Z)-10-Hydroxy Nortriptyline) is a norepinephrine reuptake inhibitor with antidepressant activity.Formule :C19H21NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.38CAY10641
CAS :cPLA2α breaks down arachidonic acid, starting prostaglandin and leukotriene synthesis. CAY10641, its inactive alcohol form, is a potent anti-inflammatory.Formule :C28H27NO6Couleur et forme :SolidMasse moléculaire :473.52GSK2945
CAS :GSK2945, a specific Rev-erbα antagonist, boosts CYP7A1 and cholesterol metabolism. EC50: 21.5 μM (mouse), 20.8 μM (human).Formule :C20H18Cl2N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.34Ciraparantag TFA
CAS :Ciraparantag TFA reverses anticoagulants by inhibiting thrombin and factor Xa.Formule :C26H50F6N12O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :740.74CGP-28014
CAS :CGP-28014 inhibits COMT, boosts renal dopamine & DOPAC excretion, lowers HVA, no effect on renal sodium.Formule :C12H19N3OCouleur et forme :SolidMasse moléculaire :221.3Razobazam
CAS :Razobazam is a benzodiazepine derivative agent. It produces nootropic (improves cognitive function) effects in animal studies.Formule :C14H14N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.29CDP 840 hydrochloride
CAS :CDP-840 (GR259653X), a potent oral PDE IV inhibitor, curbs early and late phase bronchoconstriction in squirrel monkeys.Formule :C25H27NO2Couleur et forme :SolidMasse moléculaire :373.49Pentamethonium bromide
CAS :Pentamethonium bromide is a vasodilator agent.Formule :C11H28Br2N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :348.16Levophencynonate HCl
CAS :Levophencynonate HCl is a muscarinic receptor antagonist.Formule :C22H32ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.95
