Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(164 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8626 produits trouvés pour "Métabolisme"
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Hydroxy ritonavir
CAS :<p>Hydroxy ritonavir, a metabolite of ritonavir, functions as an inhibitor of the HIV protease, thereby serving as a treatment for HIV infection and AIDS [1].</p>Formule :C37H48N6O6S2Couleur et forme :SolidMasse moléculaire :736.94Seco Rapamycin sodium salt
CAS :<p>Seco Rapamycin sodium salt is a ring-opened product of Rapamycin.</p>Formule :C51H79NNaO13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :937.177Aldosterone 21-sulfate sodium salt
<p>Aldosterone 21-sulfate sodium salt is a cholesterol metabolite found in urine.</p>Formule :C21H28NaO8SCouleur et forme :SolidMasse moléculaire :463.5Cyperine
CAS :<p>Cyperine is a useful organic compound for research related to life sciences. The catalog number is T125020 and the CAS number is 33716-82-4.</p>Formule :C15H16O4Couleur et forme :SolidMasse moléculaire :260.289TDI-11055
<p>TDI-11055 is a chromatin reader 11-19 leukemia inhibitor and can be used to study acute myeloid leukemia (AML).</p>Formule :C22H24N6ODegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :388.47trans-2-Hexadecenoyl-L-carnitine
CAS :<p>trans-2-Hexadecenoyl-L-carnitine is an endogenous metabolite in urine[1].</p>Formule :C23H43NO4Couleur et forme :SolidMasse moléculaire :397.59L-Amino acid oxidase
CAS :<p>L-Amino acid oxidase catalyzes the oxidative deamination of L-amino acids, which have local oxidative effects as well as potent antimicrobial effects.</p>Couleur et forme :Solid4,12-Dimethoxy-6-(7,8-dihydroxy-7,8-dihydrostyryl)-2-pyrone
CAS :<p>4,12-Dimethoxy-6-(7,8-dihydroxy-7,8-dihydrostyryl)-2-pyrone is a microbial metabolism of yangonin, a major styryl lactone from Piper methysticum.</p>Formule :C14H12O5Degré de pureté :99.67%Couleur et forme :SoildMasse moléculaire :260.24TPT-004
<p>TPT-004, a TPH inhibitor, exhibits superior pharmacokinetic and pharmacodynamic properties, and demonstrates efficacy in preclinical models for attenuating</p>Couleur et forme :Odour SolidD-myo-Inositol-1,4,5-triphosphate tripotassium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate tripotassium is a second messenger in the intracellular signaling system that induces Ca2+ mobilization.</p>Formule :C6H12K3O15P3Couleur et forme :SolidMasse moléculaire :534.37DSPE-PEG5000-LTLRWVGLMS
<p>DSPE-PEG5000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). Chondroitin sulfate proteoglycan NG2 serves as a receptor for LLRWVGLMS. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG5000-LTLRWVGLMS can be utilized for drug delivery.</p>Couleur et forme :Odour Solid4-Phytase
CAS :<p>4-Phytase is a phosphohydrolase of inositol hexaphosphate [1] .</p>Couleur et forme :SolidIPI-9119
CAS :<p>IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).</p>Formule :C24H19F2N5O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :495.43ACSS2-IN-2
CAS :<p>MTB-9655 inhibits ACSS2 with 3.8 nM IC50, useful in research of viral, metabolic, neuropsychiatric diseases, inflammation, and cancer.</p>Formule :C21H19F2N3O4Degré de pureté :99.5%Couleur et forme :SoildMasse moléculaire :415.39Herbicidal agent 6
<p>Herbicidal agent 6 (D15) functions as a Transketolase (TKL) inhibitor and exhibits herbicidal activity.</p>Couleur et forme :Odour SolidPF-1355
CAS :<p>PF-1355 (PF 06281355) is a selective 2-thiouracil mechanism-based MPO inhibitor. PF-1355 is used for treatment of vasculitic diseases.</p>Formule :C14H15N3O4SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :321.35(±)14-HDHA
CAS :<p>(±)14-HDHA is an oxidized metabolite of DHA and can be further oxidized to the 14-oxoDHA, 14-HDoHE inhibits LPS-induced IL-6 mRNA expression.</p>Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.49Fasnall HCl
<p>Fasnall HCl is a selective FASN inhibitor that acts through its co-factor binding sites.</p>Formule :C19H23ClN4SDegré de pureté :99.9%Couleur et forme :SoildMasse moléculaire :374.93Isodihydroauroglaucin
CAS :<p>Isodihydroauroglaucin is a useful organic compound for research related to life sciences. The catalog number is T124274 and the CAS number is 74886-31-0.</p>Formule :C19H24O3Couleur et forme :SolidMasse moléculaire :300.398Pseudoerythromycin A enol ether
CAS :<p>Pseudoerythromycin A enol ether, a non-antibiotic erythromycin degradation product, serves as a standard in stability studies.</p>Formule :C37H65NO12Couleur et forme :SolidMasse moléculaire :715.91Glisoprenin D
CAS :<p>Glisoprenin D is a useful organic compound for research related to life sciences. The catalog number is T125390 and the CAS number is 205594-89-4.</p>Formule :C45H84O7Couleur et forme :SolidMasse moléculaire :737.16H-Met-Val-OH
CAS :<p>H-Met-Val-OH is a dipeptide inhibiting FMO1 and FMO3 and promoting neurite outgrowth, relevant for neuroregenerative and enzymatic modulation studies.</p>Formule :C10H20N2O3SCouleur et forme :SolidMasse moléculaire :248.34Dihydrozeatin riboside
CAS :<p>Dihydrozeatin riboside is a cytokinin that can be isolated from Phaseolus vulgaris L.</p>Formule :C15H23N5O5Couleur et forme :SolidMasse moléculaire :353.37hCAI/II/IV-IN-28
CAS :<p>hCAI/II/IV-IN-28(WAY-638358) is a potent carbonic anhydrase inhibitor with potential anticonvulsant activity.</p>Formule :C14H15N3O3SDegré de pureté :96.48%Couleur et forme :SolidMasse moléculaire :305.35DSPE-PEG1000-octreotide
<p>DSPE-PEG1000-Octreotide, a PEG compound formed from DSPE and Octreotide, acts as a somatostatin receptor agonist. Octreotide exhibits antitumor properties and induces apoptosis, making it useful in researching acromegaly. Additionally, DSPE-PEG1000-Octreotide is applicable in drug delivery.</p>Couleur et forme :Odour Solid3,5,6,7,8,4′-hexamethoxyflavone
CAS :<p>3,5,6,7,8,4′-hexamethoxyflavone is a natural product for research related to life sciences. The catalog number is TN7114 and the CAS number is 34170-18-8.</p>Formule :C21H22O8Couleur et forme :SolidMasse moléculaire :402.399Guignardone J
CAS :<p>Guignardone J, a secondary metabolite, is isolated from the endophytic fungus Phyllosticta capitalensis [1].</p>Formule :C17H24O5Couleur et forme :SolidMasse moléculaire :308.37POPG sodium salt
CAS :<p>POPG sodium salt is a phospholipid and a component of biological membranes and can be used to study the function of biological membranes.</p>Formule :C40H76NaO10PDegré de pureté :98.21%Couleur et forme :SolidMasse moléculaire :770.99Antiproliferative agent-13
CAS :<p>Antiproliferative agent-13 is a compound with antiproliferative activity.</p>Formule :C20H18N2O6Degré de pureté :99.723%Couleur et forme :SolidMasse moléculaire :382.37(Rac)-sn-Glycerol 3-phosphate sodium
CAS :<p>(Rac)-sn-Glycerol 3-phosphate sodium, an a-site substrate analogue, inhibits indole reactions with E(A-A).</p>Formule :C3H7Na2O6PCouleur et forme :SolidMasse moléculaire :216.04DSPE-PEG-Maleimide ammonium (MW 2000)
<p>DSPE-PEG-Maleimide (ammonium) (MW 2000) is a compound containing DSPE phospholipids and maleimide, designed for the preparation of nanoscale lipid carriers. It is applicable in the study of drug delivery systems.</p>Couleur et forme :Odour SolidEstriol 3-glucuronide
CAS :<p>Estriol-3-glucuronide, a natural compound found in urine, is also present in amniotic fluid during normal pregnancy [1][2].</p>Formule :C24H32O9Couleur et forme :SolidMasse moléculaire :464.511(Iso)-Dehydroemetine
CAS :<p>(Iso)-Dehydroemetine (Dehydroisoemetine, (+/-)-) is a compound with antispasmolytic effect on smooth muscle.</p>Formule :C29H38N2O4Degré de pureté :98.26% - 98.31%Couleur et forme :SoildMasse moléculaire :478.625,7-Dichloropyrazolo[1,5-a]pyrimidine
CAS :<p>5,7-Dichloropyrazolo[1,5-a]pyrimidine (fragment 5) is an inhibitor of the enzyme phosphodiesterase 10A (PDE10A) with a Ki value of 24 μM. This compound can be employed in research related to schizophrenia.</p>Formule :C6H3Cl2N3Couleur et forme :SolidMasse moléculaire :188.0124R-Calcipotriol
CAS :<p>24R-Calcipotriol(PRI 2202) is an impurity of Calcipotriol which is a ligand of VDR-like receptors.</p>Formule :C27H40O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :412.60(±)-Equol 4'-sulfate (sodium salt)
CAS :<p>(±)-Equol 4’-sulfate is a gut-mediated phase II metabolite of the isoflavonoid phytoestrogen (±)-equol .[1] It has been used as a standard for the</p>Formule :C15H13NaO6SCouleur et forme :SolidMasse moléculaire :344.32Trifluoperazine N-Glucuronide
CAS :<p>Trifluoperazine N-Glucuronide is a metabolite of Trifluoperazine with antidepressant and antipsychotic activity.</p>Formule :C27H32F3N3O6SCouleur et forme :SolidMasse moléculaire :583.62CHEMBL1276927
CAS :<p>CHEMBL1276927 (N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide) shows antibacterial and antiparasitic activities against Chlamydia pneumoniae and</p>Formule :C21H17N3ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :327.38LL P880 β
CAS :<p>LL P880 beta is a fungal metabolite.</p>Formule :C11H18O5Couleur et forme :SolidMasse moléculaire :230.26DSPE-PEG5000-GRGDS
<p>DSPE-PEG5000-GRGDS is a PEG compound composed of DSPE and the anti-adhesion peptide (GRGDS). GRGDS can inhibit the binding and adhesion between the extracellular matrix and cell surface integrins. DSPE-PEG5000-GRGDS is applicable for drug delivery.</p>Couleur et forme :Odour SolidZymostenol
CAS :<p>Zymostenol (5a-Cholest-8-en-3b-ol) is a RORγ agonist with an EC50 of 1 μM.Zymostenol is a late stage precursor of cholesterol biosynthesis.</p>Formule :C27H46ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.65WAY-620472
CAS :<p>WAY-620472 is a PPAR regulator that can be used to alter the lifespan of eukaryotes.</p>Formule :C23H21N5OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :415.51RORγ agonist 1
CAS :<p>RORγ agonist 1 is a highly potent and orally bioavailable compound that activates the RORγ receptor.</p>Formule :C29H27ClF4N2O4SCouleur et forme :SolidMasse moléculaire :611.05ML171
CAS :<p>Compound PDK0326, with CAS No. 6631-94-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0326 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C14H11NOSCouleur et forme :Mustard-Colored PowderMasse moléculaire :241.3IGUANA-1 free base
CAS :<p>IGUANA-1: selective ALDH1 B1 inhibitor, IC50=30 nM, hinders SW480 cell growth with IC50=2.46/0.39 μM in adherent/spheroid forms, for cancer research.</p>Formule :C26H24ClN3O2Couleur et forme :SolidMasse moléculaire :445.94Transketolase-IN-6
<p>Transketolase-IN-6 (Compound 6bj) serves as a lead compound for herbicides. It achieves approximately 80% root inhibition in redroot pigweed (Amaranthus retroflexus) and green foxtail (Setaria viridis). Moreover, Transketolase-IN-6 is an effective inhibitor of transketolase (TK).</p>Formule :C23H27ClN6OMasse moléculaire :438.19349AMK318
AMK318 (Immobilized cephalexin acylase) is a biocatalyst and a critical enzyme in novel biocatalyst technology. Enzyme engineering focuses on improving enzyme reaction kinetics, substrate selectivity, and activity under harsh conditions (such as low or high pH). By incorporating stimulus responsiveness into these enzyme modifications, dynamic control of activity becomes feasible.BAY-277
<p>BAY-277 is a degrader of METAP2, with IC50 values of 5.8 nM for human METAP2 (hMETAP2) and 5.9 nM for mouse METAP2 (mMETAP2).</p>Formule :C44H52N8O5Couleur et forme :SolidMasse moléculaire :772.93ROR1 ligand-1
<p>ROR1ligand-1 (9-1) serves as the ligand for PROTAC ROR1 degrader-1. By linking with ligands of either the VHL type or CRBN, the first selective and efficient ROR1 PROTAC molecule was designed and synthesized.</p>Formule :C23H30BrN7Couleur et forme :SolidMasse moléculaire :484.44N-β-alanyldopamine hydrochloride
CAS :<p>N-β-Alanyldopamine hydrochloride (NBAD hydrochloride) represents the primary dopamine derivative found in haemolymph [1].</p>Formule :C11H17ClN2O3Couleur et forme :SolidMasse moléculaire :260.72DSPE-PEG1000-MPG
<p>DSPE-PEG1000-MPG is a PEG compound composed of DSPE and the peptide carrier (MPG). MPG is derived from the nuclear localization sequence (NLS) of the SV40 large T antigen and the fusion peptide domain of HIV-1 gp41. MPG efficiently delivers short oligonucleotides into cells, operating independently of endosomal pathways.</p>Couleur et forme :Odour SolidEdoxaban Isomer
CAS :<p>Edoxaban Isomer is an impurity of Edoxaban, which is a novel inhibitor of factor Xa.</p>Formule :C24H30ClN7O4SCouleur et forme :SolidMasse moléculaire :548.067-Hydroxydichloromethotrexate
CAS :<p>7-Hydroxydichloromethotrexate is a methotrexate metabolite.</p>Formule :C20H20Cl2N8O6Couleur et forme :SolidMasse moléculaire :539.33N-Pivaloyl-L-tyrosine
CAS :<p>N-Pivaloyl-L-tyrosine is an N-pivaloyl amino acid ester.</p>Formule :C14H19NO4Couleur et forme :SolidMasse moléculaire :265.30Febuxostat impurity 7
CAS :<p>Febuxostat impurity 7 is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1] .</p>Formule :C16H18N2O4SCouleur et forme :SolidMasse moléculaire :334.39Atocalcitol
CAS :<p>Atocalcitol is a vitamin D analog. It also acts as an agonist of alcitriol receptor.</p>Formule :C32H46O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :494.71TEI-9647
CAS :<p>TEI-9647 is a vitamin D3 analog and VDR/DRE genomic antagonist.</p>Formule :C27H38O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.59Mycophenolic acid-β-D-glucuronide
CAS :<p>Mycophenolic acid glucuronide is the glucuronide metabolite of mycophenolic acid in human plasma.</p>Formule :C23H28O12Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :496.46Febuxostat impurity 6
CAS :<p>Febuxostat impurity 6 is an impurity of Febuxostat. Febuxostat is selective xanthine oxidase inhibitor with a K i of 0.6 nM [1] .</p>Formule :C18H22N2O4SCouleur et forme :SolidMasse moléculaire :362.44DSPE-PEG2000-CREKA
<p>DSPE-PEG3000-CREKA is a PEG compound composed of DSPE and the fibrin-targeting peptide (CREKA). The CREKA peptide targets tumor cells and tumor vasculature, exhibiting antitumor activity. DSPE-PEG3000-CREKA is useful in drug delivery applications.</p>Couleur et forme :Odour Solid2,3-Dehydrosilybin B
CAS :<p>2,3-Dehydrosilybin B is a useful organic compound for research related to life sciences and the catalog number is T125883.</p>Formule :C25H20O10Couleur et forme :SolidMasse moléculaire :480.425′-Nucleotidase
CAS :<p>5′-Nucleotidase (CD73), an ectoenzyme and intrinsic membrane glycoprotein, catalyzes the hydrolysis of 5-nucleotides into their corresponding nucleosides [1].</p>Couleur et forme :SolidT3 Acyl glucuronide
CAS :<p>T3 Acyl glucuronide is the acyl glucuronide formation of triiodothyronine (T3). T3 Acyl glucuronide is an endogenous metabolite</p>Formule :C21H20I3NO10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :827.1DSPE-PEG5000-KAA
<p>DSPE-PEG5000-KAA is a PEG compound composed of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically targets the tumor vasculature of RIP-Tag2 transgenic mice. DSPE-PEG5000-KAA can be utilized for drug delivery purposes.</p>Couleur et forme :Odour SolidH-Pro-Phe-OH
CAS :<p>H-Pro-Phe-OH is a dipeptide formed from proline and phenylalanine, serving as a substrate for prolylase and in peptide synthesis.</p>Formule :C14H18N2O3Couleur et forme :SolidMasse moléculaire :262.30Streptolysin O
CAS :<p>Streptolysin O: lyses cells, cardiotoxic, used for cell permeabilization, has active and inactive states.</p>Degré de pureté :98%Couleur et forme :SolidUrate oxidase
CAS :<p>Uricase catalyzes uric acid to allantoin in many mammals' peroxisomes, used in biochemistry.</p>Couleur et forme :SolidGlucuronokinase (AtGlcAK)
CAS :<p>AtGlcAK: GHMP-kinase family, specific for D-glucuronic acid, Km 0.7 mM, converts it with ATP to D-glucuronic-1-phosphate and ADP.</p>Couleur et forme :SolidHPA-IN-1
<p>HPA-IN-1: potent human pancreatic α-amylase inhibitor; IC50: 12.0 μM for HPA, 410.4 μM for α-glucosidase.</p>Formule :C33H32N4O11Couleur et forme :SolidMasse moléculaire :660.63DKI5
CAS :<p>DKI5, a LOX-1 inhibitor with 22.5 μM IC50, may exhibit anti-inflammatory, antioxidant, and anti-lipid peroxidation effects in vitro.</p>Formule :C8H10N4SDegré de pureté :98%Couleur et forme :SoildMasse moléculaire :194.26Phosphodiesterase II
CAS :<p>Phosphodiesterase II (PDE2) breaks down cAMP and cGMP, important in cellular regulation and widespread in tissues for biochemical research.</p>Couleur et forme :SolidRitonavir metabolite
CAS :<p>Ritonavir metabolite is a Ritonavir metabolite, which is a inhibitor of HIV protease.</p>Formule :C32H45N5O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :579.80(25R)-12α-Hydroxyspirost-4-en-3-one
CAS :<p>'(25R)-12α-Hydroxyspirost-4-en-3-one is a minor metabolite resulting from Nocardia globerula's metabolization of Hecogenin [1].'</p>Formule :C27H40O4Couleur et forme :SolidMasse moléculaire :428.6Neo-inositol
CAS :<p>Neo-Inositol, a stable, polar compound, is a rare natural inositol stereoisomer.</p>Formule :C6H12O6Couleur et forme :SolidMasse moléculaire :180.16N-Decanoyl p-Nitroaniline
CAS :<p>DepNA, a nitroaniline fatty acid amide, measures FAAH activity by releasing yellow dye p-nitroaniline upon exposure, detectable via spectrophotometer.</p>Formule :C16H24N2O3Couleur et forme :SolidMasse moléculaire :292.379Diacetinase
Diacetinase, a member of the esterase family, catalyzes the hydrolysis of glyceryl diacetate (Diacetin). It is utilized in the measurement of lipase activity.Couleur et forme :Odour SolidTKL-IN-1
<p>TKL-IN-1 (compound 7r) serves as an inhibitor of transketolase (Transketolase) and can be utilized as an herbicide. This compound effectively hampers the growth of Digitaria sanguinalis (Ds) and Amaranthus retroflexus (Ar).</p>Formule :C20H12ClN5OS2Couleur et forme :SolidMasse moléculaire :437.93MS1262-C3-amide-C10-amine
<p>MS1262-C3-amide-C10-amine is an E3 Ligase Ligand-Linker conjugate. It includes a GLP ligand targeting the E3 ligase SPOP and a PROTAC linker. This compound can be utilized in designing PROTACs such as example [MS479].</p>Couleur et forme :Odour SolidACAT-IN-7
CAS :<p>ACAT-IN-7 inhibits ACAT enzyme; blocks NF-κB mediated transcription.</p>Formule :C32H49N3O5SCouleur et forme :SolidMasse moléculaire :587.82PKM2 inhibitor G
CAS :<p>PKM2 inhibitor G is a inhibitor of pyruvate kinase.</p>Formule :C16H15NO3SDegré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :301.36BMS 195614
CAS :<p>BMS 195614 (BMS614) is a selective RARα antagonist. BMS 195614 can bind to the RARα subunit.</p>Formule :C29H24N2O3Degré de pureté :97.7%Couleur et forme :SolidMasse moléculaire :448.51PDE2A-IN-1
CAS :<p>PDE2A-IN-1 is a phosphodiesterase 2A (PDE2A) inhibitor with an IC 50 value of 1.3 nM.</p>Formule :C23H22F2N6Couleur et forme :SolidMasse moléculaire :420.468IETP2
CAS :<p>IETP2 targets low-density lipoprotein receptor-related protein 1 (LRP1) with a KD of 738 nM, making it useful for delivering drugs and imaging agents across the blood-labyrinth barrier (BLB).</p>Formule :C107H171N39O29Couleur et forme :SolidMasse moléculaire :2467.7528-Epirapamycin
CAS :<p>28-Epirapamycin, an impurity of Rapamycin, serves as a potent and specific mTOR inhibitor, exhibiting an IC50 value of 0.1 nM in HEK293 cells [1].</p>Formule :C51H79NO13Couleur et forme :SolidMasse moléculaire :914.17H-Arg-Lys-OH TFA
<p>H-Arg-Lys-OH TFA is a dipeptide formed from L-arginyl and L-lysine residues [1] .</p>Formule :C14H27F3N6O5Couleur et forme :SolidMasse moléculaire :416.41-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphoinositol
CAS :<p>1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphoinositol is an intrinsic metabolite and a component of the cell membrane [1].</p>Formule :C47H83O13PCouleur et forme :SolidMasse moléculaire :887.13VDR agonist 2
<p>VDR agonist 2 (compound 16i), a vitamin D receptor (VDR) agonist, effectively inhibits TGF-β1-induced hepatic stellate cell (HSC) activation, demonstrating</p>Formule :C20H21F3O3Couleur et forme :SolidMasse moléculaire :366.37RORγ inverse agonist 1
CAS :<p>RORγ inverse agonist 1 has anti-inflammatory activity and can be used to treat rheumatism and psoriasis.</p>Formule :C22H20F3N3O3SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :463.478-iso Prostaglandin A1
CAS :<p>8-iso PGA1: an isoprostane, non-COX prostanoid, minor PGE1 impurity, biological effects unstudied.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472SDUY817
<p>SDUY817 is a dual APN/NEP inhibitor with IC50 values of 0.29 μM for APN and 7.4 μM for NEP. It exhibits analgesic effects in a concentration- and time-dependent manner, making it a potential candidate for research in the field of neuropathic pain disorders.</p>Formule :C18H16IN3O3Couleur et forme :SolidMasse moléculaire :449.24Sucrose phosphorylase
CAS :Sucrose phosphorylase, a bacterial enzyme, transforms sucrose and phosphate into α-D-glucose-1-phosphate and D-fructose.Couleur et forme :SolidHexokinase II VDAC binding domain peptide, cell-permeable
HexokinaseIIVDACbinding domain peptide (Hxk2VBD peptide) is a cell-permeable peptide derived from the hexokinase II VDAC binding domain. This peptide inhibits the mitochondrial localization of hexokinase 2 (HXK2) and also suppresses neurotrophic factor-induced axon growth.Formule :C188H291N53O40S2Masse moléculaire :3995.18073Eflucimibe
CAS :<p>Eflucimibe (L0081), an ACAT inhibitor, treats cardiovascular, endocrine, and metabolic diseases, and helps in atherosclerosis and hyperlipidemia research.</p>Formule :C29H43NO2SDegré de pureté :99.17% - 99.43%Couleur et forme :SolidMasse moléculaire :469.72DSPE-PEG3000-R6H4
<p>DSPE-PEG3000-R6H4 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (R6H4). R6H4 is applicable for pH-responsive anticancer drug delivery. DSPE-PEG3000-R6H4 can be utilized for drug delivery purposes.</p>Couleur et forme :Odour SolidFUT8-IN-1
<p>FUT8-IN-1 (Compound 37) is an inhibitor of α-1,6-fucosyltransferase (FUT8), with a dissociation constant (KD) of 49 nM and an IC50 around 50 µM. In the presence of FUT8, FUT8-IN-1 forms a highly active naphthoquinone imine intermediate, thereby inhibiting FUT8's enzymatic activity.</p>Formule :C23H25ClN2OCouleur et forme :SolidMasse moléculaire :380.91(Rac)-Azide-phenylalanine
CAS :<p>(Rac)-Azide-phenylalanine: racemate, non-natural amino acid derivative for protein labeling.</p>Formule :C9H10N4O2Couleur et forme :SolidMasse moléculaire :206.20Menthol glucuronide
CAS :<p>Menthol glucuronide is a metabolite of L-(-)-Menthol, the natural form of Methanol.</p>Formule :C16H28O7Couleur et forme :SolidMasse moléculaire :332.39NLG802
CAS :<p>NLG802 is a prodrug of indoximod, an orally active indoleamine 2,3-dioxygenase (IDO) inhibitor.</p>Formule :C20H30ClN3O3Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :395.92MDNI-caged-L-glutamate
CAS :<p>MDNI-glu: photosensitive, bio-inert L-glutamate derivative with enhanced light utilization.</p>Formule :C14H16N4O8Couleur et forme :SolidMasse moléculaire :368.302Fumiquinazoline D
CAS :<p>Fumiquinazoline D, from A. fumigatus, inhibits Gram-positive/negative bacteria (MIC 8-16 μg/ml) and F. solani, C. albicans (MIC 32, 64 μg/ml).</p>Formule :C24H21N5O4Couleur et forme :SolidMasse moléculaire :443.463CBS-1114 HCl
CAS :<p>CBS-1114 HCl: 5-lipoxygenase inhibitor, anti-inflammatory, improves heart function, reduces heart's fat.</p>Formule :C13H14ClN3Degré de pureté :99.36%Couleur et forme :SoildMasse moléculaire :247.72N-Desbutyl Dronedarone-d7 HCl
<p>N-Desbutyl Dronedarone-d7 HCl is the deuterium-labelled isomer of N-Desbutyl Dronedarone HCl, used for isotope tracing. N-Desbutyl Dronedarone is a metabolite of the antiarrhythmic drug Dronedarone.</p>Formule :C27H30D7ClN2O5SCouleur et forme :SolidMasse moléculaire :544.15Porfimer Sodium
CAS :<p>Porfimer sodium, a sodium salt with photodynamic properties, targets tumor cells and induces cytotoxicity with 630 nm laser activation.</p>Formule :C68H74N8O11Couleur et forme :SolidMasse moléculaire :1179.385L-Lysine, sulfite (2:1)
CAS :<p>L-Lysine, sulfite (2:1) is a drug/ therapeutic agent.</p>Formule :C6H14N2O2H2O3SCouleur et forme :SolidMasse moléculaire :187.23Seco Rapamycin ethyl ester
<p>Seco Rapamycin ethyl ester, an open-ring metabolite of the Rapamycin derivative, reportedly does not impact mTOR function [1].</p>Formule :C53H83NO13Couleur et forme :SolidMasse moléculaire :942.239(R)-HODE cholesteryl ester
CAS :<p>9(R)-HODE cholesteryl ester, from atherosclerotic lesions, may form enzymatically or by lipid peroxidation; used as a chiral analysis standard.</p>Formule :C45H76O3Couleur et forme :SolidMasse moléculaire :665.1BAY-588
CAS :<p>BAY-588 is an inactive control probe of BAY-876 which is an inhibitor of GLUT1.</p>Formule :C27H25F4N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.51Orotidine 5′-monophosphate
CAS :<p>Orotidine 5′-monophosphate, a pyrimidine ribonucleoside, functions as an endogenous metabolite in human, E.</p>Formule :C10H13N2O11PCouleur et forme :SolidMasse moléculaire :368.191Asundexian
CAS :<p>Asundexian (BAY-2433334) is a potent and orally active inhibitor of the coagulation factor FXIa that directly and reversibly binds to the active site of FXIa,</p>Formule :C26H21ClF4N6O4Degré de pureté :99.89% - 99.90%Couleur et forme :SolidMasse moléculaire :592.93Tetomilast
CAS :<p>Tetomilast (OPC-6535) is a phosphodiesterase-4 (PDE4) inhibitor, potentially effective in treating inflammatory bowel disease (IBD) and chronic obstructive</p>Formule :C19H18N2O4SCouleur et forme :SolidMasse moléculaire :370.42Acesulfame
CAS :<p>Acesulfame inhibits CA9/12 and can be used to study inflammation-related diseases.</p>Formule :C4H5NO4SCouleur et forme :SolidMasse moléculaire :163.15α-Lactose hydrate
CAS :<p>α-Lactose (hydrate) (α-D-Lactose (hydrate)), the main carbohydrate in mammalian milk, comprises two sugar units: glucose and galactose, and occurs as two</p>Formule :C12H24O12Couleur et forme :SolidMasse moléculaire :360.31DL-TBOA ammonium
CAS :<p>DL-TBOA ammonium is a potent EAAT inhibitor with IC50 (6-70 μM) and Ki (3.2-42 μM) against EAAT1-5, blocking [14C]glutamate uptake.</p>Formule :C11H16N2O5Couleur et forme :SolidMasse moléculaire :256.2582-Aminoflubendazole
CAS :<p>2-Aminoflubendazole, a metabolite of benzimidazoles (BZ), belongs to a class of drugs effective against fungi, protozoa, and helminths.</p>Formule :C14H10FN3OCouleur et forme :SolidMasse moléculaire :255.25DSPE-PEG2000-LyP-1
<p>DSPE-PEG2000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). LyP-1 specifically targets tumor-associated lymphatic vessels and macrophages.</p>Couleur et forme :Odour SolidGeranylgeranyl pyrophosphate
CAS :<p>Geranylgeranyl pyrophosphate: a metabolite for protein modification and diterpenoid precursor, used in cancer research.</p>Formule :C20H36O7P2Couleur et forme :SolidMasse moléculaire :450.44Z-Asp(OBzl)-OH
CAS :<p>Z-Asp(OBzl)-OH (N-Cbz-L-Aspartic acid 4-benzyl ester) is an aspartic acid derivative.</p>Formule :C19H19NO6Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :357.36(±)7(8)-EpDTE
CAS :<p>(±)7(8)-EpDTE is an oxylipin and an oxidative metabolite of docosapentaenoic acid .</p>Formule :C22H34O3Couleur et forme :SolidMasse moléculaire :346.511α-Hydroxyglutaric Acid Lithium
<p>α-Hydroxyglutaric Acid Lithium is an α-ketoglutarate-dependent dioxygenase and 5-methylcytosine hydroxylase inhibitor of ATP synthase.</p>Formule :C5H6Li2O5Degré de pureté :≥98%Couleur et forme :SoildMasse moléculaire :159.98Methionylserine
CAS :<p>Methionylserine (H-MET-SER-OH), a dipeptide, binds hPEPT1 (Km 0.2 mM), inhibits ACE, used in hypertension research.</p>Formule :C8H16N2O4SCouleur et forme :SolidMasse moléculaire :236.29MK-8245 Trifluoroacetate
CAS :<p>MK-8245 trifluoroacetate: Potent liver-targeting SCD inhibitor, IC50=1nM (human). Anti-diabetic/anti-dyslipidemic. Selective, with low adverse event exposure.</p>Formule :C19H17BrF4N6O6Couleur et forme :SolidMasse moléculaire :581.27KKII5
CAS :<p>KKII5 is a potent inhibitor of the lipoxygenase LOX-1 with an IC50 of 19 μM.KKII5 inhibits lipid peroxidation and enhances the ability of the active centers of</p>Formule :C16H14N2SDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :266.36Spaglumic acid acetate
Spaglumic acid acetate (Isospaglumic acid acetate) is a neuropeptide found in millimolar concentrations in brain.Formule :C13H20N2O10Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :364.31α-Pyrone
CAS :<p>Alpha-Pyrone exhibits inhibitory activity against tyrosinase, carbonic anhydrase 1, and carbonic anhydrase 9</p>Formule :C5H4O2Couleur et forme :SolidMasse moléculaire :96.08Enpp-1-IN-21
CAS :<p>Enpp-1-IN-21 (compound 4g) is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1), with IC50 values of 0.45 μM for ENPP1 and 0.19 μM for ENPP3.</p>Formule :C21H16F3NO5SCouleur et forme :SolidMasse moléculaire :451.42Tetrahydropteroylpentaglutamate
CAS :<p>H4PteGlu5 strongly inhibits itself and tightly binds in vivo, almost irreversibly, as a coenzyme.</p>Formule :C39H51N11O18Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :961.89Phosphodiesterase
CAS :<p>PDE enzyme hydrolyzes cyclic nucleotides, regulates signal transduction, and varies in type (PDE1-PDE11) with disease research potential.</p>Couleur et forme :Solid3-Oxocholic acid
CAS :<p>3-Oxocholic acid(3-Ketocholic acid) is the metabolite of bile acid and the main product of bile degradation by Clostridium perfringens in the intestine.3-</p>Formule :C24H38O5Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :406.56L-739750 2HCl
<p>L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.</p>Formule :C23H41Cl2N3O6S2Degré de pureté :98.69% - 99.16%Couleur et forme :SoildMasse moléculaire :590.62Acanthifolicin
CAS :Acanthifolicin, an okadaic acid derivative, has been shown top inhibit protein phosphatase 1 with an IC50= 20 nM (similar to that of okadaic acid at 19 nM).Formule :C44H68O13SCouleur et forme :SolidMasse moléculaire :837.08FCPR03
CAS :FCPR03 is a selective inhibitor of phosphodiesterase 4 (PDE4) with IC50s of 31 nM, 47 nM, and 60 nM for PDE4B1, PDE4D7, and PDE4 catalytic domain, respectively.Formule :C15H19F2NO3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :299.31(±)13(14)-EpDPA
CAS :<p>Cytochrome P450 metabolism of polyunsaturated fatty acids produces numerous bioactive epoxide regioisomers.</p>Formule :C22H32O3Couleur et forme :SolidMasse moléculaire :344.495THX6
<p>THX6 is an activator of human mitochondrial protease ClpP, with an EC50 of 1.18 μM. It displays cytotoxicity in ONC201-resistant SU-DIPG-VI cells, with an IC50 of 0.13 μM. THX6 inhibits the expression of mitochondria-related proteins (such as parkin, TFAM, NRF1, SDHA), leading to impaired mitochondrial function. Additionally, THX6 affects cell membrane lipid metabolism and exhibits antitumor potential.</p>Formule :C22H18Cl2N4O2Couleur et forme :SolidMasse moléculaire :441.31Ethyl gentisate
CAS :<p>Ethyl gentisate acts as a dual regulator of cell differentiation, promoting osteoblast differentiation while inhibiting osteoclast differentiation.</p>Formule :C9H10O4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :182.17Galactosylhydroxylysine hydrochloride
<p>Galactosylhydroxylysine hydrochloride, found in bone collagen, is higher in metabolic bone loss due to resorption.</p>Formule :C12H25ClN2O8Couleur et forme :SolidMasse moléculaire :360.79IDO1/TDO-IN-8
<p>IDO1/TDO-IN-8 (Compound CZ-17) is a dual IDO1 and TDO inhibitor capable of crossing the blood-brain barrier, with EC50 values of 0.33 μM and 1.78 μM, respectively. It modulates the kynurenine pathway of tryptophan metabolism, reducing the kynurenine/tryptophan ratio. IDO1/TDO-IN-8 has neuroprotective effects, alleviating motor dysfunction and improving depressive behavior, making it relevant for research into Parkinson's disease with comorbid depression.</p>Formule :C17H14N2SCouleur et forme :SolidMasse moléculaire :278.37Daclatasvir Impurity C
CAS :<p>Daclatasvir Impurity C is an impurity found in Daclatasvir, a robust inhibitor of the HCV NS5A protein [1].</p>Formule :C29H32N6O3Couleur et forme :SolidMasse moléculaire :512.6Meproscillarin
CAS :<p>Meproscillarin is a glycoside with high bioavailability (about 70%) and an elimination independent of renal function.</p>Formule :C31H44O8Couleur et forme :SolidMasse moléculaire :544.68PtdIns-(3,4,5)-P3 (1,2-dihexanoyl) (ammonium salt)
CAS :<p>PIP3, a minor yet critical phospholipid for cell signaling, resists PLC cleavage and anchors PH domain proteins, affecting cytoskeletal and membrane dynamics.</p>Formule :C21H45NO22P4Couleur et forme :SolidMasse moléculaire :787.471α-Glucosidase-IN-46
<p>α-Glucosidase-IN-46 is a potent inhibitor of α-glucosidase, with an IC50 of 26.0 μM. This compound is applicable in the research of Type 2 diabetes.</p>Formule :C35H32N4O5Masse moléculaire :588.23727LEI110
CAS :<p>LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.</p>Formule :C25H23F3N2O3Degré de pureté :98.66% - 98.8%Couleur et forme :SolidMasse moléculaire :456.46FA-Ala-Arg
CAS :<p>FA-Ala-Arg is a dipeptide featuring a furylacryloyl group that degrades to yield arginine.</p>Formule :C16H23N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :365.38Impurity B of Calcitriol
CAS :<p>Impurity B is a byproduct of Calcitriol, the active hormone form of vitamin D3 and VDR activator.</p>Formule :C27H44O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.64PDE1-IN-5
<p>PDE1-IN-5 (Compound 10c) is a selective PDE1C inhibitor with an IC50 of 15 nM, exhibiting anti-inflammatory properties through the inhibition of iNOS, TNF-α, IL</p>Formule :C27H29FN4OCouleur et forme :SolidMasse moléculaire :444.54Butyrolactone II
CAS :<p>Butyrolactone II is a useful organic compound for research related to life sciences. The catalog number is T124034 and the CAS number is 87414-44-6.</p>Formule :C19H16O7Couleur et forme :SolidMasse moléculaire :356.33Cholesterol esterase
CAS :<p>Cholesterol esterase breaks down cholesterol ester into cholesterol and free fatty acids, aiding absorption.</p>Couleur et forme :SolidHLF1-11
CAS :<p>HLF1-11: human lactoferrin peptide, antimicrobial, inhibits MPO, steers monocytes to macrophages, boosts immunity.</p>Formule :C56H95N25O14SCouleur et forme :SolidMasse moléculaire :1374.58Casein Kinase 2 Substrate Peptide
CAS :<p>CK2 Substrate Peptide, C-terminus linked to EDANS, used for CK2 activity assays.</p>Formule :C45H73N19O24Couleur et forme :SolidMasse moléculaire :1264.17PDE1-IN-8
<p>PDE1-IN-8 (Compound 3f) acts as an inhibitor of PDE1, with an IC50 of 11 nM. It hinders cAMP and cGMP signaling pathways, impeding the differentiation and proliferation of cells into myofibroblasts, and demonstrates antifibrotic effects in the Bleomycin-induced rat model of pulmonary fibrosis.</p>Formule :C17H11Cl2N3OS2Couleur et forme :SolidMasse moléculaire :408.32Methylcardol triene
CAS :<p>Methylcardol triene, a phenolic compound present in cashew nut shell liquid, demonstrates α-glucosidase inhibition (IC50= 39.6 µM) and exhibits schistosomicidal properties by eliminating 100% of adult S. mansoni worms within 24 hours at 100 and 200 µM concentrations. Moreover, it serves as a precursor for synthesizing mono- and bis-benzoxazines.</p>Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.496tetranor-12(S)-HETE
CAS :<p>12(S)-HETE, from arachidonic acid via 12-lipoxygenase, is found in platelets and leukocytes, aids tumor cell adhesion, with a derivative used in research.</p>Formule :C16H26O3Couleur et forme :SolidMasse moléculaire :266.3811-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine
CAS :<p>Endogenous metabolite: 1-myristoyl-2-stearoyl-sn-glycero-3-phosphocholine, a phosphatidylcholine example.</p>Formule :C40H80NO8PDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :734.04NPE-caged-proton
CAS :<p>Generates rapid acidifications down to pH 2</p>Formule :C8H9NNaO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.22α-glucosidase/PTP1B-IN-1
<p>α-glucosidase/PTP1B-IN-1 (compound 8a) is an effective inhibitor of both α-glucosidase and PTP1B, with IC50 values of 66.3 μM and 47.0 μM, respectively. It also exhibits strong inhibitory activity against α-amylase, having an IC50 of 30.62 μM. This compound is capable of binding to the active sites of α-glucosidase and PTP1B. α-glucosidase/PTP1B-IN-1 holds potential for reducing postprandial blood glucose levels and may be useful in managing type 2 diabetes.</p>Formule :C23H20Cl2O5Couleur et forme :SolidMasse moléculaire :447.31SR-4995
CAS :<p>SR-4995 (CID 16016685) is an ABHD5 ligand, directly binding to ABHD5 and stimulating lipolysis by releasing it from PLIN.</p>Formule :C19H21N3O2SCouleur et forme :SoildMasse moléculaire :355.45Vitamin K5
CAS :<p>Vitamin K5, a photosensitizer & antimicrobial, inhibits PKM2, PKM1 & PKL, induces apoptosis in colon cells, and preserves food & medicine.</p>Formule :C11H11NOCouleur et forme :SolidMasse moléculaire :173.21Carboxylesterase
CAS :<p>CESs are enzymes in mammalian liver hydrolyzing esters and other substrates in biochemical studies.</p>Couleur et forme :SolidHydroxypyruvic acid lithium hydrate
CAS :<p>Hydroxypyruvic acid lithium hydrate is a metabolic intermediate for serine, glycine, threonine, and a substrate for specific aminotransferases.</p>Formule :C3H5LiO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :128.01Arofylline
CAS :<p>Arofylline (LAS 31025) is a PDE4 inhibitor and can be used for asthma studies.</p>Formule :C14H13ClN4O2Degré de pureté :98.19%Couleur et forme :SolidMasse moléculaire :304.73NGR peptide
CAS :<p>Cell-penetrating peptide</p>Formule :C20H36N10O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.69Anti-osteoporosis agent-10
<p>Anti-osteoporosis agent-10 is an inhibitor of osteoporosis that suppresses the formation of osteoclasts with an IC50 of 0.042 μM. It also exhibits antagonistic activity towards PPARγ, with an EC50 value of 0.75 μM.</p>Couleur et forme :Odour SolidTRH Precursor Peptide
<p>Thyrotropin Releasing Hormone Precursor Peptide</p>Formule :C42H75N19O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1006.17CNBCA
<p>CNBCA, a selective and potent competitive inhibitor of the SHP2 enzyme, exhibits an IC50 value of 0.87 μM.</p>Formule :C26H34O5Couleur et forme :SolidMasse moléculaire :426.55SMS2-IN-1
CAS :<p>SMS2-IN-1: potent SMS2 inhibitor; IC50: 6.5 nM, Kd: 37 nM; 150x selectivity over SMS1.</p>Formule :C34H37F6N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :681.67BI 1015550
CAS :<p>Nerandomilast (BI 1015550) is an orally active PDE4B inhibitor with IC50 of 7.2 nM.Cost-effective and quality-assured.</p>Formule :C20H25ClN6O2SDegré de pureté :98.06% - 99.71%Couleur et forme :SoildMasse moléculaire :448.97IRC-083864
CAS :<p>IRC-083864 is a novel bis quinone CDC25 phosphatase active inhibitor against human cancer cells.</p>Formule :C28H25F2N5O5SCouleur et forme :SolidMasse moléculaire :581.59Evinacumab
CAS :<p>Evinacumab (REGN1500) is a humanized monoclonal antibody targeting ANGPTL3. It is useful for studying cardiovascular diseases.</p>Degré de pureté :100% (SEC-HPLC) - 99.43% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.5 kDaFibrostatin C
CAS :<p>Fibrostatin C is an inhibitor of prolyl 4-hydroxylase. It is produced by Streptomyces catenulae subsp.</p>Formule :C18H19NO8SCouleur et forme :SolidMasse moléculaire :409.41Systemin
CAS :<p>Systemin is an 18-amino acid polypeptide with the sequence AVQSKPPSKRDPPKMQTD that is found in Solanaceae plants (such as tomato and potato).</p>Formule :C85H144N26O28SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2010.28Trimipramine N-oxide
CAS :<p>Trimipramine N-oxide, a trimipramine metabolite, inhibits hNAT, hSERT, hDAT, and hOCT1/2 with IC50s 11.7-27.4 nM; for depression/anxiety research.</p>Formule :C20H26N2OCouleur et forme :SolidMasse moléculaire :310.43BAY 2666605
CAS :<p>BAY 2666605 is an orally active inhibitor of PDE3A and PDE3B with IC50s of 87 nM and 50 nM, respectively. BAY 2666605 has anticancer effects.</p>Formule :C17H12F4N2O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :352.28Nodularin
CAS :<p>Nodularin from N. spumigena is a hepatotoxic pentapeptide that inhibits PP1 and PP2A with IC50s of 1.8 nM and 0.026 nM, respectively.</p>Formule :C41H60N8O10Couleur et forme :SolidMasse moléculaire :824.977Canine Factor Xa
<p>CanineFactor Xa is derived from purified Canine Factor X through activation by Russell's Viper Venom, after which the venom is removed.</p>Couleur et forme :Odour Solid1-Palmitoyl-2-linoleoyl PE
CAS :<p>Phosphatidylethanolamine PLPE: a cell membrane component, studied for anandamide biosynthesis, sPLA2-IIA activity substrate.</p>Formule :C39H74NO8PCouleur et forme :SolidMasse moléculaire :715.9941,3-Diphenethylurea
CAS :<p>1,3-Diphenethylurea (N,N'-Bis(phenethyl)urea) is a marine derived natural products found in Lissoclinum patella.</p>Formule :C17H20N2ODegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :268.35α-1,3-N-Acetylgalactosaminyltransferase (Pm1138)
CAS :<p>Alpha-1,3-N-Acetylgalactosaminyltransferase (Pm1138) (EC 2.4.1.40(Pm1138)), also known as the ABO system transferase, exhibits glycosyl transferase activity [1</p>Couleur et forme :SolidPLA2-IN-1
<p>PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.</p>Couleur et forme :Odour SolidCarbonic anhydrase inhibitor 30
<p>Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].</p>Formule :C23H22FN3O5SCouleur et forme :SolidMasse moléculaire :471.12642Cyclohexanoyl Coenzyme A
CAS :<p>"Cyclohexanoyl CoA (CHCoA) activates CHC in R. palustris, converts to hippuric acid in guinea pig liver."</p>Formule :C28H46N7O17P3SCouleur et forme :SolidMasse moléculaire :877.6913-epi-12-oxo Phytodienoic Acid
CAS :<p>13-epi-12-oxo PDA is a lipoxygenase derivative of α-linolenic acid in green plant leaves, often isomerizing during extraction and storage.</p>Formule :C18H28O3Couleur et forme :SolidMasse moléculaire :292.41Microginin 527
CAS :<p>Microginin 527, a compound found in Microcystis, is an inhibitor of protein phosphatase, ACE, and leucine aminopeptidase.</p>Formule :C25H41N3O7SCouleur et forme :SolidMasse moléculaire :527.675-hydroxy Omeprazole
CAS :<p>5-hydroxy omeprazole, major omeprazole metabolite, formed by CYP2C19, affects gastric H+/K+ pump inhibition.</p>Formule :C17H19N3O4SCouleur et forme :SolidMasse moléculaire :361.42Pepticinnamin E
CAS :<p>Pepticinnamin E is a naturally occurring bisubstrate farnesyltransferase inhibitor.</p>Formule :C49H54ClN5O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :908.43Coformycin
CAS :<p>Coformycin is a ribonucleoside antibiotic synergist and adenosine deaminase inhibitor.</p>Formule :C11H16N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.27TDO-IN-2
<p>TDO-IN-2 is an orally active TDO inhibitor with an IC50 of 1.25 μM. It exhibits antitumor activity in a Hepa1-6 liver cancer allograft mouse model. Additionally, TDO-IN-2 works synergistically with PD-1/PD-L1 inhibitor BMS-202, making it useful for studying tumor immune tolerance.</p>Formule :C20H15N3O3Couleur et forme :SolidMasse moléculaire :345.11134TEI-9648
CAS :<p>TEI-9648: Potent, specific VDR antagonist, blocks 1α,25(OH)2D3 effects, may aid bone metabolism study.</p>Formule :C27H38O4Couleur et forme :SolidMasse moléculaire :426.597A 58365 A
CAS :<p>A 58365 A, an ACE inhibitor from Streptomyces chromofuscus, treats heart failure and hypertension.</p>Formule :C12H13NO6Couleur et forme :SolidMasse moléculaire :267.23CAY10640
CAS :<p>CAY10640 (sEH inhibitor-1) is a potent, orally active, water-soluble epoxide hydrolase (sEH) inhibitor that inhibits sEH in humans and mice with IC50s of 0.4</p>Formule :C17H20F3N3O3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :371.35CK1-IN-4
<p>CK1-IN-4 (Compound 59) is an inhibitor of casein kinase CK1δ with an IC50 of 2.74 μM. It exhibits neuroprotective activity in SH-SY5Y cells treated with Ethacrynic acid.</p>Couleur et forme :Odour SolidPhytin
CAS :<p>Phytin has a wide range of applications in life science related research.</p>Formule :C6H6CaMgO24P6Couleur et forme :White PowderMasse moléculaire :712.32Sandosaponin A
CAS :<p>Sandosaponin A, an olean-12-ene-type triterpene oligoglycoside, is isolated from kidney bean, the seed of Phaseolus vulgaris L.</p>Formule :C48H76O19Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :957.11Imatinib Impurity E
CAS :<p>Imatinib Impurity E, a derivative of orally taken Imatinib, inhibits tyrosine kinases BCR/ABL, PDGFR, c-kit, and SARS/MERS-CoV.</p>Formule :C52H48N12O2Couleur et forme :SolidMasse moléculaire :873.021-Heptadecanoyl-2-hydroxy-sn-glycero-3-phosphocholine
CAS :<p>An endogenous blood metabolite, 1-heptadecanoyl-glycerophosphocholine, researches pregnancy/sepsis.</p>Formule :C25H52NO7PCouleur et forme :SolidMasse moléculaire :509.66Mesembrenone
CAS :<p>Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum.</p>Formule :C17H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :287.35SPL-334
CAS :<p>SPL-334 is an inhibitor of S-nitrosoglutathione reductase.</p>Formule :C22H15N3O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.505β-Androstan-3β-ol-17-one
CAS :<p>5β-Androstan-3β-ol-17-one (3β-Etiocholanolone; 5β-Epiandrosterone), a 5β-reduced steroid and a significant metabolic derivative of dehydroepiandrosterone (DHEA</p>Formule :C19H30O2Couleur et forme :SolidMasse moléculaire :290.44α-Muricholic acid
CAS :<p>α-Muricholic acid is the most abundant primary bile acid in rodents.</p>Formule :C24H40O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.57O-Demethyl Lenvatinib hydrochloride
<p>O-Demethyl Lenvatinib HCl is a Lenvatinib metabolite; an oral inhibitor targeting VEGFR, FGFR, PDGFR, KIT, RET with antitumor properties.</p>Formule :C20H18Cl2N4O4Couleur et forme :SolidMasse moléculaire :449.29UCM-13207
CAS :UCM-13207 is a specific ICMT inhibitor that improves progeria.Formule :C24H32N2O2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :380.52Desbutyl Lumefantrine
CAS :<p>Desbutyl Lumefantrine is a metabolite of lumefantrine with antimalarial activity.</p>Formule :C26H24Cl3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.83
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