
Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(41 produits)
- Aminopeptidase(67 produits)
- CETP(18 produits)
- Anhydrase carbonique(178 produits)
- Caséine Kinase(130 produits)
- DHFR(33 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(271 produits)
- FAAH(64 produits)
- FXR(58 produits)
- Facteur Xa(80 produits)
- Synthase des acides gras(33 produits)
- Ferroptose(215 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(54 produits)
- Prolyl-Hydroxylase de HIF/HIF(142 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(30 produits)
- IDO(82 produits)
- LDL(8 produits)
- Lipase(98 produits)
- Lipides(58 produits)
- Lipoxygénase(124 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(36 produits)
- P450(6 produits)
- PAI-1(25 produits)
- PDE(166 produits)
- PED(1 produits)
- PKM(15 produits)
- PPAR(165 produits)
- Phospholipase(82 produits)
- ROR(42 produits)
- Récepteur de rétinoïdes(29 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(30 produits)
- Tansporteur(42 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
8628 produits trouvés pour "Métabolisme"
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Nitrofurazone
CAS :<p>Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria.</p>Formule :C6H6N4O4Degré de pureté :99.87%Couleur et forme :Pale Yellow Needles Solution) 6 0 - 6 5 Alkaline Solutions Are Dark Orange (Ntp 1992)Masse moléculaire :198.14Linrodostat
CAS :Linrodostat (BMS-986205) is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.Formule :C24H24ClFN2ODegré de pureté :99.54% - 99.71%Couleur et forme :SolidMasse moléculaire :410.91PF-06282999
CAS :<p>PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potentially useful for the treatment of cardiovascular diseases.</p>Formule :C13H12ClN3O3SDegré de pureté :98.15% - 98.28%Couleur et forme :SolidMasse moléculaire :325.77NS-638
CAS :<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Formule :C15H11ClF3N3Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :325.72Pentamidine
CAS :<p>Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor</p>Formule :C19H24N4O2Degré de pureté :98.64% - 99.67%Couleur et forme :Crystallizes As Colorless Plates From Water SolidMasse moléculaire :340.422-hydroxymethyl benzoic acid
CAS :<p>2-hydroxymethyl benzoic acid is a principal metabolite of the phthalidyl moiety in man.</p>Formule :C8H8O3Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :152.15Alrestatin
CAS :<p>Alrestatin (AY-22284) is a specific inhibitor of aldose reductase and attenuates glucose-induced angiotensin II production in rat vascular smooth muscle in</p>Formule :C14H9NO4Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :255.2256GOT1 inhibitor-1
CAS :<p>GOT1 inhibitor-1 (GOT1 inhibitor 2c) is a novel, potent and non-covalent inhibitor of glutamate oxaloacetate transaminase 1 (GOT1) with an IC50 of 8.2 uM.</p>Formule :C19H19ClN4ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :354.83SR3335
CAS :<p>SR3335 (ML 176) is a selective inverse agonist of RORα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (Ki: 220 nM).</p>Formule :C13H9F6NO3S2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :405.34AZ876
CAS :<p>AZ876 is a potent, highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.</p>Formule :C24H29N3O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :439.57SR8278
CAS :<p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>Formule :C18H19NO3S2Degré de pureté :99.44% - 99.73%Couleur et forme :SolidMasse moléculaire :361.48BRL-50481
CAS :<p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>Formule :C9H12N2O4SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :244.27Toloxatone
CAS :<p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>Formule :C11H13NO3Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :207.23Obafistat
CAS :<p>Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.</p>Formule :C15H16FN5O3SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :365.38BI-187004
CAS :<p>BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.</p>Formule :C21H18N4ODegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :342.39U-104
CAS :<p>U-104 (NSC-213841) is an effective carbonic anhydrase (CA) inhibitor for CA IX( Ki=45.1 nM) and CA XII(Ki=4.5 nM).</p>Formule :C13H12FN3O3SDegré de pureté :98.76% - 99.88%Couleur et forme :SolidMasse moléculaire :309.32Gonadorelin Acetate (33515-09-2 free base)
CAS :<p>Gonadorelin Acetate (33515-09-2 free base) (Luteinizing Hormone Releasing Hormone (LH-RH)) is hypothalamic neuropeptide which plays a key role in the control of</p>Formule :C59H83N17O17Degré de pureté :99.42% - 99.46%Couleur et forme :White Or Off-White PowderMasse moléculaire :1302.39AUDA
CAS :<p>AUDA is an inhibitor of sEH(IC50 values of 18 and 69 nM for the mouse and human enzymes, respectively)</p>Formule :C23H40N2O3Degré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :392.58p-Fluoro-L-phenylalanine
CAS :<p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>Formule :C9H10FNO2Degré de pureté :99.63%Couleur et forme :White To Off-White PowderMasse moléculaire :183.18BW-A 78U
CAS :<p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>Formule :C13H12FN5Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :257.27GSK805
CAS :<p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>Formule :C23H18Cl2F3NO4SDegré de pureté :98% - ≥95%Couleur et forme :SolidMasse moléculaire :532.362-Bromo-4'-hydroxyacetophenone
CAS :<p>2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).</p>Formule :C8H7BrO2Degré de pureté :98.64%Couleur et forme :Clear Colorless To Light Yellow LiquidMasse moléculaire :215.04Telaglenastat
CAS :<p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>Formule :C26H24F3N7O3SDegré de pureté :97.57% - 99.89%Couleur et forme :SolidMasse moléculaire :571.57Pargyline
CAS :<p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>Formule :C11H13NDegré de pureté :95.64% - 97.21%Couleur et forme :SolidMasse moléculaire :159.23PfDHODH-IN-2
CAS :<p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>Formule :C13H12ClNO3SDegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :297.76Pentamidine isethionate
CAS :<p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>Formule :C23H36N4O10S2Degré de pureté :98% - 99.83%Couleur et forme :Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)Masse moléculaire :592.68FG-2216
CAS :<p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>Formule :C12H9ClN2O4Degré de pureté :97.1% - >99.99%Couleur et forme :SolidMasse moléculaire :280.66JZL 184
CAS :<p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>Formule :C27H24N2O9Degré de pureté :97.56% - 99.31%Couleur et forme :SolidMasse moléculaire :520.49RGX-104
CAS :<p>RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)</p>Formule :C34H33ClF3NO3Degré de pureté :98.79% - 99.53%Couleur et forme :SolidMasse moléculaire :596.08KPT9274
CAS :KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.Formule :C35H29F3N4O3Degré de pureté :99.75% - 99.93%Couleur et forme :SolidMasse moléculaire :610.62LOX-IN-3 dihydrochloride
CAS :<p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>Formule :C13H15Cl2FN2O2SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :353.24Cobicistat
CAS :Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.Formule :C40H53N7O5S2Degré de pureté :97.36% - 99.62%Couleur et forme :SolidMasse moléculaire :776.02Glycerol 3-phosphate biscyclohexylammonium salt
CAS :<p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>Formule :C15H35N2O6PDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :370.42ARM1
CAS :<p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>Formule :C16H14N2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :266.36(±)-Amiflamine
CAS :<p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>Formule :C12H20N2Degré de pureté :97.24%Couleur et forme :SolidMasse moléculaire :192.3Cecropin P1, porcine acetate
<p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>Formule :C149H257N45O45Degré de pureté :95.4% - 98%Couleur et forme :SolidMasse moléculaire :3398.91Bempedoic acid
CAS :<p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>Formule :C19H36O5Degré de pureté :99.85% - 99.94%Couleur et forme :SolidMasse moléculaire :344.49Efonidipine hydrochloride monoethanolate
CAS :<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formule :C36H45ClN3O8PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :714.181-Ethynylpyrene
CAS :<p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>Formule :C18H10Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :226.27Suvecaltamide
CAS :Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.Formule :C20H23F3N2O2Degré de pureté :99.29% - 99.70%Couleur et forme :SolidMasse moléculaire :380.4SGC-GAK-1
CAS :<p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>Formule :C18H17BrN2O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :389.24GSK1016790A
CAS :<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formule :C28H32Cl2N4O6S2Degré de pureté :97.37% - 99.38%Couleur et forme :SolidMasse moléculaire :655.61DHBP dibromide
CAS :<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formule :C24H38Br2N2Degré de pureté :99.73%Couleur et forme :Yellow To Yellow-Green Powder Or FlakesMasse moléculaire :514.38(Rac)-LB-100
CAS :<p>LB-100, a novel Protein Phosphatase 2A (PP2A) inhibitor, sensitizes malignant meningioma cells to the therapeutic effects of radiation</p>Formule :C13H20N2O4Degré de pureté :97.11% - 99.77%Couleur et forme :SolidMasse moléculaire :268.31Pep 2-8 ammonium salt(1541011-97-5 free base)
<p>Pep 2-8 ammonium salt inhibits PCSK9-LDL receptor binding (IC50 = 0.8 μM), boosting LDL uptake in HepG2 cells.</p>Formule :C83H113N17O24Degré de pureté :95.76% - 99.87%Couleur et forme :SolidMasse moléculaire :1732.912,5-Di-tert-butylhydroquinone
CAS :<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formule :C14H22O2Degré de pureté :97.11%Couleur et forme :PelletslargecrystalsMasse moléculaire :222.32kb NB 142-70
CAS :<p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>Formule :C11H9NO2S2Degré de pureté :98.15% - ≥95%Couleur et forme :SolidMasse moléculaire :251.32AGN 193109
CAS :<p>AGN 193109, a retinoid analog, is a potent and specific antagonist of RARs (Kds: 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ).</p>Formule :C28H24O2Degré de pureté :99.87% - 99.89%Couleur et forme :SolidMasse moléculaire :392.49D-Valine
CAS :<p>D-Valine (H-D-Val-OH) is the enantiomer of L-Valine.</p>Formule :C5H11NO2Degré de pureté :99.93%Couleur et forme :White CrystalsMasse moléculaire :117.15GSK2033
CAS :<p>GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).</p>Formule :C29H28F3NO5S2Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :591.66Efonidipine
CAS :Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Formule :C34H38N3O7PDegré de pureté :98.35% - 99.47%Couleur et forme :SolidMasse moléculaire :631.66IDO5L
CAS :IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).Formule :C9H7ClFN5O2Degré de pureté :99.49% - 99.75%Couleur et forme :SolidMasse moléculaire :271.64Tedizolid
CAS :<p>Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of</p>Formule :C17H15FN6O3Degré de pureté :96.97% - 99.89%Couleur et forme :SolidMasse moléculaire :370.34Pimecrolimus
CAS :<p>Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.</p>Formule :C43H68ClNO11Degré de pureté :99.53% - 99.87%Couleur et forme :White Crystalline PowderMasse moléculaire :810.45SI-113
CAS :<p>SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.</p>Formule :C23H24N6ODegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :400.48BAY-876
CAS :<p>BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.</p>Formule :C24H16F4N6O2Degré de pureté :98.61% - 99.78%Couleur et forme :SolidMasse moléculaire :496.42Benzenesulfonamide
CAS :<p>Benzenesulfonamide (Benzosulfonamide) ia an inhibitor of carbonic anhydrases.</p>Formule :C6H7NO2SDegré de pureté :99.42% - 99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :157.19IDF-11774
CAS :<p>IDF-11774 is a HIF-1 inhibitor.It reduces hif-1α HRE luciferase activity (IC50 = 3.65 μM).</p>Formule :C23H32N2O2Degré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :368.51Z-HA155
CAS :<p>Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.</p>Formule :C24H19BFNO5SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :463.29Raphin1
CAS :Raphin1 is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B).Formule :C8H8Cl2N4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :231.08IOX2
CAS :<p>IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.</p>Formule :C19H16N2O5Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :352.34Tepoxalin
CAS :<p>Tepoxalin (RWJ 20485), potential asthma and osteoarthritis drug, inhibits COX-1, COX-2, and 5-LOX with low IC50 values.</p>Formule :C20H20ClN3O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :385.84ZINC13466751
CAS :<p>ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).</p>Formule :C20H21N5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :363.41Olumacostat Glasaretil
CAS :<p>Olumacostat glasaretil is a small molecule inhibitor of acetyl coenzyme A carboxylase (ACC). It has been used in trials studying the treatment of Acne Vulgaris.</p>Formule :C26H43NO7Degré de pureté :97.79% - 99.34%Couleur et forme :SolidMasse moléculaire :481.622-Aminoethyl diphenylborinate
CAS :<p>2-Aminoethyl diphenylborinate (2-APB) is a chemical that acts to inhibit both IP3 receptors and TRP channels.</p>Formule :C14H16BNODegré de pureté :98.74% - 99.92%Couleur et forme :WhiteMasse moléculaire :225.09MBCQ
CAS :<p>MBCQ is an inhibitor of cGMP-specific phosphodiesterase PDE5.</p>Formule :C16H12ClN3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :313.74Ingliforib
CAS :<p>Ingliforib (CP 368296) is a novel glycogen phosphorylase inhibitor,has antihyperglycemic and cardioprotective properties.</p>Formule :C23H24ClN3O5Degré de pureté :99.04% - 99.30%Couleur et forme :SolidMasse moléculaire :457.91Cyfluthrin
CAS :<p>Cyfluthrin binds to voltage-sensitive sodium channel such as Nav 1.8 sodium channel and modify their gating kinetics, thereby disrupting nerve function of pests</p>Formule :C22H18Cl2FNO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :434.29Biotin sulfone
CAS :<p>Biotin sulfone is an oxidized form of biotin.</p>Formule :C10H16N2O5SDegré de pureté :95.51%Couleur et forme :SolidMasse moléculaire :276.31Lactisole
CAS :<p>Lactisole (na-PMP) is an inhibitor of the glucose-sensing receptor</p>Formule :C10H11NaO4Degré de pureté :99.9%Couleur et forme :White To Pale Cream Crystalline SolidMasse moléculaire :218.18BCI hydrochloride
CAS :<p>BCI hydrochloride ((E)-BCI hydrochloride) is a DUSP6 inhibitor that inhibits RANKL-mediated osteoclastogenesis and attenuates oophorectomy-induced bone loss.</p>Formule :C22H24ClNODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :353.89PKM2-IN-1
CAS :<p>PKM2-IN-1 (compound 3k) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.</p>Formule :C18H19NO2S2Degré de pureté :99.49% - 99.68%Couleur et forme :SolidMasse moléculaire :345.48Glucosamine sulfate
CAS :<p>Glucosamine sulfate (D-Glucosaminesulfate) was extracted from synthetic product;Store the product in sealed, cool and dry condition.</p>Formule :C6H13NO5·H2SO4Degré de pureté :99.64%Couleur et forme :White CrystalMasse moléculaire :277.25GW604714X
CAS :<p>GW604714X (2,4-Thiazolidinedione, 5-[[5-[6-(4-acetyl-1-piperazinyl)-3-nitro-2-pyridinyl]-2-fluorophenyl]methylene]-) were found to be potent inhibitors of</p>Formule :C21H18FN5O5SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :471.46Ned 19
CAS :<p>Ned 19 inhibits tumor growth, vascularization, lung metastases in mice, and is a selective NAADP antagonist.</p>Formule :C30H31FN4O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :514.59SDZ285428
CAS :<p>SDZ285428 is a CYP24A1 inhibitor.</p>Formule :C24H20ClN3ODegré de pureté :97.51%Couleur et forme :SolidMasse moléculaire :401.891-Ethynylnaphthalene
CAS :<p>1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 IB1</p>Formule :C12H8Degré de pureté :99.05%Couleur et forme :Yellow To Brown LiquidMasse moléculaire :152.19SR9243
CAS :<p>SR9243, an LXR inverse agonist, can induce LXR-corepressor interaction; shows anticancer activity and selectively targets the lipogenesis and Warburg effect.</p>Formule :C31H32BrNO4S2Degré de pureté :98% - 99.03%Couleur et forme :SolidMasse moléculaire :626.62Alendronate sodium trihydrate
CAS :<p>Alendronate sodium hydrate (MK 217), a nitrogen bisphosphonate, inhibits bone loss, treats and prevents osteoporosis.</p>Formule :C4H12NO7P2·3H2O·NaDegré de pureté :99.66% - 99.90%Couleur et forme :White Crystalline SolidMasse moléculaire :325.121-NM-PP1
CAS :<p>1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.</p>Formule :C20H21N5Degré de pureté :98% - 98.93%Couleur et forme :White Cyrstalline SolidMasse moléculaire :331.41F1063-0967
CAS :<p>F1063-0967 is a Dual-specificity phosphatase 26 (DUSP26) inhibitor with an IC50 of 11.62 μM.</p>Formule :C24H24N2O5S2Degré de pureté :97.77%Couleur et forme :SolidMasse moléculaire :484.59M1001
CAS :<p>M1001 is a HIF-2α agonist.</p>Formule :C17H17N3O2SDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :327.4SHP099 hydrochloride
CAS :<p>SHP099 hydrochloride is a potent, selective, orally bioavailable SHP2 inhibitor with IC50 of 70 nM, which inhibits ERK1/2 activation in cancer cells.Cost-effective and quality-assured.</p>Formule :C16H20Cl3N5Degré de pureté :99.13% - 99.62%Couleur et forme :SolidMasse moléculaire :388.72CDC25B-IN-2
CAS :<p>BIA is an inhibitor of the interaction between TMBIM6 and mTORC2, which ultimately blocks AKT activation and cancer progression.</p>Formule :C15H12N2O3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :268.27GW 501516
CAS :<p>GW 501516 (Endurobol) is a effective and highly specifc PPARβ/δ agonist (EC50: 1 nM), with 1000-fold selectivity over hPPARα/γ.</p>Formule :C21H18F3NO3S2Degré de pureté :98.91% - 99.64%Couleur et forme :White SolidMasse moléculaire :453.50CDD3505
CAS :CDD3505 (4-nitro-1-trityl-1H-imidazole) increases high-density lipoprotein cholesterol by targeting hepatic CYP3A.Formule :C22H17N3O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :355.39FPL 62064
CAS :<p>FPL 62064 is a potent dual inhibitor of 5-lipoxygenase (5-LOX) and COX (IC50 of 3.5 μM and 3.1 μM for RBL-1 cytosolic 5-lipoxygenase and prostaglandin</p>Formule :C16H15N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :265.31GSK2981278
CAS :<p>GSK2981278 (ROR gama modulator 1) is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).</p>Formule :C25H35NO5SDegré de pureté :99.31% - 99.67%Couleur et forme :SolidMasse moléculaire :461.61all-trans-4-Oxoretinoic acid
CAS :all-trans-4-Oxoretinoic acid (all-trans 4-Keto Retinoic Acid) is an active metabolite of vitamin A.Formule :C20H26O3Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :314.42Entacapone
CAS :<p>Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).</p>Formule :C14H15N3O5Degré de pureté :98.80% - >99.99%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :305.29Ervogastat
CAS :<p>Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.</p>Formule :C21H21N5O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :407.42Galeterone
CAS :<p>Galeterone (VN 124) is an oral androgen receptor modulator/CYP17 inhibitor with antiandrogen properties, targeting prostate cancer growth.</p>Formule :C26H32N2ODegré de pureté :99.47% - 99.773%Couleur et forme :SolidMasse moléculaire :388.55AR7
CAS :<p>AR7 is a retinoic acid receptor α (RARα) antagonist.</p>Formule :C15H12ClNODegré de pureté :98.12% - 99.86%Couleur et forme :SolidMasse moléculaire :257.71Heparin sodium salt
CAS :<p>Heparin sodium, a sulfated glycosaminoglycan, acts as an anticoagulant and inhibits exosome-cell interactions.</p>Formule :C26H42N2NaO37S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1157.89BMS-687453
CAS :<p>BMS-687453 is a potent and selective PPAR alpha agonist, with an EC(50) of 10 nM for human PPARalpha and approximately 410-fold selectivity vs human PPARgamma</p>Formule :C22H21ClN2O6Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :444.86PF-06840003
CAS :<p>PF-06840003 (EOS200271) is a specific and oral active IDO-1 inhibitor.</p>Formule :C12H9FN2O2Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :232.21RORγt inverse agonist 13
CAS :<p>RORγt inverse agonist 13 (Compound 3i) is a potent, orally active and selective RORγt inverse agonist (IC50=63.8 nM), with improved drug-like properties[1].</p>Formule :C23H17Cl2F3N2O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :513.29SB 204990
CAS :<p>SB 204990 is a lactone prodrug of SB-201076, a potent and specific ATP citrate lyase inhibitor.Cost-effective and quality-assured.</p>Formule :C18H22Cl2O5Degré de pureté :96.32% - 99.6%Couleur et forme :SolidMasse moléculaire :389.27Tosedostat
CAS :<p>Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.</p>Formule :C21H30N2O6Degré de pureté :98.14% - 99.4%Couleur et forme :SolidMasse moléculaire :406.47Homo Sildenafil
CAS :<p>Homo Sildenafil is an analog of Sildenafil, It acts as a phosphodiesterase inhibitor.</p>Formule :C23H32N6O4SDegré de pureté :99.88%Couleur et forme :White SolidMasse moléculaire :488.6TCS 401
CAS :TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B; Ki = 0.29 μM)Formule :C10H11ClN2O5SDegré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :306.72GEBR-7b
CAS :<p>GEBR-7b (3-(Cyclopentyloxy)-4-methoxybenzaldehyde) is a phosphodiesterase-4 (PDE4) inhibitor.</p>Formule :C13H16O3Degré de pureté :99.533%Couleur et forme :SolidMasse moléculaire :220.26α-Amylase
CAS :<p>α-Amylase, a hydrolase enzyme, catalyzes the hydrolysis of internal α-1,4-glycosidic linkages in starch, producing glucose and maltose.</p>Degré de pureté :98%Couleur et forme :SolidDeoxyshikonin
CAS :<p>1.</p>Formule :C16H16O4Degré de pureté :99.36% - ≥95%Couleur et forme :SolidMasse moléculaire :272.3Ro 61-8048
CAS :Ro 61-8048 is a potent and selective inhibitor of kynurenine hydroxylase with an IC50 value of 37 nM.Formule :C17H15N3O6S2Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :421.45palovarotene
CAS :<p>Palovarotene (Ro 3300074) is an agonist of nuclear retinoic acid receptor γ (RAR-γ).</p>Formule :C27H30N2O2Degré de pureté :97.88% - 98.05%Couleur et forme :SolidMasse moléculaire :414.54Sapropterin dihydrochloride
CAS :Sapropterin dihydrochloride (6R-BH4 dihydrochloride) is phenylalanine hydroxylase agonist that is approved for the treatment of BH4 responsive PKU.Formule :C9H17Cl2N5O3Degré de pureté :98% - 99.88%Couleur et forme :White Crystalline SolidMasse moléculaire :314.17Malotilate
CAS :<p>Malotilate (Kantec) is a medicine used for the therapy of liver cirrhosis.</p>Formule :C12H16O4S2Degré de pureté :99.79% - 99.79%Couleur et forme :SolidMasse moléculaire :288.38GW4869
CAS :<p>GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).</p>Formule :C30H30Cl2N6O2Degré de pureté :98.12% - 98.47%Couleur et forme :SolidMasse moléculaire :577.5NSC 65809
CAS :<p>NSC-65809 (Raphin1) is a selective inhibitor of R15B.</p>Formule :C8H8Cl2N4Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :231.08FT113
CAS :<p>FT113 is a novel potent inhibitor of fatty acid synthase (fasn, IC50 : 213 nM),and exhibits anti-cancer activity</p>Formule :C22H20FN3O4Degré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :409.41Anacetrapib
CAS :<p>Anacetrapib (MK-0859) inhibits rhCETP/CETP(C13S) (IC50: 7.9/11.8 nM), boosts HDL, lowers LDL cholesterol.</p>Formule :C30H25F10NO3Degré de pureté :98.40% - 99.87%Couleur et forme :SolidMasse moléculaire :637.51Anti-Inflammatory Peptide 1 Acetate
<p>Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.</p>Formule :C47H86N12O16S2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :1139.39LDHA-IN-4
CAS :<p>LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.</p>Formule :C25H27N3O6SDegré de pureté :98.17% - 99.68%Couleur et forme :SolidMasse moléculaire :497.56H2S Donor 5a
CAS :<p>H2S Donor 5a is a H2S donor that could mimic the slow and continuous H(2)S generation process.</p>Formule :C14H11NO2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :257.31Indisulam
CAS :<p>Indisulam (E 7070) is a dual-action anticancer drug, blocking G1/S cell cycle transition by degrading cyclin E and activating p53/p21.</p>Formule :C14H12ClN3O4S2Degré de pureté :98.68% - 99.77%Couleur et forme :SolidMasse moléculaire :385.85(E,E)-RAMB4
CAS :<p>PTP1B-IN-8 is a potent and selective inhibitor of protein tyrosine phosphatase-1B (PTP1B).</p>Formule :C19H13Cl4NODegré de pureté :96.03%Couleur et forme :SolidMasse moléculaire :413.12Levamlodipine besylate
CAS :<p>Levamlodipine besylate, or S-amlodipine (CAS 103129-82-4), is the active enantiomer of amlodipine, used to treat hypertension and angina.</p>Formule :C26H31ClN2O8SDegré de pureté :99.78% - 99.79%Couleur et forme :SolidMasse moléculaire :567.05Ziconotide Acetate (107452-89-1 free base)
CAS :<p>Ziconotide Acetate (Prialt, 107452-89-1) is an analgesic for neuropathic pain, acting on N-type calcium channels to block pain signals.</p>Formule :C102H172N36O32S7Degré de pureté :99.52% - 99.87%Couleur et forme :SolidMasse moléculaire :2639.2Bay K 8644
CAS :<p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>Formule :C16H15F3N2O4Degré de pureté :99.41%Couleur et forme :Yellow PowderMasse moléculaire :356.3PHD-1-IN-1
CAS :PHD-1-IN-1 is a potent inhibitor of hypoxia-inducible factor prolylhydroxylase domain-1 (PHD-1) enzyme(IC50 = 0.034 μM).Formule :C13H8N4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :220.23Fabomotizole hydrochloride
CAS :<p>Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。</p>Formule :C15H22ClN3O2SDegré de pureté :99.54% - >99.99%Couleur et forme :SolidMasse moléculaire :343.87Pyridaben
CAS :<p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>Formule :C19H25ClN2OSDegré de pureté :97.11% - 99.75%Couleur et forme :SolidMasse moléculaire :364.93Betrixaban hydrochloride(330942-05-7(free base))
<p>Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5</p>Formule :C23H23Cl2N5O3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :488.36VY-3-135
CAS :<p>VY-3-135 is an orally active, stable and specific acetyl-CoA synthetase 2 (ACSS2) inhibitor.Cost-effective and quality-assured.</p>Formule :C26H27N3O3Degré de pureté :99.25% - 99.79%Couleur et forme :SolidMasse moléculaire :429.51A939572
CAS :<p>A939572 is stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of <4 nM for mSCD1 and 37 nM for hSCD1.</p>Formule :C20H22ClN3O3Degré de pureté :99.96% - ≥95%Couleur et forme :SolidMasse moléculaire :387.86Verdiperstat
CAS :Verdiperstat (AZD 3241) is a selective, irreversible, orally active myeloperoxidase inhibitor for neurodegenerative brain diseases.Formule :C11H15N3O2SDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :253.32GW3965 hydrochloride
CAS :<p>GW3965 hydrochloride (GW3965 HCl) is an effective and specific LXR agonist for hLXRα/β (EC50: 190/30 nM).</p>Formule :C33H31ClF3NO3·HClDegré de pureté :98.9% - 99.51%Couleur et forme :SolidMasse moléculaire :618.51YM976
CAS :YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)Formule :C17H16ClN3ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :313.78L-Homocystine
CAS :<p>Homocystine briefly forms before turning into cystathionine via vitamin B6; linked to schizophrenia and neural tube defects; folic acid lowers risk.</p>Formule :C8H16N2O4S2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :268.35UK-5099
CAS :<p>UK-5099 (PF-1005023) is a potent MPC inhibitor with an IC50 of 50 nM in rat heart mitochondria.</p>Formule :C18H12N2O2Degré de pureté :97.39% - >99.99%Couleur et forme :SolidMasse moléculaire :288.3TEPP-46
CAS :<p>TEPP-46 (ML265) is an activator of pyruvate kinase M2 (PKM2), selective for PKM1, PKL and PKR. TEPP-46 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C17H16N4O2S2Degré de pureté :98.21% - 98.77%Couleur et forme :SolidMasse moléculaire :372.46(R)-3-Hydroxy-4,4-dimethyldihydrofuran-2(3H)-one
CAS :<p>Pantolactone belongs to the class of organic compounds known as gamma-butyrolactones. gamma-Butyrolactones are compounds containing a gamma-butyrolactone moiety, which consists of an aliphatic five-member ring with four carbon atoms, one oxygen atom, and </p>Formule :C6H10O3Degré de pureté :99.41%Couleur et forme :White Crystalline Powder Or CrystalsMasse moléculaire :130.14Nepicastat hydrochloride
CAS :<p>Nepicastat hydrochloride (RS-25560-197 hydrochloride) is a selective, orally active, dopamine-beta-hydroxylase inhibitor that crosses the blood-brain barrier.</p>Formule :C14H15F2N3S·HClDegré de pureté :98.35% - 99.74%Couleur et forme :SolidMasse moléculaire :331.81ML-095 hydrochloride
CAS :ML-095 hydrochloride (CID-25067483 hydrochloride) is a specific placental alkaline phosphatase inhibitor.Formule :C13H15ClN2O3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :282.72Biocytin
CAS :<p>Biocytin, a D-biotin and L-lysine conjugate, maps brain connections via a secondary amide bond.</p>Formule :C16H28N4O4SDegré de pureté :97.23%Couleur et forme :White SolidMasse moléculaire :372.48Cilostamide
CAS :<p>Cilostamide (OPC3689) is a selective phosphodiesterase (PDE)3A and PDE3B inhibitor(IC50 values of 27 and 50 nM, respectively)</p>Formule :C20H26N2O3Degré de pureté :98.87%Couleur et forme :White To Off-White SolidMasse moléculaire :342.43Captopril hydrochloride
CAS :<p>Captopril hydrochloride: an oral ACE inhibitor (IC50: 0.025 μM), treats hypertension/heart failure, and blocks NDM-1 (IC50: 7.9 μM).</p>Formule :C9H16ClNO3SCouleur et forme :SolidMasse moléculaire :253.74Hexacosanoic acid
CAS :Hexacosanoic acid, a very long-chain fatty acid, is related to adrenoleukodystrophy (ALD), adrenomyeloneuropathy (AMN) and atherosclerosis.Formule :C26H52O2Degré de pureté :99.41% - ≥95%Couleur et forme :SolidMasse moléculaire :396.69FIPI
CAS :<p>FIPI, a halopemide derivative, strongly blocks PLD1 and PLD2 (IC50s: 25 nM, 20 nM) and hinders PLD-mediated cell activity.</p>Formule :C23H24FN5O2Degré de pureté :97.21% - 98.68%Couleur et forme :SolidMasse moléculaire :421.474-Hydroxyquinoline
CAS :<p>4-Hydroxyquinoline, aka 4-Quinolinol, is a quinoline with antimicrobial properties, inhibiting gut bacteria, and scavenges photogenerated oxygen species.</p>Formule :C9H7NODegré de pureté :97.50%Couleur et forme :Light Yellow And Off-White Crystal PowderMasse moléculaire :145.16Nicotinamide riboside chloride
CAS :<p>NR, also SRT647, is a B3 vitamin form; precursor to NAD+.</p>Formule :C11H15ClN2O5Degré de pureté :98.92% - 99.86%Couleur et forme :SolidMasse moléculaire :290.7Fmoc-Phe(4-CN)-OH
CAS :<p>Fmoc-Phe(4-CN)-OH is an N-Fmoc protected phenylalanine derivative and potentially useful synthetic intermediate</p>Formule :C25H20N2O4Degré de pureté :99.45%Couleur et forme :White PowderMasse moléculaire :412.44Safinamide mesylate
CAS :<p>Safinamide mesylate (EMD 1195686 mesylate) , a mesylate salt of Safinamide, can reversibly and specifically inhibit MAO-B (IC50: 98 nM), has 5918-fold</p>Formule :C18H23FN2O5SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :398.45Doxercalciferol
CAS :<p>Doxercalciferol, a synthetic vitamin D2, curbs parathyroid activity for treating secondary hyperparathyroidism and bone disorders.</p>Formule :C28H44O2Degré de pureté :99.03% - 99.69%Couleur et forme :White Crystalline PowderMasse moléculaire :412.65URB937
CAS :<p>URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).</p>Formule :C20H22N2O4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :354.4SEA0400
CAS :<p>SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.</p>Formule :C21H19F2NO3Degré de pureté :98.88% - 99.55%Couleur et forme :SolidMasse moléculaire :371.38Oxaceprol
CAS :<p>Oxaceprol (N-Acetyl-L-hydroxyproline) is an established therapeutic agent for osteoarthritis.</p>Formule :C7H11NO4Degré de pureté :99.21%Couleur et forme :White Fine CrystalsMasse moléculaire :173.17N-Benzyllinoleamide
CAS :<p>N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) is a natural product isolated from Lepidium meyenii Walp, has pharmaceutical property against</p>Formule :C25H39NODegré de pureté :95%Couleur et forme :SolidMasse moléculaire :369.58TAK-700
CAS :<p>TAK-700 (Orteronel) is a selective 17, 20-lyase inhibitor, IC50 38 nM, with >1000x specificity vs other CYPs. Phase 3.</p>Formule :C18H17N3O2Degré de pureté :97.26%Couleur et forme :SolidMasse moléculaire :307.35N-Biotinyl-6-aminohexanoic acid
CAS :<p>N-Biotinyl-6-aminohexanoic acid (N-(+)-Biotinyl-6-aminohexanoic acid) can be used to perform N-terminal biotinylation.</p>Formule :C16H27N3O4SDegré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :357.47Sildenafil Mesylate
CAS :<p>Sildenafil Mesylate is a mesylate form of Sildenafil, an inhibitor of Phosphodiesterase 5.</p>Formule :C22H30N6O4S·xCH4O3SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :570.68ML-298
CAS :<p>ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).</p>Formule :C22H23F3N4O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :432.44GSK 2830371
CAS :<p>GSK 2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.</p>Formule :C23H29ClN4O2SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :461.02Antimalarial agent 14
CAS :<p>Antimalarial agent 14 (NSC-102533) is a bioactive chemical.</p>Formule :C16H10O3Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :250.251H-1-ethyl Candesartan Cilexetil
CAS :1H-1-ethyl Candesartan Cilexetil is an impurity in candesartan bulk synthesis, a strong, lasting AT1 blocker.Formule :C35H38N6O6Degré de pureté :98.19%Couleur et forme :SolidMasse moléculaire :638.71BSBM7
CAS :<p>BSBM7 is an inhibitor of Aβ aggregation and neuronal toxicity.</p>Formule :C22H24N2O8S2Degré de pureté :97.27%Couleur et forme :SolidMasse moléculaire :508.56Furagin
CAS :<p>Furagin (Furazidine) is a Nitrofuran derivative with anti-infective activity used for urinary tract infections.</p>Formule :C10H8N4O5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :264.19Ethionine
CAS :<p>Ethionine (NSC-82393) is an antimetabolite and methionine antagonist. It also produces liver neoplasms.</p>Formule :C6H13NO2SDegré de pureté :99.28% - ≥95%Couleur et forme :Crystals White SolidMasse moléculaire :163.24Guanoclor
CAS :<p>Guanoclor (VATENSOL) (INN), also known as guanochlor, is a sympatholytic drug. It is known to bind to non-adrenergic sites in pig kidney membranes.</p>Formule :C9H12Cl2N4ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :263.12PDE4-IN-20
CAS :<p>EAPT, a selective PDE4 inhibitor, controls cAMP levels and has potential for treating inflammatory diseases.</p>Formule :C13H12F3N3O2Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :299.25Nicosulfuron
CAS :<p>Nicosulfuron is a non-mutagenic herbicide that protects corn by blocking acetolactate synthase.</p>Formule :C15H18N6O6SDegré de pureté :97.16%Couleur et forme :White SolidMasse moléculaire :410.40Ezutromid
CAS :<p>Ezutromid (BMN 195) upregulates utrophin gene, enhancing muscle function in MDX mice. EC50: 0.4 uM, orally bioavailable.</p>Formule :C19H15NO3SDegré de pureté :97.57% - 99.76%Couleur et forme :SolidMasse moléculaire :337.39Fmoc-N-Me-Leu-OH
CAS :Fmoc-N-Me-Leu-OH is available for the peptide-coupling reaction.Formule :C22H25NO4Degré de pureté :99.51%Couleur et forme :White PowderMasse moléculaire :367.444-Methylumbelliferyl-β-D-Glucopyranoside
CAS :<p>4-Methylumbelliferyl-β-D-Glucopyranoside (4-MU-GLU) is used in the GCase activity assay based on the catalytic hydrolysis of 4-methylumbelliferyl β-D-</p>Formule :C16H18O8Degré de pureté :99.89%Couleur et forme :White PowderMasse moléculaire :338.31BMS-823778 hydrochloride
CAS :<p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>Formule :C18H19Cl2N3OCouleur et forme :SolidMasse moléculaire :364.27β-Nicotyrine
CAS :<p>beta-Nicotyrine is a tobacco alkaloids Metabolite in the liver.</p>Formule :C10H10N2Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :158.2Turofexorate Isopropyl
CAS :<p>Turofexorate Isopropyl (XL335) is a potent, selective, and orally bioavailable FXR agonist with EC50 of 4 nM</p>Formule :C25H24F2N2O3Degré de pureté :98.55% - 99.73%Couleur et forme :SolidMasse moléculaire :438.47Carbamazepine 10,11-epoxide
CAS :<p>Carbamazepine 10,11-epoxide, an active metabolite with anticonvulsant properties, is created by CYP3A4 and CYP2C8.</p>Formule :C15H12N2O2Degré de pureté :98.64% - 99.75%Couleur et forme :SolidMasse moléculaire :252.27Z-Glycine
CAS :N-Benzyloxycarbonylglycine is a lipid-like drug designed for enhanced brain penetration.Formule :C10H11NO4Degré de pureté :99.88%Couleur et forme :Slightly Beige PowderMasse moléculaire :209.27-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS :<p>7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).</p>Formule :C15H16N4Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :252.31Chondroitine sulfate
CAS :<p>Chondroitin sulfate is an important structural component of cartilage and has been used as a dietary supplement for the treatment of joint discomfort.</p>Formule :C13H21NO15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :463.36Hydramethylnon
CAS :<p>Hydramethylnon (AC217300) is an insecticide primarily. Hydramethylnon is used for fire ants.</p>Formule :C25H24F6N4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :494.48RO6889678
CAS :RO6889678 is HBV inhibitor with a complex ADME profile.Formule :C21H20ClFN4O5SDegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :494.92Xanthine dehydrogenase Inhibitor 1
CAS :5-Amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile is an enzyme inhibitor with antitumor, anti-inflammatory, and antioxidant properties.Formule :C11H7F3N4Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :252.2HET0016
CAS :<p>HET0016: potent, selective 20-HETE synthase/CYP450 inhibitor; IC50s: 17.7-20.6 nM; inhibits angiogenesis, tumor growth.</p>Formule :C12H18N2ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :206.28N-desmethylmirtazapine
CAS :N-desmethylmirtazapine: mirtazapine metabolite; used for anxiety, sleep, nausea, appetite.Formule :C16H17N3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :251.33CD00509
CAS :<p>CD00509 is a tyrosyl-DNA phosphodiesterase inhibitor.</p>Formule :C9H6N2O3SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :222.22Kyotorphin acetate
<p>Kyotorphin acetate is an endogenous peptide with analgesia activity and can be used as a biomarker of Alzheimer disease.</p>Formule :C17H27N5O6Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :397.43Anecortave Acetate
CAS :<p>Anecortave Acetate (NSC-24345), an angiostatic steroid, is used for proteomics research.</p>Formule :C23H30O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :386.48W 36017
CAS :W36017 is an impurity of lidocaine with a PKA of 7.4 for blocking neurologic activity.Formule :C12H18N2ODegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :206.28BISMUTH SUBGALLATE
CAS :<p>Bismuth subgallate (Dermatol Puder) is an astringent and antiseptic and is applied to skin diseases such as eczema.</p>Formule :C7H5BiO6Degré de pureté :98.7%Couleur et forme :White To Yellow CrystalsMasse moléculaire :394.09Teriflunomide
CAS :<p>Teriflunomide (A 77-1726) is the principal active metabolite of leflunomide, an approved therapy for rheumatoid arthritis and multiple sclerosis.</p>Formule :C12H9F3N2O2Degré de pureté :99.54% - 99.95%Couleur et forme :SolidMasse moléculaire :270.21Jalapinolic acid
CAS :<p>Jalapinolic acid (Builic Acid) is a hydroxypalmitic acid.</p>Formule :C16H32O3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :272.42L-Cysteinesulfinic acid monohydrate
CAS :<p>L-Cysteinesulfinic acid monohydrate activates rat mGluR1/2/4/5/6/8 with pEC50s of 3.92, 3.9, 2.7, 4.6, 4.0, 3.94 respectively.</p>Formule :C3H9NO5SDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :171.17S18-000003
CAS :<p>S18-000003: Oral retinoic acid receptor gamma-t inhibitor, IC50 29 nM, reduces IL-17 production.</p>Formule :C26H25F3N2O4SDegré de pureté :99.24% - 99.31%Couleur et forme :SolidMasse moléculaire :518.55GNE-617 hydrochloride
CAS :<p>GNE-617 hydrochloride is a specific inhibitor of NAMPT and inhibits NAMPT activity (IC50: 5 nM).</p>Formule :C21H16ClF2N3O3SCouleur et forme :SolidMasse moléculaire :463.88(S)-Mephenytoin
CAS :<p>(S)-Mephenytoin: (+)-enantiomer, anticonvulsant, CYP2C19 substrate for analyzing CYP450 metabolism.</p>Formule :C12H14N2O2Degré de pureté :98.73% - 99.82%Couleur et forme :SolidMasse moléculaire :218.25GN44028
CAS :<p>GN44028 is a HIF-1 inhibitor with an IC50 of 14 nM, stopping HIF-1α activity but not mRNA or protein levels, or dimerization.</p>Formule :C18H15N3O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :305.334-Oxoisotretinoin
CAS :4-Oxoisotretinoin (Ro 22-6595) is the major blood metabolite.Formule :C20H26O3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :314.42H-L-Lys(Poc)-OH HCl
CAS :<p>N-ε-propargyloxycarbonyl-L-lysine hydrochloride (N6-((Prop-2-yn-1-yloxy)carbonyl)-L-lysine hydrochloride) is a modified amino acid for cancer therapy</p>Formule :C10H17ClN2O4Degré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :264.71OGT-IN-2
CAS :<p>OGT-IN-2: Potent OGT inhibitor, IC50: sOGT 30μM, ncOGT 53μM, for articular disease research.</p>Formule :C23H27ClN2O3SDegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :446.99SR1664
CAS :<p>SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity.</p>Formule :C33H29N3O5Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :547.6Eflornithine hydrochloride hydrate
CAS :Eflornithine hydrochloride hydrate (DFMO hydrochloride hydrate) is an ornithine decarboxylase (ODC) inhibitor with antitumor activity. Cost-effective and quality-assured.Formule :C6H15ClF2N2O3Degré de pureté :99% - 99.61%Couleur et forme :White SolidMasse moléculaire :236.64DIPQUO
CAS :<p>DIPQUO activates ALP and osteoblasts via p38MAPK-β; EC50 in C2C12 cells is 6.27 μM.</p>Formule :C20H17N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.37Celgosivir hydrochloride
CAS :<p>Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).</p>Formule :C12H22ClNO5Couleur et forme :SolidMasse moléculaire :295.76Umbralisib hydrochloride
CAS :<p>Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.</p>Formule :C31H25ClF3N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :608.01Inulin
CAS :<p>Inulin(Inulin and sodium chloride), a starch found in the tubers and roots of many plants.</p>Formule :C6nH10nO5nDegré de pureté :99% - ≥95%Couleur et forme :White PowderMasse moléculaire :490.411RS-25344 hydrochloride
CAS :<p>RS 25344 hydrochloride is a phosphodiesterase (PDE) 4 inhibitor</p>Formule :C19H14ClN5O4Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :411.8WWL229
CAS :<p>WWL229 selectively inhibits Ces3 without affecting Ces1f, ABHD6, or other serine hydrolases, mimicking WWL113 in adipocytes.</p>Formule :C16H22N2O5Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :322.36
