Métabolisme

Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.

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9007 produits trouvés pour "Métabolisme"

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FCPR03
CAS :
- 1917347-65-9
FCPR03 is a selective inhibitor of phosphodiesterase 4 (PDE4) with IC50s of 31 nM, 47 nM, and 60 nM for PDE4B1, PDE4D7, and PDE4 catalytic domain, respectively.
Formule :C₁₅H₁₉F₂NO₃
Degré de pureté :99.94%
Couleur et forme :Solid
Masse moléculaire :299.31
Ref: TM-T39341
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IPI-9119
CAS :
- 1346564-56-4
IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).
Formule :C₂₄H₁₉F₂N₅O₅
Degré de pureté :99.81%
Couleur et forme :Solid
Masse moléculaire :495.43
Ref: TM-T36841
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ACSS2-IN-2
CAS :
- 2332820-04-7
MTB-9655 inhibits ACSS2 with 3.8 nM IC50, useful in research of viral, metabolic, neuropsychiatric diseases, inflammation, and cancer.
Formule :C₂₁H₁₉F₂N₃O₄
Degré de pureté :99.5%
Couleur et forme :Soild
Masse moléculaire :415.39
Ref: TM-T60060
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L-Hisidine monohydrocholoride
CAS :
- 645-35-2
L-Hisidine is an essential amino acid for infants and acts as an inhibitor of mitochondrial glutamine transport.
Formule :C₆H₁₀ClN₃O₂
Couleur et forme :Solid
Masse moléculaire :191.62
Ref: TM-TN8219
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α-Glucosidase-IN-87
α-Glucosidase-IN-87 (Compound 11c) is an orally active inhibitor of α-glucosidase with an IC50 of 119.7 μM. It exhibits hypoglycemic properties and is applicable in research on metabolic diseases such as diabetes.
Couleur et forme :Odour Solid
Ref: TM-T206086
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BC 11-38
CAS :
- 686770-80-9
BC 11-38 is a potent, selective PDE biodepressant which is mainly effective against PDE11 (IC50 : 0.28 μM).
Formule :C₁₅H₁₆N₂OS₂
Degré de pureté :98.95% - 99.28%
Couleur et forme :Solid
Masse moléculaire :304.43
Ref: TM-T21865
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α-glucosidase/PTP1B-IN-1
α-glucosidase/PTP1B-IN-1 (compound 8a) is an effective inhibitor of both α-glucosidase and PTP1B, with IC50 values of 66.3 μM and 47.0 μM, respectively. It also exhibits strong inhibitory activity against α-amylase, having an IC50 of 30.62 μM. This compound is capable of binding to the active sites of α-glucosidase and PTP1B. α-glucosidase/PTP1B-IN-1 holds potential for reducing postprandial blood glucose levels and may be useful in managing type 2 diabetes.
Formule :C₂₃H₂₀Cl₂O₅
Couleur et forme :Solid
Masse moléculaire :447.31
Ref: TM-T201678
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Myristelaidic Acid
CAS :
- 50286-30-1
Myristelaidic Acid is a natural product for research related to life sciences. The catalog number is T37358 and the CAS number is 50286-30-1.
Formule :C₁₄H₂₆O₂
Couleur et forme :Solid
Masse moléculaire :226.35
Ref: TM-T37358
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Vardenafil dihydrochloride
CAS :
- 224789-15-5
Vardenafil dihydrochloride (Levitra) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.
Formule :C₂₃H₃₄Cl₂N₆O₄S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :561.52
Ref: TM-T4480
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SR-4995
CAS :
- 891509-95-8
SR-4995 (CID 16016685) is an ABHD5 ligand, directly binding to ABHD5 and stimulating lipolysis by releasing it from PLIN.
Formule :C₁₉H₂₁N₃O₂S
Couleur et forme :Soild
Masse moléculaire :355.45
Ref: TM-T200801
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Lalistat 2
CAS :
- 1234569-09-5
Lalistat 2: selective lysosomal acid lipase inhibitor, IC50 152 nM, no effect on pancreatic/milk lipase <10 μM.
Formule :C₁₃H₂₀N₄O₂S
Degré de pureté :99.84%
Couleur et forme :Solid
Masse moléculaire :296.39
Ref: TM-T41160
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1-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine
CAS :
- 76343-22-1
Endogenous metabolite: 1-myristoyl-2-stearoyl-sn-glycero-3-phosphocholine, a phosphatidylcholine example.
Formule :C₄₀H₈₀NO₈P
Degré de pureté :99.23%
Couleur et forme :Solid
Masse moléculaire :734.04
Ref: TM-T10022
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(Ile8)-Oxytocin acetate
(Ile8)-Oxytocin acetate is a neurohypophysial hormone analog of oxytocin produced in marsupials.
Formule :C₄₅H₇₀N₁₂O₁₄S₂
Couleur et forme :Solid
Masse moléculaire :1067.24
Ref: TM-TP2929
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(rac./meso)-Astaxanthin
CAS :
- 7542-45-2
(rac./meso)-Astaxanthin (AstaREAL; AstaXin) is a carotenoid pigment primarily found in marine animals such as shrimp and salmon. It serves as an effective fat-soluble antioxidant.
Formule :C₄₀H₅₂O₄
Couleur et forme :Solid
Masse moléculaire :596.84
Ref: TM-TN8210
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2,4-Dimethylquinoline
CAS :
- 1198-37-4
2,4-Dimethylquinoline is a potential CYP1A2 inhibitor , and it also exhibits weak inhibitory activity against CYP2A5, CYP2A6, and CYP2B6.
Formule :C₁₁H₁₁N
Degré de pureté :99.81%
Couleur et forme :Solid
Masse moléculaire :157.21
Ref: TM-TN9268
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H-Pro-Phe-OH
CAS :
- 13589-02-1
H-Pro-Phe-OH is a dipeptide formed from proline and phenylalanine, serving as a substrate for prolylase and in peptide synthesis.
Formule :C₁₄H₁₈N₂O₃
Couleur et forme :Solid
Masse moléculaire :262.30
Ref: TM-T76613
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IETP2
CAS :
- 2314338-36-6
IETP2 targets low-density lipoprotein receptor-related protein 1 (LRP1) with a KD of 738 nM, making it useful for delivering drugs and imaging agents across the blood-labyrinth barrier (BLB).
Formule :C₁₀₇H₁₇₁N₃₉O₂₉
Couleur et forme :Solid
Masse moléculaire :2467.75
Ref: TM-TP3115
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α-Glucosidase-IN-32
α-Glucosidase-IN-32 (compound f26) is a reversible, noncompetitive inhibitor of α-glucosidase that is orally active and exhibits an IC50 of 3.07 μM.
Formule :C₃₂H₂₂N₄OS
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :510.61
Ref: TM-T79700
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BAY-277
BAY-277 is a degrader of METAP2, with IC50 values of 5.8 nM for human METAP2 (hMETAP2) and 5.9 nM for mouse METAP2 (mMETAP2).
Formule :C₄₄H₅₂N₈O₅
Couleur et forme :Solid
Masse moléculaire :772.93
Ref: TM-T205262
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Vitamin K5
CAS :
- 83-70-5
Vitamin K5, a photosensitizer & antimicrobial, inhibits PKM2, PKM1 & PKL, induces apoptosis in colon cells, and preserves food & medicine.
Formule :C₁₁H₁₁NO
Couleur et forme :Solid
Masse moléculaire :173.21
Ref: TM-T75317
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NGR peptide
CAS :
- 651328-78-8
Cell-penetrating peptide
Formule :C₂₀H₃₆N₁₀O₈S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :608.69
Ref: TM-TP2185
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Isobutyl Butyrate
CAS :
- 539-90-2
Isobutyl Butyrate is a butyrate ester formed by the condensation of butyric acid with isobutyl alcohol, which is a metabolite of rifampicin.
Formule :C₈H₁₆O₂
Degré de pureté :99.58%
Couleur et forme :Solid
Masse moléculaire :144.21
Ref: TM-T203881
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O-Demethyl Lenvatinib
CAS :
- 417717-04-5
O-Demethyl Lenvatinib, a Lenvatinib metabolite, is an oral TKI targeting VEGFR, FGFR, PDGFR, KIT & RET with potent antitumor effects.
Formule :C₂₀H₁₇ClN₄O₄
Couleur et forme :Solid
Masse moléculaire :412.83
Ref: TM-T74020
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DSPE-PEG1000-ESBP
DSPE-PEG1000-ESBP is a PEG compound composed of DSPE and an E-selectin binding peptide (ESBP). As a tumor-targeting peptide, ESBP can specifically recognize and bind to receptors or markers on the surface of tumor cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01151
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ZD-2138
CAS :
- 140841-32-3
ZD-2138: Selective 5-LOX inhibitor, eases allergen-induced asthma attacks and airway constriction in guinea pigs.
Formule :C₂₃H₂₄FNO₄
Degré de pureté :99.68% - >99.99%
Couleur et forme :Solid
Masse moléculaire :397.44
Ref: TM-T68173
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2-oxo Clopidogrel
CAS :
- 109904-27-0
2-oxo Clopidogrel SR-121683 is a metabolite of Clopidogrel,catalyzed by P450 enzyme via CYP3A oxidation, ydrolysis to the active metabolite CAM.antithrombotic.
Formule :C₁₆H₁₆ClNO₃S
Couleur et forme :Solid
Masse moléculaire :337.82
Ref: TM-T36222
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Chlorothiazide
CAS :
- 58-94-6
Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.
Formule :C₇H₆ClN₃O₄S₂
Degré de pureté :98.46% - 98.91%
Couleur et forme :Crystals Physical Description Crystals; White Powder (Ntp 1992)
Masse moléculaire :295.72
Ref: TM-T0677
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Acetoacetic acid
CAS :
- 541-50-4
Acetoacetic acid(3-oxobutanoic acid) is a oxidative stress inducer, gluconeogenesis, and can be used as an indicator of in ketoacidosis.
Formule :C₄H₆O₃
Degré de pureté :99.59% - 99.85%
Couleur et forme :Solid
Masse moléculaire :102.09
Ref: TM-T73734
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α-Glucosidase-IN-42
α-Glucosidase-IN-42 (Compound 26), a 9-O-berberrubine carboxylate derivative, exhibits potent α-glucosidase inhibitory activity with an IC50 value of 1.61 μM
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T80708
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CALP3 TFA(261969-05-5 free base)
CALP3 TFA is a potent Ca2+ channel blocker that activates EF-hand motifs of Ca2+-binding proteins.
Formule :C₄₆H₆₉F₃N₁₀O₁₁
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :995.1
Ref: TM-TP2170
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2-Methylnicotinamide
CAS :
- 58539-65-4
2-Methylnicotinamide is an endogenous metabolite of nicotinamide and can be used for related research in the life sciences.
Formule :C₇H₈N₂O
Degré de pureté :99.84%
Couleur et forme :Solid
Masse moléculaire :136.15
Ref: TM-TN9444
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BVT-2733 hydrochloride
CAS :
- 376641-65-5
BVT-2733 hydrochloride is a potent, selective, and orally active non-steroidal 11β-HSD1 inhibitor. It exhibits stronger inhibition on mouse 11β-HSD1 enzyme (IC50=96 nM) compared to the human 11β-HSD1 enzyme (IC50=3341 nM). BVT-2733 hydrochloride shows potential for research in arthritis and obesity-related diseases.
Formule :C₁₇H₂₂Cl₂N₄O₃S₂
Couleur et forme :Solid
Masse moléculaire :465.42
Ref: TM-T203621
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FABP4-IN-4
FABP4-IN-4 (Compound 30) is an orally effective inhibitor of FABP, with an IC50 value of 1.18 μM against FABP1. In a mouse model of diet-induced obesity, FABP4-IN-4 improves glucose tolerance, reduces levels of blood sugar, lipids, and liver inflammation markers, alleviates hepatic steatosis, and exhibits anti-inflammatory activity.
Couleur et forme :Odour Solid
Ref: TM-T89572
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Octapeptide-2
CAS :
- 1374396-34-5
Octapeptide-2 is a bioactive peptide known for its hair growth-promoting effects and is reported to be used as a cosmetic ingredient [1].
Formule :C₃₈H₆₀N₁₀O₁₆S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :945.01
Ref: TM-T80204
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PCSK9-IN-11
PCSK9-IN-11, an oral potent PCSK9 inhibitor; IC50=5.7μM in HepG2; boosts LDLR; for atherosclerosis study.
Formule :C₁₆H₁₇ClFN₅O₃
Degré de pureté :99.1%
Couleur et forme :Soild
Masse moléculaire :381.79
Ref: TM-T67776
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FABP4-IN-2
FABP4-IN-2 (Compd 10g), a selective and orally active FABP4 inhibitor, exhibits K i values of 0.51 μM for FABP4 and 33.01 μM for FABP3, demonstrating its
Formule :C₂₂H₁₄ClF₃O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :418.79
Ref: TM-T78960
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α-Amylase-IN-11
α-Amylase-IN-11 (compound C5f) is an α-amylase inhibitor with an IC50 of 0.56 μM, effective in reducing glucose levels in vivo. Additionally, it exhibits moderate inhibitory activity against α-glucosidase with an IC50 of 11.03 μM. In mouse models, α-Amylase-IN-11 significantly decreases glucose concentrations, indicating its potential for diabetes research.
Formule :C₂₂H₁₈N₄OS
Couleur et forme :Solid
Masse moléculaire :386.47
Ref: TM-T205363
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WAY-311610
CAS :
- 314051-55-3
WAY-311610 is an HSD11B1 inhibitor targeting 11β-HSD1 enzyme with 0.34 μM IC; used for neuropathic and inflammatory pain research.
Formule :C₁₆H₁₃F₃N₄O₂
Degré de pureté :99.75%
Couleur et forme :Solid
Masse moléculaire :350.3
Ref: TM-T77606
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α-Glucosidase-IN-33
α-Glucosidase-IN-33 (compound 7c), with an IC50 of 2.39 μM, is a potent inhibitor of α-glucosidase and is relevant in research on type 2 diabetes and
Formule :C₂₆H₁₉F₃N₂O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :480.44
Ref: TM-T78864
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γ-Glutamylserine TFA
γ-Glutamylserine TFA (γ-Glu-Ser TFA) serves as a calcium receptor activator and is utilized in research focused on Parkinson's disease, diabetes, and obesity [1
Formule :C₁₀H₁₅F₃N₂O₈
Degré de pureté :98%
Couleur et forme :Soild
Masse moléculaire :348.23
Ref: TM-T80681
+ Info
γ-Glu-Phe
CAS :
- 7432-24-8
γ-Glu-Phe (γ-Glutamylphenylalanine) is a γ-3 glutamyl dipeptide found in sourdough.it is synthesized by Bacillus amyloliquefaciens (GBA) and Aspergillus oryzae
Formule :C₁₄H₁₈N₂O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :294.3
Ref: TM-TP1001
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A4333
A4333, a biotinylated derivative of A3373, selectively inhibits Phospholipase D1 (PLD1) while sparing PLD2.
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T83225
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FS-2
FS-2 is a potent, specific inhibitor of L-type CaV channels, effectively impeding high K+ or glucose-induced L-type Ca2+ influx in RIN beta cells [1].
Formule :C₂₉₇H₄₆₂N₉₂O₈₆S₁₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :7018.06
Ref: TM-T80441
+ Info
WAY-620472
CAS :
- 686769-90-4
WAY-620472 is a PPAR regulator that can be used to alter the lifespan of eukaryotes.
Formule :C₂₃H₂₁N₅OS
Degré de pureté :98.07%
Couleur et forme :Solid
Masse moléculaire :415.51
Ref: TM-T77612
+ Info
ω-Hexatoxin-Hv1a
CAS :
- 193981-10-1
ω-Hexatoxin-Hv1a, a neurotoxin extracted from the venom of the spider Hadronyche versuta, inhibits voltage-gated calcium channels [1] [2].
Formule :C₁₆₂H₂₄₇N₄₉O₆₁S₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :4049.38
Ref: TM-T80160
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hCAI/II/IV-IN-28
CAS :
- 78659-11-7
hCAI/II/IV-IN-28(WAY-638358) is a potent carbonic anhydrase inhibitor with potential anticonvulsant activity.
Formule :C₁₄H₁₅N₃O₃S
Degré de pureté :96.48%
Couleur et forme :Solid
Masse moléculaire :305.35
Ref: TM-T80663
+ Info
DJ-53
DJ-53 (compound 68) is an orally active, phenyl-quinoline-based soluble epoxide hydrolase inhibitor.
Couleur et forme :Odour Solid
Ref: TM-T200655
+ Info
CBS-1114 HCl
CAS :
- 33244-00-7
CBS-1114 HCl: 5-lipoxygenase inhibitor, anti-inflammatory, improves heart function, reduces heart's fat.
Formule :C₁₃H₁₄ClN₃
Degré de pureté :99.93%
Couleur et forme :Soild
Masse moléculaire :247.72
Ref: TM-T68037L
+ Info
hCAIX-IN-19
hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/
Couleur et forme :Odour Solid
Ref: TM-T82234
+ Info
Histone acetyltransferase p300 Inhibitor 4c
CAS :
- 2103-99-3
2-Amino-4-(4-chlorophenyl)thiazole blocks hCA I/II, AChE, BChE with Ki: ~0.008, 0.124, 0.129, 0.083 µM.
Formule :C₉H₇ClN₂S
Degré de pureté :99.76%
Couleur et forme :Solid
Masse moléculaire :210.68
Ref: TM-T77560
+ Info
Galactosylhydroxylysine hydrochloride
Galactosylhydroxylysine hydrochloride, found in bone collagen, is higher in metabolic bone loss due to resorption.
Formule :C₁₂H₂₅ClN₂O₈
Couleur et forme :Solid
Masse moléculaire :360.79
Ref: TM-T73770
+ Info
Izilendustat
CAS :
- 1303512-02-8
Tert-butyl compound inhibits human EGLN-1; confirmed by spectrometry after 20 mins.
Formule :C₂₂H₂₈ClN₃O₄
Degré de pureté :99.95%
Couleur et forme :Solid
Masse moléculaire :433.93
Ref: TM-T64336
+ Info
1α, 24, 25-Trihydroxy VD2
CAS :
- 457048-34-9
1alpha, 24, 25-Trihydroxy VD2 is a vitamin D analog.
Formule :C₂₈H₄₄O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :444.65
Ref: TM-T19090
+ Info
E 6080 HCl
CAS :
- 120164-49-0
E 6080 HCl is a 5-lipoxygenase inhibitor and can be used to study bronchial diseases.
Formule :C₁₇H₂₀ClN₃O₃S₂
Degré de pureté :99.80%
Couleur et forme :Soild
Masse moléculaire :413.94
Ref: TM-T10508L
+ Info
CJ-13,610 hydrochloride
CAS :
- 179420-27-0
CJ-13,610 hydrochloride is an orally active nonredox-type inhibitor of 5-LOX and can be used in studies about the prevention of untoward pathophysiological
Formule :C₂₂H₂₄ClN₃O₂S
Degré de pureté :98.5%
Couleur et forme :Soild
Masse moléculaire :429.96
Ref: TM-T27026L
+ Info
EN3356
CAS :
- 1429329-63-4
EN3356 is an orally available and selective inhibitor of steroidal 17-alpha-hydroxylase/C17,20 cleavage enzyme (CYP17A1 or CYP17), a non-steroidal cleavage
Formule :C₁₆H₁₃FN₂OS
Degré de pureté :99.78%
Couleur et forme :Soild
Masse moléculaire :300.35
Ref: TM-T30161
+ Info
ROS-IN-2
ROS-IN-2 (compound 85), a seco-lupane triterpenoid derivative, inhibits reactive oxygen species (ROS) production and shields mitochondria from oxidative damage
Formule :C₄₂H₆₂ClNO₈S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :776.46
Ref: TM-T78887
+ Info
PROTAC PTPN2 degrader-2 TFA
CAS :
- 2912307-39-0
PROTAC PTPN2 degrader-2 (example 187B) TFA is a potent degrader of Protein Tyrosine Phosphatase Non-receptor Type 2 (PTPN2), with potential applications in
Formule :C₅₁H₅₀ClF₃N₆O₁₃S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :1111.55
Ref: TM-T79161
+ Info
DSPE-PEG1000-ANG
DSPE-PEG1000-ANG is a PEG compound composed of DSPE and a dual-targeting ligand (Angiopep-2, ANG). ANG demonstrates high LRP1 binding efficiency and has been utilized for targeting glioma delivery. DSPE-PEG1000-ANG is suitable for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01158
+ Info
MAGL-IN-10
MAGL-IN-10, a reversible monoacylglycerol lipase (MAGL) inhibitor, exhibits favorable ADME properties and low in vivo toxicity.
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T81881
+ Info
DSPE-PEG1000-CCK8
DSPE-PEG1000-CCK8 is a PEG compound composed of DSPE and Cholecystokinin-8 (CCK8). Cholecystokinin-8 exhibits peptide activity that regulates gallbladder contraction and the functions of the digestive system. DSPE-PEG1000-CCK8 can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01170
+ Info
DSPE-PEG5000-R9
DSPE-PEG5000-R9 is a PEG compound composed of DSPE and the polyarginine-9 peptide (R9) peptide, applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01086
+ Info
Ovotransferrin (328-332)
CAS :
- 1226776-54-0
Ovotransferrin (328-332), with an IC50 of 20 μM, exhibits protective activity against hypertension by inhibiting the Angiotensin-Converting Enzyme (ACE) and
Formule :C₂₅H₄₆N₈O₇
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :570.68
Ref: TM-T80100
+ Info
DSPE-PEG5000-RVG29
DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.
Couleur et forme :Odour Solid
Ref: TM-TCL-01074
+ Info
DSPE-PEG1000-R8
DSPE-PEG1000-R8 is a PEG compound composed of DSPE and the cell-penetrating peptide (R8). It is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01082
+ Info
DSPE-PEG2000-WYRGRL
DSPE-PEG2000-WYRGRL is a PEG compound composed of DSPE and the cartilage-targeting peptide (WYRGRL). The peptide WYRGRL can specifically bind to type II collagen α1. DSPE-PEG2000-WYRGRL is utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01128
+ Info
DSPE-PEG2000-EB1
DSPE-PEG2000-EB1 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (EB1). It is utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01126
+ Info
DSPE-PEG5000-KAA
DSPE-PEG5000-KAA is a PEG compound composed of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically targets the tumor vasculature of RIP-Tag2 transgenic mice. DSPE-PEG5000-KAA can be utilized for drug delivery purposes.
Couleur et forme :Odour Solid
Ref: TM-TCL-01116
+ Info
α-Glucosidase-IN-36
α-Glucosidase-IN-36 (compound 5g) is a potent inhibitor of α-glucosidase, exhibiting an IC50 value of 6.69 ± 0.18 μM and inhibition constants Ki and Kis of 1.65
Formule :C₂₆H₂₄BrN₅O₃S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :566.47
Ref: TM-T78881
+ Info
DSPE-PEG1000-R9
DSPE-PEG1000-R9 is a PEG compound composed of DSPE and the polyarginine-9 peptide (R9). It can be utilized in drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01190
+ Info
DSPE-PEG5000-THRPPMWSPVWP
DSPE-PEG5000-THRPPMWSPVWP is a PEG compound composed of DSPE and a transferrin receptor (TfR) peptide. The peptide sequence THRPPMWSPVWP binds to the TfR and is subsequently internalized into cells that express the receptor.
Couleur et forme :Odour Solid
Ref: TM-TCL-01110
+ Info
DSPE-PEG5000-CTT2
DSPE-PEG5000-CTT2 is a PEG compound composed of DSPE and the gelatinase inhibitor CTT2 (CTTHWGFTLC). CTT2 (CTTHWGFTLC) has the capability to specifically target tumors. DSPE-PEG5000-CTT2 is applicable for drug delivery purposes.
Couleur et forme :Odour Solid
Ref: TM-TCL-01089
+ Info
DSPE-PEG5000-CCK8
DSPE-PEG5000-CCK8 is a PEGylated compound comprised of DSPE and Cholecystokinin-8 (CCK8). Cholecystokinin-8 exhibits peptide activity that regulates gallbladder contraction and the functioning of the digestive system. DSPE-PEG5000-CCK8 can be applied in drug delivery systems.
Couleur et forme :Odour Solid
Ref: TM-TCL-01172
+ Info
Myoregulin TFA
Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics.
Formule :C₂₃₉H₃₉₁N₅₃O₆₇S₃·xC₂HF₃O₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :5175.17 (free base)
Ref: TM-T80555
+ Info
DSPE-PEG2000-TH
DSPE-PEG2000-TH is a PEG conjugate made from DSPE and a pH-responsive cell-penetrating peptide (TH). In acidic environments—such as the tumor microenvironment—TH becomes activated, allowing for the selective delivery of small molecules, oligonucleotides, and proteins into tumor cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01169
+ Info
DSPE-PEG1000-GRGDS
DSPE-PEG1000-GRGDS is a PEG compound composed of DSPE and the anti-adhesion peptide (GRGDS). GRGDS can inhibit the binding and adhesion between the extracellular matrix and cell surface integrins. The compound is useful for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01174
+ Info
DSPE-PEG5000-K237
DSPE-PEG5000-K237 is a PEG compound composed of DSPE and the KDR-targeting peptide (K237). K237 effectively disrupts the interaction between VEGF and KDR receptors, yielding significant biological effects, such as inhibiting angiogenesis and tumor growth. DSPE-PEG5000-K237 is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01168
+ Info
DSPE-PEG2000-THRPPMWSPVWP
DSPE-PEG2000-THRPPMWSPVWP is a PEG compound composed of DSPE and transferrin receptor (TfR) peptide. The sequence THRPPMWSPVWP binds to TfR and is subsequently internalized into cells expressing TfR.
Couleur et forme :Odour Solid
Ref: TM-TCL-01117
+ Info
DSPE-PEG1000-CTT2
DSPE-PEG1000-CTT2 is a PEG compound comprised of DSPE and a gelatinase inhibitor [CTT2 (CTTHWGFTLC)]. The CTT2 (CTTHWGFTLC) peptide is capable of specifically targeting tumors. DSPE-PEG1000-CTT2 can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01113
+ Info
DSPE-PEG5000-CGKRK
DSPE-PEG5000-CGKRK is a PEG compound composed of DSPE and the cell-penetrating peptide (CGKRK). It is utilized for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01124
+ Info
PTP Inhibitor IV
CAS :
- 329317-98-8
PTP Inhibitor IV selectively inhibits DUSP14 (IC50=5.21µM) and other PTPs, affecting cellular signaling.
Formule :C₂₆H₂₆F₆N₂O₄S₂
Degré de pureté :99.76%
Couleur et forme :Solid
Masse moléculaire :608.62
Ref: TM-T22137
+ Info
DSPE-PEG2000-GRGDS
DSPE-PEG2000-GRGDS is a PEG-based compound formed from DSPE and the anti-adhesion peptide (GRGDS). GRGDS serves to inhibit the binding and adhesion between the extracellular matrix and cell surface integrins. This compound is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01162
+ Info
DSPE-PEG2000-R9
DSPE-PEG2000-R9 is a PEG compound composed of DSPE and polyarginine-9 peptide (R9) peptide. It can be used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01119
+ Info
DSPE-PEG2000-SP94
DSPE-PEG2000-SP94 is a PEG compound composed of DSPE and the cell-penetrating peptide (SP94). SP94 exhibits specific binding to hepatocellular carcinoma (HCC) cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01167
+ Info
Pyrocatechol
CAS :
- 120-80-9
Pyrocatechol, often known as catechol or benzene-1,2-diol, is a benzenediol, Pyrocatechol was produced at a large scale industrially, mainly as precursors to pesticides, flavors, and fragrances. Its sulfonic acid is often present in the urine of many mammals.
Formule :C₆H₆O₂
Degré de pureté :99.96%
Couleur et forme :Solid
Masse moléculaire :110.11
Ref: TM-T4847
+ Info
DSPE-PEG1000-F3
DSPE-PEG1000-F3 is a PEG compound made from DSPE and a targeting peptide called nucleolin (F3). The F3 peptide can specifically bind to cell surface nucleolin, enabling efficient transport from the cell surface to the nucleus. DSPE-PEG1000-F3 is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01187
+ Info
DSPE-PEG5000-WYRGRL
DSPE-PEG5000-WYRGRL is a PEG compound composed of DSPE and a cartilage-targeting peptide (WYRGRL). The WYRGRL peptide targets type II collagen and can bind to type II collagen α1. DSPE-PEG5000-WYRGRL is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01164
+ Info
DSPE-PEG5000-CSTSMLKAC
DSPE-PEG5000-CSTSMLKAC is a PEG compound consisting of DSPE and CSTSMLKAC. CSTSMLKAC facilitates targeted homing of phages to ischemic heart tissue. This compound can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01102
+ Info
DSPE-PEG2000-MPG
DSPE-PEG2000-MPG is a PEG compound composed of DSPE and the peptide carrier (MPG). The MPG component is derived from the nuclear localization sequence (NLS) of the SV40 large T antigen and the fusion peptide domain of HIV-1gp41. It effectively delivers short oligonucleotides into cells independently of the endosomal pathway.
Couleur et forme :Odour Solid
Ref: TM-TCL-01130
+ Info
DSPE-PEG1000-KAA
DSPE-PEG1000-KAA is a PEG compound comprised of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically binds to tumor vasculature in RIP-Tag2 transgenic mice. DSPE-PEG1000-KAA is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01189
+ Info
CT140
CT140 is a human IgG4 monoclonal antibody (mAb) that specifically targets PAI-1. The suggested isotype control for this compound is Human IgG4 kappa, Isotype Control.
Couleur et forme :Odour Liquid
Ref: TM-T9901A-1069
+ Info
DSPE-PEG3000-TAASGVRSMH
DSPE-PEG3000-TAASGVRSMH is a PEG compound composed of DSPE and TAASGVRSMH. TAASGVRSMH exhibits a strong affinity for the NG2 proteoglycan on the PC membrane. DSPE-PEG3000-TAASGVRSMH can be utilized in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01143
+ Info
DSPE-PEG3000-LyP-1
DSPE-PEG3000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). The LyP-1 component specifically targets tumor-associated lymphatics and macrophages.
Couleur et forme :Odour Solid
Ref: TM-TCL-01091
+ Info
DSPE-PEG5000-octreotide
DSPE-PEG5000-Octreotide is a PEG compound composed of DSPE and Octreotide. Octreotide serves as a somatostatin receptor agonist and exhibits anti-tumor properties, induces apoptosis, and is applicable for acromegaly research. DSPE-PEG5000-Octreotide can be utilized in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01159
+ Info
DSPE-PEG1000-K237
DSPE-PEG1000-K237 is a PEG compound composed of DSPE and the KDR-targeting peptide (K237). K237 functionally disrupts the interaction between VEGF and KDR receptors, producing significant biological effects such as inhibiting angiogenesis and tumor growth. DSPE-PEG1000-K237 is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01181
+ Info
DSPE-PEG5000-pPB
DSPE-PEG5000-pPB is a PEG compound composed of DSPE and the cyclic oligopeptide (pPB). The pPB component has high binding affinity to PDGFRβ, which is overexpressed on activated hepatic stellate cells (HSC). DSPE-PEG5000-pPB is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01144
+ Info
DSPE-PEG1000-SP94
DSPE-PEG1000-SP94 is a PEG compound composed of DSPE and the cell-penetrating peptide (SP94). SP94 exhibits specific binding affinity to hepatocellular carcinoma (HCC) cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01078
+ Info
DSPE-PEG2000-M2pep
DSPE-PEG2000-M2pep is a PEG compound formed from DSPE and the M2-polarized macrophage-targeting peptide (M2pep). M2pep acts as a monovalent or multivalent ligand conjugated with pro-apoptotic peptides to specifically target M2 macrophages with toxic effects. DSPE-PEG2000-M2pep is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01085
+ Info
DSPE-PEG1000-TAASGVRSMH
DSPE-PEG1000-TAASGVRSMH is a PEG compound composed of DSPE and TAASGVRSMH. The TAASGVRSMH sequence exhibits high affinity for the NG2 proteoglycan on PC membranes. DSPE-PEG1000-TAASGVRSMH is useful for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01152
+ Info
DSPE-PEG1000-VIP
DSPE-PEG1000-VIP is a PEG compound composed of DSPE and the vasoactive intestinal peptide (VIP). It can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01081
+ Info
VHL-IN-1
VHL-IN-1 (compound 30), a ubiquitin E3 ligase von Hippel-Lindau (VHL) inhibitor with a dissociation constant (Kd) of 37 nM, potently stabilizes HIF-1α and
Formule :C₂₈H₃₇FN₄O₄S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :544.68
Ref: TM-T79720
+ Info
DSPE-PEG5000-PP1
DSPE-PEG5000-PP1 is a PEG compound composed of DSPE and the PP1 peptide, which targets inflammatory atherosclerotic plaques. It can be used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01147
+ Info
DSPE-PEG2000-VIP
DSPE-PEG2000-VIP is a PEG-based compound composed of DSPE and the vasoactive intestinal peptide (VIP). This compound is useful for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01125
+ Info
Alternaphenol B2
Alternaphenol B2, a selective inhibitor of mutant isocitrate dehydrogenase 1 (IDH1m), is sourced from the coral-derived fungus Parengyodontium album SCSIO
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T83133
+ Info
DSPE-PEG5000-F3
DSPE-PEG5000-F3 consists of DSPE and the nucleolin-targeting peptide (F3) and is a PEGylated compound. The F3 peptide specifically binds to nucleolin on the cell surface, facilitating efficient transport from the cell surface to the nucleus. DSPE-PEG5000-F3 is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01084
+ Info
DSPE-PEG2000-pPB
DSPE-PEG2000-pPB is a PEG compound comprised of DSPE and the cyclic oligopeptide (pPB). The pPB component exhibits a high binding affinity for PDGFRβ, which is overexpressed on activated hepatic stellate cells (HSC). DSPE-PEG2000-pPB is utilizable for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01135
+ Info
DSPE-PEG2000-ESBP
DSPE-PEG2000-ESBP is a PEGylated compound composed of DSPE and E-selectin binding peptide (ESBP). As a tumor-targeting peptide, ESBP can specifically recognize and bind to receptors or markers on the surface of tumor cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01173
+ Info
DSPE-PEG5000-T7
DSPE-PEG5000-T7 is a PEG-based compound composed of DSPE and transferrin receptor peptide (T7). T7 (HAIYPRH) specifically binds to TfR. DSPE-PEG5000-T7 is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01079
+ Info
C12 DG PEG (MW 2000)
C12 DG PEG (1,2-Didodecanoyl-rac-glycero-3-methoxypolyethylene glycol) (MW 2000) is a polyethylene glycol lipid that can be utilized in the formation of lipid nanoparticles and liposomes. C12 DG PEG (MW 2000) shows potential for use in cancer research.
Couleur et forme :Odour Solid
Ref: TM-TCL-01219
+ Info
DSPE-PEG5000-SP94
DSPE-PEG5000-SP94 is a PEGylated compound composed of DSPE and the cell-penetrating peptide (SP94). SP94 demonstrates specific binding affinity to hepatocellular carcinoma (HCC) cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01077
+ Info
DSPE-PEG1000-CSTSMLKAC
DSPE-PEG1000-CSTSMLKAC is a PEG compound composed of DSPE and CSTSMLKAC. The CSTSMLKAC component facilitates phage-mediated targeting to ischemic cardiac tissue. DSPE-PEG1000-CSTSMLKAC is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01104
+ Info
DSPE-PEG2000-ANG
DSPE-PEG2000-ANG is a PEG compound composed of DSPE and the dual-targeting ligand (Angiopep-2, ANG). ANG exhibits high binding efficiency to LRP1 and has been used for targeted delivery to gliomas. DSPE-PEG2000-ANG can be utilized in drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01087
+ Info
DSPE-PEG1000-YIGSR
DSPE-PEG1000-YIGSR is a PEG compound consisting of DSPE and the biomimetic peptide YIGSR. YIGSR interacts with the 67 kDa laminin-binding protein (LBP) to enhance adhesion and spreading of various cell types, including endothelial cells, fibroblasts, and smooth muscle cells. DSPE-PEG1000-YIGSR is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01157
+ Info
DSPE-PEG5000-ANG
DSPE-PEG5000-ANG is a PEGylated compound formed by DSPE and the dual-targeting ligand (Angiopep-2, ANG). ANG exhibits high binding efficacy to LRP1 and has been utilized for targeting glioma delivery. DSPE-PEG5000-ANG is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01140
+ Info
DSPE-PEG1000-T7
DSPE-PEG1000-T7 is a PEG compound composed of DSPE and transferrin receptor peptide (T7). The T7 peptide (HAIYPRH) specifically binds to TfR. DSPE-PEG1000-T7 is applicable in drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01076
+ Info
DSPE-PEG5000-M2pep
DSPE-PEG5000-M2pep is a PEG compound composed of DSPE and the M2 macrophage-targeting peptide (M2pep). Serving either as a monovalent or multivalent ligand, M2pep is conjugated with pro-apoptotic peptides to direct toxicity specifically toward M2 macrophages. DSPE-PEG5000-M2pep is applicable for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01080
+ Info
DSPE-PEG5000-TH
DSPE-PEG5000-TH is a PEG compound formed from DSPE and the pH-responsive cell-penetrating peptide (TH). In acidic environments like the tumor microenvironment, TH is activated, allowing it to selectively deliver small molecules, oligonucleotides, proteins, and similar substances into tumor cells.
Couleur et forme :Odour Solid
Ref: TM-TCL-01120
+ Info
DSPE-PEG1000-EB1
DSPE-PEG1000-EB1 is a PEG compound composed of DSPE and a pH-responsive cell-penetrating peptide (EB1). It is utilized for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01134
+ Info
DSPE-PEG3000-TAT
DSPE-PEG3000-TAT is a PEG compound composed of DSPE and a cell-penetrating peptide (TAT). It is used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01118
+ Info
DSPE-PEG2000-PP1
DSPE-PEG2000-PP1 is a PEG compound composed of DSPE and the PP1 peptide. The PP1 peptide specifically targets inflammatory atherosclerotic plaques. DSPE-PEG2000-PP1 is utilized in drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01179
+ Info
DSPE-PEG1000-LTLRWVGLMS
DSPE-PEG1000-LTLRWVGLMS is a PEG compound composed of DSPE and the decapeptide (LTLRWVGLMS). The receptor for LLRWVGLMS is the chondroitin sulfate proteoglycan NG2. LLRWVGLMS demonstrates homing to pericytes associated with tumor vasculature. DSPE-PEG1000-LTLRWVGLMS can be utilized for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01105
+ Info
DSPE-PEG2000-NGR
DSPE-PEG2000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide specifically targets the tumor vasculature antigen CD13. This compound is suitable for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01182
+ Info
LY 135114
CAS :
- 126254-82-8
LY 135114 is a metabolite of LY 195448, which is a phenethanolamine with anti-tumour activity.
Formule :C₂₀H₂₆N₂O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :342.43
Ref: TM-T27873
+ Info
GGACK hydrochloride
GGACK (H-Glu-Gly-Arg-CMK) hydrochloride is an irreversible substrate-like inhibitor of the serine protease urokinase-type plasminogen activator (uPA).
Formule :C₁₄H₂₆Cl₂N₆O₅
Couleur et forme :Solid
Masse moléculaire :428.13417
Ref: TM-T207613
+ Info
FXIIa-IN-1 HCl
CAS :
- 3052551-20-6
FXIIa-IN-1 HCl is a selective inhibitor of Factor XIIa,and can be used to study thrombosis and inflammation induced by artificial surfaces.
Formule :C₂₁H₁₇ClN₂O₆
Degré de pureté :99.61%
Couleur et forme :Soild
Masse moléculaire :428.82
Ref: TM-T82361L
+ Info
DSPE-PEG2000-T7
DSPE-PEG2000-T7 is a PEG compound composed of DSPE and the transferrin receptor peptide (T7). The T7 peptide (HAIYPRH) specifically binds to TfR, making DSPE-PEG2000-T7 useful for drug delivery applications.
Couleur et forme :Odour Solid
Ref: TM-TCL-01139
+ Info
CP-LC-1422
CP-LC-1422 is a homocysteine-derived ionizable amino lipid known for its efficient RNA delivery capabilities, enabling high-level protein expression in vivo. When formulated in lipid nanoparticles (LNP) and administered intravenously, it demonstrates significant spleen-targeting properties without observed notable toxicity.
Formule :C₅₁H₉₇N₃O₈S₃
Couleur et forme :Solid
Masse moléculaire :975.64378
Ref: TM-TCL-01213
+ Info
MK-8245 Trifluoroacetate
CAS :
- 1415559-41-9
MK-8245 trifluoroacetate: Potent liver-targeting SCD inhibitor, IC50=1nM (human). Anti-diabetic/anti-dyslipidemic. Selective, with low adverse event exposure.
Formule :C₁₉H₁₇BrF₄N₆O₆
Couleur et forme :Solid
Masse moléculaire :581.27
Ref: TM-T38844
+ Info
Aminopeptidase N inhibitor 2
AminopeptidaseN inhibitor 2 is an APN inhibitor (IC50: 4.3 μM) with antitumor properties.
Formule :C₁₂H₁₆F₂N₂O₄S
Couleur et forme :Solid
Masse moléculaire :322.07988
Ref: TM-T207518
+ Info
Xanthine oxidase-IN-11
Xanthine Oxidase-IN-11, an analog of XO8, is an inhibitor of xanthine oxidase (XO) [1].
Formule :C₁₀H₈N₂OS
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :204.25
Ref: TM-T78985
+ Info
H-Ile-Pro-Pro-OH acetate
H-Ile-Pro-Pro-OH acetate is a angiotensin-converting enzyme inhibitor (ACE) of milk-derived tripeptides.
Formule :C₁₈H₃₁N₃O₆
Degré de pureté :97.15%
Couleur et forme :Solid
Masse moléculaire :385.46
Ref: TM-TP1750L
+ Info
1'-Hydroxy bufuralol
CAS :
- 57704-16-2
1'-Hydroxy bufuralol is a metabolite of bufuralol, an orally active β-adrenoceptor blocker used in the study of hypertension and cardiac arrhythmias.
Formule :C₁₆H₂₃NO₃
Couleur et forme :Solid
Masse moléculaire :277.36
Ref: TM-T41364
+ Info
BTT-266
CAS :
- 2413939-89-4
BTT-266 is a blocker of voltage-gated calcium channel for pain management.
Formule :C₃₄H₂₈N₄O₄
Degré de pureté :98.34%
Couleur et forme :Solid
Masse moléculaire :556.61
Ref: TM-T60010
+ Info
SHO1122147
SHO1122147 (Compound 7m) disrupts the mitochondrial electron transport chain, demonstrating mitochondrial uncoupling activity (EC50=3.6 μM). It increases the cellular oxygen consumption rate (OCR=69%) and enhances cellular respiration. Additionally, SHO1122147 is orally active and can be utilized in research related to obesity and metabolic dysfunction-associated steatohepatitis (MASH).
Formule :C₁₇H₁₁ClN₄O₂
Couleur et forme :Solid
Masse moléculaire :338.748
Ref: TM-T204360
+ Info
Equilenin
CAS :
- 517-09-9
Equilenin (E 400) is a natural estrogen that is an endocrine disruptor and has been used in breast cancer research.
Formule :C₁₈H₁₈O₂
Degré de pureté :99.4%
Couleur et forme :Solid
Masse moléculaire :266.33
Ref: TM-T19776
+ Info
Zaragozic acid D
CAS :
- 155179-14-9
Zaragozic acid D inhibits squalene synthase and ras farnesyl-protein transferase isolated from the keratinophilic fungus Amauroascus niger.
Formule :C₃₄H₄₆O₁₄
Couleur et forme :Solid
Masse moléculaire :678.72
Ref: TM-T26347
+ Info
1-epi-Regadenoson
CAS :
- 2015222-31-6
1-epi-Regadenoson is an α-isomer impurity of Regadenoson, a highly selective adenosine A2A receptor agonist [1].
Formule :C₁₅H₁₈N₈O₅
Couleur et forme :Solid
Masse moléculaire :390.35
Ref: TM-T77294
+ Info
AY 9944 dihydrochloride
CAS :
- 1245-84-7
AY 9944 dihydrochloride is a intermediate.
Formule :C₂₂H₃₀Cl₄N₂
Degré de pureté :99.22% - 99.82%
Couleur et forme :Soild
Masse moléculaire :464.3
Ref: TM-T14362L
+ Info
HLF1-11
CAS :
- 183623-03-2
HLF1-11: human lactoferrin peptide, antimicrobial, inhibits MPO, steers monocytes to macrophages, boosts immunity.
Formule :C₅₆H₉₅N₂₅O₁₄S
Couleur et forme :Solid
Masse moléculaire :1374.58
Ref: TM-T73659
+ Info
Z-Asp(OBzl)-OH
CAS :
- 3479-47-8
Z-Asp(OBzl)-OH (N-Cbz-L-Aspartic acid 4-benzyl ester) is an aspartic acid derivative.
Formule :C₁₉H₁₉NO₆
Degré de pureté :98.71%
Couleur et forme :Solid
Masse moléculaire :357.36
Ref: TM-T64326
+ Info
IYPTNGYTR acetate
IYPTNGYTR acetate, a deamidation-sensitive peptide derived from Trastuzumab, is a suitable tool for monitoring the metabolism of Trastuzumab in vivo [1].
Couleur et forme :Liquid
Ref: TM-T36669
+ Info
Acremonidin A
CAS :
- 701914-77-4
Acremonidin A, from Purpureocillium lilacinum, is a strong CaM inhibitor binding to hCaM M124C-mBBr with a Kd of 19.40 nM.
Formule :C₃₃H₂₆O₁₂
Couleur et forme :Solid
Masse moléculaire :614.55
Ref: TM-T72902
+ Info
2,6-Diphenylpyridine
CAS :
- 3558-69-8
2,6-Diphenylpyridine is toxic to MDA-MB-231 cells and has anticancer potential.
Formule :C₁₇H₁₃N
Degré de pureté :99.21%
Couleur et forme :Solid
Masse moléculaire :231.29
Ref: TM-TN9491
+ Info
ω-Conotoxin Bu8
ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges.
Formule :C₁₀₃H₁₇₄N₄₂O₃₅S₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :2753.13
Ref: TM-T80457
+ Info
9AzNue5Ac
CAS :
- 76487-51-9
9AzNue5Ac is a Neu5Ac analog that is metabolized in vivo in living cells and in mice.9AzNue5Ac binds to sialoglycans.
Formule :C₁₁H₁₈N₄O₈
Degré de pureté :≥98%
Couleur et forme :Solid
Masse moléculaire :334.28
Ref: TM-T74989
+ Info
BDM_92499
BDM_92499 is a nanomolar, selective IRAP inhibitor with an IC50 of 3.4 nM. It also inhibits ERAP1 and ERAP2, with IC50 values of 0.46 μM and 4.2 μM, respectively.
Couleur et forme :Odour Solid
Ref: TM-T206956
+ Info
α-Glucosidase-IN-27
α-Glucosidase-IN-27 (compound 8l), an α-glucosidase inhibitor with an IC50 value of 25.78 μM, demonstrates potential for research into type 2 diabetes (D2M) [1
Formule :C₂₂H₂₀N₄O₄S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :436.48
Ref: TM-T79237
+ Info
Bz-Ala-Arg
CAS :
- 71448-11-8
Bz-Ala-Arg, a dipeptide, serves as a spectrophotometric substrate (0.4 M pyridine formate, pH 4.25) for human pancreatic carboxypeptidase B and plasma
Formule :C₁₆H₂₃N₅O₄
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :349.38
Ref: TM-T80113
+ Info
ω-Conotoxin CVIE
ω-Conotoxin CVIE selectively inhibits voltage-gated Ca^2+ channels (Ca_v 2.2) [1].
Formule :C₉₈H₁₆₄N₄₀O₃₄S₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :2638.99
Ref: TM-T80449
+ Info
10 FTHF disodium
CAS :
- 914800-65-0
10 FTHF disodium (10-Formyltetrahydrofolic acid disodium) is a form of tetrahydrofolate that is involved in the synthesis of purine compounds.
Formule :C₂₀H₂₁N₇Na₂O₇
Couleur et forme :Solid
Masse moléculaire :517.4
Ref: TM-T73731
+ Info
Maurocalcine
CAS :
- 269745-22-4
Maurocalcine is a cell-permeable agonist for ryanodine receptor (RyR) subtypes 1, 2, and 3.
Formule :C₁₅₆H₂₇₀N₅₆O₄₆S₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :3858.55
Ref: TM-T80153
+ Info
PPARγ-IN-3
PPARγ-IN-3 (compound 9ga), a potent and orally active PPARγ inhibitor, effectively reduces triglyceride (TG) accumulation and exhibits low cytotoxicity. Additionally, it prevents excessive body weight gain, lessens fat and liver mass, and decreases lipid accumulation in both the liver and blood. PPARγ-IN-3 holds promise for research into diet-induced obesity.
Formule :C₂₃H₂₈FN₇O₃
Couleur et forme :Solid
Masse moléculaire :469.51
Ref: TM-T89904
+ Info
Monoglyceride lipase
CAS :
- 9040-75-9
Monoglyceridelipase is a crucial enzyme involved in lipid metabolism, catalyzing the hydrolysis of monoglycerides (especially 2-AG, or 2-arachidonoylglycerol) into glycerol and free fatty acids. By regulating the levels of 2-AG, this enzyme impacts neural signaling, pain perception, inflammatory responses, and metabolic processes.
Couleur et forme :Solid
Ref: TM-T200072
+ Info
α-Glucosidase-IN-72
α-Glucosidase-IN-72 (compound 5i), a 2,4-dichloro-N-phenylacetamide derivative, functions as an α-glucosidase inhibitor with an inhibitory concentration (IC 50) of 6 μM. Notably, it does not adhere to Lipinski's "rule of five" and is not a cancer inducer.
Formule :C₃₇H₂₆Cl₂N₄O₉
Couleur et forme :Solid
Masse moléculaire :741.53
Ref: TM-T200200
+ Info
PP5-IN-2
PP5-IN-2, a selective and orally active inhibitor of protein phosphatase 5 (PP5), exhibits an IC 50 of 0.9 μM. This compound activates p53 and leads to the downregulation of cyclin D1 and MGMT, thereby inducing cell cycle arrest and reversing Temozolomide (TMZ) resistance in the U87 MG cell line. Additionally, PP5-IN-2 has demonstrated effective inhibition of tumor growth in the xenograft mouse model.
Formule :C₁₆H₁₅NO₄
Couleur et forme :Solid
Masse moléculaire :285.29
Ref: TM-T89967
+ Info
Penicillinase
CAS :
- 9001-74-5
Penicillinase is a β-lactamase and secretory enzyme capable of degrading and inactivating penicillin and similar compounds.
Couleur et forme :Solid
Ref: TM-T75391
+ Info
C-Type Natriuretic Peptide (1-53), Porcine, Rat,mouse
CAS :
- 129405-72-7
C-Type Natriuretic Peptide (1-53), from porcine, rat, and mouse sources, serves as an activator of particulate guanylate cyclase B (pGC-B), prominently found in endothelial cells, kidneys, and the heart. This peptide efficiently mediates a potent anti-fibrotic effect in human cardiac and renal fibroblasts through the production of the second messenger cGMP.
Couleur et forme :Solid
Ref: TM-TP2855
+ Info
PF-07247685
PF-07247685, a potent BCKDC kinase (BDK) inhibitor (EC 50 = 2.2 nM), enhances the binding between BDK and the BCKDH E2 core subunit to block E1 phosphorylation.
Formule :C₂₁H₂₀N₂O₃S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :380.46
Ref: TM-T79358
+ Info
α-Glucosidase-IN-73
α-Glucosidase-IN-73 (compound 16b), an α-Glucosidase inhibitor, exhibits an IC 50 value of 0.158 μM and possesses the ability to activate PPAR γ. This compound is applicable in studies focusing on anti-diabetic and anti-inflammatory treatments.
Formule :C₂₄H₂₁N₃O₂S
Couleur et forme :Solid
Masse moléculaire :415.51
Ref: TM-T200247
+ Info
Stevisalioside A
Stevisalioside A (Compound 2), isolated from the roots of Stevia serrata, is an orally active antidiabetic agent that inhibits Protein Tyrosine Phosphatase 1B (
Formule :C₃₅H₅₀O₁₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :710.76
Ref: TM-T80007
+ Info
ITH12711
ITH12711, a PP2A ligand, can traverse the blood-brain barrier (BBB) and exerts neuroprotection by restoring PP2A-phosphatase activity [1].
Formule :C₁₂H₂₀O₅
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :244.28
Ref: TM-T78681
+ Info
Cryptosporioptide A
CAS :
- 1647101-05-0
Cryptosporioptide A (Compound 3), a protein tyrosine phosphatase inhibitor, originates from the insect-parasitic fungus Cordyceps gracilioides.
Formule :C₁₈H₁₇NO₁₀
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :407.33
Ref: TM-T79985
+ Info
3-O-Dihydro-p-coumaroyltohogenol
3-O-Dihydro-p-coumaroyltohogenol functions as a PTP1B inhibitor (IC50 = 6.27 μM), exhibiting anti-diabetic and anti-obesity activities.
Formule :C₃₉H₆₀O₅
Couleur et forme :Solid
Masse moléculaire :608.89
Ref: TM-T200206
+ Info
ADP-specific glucokinase
CAS :
- 173585-07-4
ADP-specific glucokinase, expressed in thermophilic archaea, is an ADP-specific enzyme that catalyzes the conversion of glucose to glucose-6-phosphate, thereby facilitating glycolysis. This enzyme can activate T cells and enhance the phagocytic activity of macrophages. It is used in research related to metabolic disorders, neurological diseases, and tumors.
Couleur et forme :Solid
Ref: TM-T89882
+ Info
Phosphofructokinase
CAS :
- 9001-80-3
Phosphofructokinase, a crucial glycolytic enzyme, catalyzes the conversion of fructose-6-phosphate to fructose-1,6-bisphosphate in the glycolysis pathway. Its activity is inhibited by the binding of Phosphoenolpyruvate (PEP), which regulates the rate of glycolysis. Additionally, Phosphofructokinase is utilized in the measurement of fructose-6-phosphate (fructose-6-phosphate) levels.
Couleur et forme :Solid
Ref: TM-T200040
+ Info
IONIS PTP1BRx
CAS :
- 1403406-29-0
IONIS PTP1BRx (ISIS 404173) acts as an antisense inhibitor of protein tyrosine phosphatase 1B (PTP-1B). This compound exhibits anti-diabetic properties, making it suitable for research into insulin resistance related to obesity and type 2 diabetes.
Couleur et forme :Solid
Ref: TM-T200394
+ Info
Antibacterial agent 237
Anti bacterial agent 237 (compound Ru-8) acts as a potent antibacterial agent against Staphylococcus aureus, exhibiting minimum inhibitory concentrations (MICs) ranging from 0.78 to 1.56 μg/mL. It works by disrupting bacterial cell membranes, altering their permeability, and inducing the production of reactive oxygen species, which leads to bacterial cell death without promoting resistance. Additionally, Anti bacterial agent 237 demonstrates low hemolytic toxicity towards rabbit erythrocytes and Raw 264.7 cells. It has shown significant antibacterial activity in models of skin wound infections in mice and larval infections by the greater wax moth, effectively combating Staphylococcus aureus infections.
Formule :C₆₅H₆₉Cl₃N₁₀RuS₂
Couleur et forme :Solid
Masse moléculaire :1261.87
Ref: TM-T89870
+ Info
Imperatoxin A TFA
Imperatoxin A TFA, a peptide toxin derived from the venom of the African scorpion Pandinus imperator, acts as an activator of Ca2+-release channels/ryanodine receptors (RyRs). It facilitates the influx of Ca2+ from the sarcoplasmic reticulum into the cell.
Formule :C₁₄₈H₂₅₄N₅₈O₄₅S₆·xC₂HF₃O₂
Couleur et forme :Solid
Masse moléculaire :3758.35 (free base)
Ref: TM-TP2838
+ Info
NAD Synthetase
CAS :
- 9032-69-3
NAD Synthetase is responsible for the final step in the synthesis of Nicotinamide Adenine Dinucleotide (NAD). The enzyme sourced from Escherichia coli exhibits Km values of 200 μM for NAD, 11 μM for ATP, and 0.65 μM for ammonia. Conversely, NAD Synthetase derived from yeast demonstrates Km values of 170 μM for NAD, 190 μM for ATP, and 64 μM for ammonia. This enzyme is applicable in enzymatic assays for ATP, ammonia, urea, or creatinine and can also be used in enzymatic recycling methods. Additionally, NAD Synthetase holds potential for research into metabolic diseases, cancer, aging, and neurodegenerative disorders.
Couleur et forme :Solid
Ref: TM-T200236
+ Info
ω-Conotoxin FVIA
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and thermal pain abnormalities in a rat model of caudal nerve
Formule :C₉₈H₁₆₄N₃₆O₃₃S₆
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :2566.96
Ref: TM-T80446
+ Info
Ledelabricin alfa
Ledelabricin alfa, an isoform A variant of human proteoglycan 4 (PRG4), functions as a lubricant for joints and boundaries.
Degré de pureté :98%
Couleur et forme :Odour Liquid
Ref: TM-T80592
+ Info
h15-LOX-2 inhibitor 2
Compound 10 (h15-LOX-2 inhibitor 2) suppresses h15-LOX activity, exhibiting IC 50 and K i values of 26.9 μM and 16.4 μM, respectively.
Formule :C₂₂H₃₀Cl₂N₆O₃
Couleur et forme :Solid
Masse moléculaire :497.42
Ref: TM-T200017
+ Info
IHMT-IDH1-053
IHMT-IDH1-053 (compound 16) is an irreversible inhibitor exhibiting high selectivity for the IDH1 R132H mutant, achieving an IC50 of 4.7 nM.
Formule :C₂₅H₃₃FN₆O₄S
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :532.63
Ref: TM-T78758
+ Info
Tpp-CAQK
Tpp-CAQK, a specially engineered mitochondrial compound, has been shown to improve phagocytosis of myelin debris by macrophages, reduce mitochondrial dysfunction and pro-inflammatory features, and enhance tissue repair and functional recovery in mice after spinal cord injury.
Formule :C₄₀H₅₄BrN₆O₇PS
Couleur et forme :Solid
Masse moléculaire :873.84
Ref: TM-TP2850
+ Info
IONIS PTP1BRx sodium
IONIS PTP1BRx (ISIS 404173) sodium, an antisense inhibitor of protein tyrene phosphatase 1B (PTP-1B), exhibits antidiabetic properties. This compound is utilzed in researching insulin resistance and type 2 diabetes mellitus associated with obesity.
Couleur et forme :Odour Solid
Ref: TM-T200242
+ Info
Maurocalcine TFA
Maurocalcine TFA acts as an agonist for ryanodine receptor (RyR) channels 1, 2, and 3, demonstrating cell-penetrating capabilities. It induces binding of [3H]ryanodine to RyR1 with an EC50 of 2558 nM and exhibits an apparent affinity of 14 nM for RyR2. This compound is applicable for in vivo cell tracking or other cellular imaging techniques.
Formule :C₁₅₆H₂₇₀N₅₆O₄₆S₆·xC₂HF₃O₂
Couleur et forme :Solid
Masse moléculaire :3858.55 (free base)
Ref: TM-TP2868
+ Info
Epoxide hydrolase
CAS :
- 9048-63-9
Epoxide hydrolase, an enzyme responsible for catalyzing the reaction of epoxides with water to convert epoxy groups into diols, plays a crucial role in the metabolism of environmental pollutants and lipids. It is instrumental in detoxification, inflammatory responses, and regulating the health of the cardiovascular system. Additionally, Epoxide hydrolase is used in asymmetric catalytic reactions, such as the asymmetric ring-opening of epoxides, which are important for the synthesis of chiral pharmaceutical molecules.
Couleur et forme :Solid
Ref: TM-T200049
+ Info
Carbonic anhydrase inhibitor 15
Carbonic Anhydrase Inhibitor 15 (Compound 8), with an inhibitory constant (K_i) of 8.5 nM for hCA II, exhibits analgesic effects [1].
Formule :C₂₇H₃₃N₅O₂S₂
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :523.71
Ref: TM-T78840
+ Info
Denecimig
CAS :
- 2488745-86-2
Denecimig (Mim8) is a bispecific and humanized IgG4κ antibody, hemophilia A, activated coagulation factors IXa (FIXa) and X (FX) arresting bleeding.
Degré de pureté :95%
Couleur et forme :Liquid
Ref: TM-T82585
+ Info
ESI1
ESI1 is a small molecule inhibitor of epigenetic silencing. This compound induces the formation of nuclear aggregates of the key lipid metabolism regulator SREBP1/2, thereby concentrating transcription co-activators to drive lipid/cholesterol biosynthesis. Additionally, ESI1 promotes myelin regeneration in demyelination animal models and facilitates de novo myelination on regenerating CNS axons, reversing age-related cognitive decline.
Formule :C₁₈H₁₈ClN₅O
Couleur et forme :Solid
Masse moléculaire :355.82
Ref: TM-T200212
+ Info
CA inhibitor 2
Compound 4H is a potent carbonic anhydrase inhibitor with an IC50 value of 0.033 μM [1].
Formule :C₇H₉N₇O₃S₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :335.39
Ref: TM-T79681
+ Info
Ovalbumin (154-159)
CAS :
- 1370698-94-4
Ovalbumin (154-159), a peptide fragment derived from ovalbumin, acts as a potent inhibitor of the angiotensin-converting enzyme (ACE) and is utilized in
Formule :C₂₈H₅₂N₁₀O₉
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :672.77
Ref: TM-T80099
+ Info
Galactose 1-dehydrogenase
Galactose 1-dehydrogenase, pseudomonas fluorescens, a dehydrogenase found in Pseudomonas fluorescens, facilitates the oxidation of L-arabinose and D-galactose, utilizing NADP+/NAD+ as a cofactor. This enzyme is employed in diagnostic assays to quantify total galactose levels and serves as a biocatalyst in the production of galacturonic acid salts.
Couleur et forme :Odour Solid
Ref: TM-T200393
+ Info
Mortatarin F
Mortatarin F (Compound 1), a renyleted flavonoid derived from mulberry leaves, functions as an α-glucosidase inhibitor with an IC50 value of 8.7 μM, making it
Formule :C₂₅H₃₀O₇
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :442.5
Ref: TM-T79937
+ Info
Glycerol-3-phosphate dehydrogenase
CAS :
- 9001-49-4
Glycerol-3-phosphate dehydrogenase from Saccharomyces cerevisiae is an enzyme that catalyzes the oxidation of glycerol-3-phosphate (G3P) to dihydroxyacetone phosphate (DHAP), playing a crucial role in glycerol metabolism and energy production. This enzyme acts as the rate-limiting step in glycerol production within Saccharomyces cerevisiae, regulating glycerol formation and accumulation to aid the yeast in adapting to hyperosmotic environments. Additionally, glycerol-3-phosphate dehydrogenase from Saccharomyces cerevisiae is relevant in research within the field of metabolic engineering.
Couleur et forme :Solid
Ref: TM-T89979
+ Info
Diacetinase
Diacetinase, a member of the esterase family, catalyzes the hydrolysis of glyceryl diacetate (Diacetin). It is utilized in the measurement of lipase activity.
Couleur et forme :Odour Solid
Ref: TM-T200253
+ Info
Autophagy inducer 5
Autophagyinducer 5 (compound 21o) serves as a potent inhibitor of MCF-7 (IC50: 2 μM), making it a potential candidate for breast cancer therapy. It induces autophagy by activating the ROS/JNK signaling pathway, which increases ROS production and JNK phosphorylation, ultimately exerting cytotoxic effects.
Formule :C₄₁H₅₂N₄O₃
Couleur et forme :Solid
Masse moléculaire :648.88
Ref: TM-T89960
+ Info
α-Amylase/α-Glucosidase-IN-5
α-Amylase/α-Glucosidase-IN-5 (compound 4l) functions as a dual inhibitor, effectively inhibiting both α-glucosidase (Glucosidase) and α-amylase (Amylases) with
Formule :C₃₀H₂₇BrN₃O₃P
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :588.43
Ref: TM-T78878
+ Info
Pregnant mare serum gonadotropin
CAS :
- 9002-70-4
Pregnant mare serum gonadotropin (PMSG) functions as a gonadotropin that enhances follicular development and ovulation in animals. This compound operates by modulating blood hormones, gonadotropins, and cytoplasmic estradiol receptors in the anterior pituitary and hypothalamus. Commonly employed in livestock to boost reproductive efficiency, PMSG is also valuable for research focused on estrous cycle regulation.
Couleur et forme :Solid
Ref: TM-T200009
+ Info
Sorbitol-6-phosphate 2-dehydrogenase
CAS :
- 37250-69-4
Sorbitol-6-phosphate 2-dehydrogenase, a dehydrogenase enzyme produced by Escherichia coli, catalyzes the interconversion of D-sorbitol 6-phosphate and D-fructose 6-phosphate. The enzyme oxidizes D-sorbitol 6-phosphate at a rate ten times faster than it reduces D-fructose 6-phosphate, playing a role in various cellular processes.
Couleur et forme :Solid
Ref: TM-T200233
+ Info
12α-Hydroxysteroid dehydrogenase
CAS :
- 61642-40-8
12α-Hydroxysteroid dehydrogenase, an NAD-dependent enzyme expressed in Bacillus sphaericus, actively processes both free and conjugated bile salts. It is utilized to determine the levels of 12α-hydroxy bile acids in serum.
Couleur et forme :Solid
Ref: TM-T200077
+ Info
Methyl (5α,7α)-7-hydroxy-3-oxocholan-24-oate
CAS :
- 14772-96-4
Compound 7a, Methyl (5α,7α)-7-hydroxy-3-oxocholan-24-oate, is a metabolite of bile acid.
Formule :C₂₅H₄₀O₄
Couleur et forme :Solid
Masse moléculaire :404.58
Ref: TM-TN8175
+ Info
MAGL-IN-11
MAGL-IN-11 (compound 29) is a selective, reversible inhibitor of monoacylglycerol lipase (MAGL), with potential in researching inflammation, cancer, and
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T81880
+ Info
α-Glucosidase-IN-25
α-Glucosidase-IN-25 (Compound (R)-8k) serves as a competitive inhibitor for α-glucosidase, demonstrating an inhibitory concentration 50 (IC50) of 1.19μM, making
Formule :C₂₉H₂₂N₆O₃
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :502.52
Ref: TM-T79259
+ Info
MPC-IN-1
MPC-IN-1 (compound 4i), a derivative of UK-5099, is a cyanocinnamate-based inhibitor of the mitochondrial pyruvate transporter (MPC). This compound selectively fosters the development of hair follicle stem cells while not impacting normal cells. It enhances cellular lactate production and has shown significant hair growth promotion in mice, suggesting its potential use in combating hair loss.
Formule :C₁₈H₁₃N₃O₂
Couleur et forme :Solid
Masse moléculaire :303.31
Ref: TM-T89896
+ Info
DDC 3′-O-β-D glucuronide
Compound 5, DDC 3′-O-β-D-glucuronide, is a drug metabolite with properties that inhibit the fibrillization and oligomerization of Aβ42, suggesting its potential
Degré de pureté :98%
Couleur et forme :Odour Solid
Ref: TM-T82599
+ Info
5-NH2-Baicalein
CAS :
- 2478604-99-6
5-NH2-Baicalein, an aminated metabolite of Baicalein, can be utilized for researching ammonia and ammonia-associated chronic diseases [1].
Formule :C₁₅H₁₁NO₄
Couleur et forme :Solid
Masse moléculaire :269.25
Ref: TM-TN7614
+ Info
ω-conotoxin MoVIA
ω-Conotoxin MVIIA is a potent, selective inhibitor of Ca_v2.2, exhibiting an IC_50 of 0.33 μM in the SH-SY5Y fluorimetric hCa_v2.2 assay [1].
Formule :C₁₄₇H₂₃₃N₄₅O₄₇S₇
Degré de pureté :98%
Couleur et forme :Solid
Masse moléculaire :3607.15
Ref: TM-T80520
+ Info
BMT-297376
CAS :
- 2251031-81-7
BMT-297376, the optimized Linrodostat, is a potent IDO1 inhibitor.
Formule :C₂₃H₂₉F₂N₃O₃
Couleur et forme :Solid
Masse moléculaire :433.5
Ref: TM-T39779
+ Info
DSPE-PEG2000-TAT
DSPE-PEG2000-TAT is a PEG compound consisting of DSPE and the cell-penetrating peptide (TAT) peptide. It can be used for drug delivery.
Couleur et forme :Odour Solid
Ref: TM-TCL-01111