Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(197 produits)
- Caséine Kinase(137 produits)
- DHFR(34 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(66 produits)
- FXR(62 produits)
- Facteur Xa(87 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(4 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(33 produits)
- Hydroxylase(35 produits)
- IDO(84 produits)
- LDL(8 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(134 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(167 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(169 produits)
- Phospholipase(83 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(28 produits)
- SGK(11 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(46 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
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9280 produits trouvés pour "Métabolisme"
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PF-06445974
CAS :PF-06445974 has good selectivity for PDE4D, excellent brain permeability, and has a high level of specific binding in the "cold tracer" study.Formule :C20H15FN4OCouleur et forme :SolidMasse moléculaire :346.365-FAM-Alkyne
CAS :5-FAM-Alkyne is a highly selective and sensitive fluorescent biosensor designed for detecting alkaline phosphatase (ALP).Formule :C24H15NO6Couleur et forme :SolidMasse moléculaire :413.38BMS-963272
CAS :BMS-963272 is a selective and potent MGAT2 inhibitor with an IC50 value of 7.1 nM used in the study of metabolic disorders and obesity.Formule :C24H21F6N5O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :525.452-Methylcitric acid trisodium
CAS :2-Methylcitric acid trisodium (Methylcitric acid) is an endogenous metabolite in the 2-methylcitric acid cycle, which accumulates in methylmalonic and propionic acidemias.Formule :C7H7Na3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :272.18-Bromo-AMP
CAS :8-Bromo-AMP, also known as 8-Bromoadenosine 5'-monophosphate, is a membrane permeable cAMP analogue. It enhances cardiac recovery from ischemia and reperfusion by elevating ATP, ADP, and total adenine nucleotide concentrations.Formule :C10H13BrN5O7PCouleur et forme :SolidMasse moléculaire :426.123-Hydroxyisobutyric acid
CAS :(S)-3-Hydroxyisobutyric acid is an important interorgan metabolite.Formule :C4H8O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :104.1045Dabigatran Acyl-β-D-Glucuronide
CAS :Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran .Formule :C31H33N7O9Couleur et forme :SolidMasse moléculaire :647.645Vitamin D3 octanoate
CAS :Vitamin D3 octanoate, an ester derived from vitamin D3, is commonly known as cholecalciferol. Cholecalciferol is a naturally occurring form of vitamin D with notable properties such as inducing cell differentiation and impeding cancer cell proliferation.Formule :C35H58O2Couleur et forme :SolidMasse moléculaire :510.8474"-C18 EGCG
<p>4"-C18 EGCG is an effective inhibitor of α-amylase and α-glucosidase, with IC50 values of 3.74 μM and 0.81 μM respectively. It inhibits carbohydrate-hydrolyzing enzymes, reducing oxidative stress and inflammation, and demonstrates anti-diabetic activity. Additionally, 4"-C18 EGCG downregulates pro-inflammatory cytokines and exhibits cytotoxicity at 50 μM in primary human peripheral blood mononuclear cells (PBMC), and non-cancerous cell lines 3T3-L1 and HEK 293.</p>L-Glyceric acid sodium
CAS :L-Glyceric acid sodium, a urinary metabolite, is predominantly found in individuals with the rare inherited metabolic disorder L-glyceric aciduria. This compound is a diagnostic tool for identifying primary hyperoxaluria type 2 (PH2) and distinguishing it from primary hyperoxaluria type 1 (PH1) based on its excretion pattern.Formule :C3H5NaO4Couleur et forme :SolidMasse moléculaire :128.063-Hydroxy-4-aminopyridine
CAS :3-Hydroxy-4-aminopyridine is a natural product for research related to life sciences. The catalog number is T66009 and the CAS number is 52334-53-9.Formule :C5H6N2OCouleur et forme :SolidMasse moléculaire :110.1164-Phenyl-1H-1,2,3-triazole
CAS :4-Phenyl-1H-1,2,3-triazole, an inhibitor of the enzyme IDO1 (IC50: 60 µM), is utilized in cancer research [1].Formule :C8H7N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :145.16HIF-PHD-IN-1
CAS :HIF-PHD-IN-1 is a pharmacological compound that acts as an orally active inhibitor of the hypoxia-inducible factor prolyl hydroxylase domain (HIF-PHD), displaying an IC50 of 54 nM for hHIF-PHD2. Its potential as a therapeutic agent for renal anemia is highly promising.Formule :C17H12Cl2N6O3Couleur et forme :SolidMasse moléculaire :419.22Mebendazole-amine
CAS :R-18986 is a biochemical substance.Formule :C14H11N3OCouleur et forme :SolidMasse moléculaire :237.26Cefadroxil (hydrate)
CAS :Cefadroxil is a first generation aminocephalosporin with good patient compliance, a long-acting therapeutic effect, high solubility and relatively broad spectrum of anti-bacterial activity. Cefadroxil is also a substrate of the intestinal peptide transporter PepT1, which is primarily responsible for the drug's uptake across the apical membrane of small intestine.Formule :C16H19N3O6SCouleur et forme :White Crystalline SolidMasse moléculaire :381.404Boc-D-His(trt)-OH
CAS :Boc-D-His(trt)-OH is an amino acid derivative and has a wide range of applications in life science related research.Formule :C30H31N3O4Couleur et forme :SolidMasse moléculaire :497.595L-N-Benzylserine
CAS :L-N-Benzylserine is a useful organic compound for research related to life sciences. The catalog number is T65056 and the CAS number is 17136-45-7.Formule :C10H13NO3Couleur et forme :SolidMasse moléculaire :195.218Dichloroiodomethane
CAS :Dichloroiodomethane is a natural compound found in human beings[1].Formule :CHCl2ICouleur et forme :SolidMasse moléculaire :210.82N1,N8-Diacetylspermidine hydrochloride
CAS :N1,N8-Diacetylspermidine hydrochloride is a polyamine found in human urine.Formule :C11H24ClN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.783,5-Dibromotyrosine
CAS :3,5-Dibromotyrosine is a useful organic compound for research related to life sciences. The catalog number is T65914 and the CAS number is 300-38-9.Formule :C9H9Br2NO3Couleur et forme :SolidMasse moléculaire :338.9833-Deoxy-galactosone
CAS :3-Deoxy-galactosone, a 1,2-dicarbonyl compound, originates from the degradation of galactose. It forms in food during Maillard and caramelization reactions.Formule :C6H10O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :162.141Z-D-Trp-OH
CAS :Z-D-Trp-OH has a wide range of applications in life science related research.Formule :C19H18N2O4Couleur et forme :SolidMasse moléculaire :338.363Elamipretide TFA
CAS :<p>Elamipretide TFA (RX-31 TFA) is a cardiolipin peroxidase inhibitor and mitochondria-targeting peptide[1].</p>Formule :C34H50F3N9O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :753.8111β-HSD1-IN-8
CAS :11β-HSD1-IN-8 is a useful organic compound for research related to life sciences. The catalog number is T65743 and the CAS number is 386704-15-0.Formule :C10H8F3NO3Couleur et forme :SolidMasse moléculaire :247.173GDP-D-mannose disodium
CAS :GDP-D-mannose disodium is a natural product for research related to life sciences and the catalog number is T65209.Couleur et forme :SoildMB-07803
CAS :MB07803 is an orally available prodrug of an effective, noncompetitive inhibitor of fructose 1,6-bisphosphatase (FBPase) (EC50: 140 nM and t1/2 of 7.6±2.9 h).Formule :C24H37N4O7PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.61cgc-11047 free base
CAS :CGC-11047 free base is a second generation polyamine analogue of N1, N12-bisethylspermine (BESpm).Formule :C14H32N4Couleur et forme :SolidMasse moléculaire :256.43CBD3063
CAS :<p>CBD3063 is a CRMP2-based peptidomimetic small molecule that can regulate Cav 2.2 and can be used to study neurological diseases.</p>Formule :C16H25N5O2Degré de pureté :99.39%Couleur et forme :SoildMasse moléculaire :319.4Ibiglustat succinate
CAS :Ibiglustat (Venglustat) succinate is an orally active, brain-penetrant inhibitor of glucosylceramide synthase (GCS) utilized in the investigation of Gaucher disease type 3, Parkinson's disease associated with GBA mutations, Fabry disease, GM2 gangliosidosis, and autosomal dominant polycystic kidney disease.Formule :C24H30FN3O6SCouleur et forme :SolidMasse moléculaire :507.58WAY-339495
CAS :WAY-339495 may have anti-tumor, anti-inflammatory and analgesic activity and can be used to study obesity, cardiovascular disease, diabetes, neurodegenerative diseases, Alzheimer's disease and stroke.Formule :C21H17N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.44MRS2802
CAS :MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.Formule :C10H14F2N2O11P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.1691-(2,3-Dichlorphenyl)-piperazine
CAS :1-(2,3-Dichlorphenyl)-piperazine (DCPP) is a potent DHCR7 inhibitor. DHCR7 is the last enzyme in cholesterol biosynthesis.Formule :C10H12Cl2N2Degré de pureté :98%Couleur et forme :Brown OilMasse moléculaire :231.121-Arachidoyl-sn-glycero-3-phosphocholine
CAS :1-Arachidoyl-sn-glycero-3-phosphocholine is a lysophospholipid (LyP).Formule :C28H58NO7PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :551.74TRC-766
CAS :TRC-766, a negative control of RTC-5 (TRC-382), is a compound that exhibits protein phosphatase 2A (PP2A) binding properties while lacking phosphatase activation capabilities.Formule :C25H24ClF3N2O3SCouleur et forme :SolidMasse moléculaire :524.98Antibiotic K 4
CAS :Antibiotic K 4 is an inhibitor of angiotensin I converting enzyme produced by Actinomadura spiculosospora.Formule :C23H32N3O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.498(Rac)-PD0299685
CAS :<p>(Rac)-PD0299685 is a potent voltage-dependent calcium channel inhibitor for the study of retina-related diseases.</p>Formule :C10H21NO2Degré de pureté :97.20%Couleur et forme :SolidMasse moléculaire :187.28Neuraminic acid
CAS :<p>Neuraminic acid: acidic amino sugar, 9 carbon chain, from pyruvic acid + D-mannosamine, in active mucoproteins.</p>Formule :C9H17NO8Couleur et forme :SolidMasse moléculaire :267.23Orismilast
CAS :LEO-32731 is a bioactive chemical.Formule :C19H15Cl2F2NO7SCouleur et forme :SolidMasse moléculaire :510.29RORγt Inverse agonist 10
CAS :RORγt Inverse agonist 10 is a highly potent, orally bioavailable compound that acts as an antagonist for the retinoic acid receptor-related orphan nuclear receptor gamma t (RORγt). With an IC50 of 51 nM, it effectively inhibits RORγt activity, a key transcription factor regulating genes linked to psoriasis pathogenesis, including [IL-17A], [IL-22], and [IL-23R].Formule :C25H26F6N6O3Couleur et forme :SolidMasse moléculaire :572.5121-Trityl-1H-imidazole
CAS :1-Trityl-1H-imidazole is a useful organic compound for research related to life sciences. The catalog number is T66710 and the CAS number is 15469-97-3.Formule :C22H18N2Couleur et forme :SolidMasse moléculaire :310.4O-allylvanillin
CAS :O-Allylvanillin, an O-allylchalcone derivative, exhibits anti-cancer properties by inhibiting the growth of THP-1, HL60, Hep-G2, and MCF-7 cells with IC50 values of 74.76 μM, 63.52 μM, 90.99 μM, and 90.11 μM, respectively [1].Formule :C11H12O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :192.21Creatinine-D3
CAS :Creatinine-D3 is a deuterium-labeled Creatinine which is a break-down product of creatine phosphate in muscle.Formule :C4H7N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :116.141,2-Dioleoyl-sn-glycero-3-phosphate, sodium salt
1,2-Dioleoyl-sn-glycero-3-phosphate, sodium salt (T64571) is a natural product utilized in life sciences research.Couleur et forme :Odour SolidBoc-His(Boc)-OH.DCHA
CAS :Boc-His(Boc)-OH.DCHA, an amino acid derivative, has a wide range of applications in life science research.Formule :C28H48N4O6Couleur et forme :SolidMasse moléculaire :536.7142-(Methoxycarbonyl)benzoic acid
CAS :2-(Methoxycarbonyl)benzoic acid is a natural product for research related to life sciences. The catalog number is T67426 and the CAS number is 4376-18-5.Formule :C9H8O4Couleur et forme :SolidMasse moléculaire :180.16Valiolamine
CAS :Valiolamine is a useful organic compound for research related to life sciences. The catalog number is T65494 and the CAS number is 83465-22-9.Formule :C7H15NO5Couleur et forme :SolidMasse moléculaire :193.199Epiquinidine
CAS :Epiquinidine, an analogue of quinine, serves as an agonist for ggTas2r1, exhibiting activation at concentrations of 10 μM or higher.Formule :C20H24N2O2Couleur et forme :SolidMasse moléculaire :324.4244-Nitrophenyl N-acetyl-β-D-galactosaminide
CAS :4-Nitrophenyl N-acetyl-β-D-galactosaminide is a useful organic compound for research related to life sciences. The catalog number is T67691 and the CAS number is 14948-96-0.Formule :C14H18N2O8Couleur et forme :SolidMasse moléculaire :342.304DSR-141562
CAS :DSR-141562 is a new compound that can be taken orally and has a specific ability to inhibit phosphodiesterase 1 (PDE1) in the brain. This compound exhibits a preference for inhibiting human PDE1B, with an IC50 value of 43.9 nM. It also shows moderate inhibition of human PDE1A (IC50 = 97.6 nM) and PDE1C (IC50 = 431.8 nM). DSR-141562 is particularly useful in the study of positive symptoms, negative symptoms, and cognitive impairments associated with schizophrenia.Formule :C19H25F3N4O3Couleur et forme :SolidMasse moléculaire :414.42Lichenase
CAS :Lichenase, an enzyme, breaks down β-glucans in grains into GOS, aiding polysaccharide degradation in cell walls.Couleur et forme :Solid
