
Métabolisme
Les inhibiteurs du métabolisme sont des composés qui interfèrent avec les voies métaboliques, modifiant ainsi la production et l'utilisation de l'énergie au sein des cellules. Ces inhibiteurs sont utilisés pour étudier la régulation du métabolisme, le rôle des voies métaboliques dans des maladies telles que le cancer et le diabète, et pour développer de nouvelles stratégies thérapeutiques. Les inhibiteurs du métabolisme peuvent cibler diverses enzymes et processus impliqués dans la glycolyse, l'oxydation des acides gras et d'autres fonctions métaboliques. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de métabolisme de haute qualité pour soutenir vos recherches en biochimie, troubles métaboliques et développement de médicaments.
Sous-catégories appartenant à la catégorie "Métabolisme"
- AhR(42 produits)
- Aminopeptidase(76 produits)
- CETP(20 produits)
- Anhydrase carbonique(196 produits)
- Caséine Kinase(138 produits)
- DHFR(32 produits)
- Décarboxylase(4 produits)
- Déshydrogénase(302 produits)
- FAAH(64 produits)
- FXR(62 produits)
- Facteur Xa(85 produits)
- Synthase des acides gras(37 produits)
- Ferroptose(226 produits)
- GR(3 produits)
- GSNOR(3 produits)
- Glucokinase(57 produits)
- Prolyl-Hydroxylase de HIF/HIF(146 produits)
- HMG-CoA Réductase(34 produits)
- Hydroxylase(36 produits)
- IDO(84 produits)
- LDL(7 produits)
- Lipase(107 produits)
- Lipides(61 produits)
- Lipoxygénase(134 produits)
- MAO(87 produits)
- MPO(2 produits)
- NAMPT(40 produits)
- P450(6 produits)
- PAI-1(26 produits)
- PDE(169 produits)
- PED(1 produits)
- PKM(17 produits)
- PPAR(170 produits)
- Phospholipase(86 produits)
- ROR(47 produits)
- Récepteur de rétinoïdes(22 produits)
- SGK(10 produits)
- Thioredoxine(12 produits)
- Transférase(29 produits)
- Tansporteur(45 produits)
- UGT(4 produits)
- Inhibiteurs de la xanthine oxydase (XO)(9 produits)
Affichez 34 plus de sous-catégories
9182 produits trouvés pour "Métabolisme"
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Fenirofibrate
CAS :Fenirofibrate is a metabolite of Fenofibrate.Formule :C17H17ClO4Couleur et forme :SolidMasse moléculaire :320.77MAGL-IN-5
CAS :MAGL-IN-5 is a non-selective lipase inhibitor.Formule :C18H17N3O5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :355.3410-hydroxy Warfarin
CAS :10-hydroxy Warfarin, a metabolite of (R)-warfarin, is created by CYP3A4 and inhibits CYP2C9 (IC50=1.6μM).Formule :C19H16O5Couleur et forme :SolidMasse moléculaire :324.332Decarbamylsaxitoxin
CAS :Decarbamylsaxitoxin is a biochemical.Formule :C9H16N6O3Couleur et forme :SolidMasse moléculaire :256.266',7'-Epoxybergamottin
CAS :6'7'-Epoxybergamottin: Found in grapefruit; inhibits CYP3A4 (IC50: 0.30 ppm); presents in juice (0.1-7.4 μM); blocks talinolol transport; is insecticidal.Formule :C21H22O5Couleur et forme :SolidMasse moléculaire :354.4Calcitriol lactone
CAS :Calcitriol lactone (1α,25-Dihydroxyvitamin D3-26,23-lactone), a vitamin D3 metabolite, serves as the active form of vitamin D, influencing bone health, cell differentiation, and immune function.Formule :C27H40O5Couleur et forme :SolidMasse moléculaire :444.60DSPE-PEG3400-NYZL1
DSPE-PEG3400-NYZL1 is a PEG compound composed of DSPE and NYZL1. NYZL1 specifically binds to bladder cancer tissues and cells, making DSPE-PEG3400-NYZL1 suitable for drug delivery applications.Couleur et forme :Odour SolidL-Mevalonic acid
CAS :L-Mevalonic acid, a cholesterol precursor, is studied in autoimmune, atherosclerosis, and Alzheimer's research.Formule :C6H12O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :148.16β-Cembrenediol
CAS :β-Cembrenediol (β-CBT) is a natural product from tobacco plants that is found in cigarette smoke condensate.Formule :C20H34O2Couleur et forme :SolidMasse moléculaire :306.49EAAT2 activator 2
EAAT2 activator2 (Compound 4(SF-2)) is a brain-penetrant modulator of excitatory amino acid transporter 2 (EAAT2) with a Ki of 28.7 nM. This compound enhances EAAT2-mediated glutamate uptake and improves synaptic glutamate clearance. EAAT2 activator2 holds potential for research into neurodegenerative diseases, such as amyotrophic lateral sclerosis and Alzheimer's disease.Couleur et forme :Odour Solid14,15-EE-5(Z)-E
CAS :EETs, derivatives of arachidonic acid, act as vasodilators. 14,15-EE-5(Z)-E, a 14,15-EET analog, inhibits EET's effect on vascular smooth muscle relaxation.Formule :C20H36O3Couleur et forme :SolidMasse moléculaire :324.505DSPE-PEG-Maleimide (MW 40000) ammonium
DSPE-PEG-Maleimide (MW 40000) ammonium possesses DSPE phospholipids and maleimide, enabling the preparation of nanoscale lipid carriers. This compound is applicable in drug delivery research.Couleur et forme :Odour SolidXenoclauxin
CAS :Xenoclauxin is a biochemical.Formule :C28H18O11Couleur et forme :SolidMasse moléculaire :530.44113,14-dihydro-15-keto Prostaglandin E1
CAS :13,14-dihydro-15-keto Prostaglandin E1 inhibits ADP-induced platelet aggregation in human isolated platelet-rich plasma (IC50=14.8 μg/mL) and is a PGE1Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.48N-desmethyl Eletriptan
CAS :N-desmethyl Eletriptan, eletriptan's metabolite, forms via CYP3A4 in human liver.Formule :C21H24N2O2SCouleur et forme :SolidMasse moléculaire :368.5Cipepofol glucuronide
Cipepofolglucuronide (Ciprofol Glucuronide) (M4) is a glucuronide metabolite of Ciprofol. This compound does not significantly inhibit P450s or UDP-glucuronosyltransferase (UGT) enzymes and poses a low risk as a perpetrator of drug-drug interactions (DDIs). Cipepofolglucuronide is used in anesthesia research.Couleur et forme :Odour SolidDSPE-PEG3400-NGR
DSPE-PEG3400-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide, which targets tumor vascular antigen CD13. DSPE-PEG3400-NGR can be employed for drug delivery.Couleur et forme :Odour SolidhPL-IN-1
CAS :hPL-IN-1 is a potent reversible pancreatic lipase (PL) inhibitor (IC50=1.86 μM) that can be used to study obesity-related diseases.Formule :C19H11Cl2F2NO3Degré de pureté :98.41%Couleur et forme :SoildMasse moléculaire :410.2VH4127 TFA
VH4127 TFA is a cyclic peptide with a KD of 18 nM for human low-density lipoprotein receptor (hLDLR). It can specifically bind to epidermal growth factor (EGF) LDLR homologous domains in both rodents and humans.Couleur et forme :Odour SolidPregnanetriol
CAS :Pregnanetriol, a metabolite from 17α-hydroxyprogesterone, indicates 21-hydroxylase deficiency when urinary levels are high.Formule :C21H36O3Couleur et forme :SolidMasse moléculaire :336.5166,15-diketo-13,14-dihydro Prostaglandin F1α
CAS :6,15-diketo-13,14-dihydro PGF1α is a metabolite of PGI2.Formule :C20H34O6Couleur et forme :SolidMasse moléculaire :370.48Habenariol
CAS :Habenariol is a substance isolated from the freshwater orchid Habenaria repens, characterized by its significant phenolic antioxidant activity.Formule :C22H26O7Couleur et forme :SolidMasse moléculaire :402.44Creatine Kinase BB (CK-BB) Isoenzyme, Porcine Brain
Creatine Kinase BB (CK-BB) Isoenzyme, derived from Porcine Brain (also known as CPK-1, CKBB isoenzyme, CK-BB), serves as a valuable biological material or organic compound for life science research.Valilactone
CAS :Valilactone is a fatty acid synthase inhibitor, which is produced by a cultured strain of soil actinomycetes.Formule :C22H39NO5Couleur et forme :SolidMasse moléculaire :397.556DSPE-PEG2000-WLSEAGPVVTVRALRGTGSW
DSPE-PEG2000-WLSEAGPVVTVRALRGTGSW is a polyethylene glycol (PEG) compound composed of DSPE and a cardiomyocyte-specific peptide (WLSEAGPVVTVRALRGTGSW). This compound can be utilized for drug delivery.Couleur et forme :Odour Solid17α,20β-Dihydroxy-4-pregnen-3-one
CAS :17α,20β-Dihydroxy-4-pregnen-3-one (17α,20β-DHP) is an endogenous, maturation-inducing steroid that stimulates oocyte maturation in females of several teleostFormule :C21H32O3Couleur et forme :SolidMasse moléculaire :332.482-[dodecyl(2-hydroxyethyl)amino]ethanol
CAS :2-[dodecyl(2-hydroxyethyl)amino]ethanol (N-Lauryldiethanolamine) is a surfactant that can also be used as an emulsifier and wetting agent in skin care products.Formule :C16H35NO2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :273.45CK2-IN-15
CK2-IN-15 (Compound Biv5) is a selective and potent inhibitor of the enzyme protein kinase CK2, with an IC50 value of 51 pM. It significantly reduces the replication of SARS-CoV-2 in HEK-ACE2-TMPRSS2 and Vero cells, and also decreases viral replication in an in vitro model of human nasal epithelial cells. CK2-IN-15 holds potential for research into diseases related to β-coronavirus infections.Couleur et forme :Odour SolidHIV-IN-9
HIV-IN-9 (Compound 2b) is an HIV inhibitor with an IC50 value of 6.65 μg/mL, demonstrating high binding affinity for HIV-RT.Couleur et forme :Odour SolidAcetaminophen Glucuronide sodium salt
CAS :Acetaminophen Glucuronide sodium salt (APAP-glu) is a compound with antipyretic and analgesic activity and potential nephrotoxicity.Formule :C14H16NNaO8Couleur et forme :Off-White Cyrstalline SolidMasse moléculaire :349.27BLX3887
CAS :BLX3887 selectively inhibits 15-LO-1 (IC50 = 32 nM), not 15-LO-2, less on 5-LO/12-LO, and affects eosinophils and dendritic cells.Formule :C10H5Cl3FN3OCouleur et forme :SolidMasse moléculaire :308.5218:1 DGS-NTA(Ni)
CAS :18:1 DGS-NTA(Ni) is a nickel-chelating lipid. It exhibits high affinity for histidine tags and can bind to the histidine tags on recombinant proteins. This compound is useful in the preparation of liposomes and nanomultilamellar vesicles (NMV), which are employed in studies of protein and peptide binding as well as for antigen delivery.Formule :C53H94N2NiO15Couleur et forme :SolidMasse moléculaire :1058.01514O6,10
CAS :514O6,10 functions as an ionizable cationic lipid utilized in creating lipid nanoparticles (LNPs) for in vivo mRNA delivery. In mice, LNPs incorporating 514O6,10 and containing an mRNA reporter primarily target the spleen, lungs, and liver.Formule :C87H172N4O8Masse moléculaire :1402.324-Nitrophenyl Phenylphosphonate
CAS :4-Nitrophenyl phenylphosphonate: stable, easy-to-make 5'-nucleotide phosphodiesterase substrate; hydrolyzes faster than natural options.Formule :C12H10NO5PCouleur et forme :SolidMasse moléculaire :279.194-methoxythio Benzamide
CAS :4-Methoxythio benzamide: synthetic pharmaceutic intermediate & potent in vivo hepatotoxin.Formule :C8H9NOSCouleur et forme :SolidMasse moléculaire :167.23Circumdatin A
CAS :Circumdatin A, a benzodiazepine alkaloid derived from the fungus A. ochraceus, is a fungal metabolite.Formule :C21H19N3O5Couleur et forme :SolidMasse moléculaire :393.399Lys-psi(CH2NH)-trp(nps)-ome
CAS :Lys-psi(CH2NH)-trp(nps)-ome peptide bond replaced by CH2NH group.Formule :C24H31N5O4SCouleur et forme :SolidMasse moléculaire :485.60Triflusulfuron-methyl
CAS :Triflusulfuron-methyl is a triazinylsulfonylurea herbicide.Formule :C17H19F3N6O6SMasse moléculaire :492.43Keto-itraconazole
CAS :Keto-itraconazole is a metabolite of Itraconazole.Formule :C35H36Cl2N8O5Couleur et forme :SolidMasse moléculaire :719.62PDE11A4-IN-1
PDE11A4-IN-1 (compound 23b) is a potent, selective inhibitor of PDE11A4, demonstrating an IC50 of 12 nM and exhibiting high selectivity against PDE1, PDE2,Couleur et forme :Odour SolidAcetoacetyl coenzyme A sodium
CAS :Acetoacetyl-CoA sodium is a key metabolite, with a Km of 1.10 mM at pH 7.5, used in PTB and PHB synthesis.Formule :C25H37N7Na3O18P3SCouleur et forme :SolidMasse moléculaire :917.55Antibacterial agent 132
CAS :Antibacterial agent 132 showed antimicrobial activity against C.Formule :C24H17ClN4OSDegré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :444.94UDP-α-D-Glucose sodium hydrate
UDP-α-D-Glucose sodium hydrate is an endogenous metabolite and a pyrimidine nucleotide sugar, involved in glycosylation reactions during metabolicFormule :C15H24N2Na2O18P2Couleur et forme :SolidMasse moléculaire :628.28γ-Glu-Phe
CAS :γ-Glu-Phe (γ-Glutamylphenylalanine) is a γ-3 glutamyl dipeptide found in sourdough.it is synthesized by Bacillus amyloliquefaciens (GBA) and Aspergillus oryzaeFormule :C14H18N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.3Sapropterin free base
CAS :Sapropterin aids in amino acid breakdown and neurotransmitter synthesis, including dopamine and serotonin, and supports nitric oxide production.Formule :C9H15N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :241.25Glutarylcarnitine lithium
Glutarylcarnitine lithium indicates malonic aciduria, glutaric aciduria I in newborn screenings.Formule :C12H20LiNO6Couleur et forme :SolidMasse moléculaire :281.23Angiotensinogen (1-14), human
CAS :Angiotensinogen (1-14), human,Liver-synthesized globulin. Precursor to angiotensin I.Formule :C83H122N24O19Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1760.01DSPE-PEG1000-THRPPMWSPVWP
DSPE-PEG1000-THRPPMWSPVWP is a PEG compound composed of DSPE and the transferrin receptor (TfR) peptide. The THRPPMWSPVWP peptide binds to TfR and is subsequently internalized into cells expressing TfR.Couleur et forme :Odour SolidAngiotensin I-13C6,15N (human, mouse, rat) TFA
Angiotensin I-13C6,15N (human, mouse, rat) TFA is a labeled version of Angiotensin I, using isotopes 13C and 15N, specifically targeted for human, mouse, and rat studies. This compound serves as a precursor to angiotensin II, which is formed through the cleavage by angiotensin-converting enzyme (ACE).Formule :C5713C6H89N1615NO14·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1303.42 (free base)Dios-Arg (trifluoroacetate salt)
CAS :Dios-Arg, a steroid cationic lipid, binds DNA for transfection, but is cytotoxic to H1299/HeLa cells at 83.5/74.1 μg/ml IC50s.
Formule :C43H67F6N5O9Couleur et forme :SolidMasse moléculaire :912.01

