
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.833 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.875 produits)
- Chromatine/Épigénétique(2.612 produits)
- Signalisation du cytosquelette(1.566 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.014 produits)
- Immunologie et Inflammation(3.900 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.256 produits)
- Transporteur membranaire/Canal ionique(3.154 produits)
- Métabolisme(10.139 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.369 produits)
- Autres inhibiteurs(35.852 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.430 produits)
- Protéases/Protéasome(1.691 produits)
- Cellules souche et Dérivés(733 produits)
- Tyrosine Kinase/Adaptateurs(1.983 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66522 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
IK-930
CAS :IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency.Formule :C19H19F3N4O2SDegré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :424.4418β-Glycyrrhetinic acid
CAS :18β-Glycyrrhetinic acid (Enoxolone) is the major bioactive component of Glycyrrhizae Radix and possesses anti-inflammatory and antiproliferative properties.Formule :C30H46O4Degré de pureté :99.03% - 99.64%Couleur et forme :SolidMasse moléculaire :470.68Hydrocortisone
CAS :Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.Formule :C21H30O5Degré de pureté :98.4% - 99.95%Couleur et forme :Plates From Alc Or Iso-Propyl Alc SolidMasse moléculaire :362.46GSK-LSD1
CAS :GSK-LSD1 is an LSD1 inhibitor that regulates the cell cycle and induces apoptosis, and can be used for the study of breast cancer.Formule :C14H20N2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :216.32Thermolysin
CAS :Thermolysin is an extracellular metalloendopeptidase from Bacillus thermolysinophilus that selectively catalyzes short peptides.Couleur et forme :SolidAdrenocorticotropic hormone TFA
Adrenocorticotropic hormone TFA is an adrenocorticotropic hormone involved in neurohormonal regulation of the body.Degré de pureté :99.71%Couleur et forme :Odour SolidMK-8719
CAS :MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .Formule :C9H14F2N2O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.28Ref: TM-T12070
1mg90,00€5mg177,00€10mg295,00€25mg502,00€50mg710,00€100mg1.009,00€1mL*10mM (DMSO)263,00€Regorafénib N-oxyde (M2)
CAS :Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.
Formule :C21H15ClF4N4O4Degré de pureté :98.03% - 98.26%Couleur et forme :SolidMasse moléculaire :498.81AP20187
CAS :AP20187: Cell-permeable ligand dimerizing FKBP fusion proteins for signaling and gene expression control.Formule :C82H107N5O20Degré de pureté :99.05% - 99.80%Couleur et forme :SolidMasse moléculaire :1482.75Docusate sodium
CAS :Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation.Formule :C20H37NaO7SDegré de pureté :99.34%Couleur et forme :White Wax-Like Solid With Water (Uscg 1999)Masse moléculaire :444.56C527
CAS :C527 is a is a pan DUB enzyme inhibitor. Which has a high potency for the USP1/UAF1 complex (IC50=0.88 μM).Formule :C17H8FNO3Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :293.25Heptaminol hydrochloride
CAS :Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.Formule :C8H20ClNODegré de pureté :98.61%Couleur et forme :White Crystalline PowderMasse moléculaire :181.71Mianserin hydrochloride
CAS :Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formule :C18H21ClN2Degré de pureté :99.63% - 99.82%Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMasse moléculaire :300.83Brivudine
CAS :Brivudine (BVDU), an antiviral medicine, is used in the therapy of herpes zoster.Formule :C11H13BrN2O5Degré de pureté :99.51% - 99.85%Couleur et forme :SolidMasse moléculaire :333.14Bromhexine hydrochloride
CAS :Bromhexine hydrochloride (Bisolvon) is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus.Formule :C14H21Br2ClN2Degré de pureté :99.98%Couleur et forme :White SolidMasse moléculaire :412.59NH2-PEG6-Boc
CAS :NH2-PEG6-Boc is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Formule :C19H39NO8Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :409.51Lonidamine
CAS :Lonidamine (Diclondazolic Acid) is an indazole carboxylic acid derivative, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-Formule :C15H10Cl2N2O2Degré de pureté :97.90%Couleur et forme :White To Light Yellow CrystalMasse moléculaire :321.16Ref: TM-T0239
1g500,00€2mg37,00€5mg50,00€10mg60,00€25mg78,00€50mg109,00€100mg141,00€500mg335,00€1mL*10mM (DMSO)52,00€Pentetic Acid
CAS :Pentetic Acid (Detarex) is an edetate and a chelating agent used in preparing radiopharmaceuticals.Formule :C14H23N3O10Degré de pureté :≥95%Couleur et forme :White Solid PowderMasse moléculaire :393.35Ascaridole
CAS :Ascaridole (NSC-406266) acts as an anthelmintic compound that repels parasitic helminths (worms) in humans and plants and has weak antimalarial activity.Formule :C10H16O2Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :168.23Diclofenac sodium
CAS :Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.
Formule :C14H10Cl2NNaO2Degré de pureté :98.21% - 99.73%Couleur et forme :White Or Off-White PowderMasse moléculaire :318.13Nacubactam
CAS :Nacubactam (OP0595 free acid) is a potent inhibitor of non-β-lactam-β-lactamase with activity against class A and class C β-lactamases.Formule :C9H16N4O7SDegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :324.31Ref: TM-T12166
1mg56,00€5mg119,00€10mg195,00€25mg391,00€50mg590,00€100mg838,00€1mL*10mM (DMSO)133,00€AR-C155858
CAS :AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).Formule :C21H27N5O5SDegré de pureté :98.96% - 99.42%Couleur et forme :SolidMasse moléculaire :461.53Ref: TM-T14316
1mg96,00€5mg283,00€10mg492,00€25mg800,00€50mg1.103,00€100mg1.491,00€1mL*10mM (DMSO)296,00€Streptomycin sulfate
CAS :Streptomycin sulfate (Phytomycin) is a sulfate salt of streptomycin that is a protein synthesis inhibitor.Formule :C21H39N7O12H2SO4Degré de pureté :99.84% - 99.86%Couleur et forme :White To Off-White PowderMasse moléculaire :728.68Fmoc-NH-PEG8-NHS ester
CAS :Fmoc-NH-PEG8-NHS ester is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Formule :C38H52N2O14Degré de pureté :94.69%Couleur et forme :SolidMasse moléculaire :760.82ALK inhibitor 1
CAS :ALK inhibitor 1 is a selective ALK kinase inhibitor.Formule :C23H28BrN7O3SDegré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :562.48Ref: TM-T10285
1mg50,00€5mg110,00€10mg166,00€25mg323,00€50mg447,00€100mg610,00€1mL*10mM (DMSO)136,00€Sodium 2-mercaptoethanesulfonate
CAS :Sodium 2-mercaptoethanesulfonate (Uromitexan) is a sulfhydryl compound used to prevent urothelial toxicity by inactivating metabolites from antineoplastic.Formule :C2H5NaO3S2Degré de pureté :99.88% - 99.89%Couleur et forme :SolidMasse moléculaire :164.18Cloroperone
CAS :Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.Formule :C22H23ClFNO2Degré de pureté :98.40%Couleur et forme :SoildMasse moléculaire :387.88Sulfamethoxypyridazine
CAS :Sulfamethoxypyridazine (CL 13494) is a sulfanilamide antibacterial agent.Formule :C11H12N4O3SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :280.3Etimizol
CAS :Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.Formule :C9H14N4O2Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :210.23PF-4878691
CAS :PF-4878691 (3M-852A) is an effective and selective Toll-like receptor 7 agonists modelled. It is used to dissociate its antiviral and inflammatory activities.Formule :C17H23N5O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :361.46Ref: TM-T16506
1mg46,00€5mg137,00€10mg222,00€25mg485,00€50mg802,00€100mg1.305,00€1mL*10mM (DMSO)150,00€Fendiline hydrochloride
CAS :Fendiline hydrochloride (Fendiline HCl) is a non-selective blocker of calcium channel.Formule :C23H26ClNDegré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :351.91PF-3450074
CAS :PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Formule :C27H27N3O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :425.52Nampt activator-1
CAS :NAMPT Activator-1, EC50: 3.3-3.7 µM, specific niacinamide phosphotransferase stimulant, shields cells, potential neuroprotectant.Formule :C16H17N3O3Degré de pureté :99.84% - 99.98%Couleur et forme :SoildMasse moléculaire :299.32Moguisteine
CAS :Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Formule :C16H21NO5SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :339.41Orelabrutinib
CAS :Orelabrutinib (ICP-022) is an orally active and irreversible inhibitor of Bruton's tyrosine kinase (BTK).Formule :C26H25N3O3Degré de pureté :97.77% - 99.54%Couleur et forme :SolidMasse moléculaire :427.49Ref: TM-T12317
1mg86,00€5mg177,00€10mg299,00€25mg492,00€50mg682,00€100mg897,00€500mg1.791,00€1mL*10mM (DMSO)205,00€CYM50308
CAS :CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).Formule :C20H21F2N3O2SDegré de pureté :99.43% - 99.77%Couleur et forme :SolidMasse moléculaire :405.46Ref: TM-T15032
1mg62,00€5mg140,00€10mg202,00€25mg324,00€50mg455,00€100mg597,00€200mg842,00€500mg1.225,00€Adenosine 5'-monophosphate monohydrate
CAS :Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.
Formule :C10H14N5O7P·H2ODegré de pureté :97.68% - 98.49%Couleur et forme :White PowderMasse moléculaire :365.24SP-8356
CAS :SP-8356 is a potent, orally active inhibitor of cluster of differentiation 147 (CD147) with anti-atherosclerotic effects.Formule :C18H20O4Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :300.35Ref: TM-T12981
1mg66,00€5mg147,00€10mg225,00€25mg425,00€50mg577,00€100mg772,00€200mg1.044,00€1mL*10mM (DMSO)166,00€Diaveridine
CAS :Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.Formule :C13H16N4O2Degré de pureté :99.10%Couleur et forme :White SolidMasse moléculaire :260.29Stachyose tetrahydrate
CAS :Stachyose tetrahydrate (D-Stachyose tetrahydrate) is a tetrasaccharide consisting of two α-D-galactose units, one α-D-glucose unit, and one β-D-fructose unitFormule :C24H50O25Degré de pureté :99.89%Couleur et forme :White To Off White Crystalline PowderMasse moléculaire :738.64Pseudobaptigenin
CAS :Pseudobaptigenin (Psi-baptigenin) is an isoflavone, a flavonoid lipid molecule that is a natural product found in Pterocarpus marsupium, Dalbergia spruceana.Formule :C16H10O5Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :282.25STAT3-IN-1
CAS :STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumorFormule :C28H29NO6Degré de pureté :95.89% - 95.89%Couleur et forme :SolidMasse moléculaire :475.53Ref: TM-T13009
1mg60,00€2mg88,00€5mg131,00€10mg192,00€25mg349,00€50mg523,00€100mg753,00€500mg1.549,00€1mL*10mM (DMSO)137,00€Maltose monohydrate
CAS :D-(+)-Maltose monohydrate (D-(+)-Maltose monohydrate), a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent inFormule :C12H2201·H2ODegré de pureté :98.41%Couleur et forme :PowderMasse moléculaire :360.31N-Acetylprocainamide
CAS :N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmicFormule :C15H23N3O2Degré de pureté :99.65% - 99.74%Couleur et forme :SolidMasse moléculaire :277.36HCV-IN-29
CAS :HCV-IN-29 is a hepatitis C virus (HCV) inhibitor.Formule :C26H32Cl4N6Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :570.38A-395
CAS :A-395 blocks PRC2 (EZH2-EED-SUZ12) interactions, strongly inhibiting the complex with an IC50 of 18 nM.Formule :C26H35FN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :486.65Chitosan oligosaccharide
CAS :Chitosan oligosaccharide (COS) is an oligomer of β-(1→4)-linked D-glucosamine.Formule :C12H24N2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :340.327AZ084
CAS :AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.Formule :C26H34N4O2Degré de pureté :97.12%Couleur et forme :SolidMasse moléculaire :434.57Ref: TM-T10425
1mg66,00€5mg142,00€10mg202,00€25mg358,00€50mg530,00€100mg745,00€1mL*10mM (DMSO)158,00€Lin28-let-7a antagonist 1
CAS :Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formule :C31H29N5O7Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :583.59Ref: TM-T11851
1mg96,00€5mg205,00€10mg313,00€25mg562,00€50mg845,00€100mg1.243,00€1mL*10mM (DMSO)266,00€Fluorothyl
CAS :Fluorothyl (Bis(2,2,2-trifluoroethyl) ether) is a convulsant used in experimental animals.Formule :C4H4F6ODegré de pureté :98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :182.06Nevanimibe hydrochloride
CAS :Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50Formule :C27H40ClN3ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :458.08Ref: TM-T12225L
1mg90,00€5mg192,00€10mg268,00€25mg416,00€50mg532,00€100mg708,00€1mL*10mM (DMSO)212,00€Dibenzosuberone
CAS :Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline.Formule :C15H12ODegré de pureté :99.83%Couleur et forme :Clear To Yellow LiquidMasse moléculaire :208.26Quinestrol
CAS :Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer andFormule :C25H32O2Degré de pureté :99.36% - 99.72%Couleur et forme :SolidMasse moléculaire :364.52Amphotericin B
CAS :Amphotericin B (NSC-527017) is a polyene antifungal agent with broad-spectrum activity against many fungal species.Formule :C47H73NO17Degré de pureté :99.75% - ≥98%Couleur et forme :Deep Yellow Prisms Or Needles From N N-Dimethylformamide Physical Description Bright Yellow Powder (Ntp 1992)Masse moléculaire :924.08Aliskiren hemifumarate
CAS :Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.Formule :C30H53N3O6C4H4O4Degré de pureté :96.18% - 99.21%Couleur et forme :SolidMasse moléculaire :1219.6Zileuton
CAS :Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.Formule :C11H12N2O2SDegré de pureté :98.72% - 99.43%Couleur et forme :Crystalline SolidMasse moléculaire :236.29Fostemsavir Tris
CAS :Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formule :C29H37N8O11PDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :704.62Ref: TM-T10570
1mg54,00€5mg114,00€10mg167,00€25mg268,00€50mg409,00€100mg580,00€1mL*10mM (DMSO)170,00€Amiselimod hydrochloride
CAS :Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Formule :C19H31ClF3NO3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :413.9Ref: TM-T10305
1mg35,00€2mg50,00€5mg75,00€10mg114,00€25mg203,00€50mg334,00€100mg485,00€200mg700,00€1mL*10mM (DMSO)84,00€Tiragolumab
CAS :Tiragolumab, a monoclonal antibody, targets TIGIT and is used with Atezolizumab to treat solid tumors like lung cancer.
Degré de pureté :SDS-PAGE:95.3%;SEC-HPLC:98.8%Couleur et forme :LiquidMasse moléculaire :148.3 kDa6-Methoxy-2-naphthoic acid
CAS :6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.Formule :C12H10O3Degré de pureté :99.25%Couleur et forme :White To Off-White Powder Crystals Crystalline Powder And/Or ChunksMasse moléculaire :202.21Pomisartan 2HCl
Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.
Formule :C31H32Cl2N4O2Degré de pureté :99.88%Couleur et forme :SoildMasse moléculaire :563.52Mometasone furoate
CAS :Mometasone furoate (Sch32088) is a pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA andFormule :C27H30Cl2O6Degré de pureté :99.43% - 99.48%Couleur et forme :Distributed As 0 1% Ointment With A Petrolatum BaseMasse moléculaire :521.43DUPA(OtBu)-OH
CAS :DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.Formule :C23H40N2O9Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :488.57Ref: TM-T11122
2mg34,00€5mg50,00€10mg82,00€25mg123,00€50mg170,00€100mg235,00€200mg334,00€1mL*10mM (DMSO)54,00€Sulfalene
CAS :Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria.Formule :C11H12N4O3SDegré de pureté :99.24% - 99.52%Couleur et forme :White Or Slightly Yellow Crystal PowderMasse moléculaire :280.3Bendamustine hydrochloride
CAS :Bendamustine hydrochloride (EP-3101) (IC50 of 50 μM) is an alkylating agent associated with DNA damage.Formule :C16H21Cl2N3O2·HClDegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :394.72Linaclotide
CAS :Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.Formule :C59H79N15O21S6Degré de pureté :97.93% - 98.71%Couleur et forme :SolidMasse moléculaire :1526.74Ref: TM-T11852
1mg50,00€5mg99,00€10mg177,00€25mg313,00€50mg465,00€100mg662,00€200mg888,00€1mL*10mM (DMSO)255,00€Zolmitriptan
CAS :Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36Deoxycholic acid
CAS :Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.Formule :C24H40O4Degré de pureté :99.91% - 99.91%Couleur et forme :Crystals From Alc SolidMasse moléculaire :392.57Procodazole
CAS :Procodazole (2-Benzimidazolepropionic acid) is a non-specific active immunoprotective agent against viral and bacterial infections.Formule :C10H10N2O2Degré de pureté :98% - 99.35%Couleur et forme :White To Tan Powder Crystals Or Crystalline Powder And/Or ChunksMasse moléculaire :190.2Dexchlorpheniramine Maleate
CAS :Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86Citalopram hydrobromide
CAS :Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, therebyFormule :C20H22BrFN2ODegré de pureté :99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :405.304L-Cycloserine
CAS :L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formule :C3H6N2O2Degré de pureté :99.75% - 99.99%Couleur et forme :Crystals White PowderMasse moléculaire :102.09ZT 52656A hydrochloride
CAS :ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Formule :C19H26ClF3N2ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :390.87FSEN1
CAS :FSEN1 is a novel and highly effective non-competitive FSP1 inhibitor with an IC50 value of 313 nM.Formule :C22H22BrN5OSDegré de pureté :99.54% - 99.97%Couleur et forme :SolidMasse moléculaire :484.41BRD4 Inhibitor-10
CAS :BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).Formule :C25H27N5O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :429.51Ref: TM-T14776
1mg44,00€5mg92,00€10mg147,00€25mg285,00€50mg414,00€100mg583,00€200mg785,00€1mL*10mM (DMSO)100,00€AZD-8529 mesylate
CAS :AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM).Formule :C25H28F3N5O6SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :583.58Nitrendipine
CAS :Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.Formule :C18H20N2O6Degré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :360.36Ref: TM-T0119
1g414,00€10mg35,00€25mg52,00€50mg67,00€100mg113,00€200mg172,00€500mg268,00€1mL*10mM (DMSO)52,00€CXCR7 antagonist-1
CAS :CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.Formule :C21H19FN6ODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :390.41Oxyclozanide
CAS :Oxyclozanide (Oxyclozanid) is a salicylanilide anthelmintic used in grazing animals for fasciola and cestode infestations.Formule :C13H6Cl5NO3Degré de pureté :99.28%Couleur et forme :White To Yellowish PowderMasse moléculaire :401.46Desmethyl Celecoxib
CAS :Demethyl celecoxib, a COX-2 inhibitor with 32 nM IC50, is an anti-inflammatory Celecoxib analog with a 75% yield.
Formule :C16H12F3N3O2SDegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :367.35Rimonabant
CAS :Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formule :C22H21Cl3N4ODegré de pureté :98% - 99.91%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :463.79Capsaicin
CAS :Capsaicin ((E)-Capsaicin) is a natural product extracted from Capsicum annuum, and is a TRPV1 agonist (EC50=0.29 μM).Formule :C18H27NO3Degré de pureté :98.24% - 99.88%Couleur et forme :Pure Dark Red Solid SolidMasse moléculaire :305.41Loxeen
CAS :Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.Formule :C20H25NO·CH4O3SDegré de pureté :99.46%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.52AZD5423
CAS :AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.Formule :C25H21F4N3O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :487.45CHK1-IN-4 hydrochloride
CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).Formule :C18H19BrClN7O2Degré de pureté :99.29%Couleur et forme :SoildMasse moléculaire :480.75PIT
CAS :PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.Formule :C20H16N2O5SDegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :396.42Desbenzyl Donepezil Hydrochloride
CAS :Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.Formule :C17H24ClNO3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :325.83Oxeladin citrate
CAS :Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.Formule :C26H41NO10Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :527.6Glimepiride
CAS :Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.Formule :C24H34N4O5SDegré de pureté :97.84% - 98.87%Couleur et forme :White Cyrstalline SolidMasse moléculaire :490.62Amoxapine
CAS :Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a lesser degree, of serotonin, at adrenergic nerveFormule :C17H16ClN3ODegré de pureté :98.25% - 99.99%Couleur et forme :SolidMasse moléculaire :313.78Procurcumadiol
CAS :Procurcumadiol (5-Hydroxyprocurcumenol) is a natural product found in Curcuma longa and Curcuma phaeocaulis.Formule :C15H22O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :250.33SAR405 R enantiomer
CAS :SAR405 R enantiomer is the less active enantiomer of SAR405. SAR405 is an inhibitor of PIK3C3/Vps34.Formule :C19H21ClF3N5O2Degré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :443.85Ref: TM-T12831
1mg46,00€5mg96,00€10mg149,00€25mg248,00€50mg359,00€100mg502,00€200mg683,00€1mL*10mM (DMSO)94,00€Fosamprenavir Calcium Salt
CAS :Fosamprenavir Calcium Salt (GW433908G) (GW433908G) is a phosphate ester prodrug of the antiretroviral protease inhibitor Amprenavir, with improved solubility.Formule :C25H34CaN3O9PSDegré de pureté :98.68% - 99.24%Couleur et forme :White Microcrystalline NeedlesMasse moléculaire :623.67Fosfomycin calcium
CAS :Fosfomycin calcium (Phosphomycin calcium salt) is a BBB penetrating, broad-spectrum antibiotic by irreversibly inhibiting an early stage in cell wall synthesis.Formule :C3H5CaO4PDegré de pureté :99%Couleur et forme :White Crystal Powder TastelessMasse moléculaire :176.12NBD-556
CAS :NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Formule :C17H24ClN3O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :337.84Ciproquazone
CAS :Ciproquazone has analgesic activity and is used to treat spondylitis.Formule :C19H18N2O2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :306.36RH1
CAS :RH1 is an effective bioreductive agent.Formule :C12H14N2O3Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :234.25Clobetasone butyrate
CAS :Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such asFormule :C26H32ClFO5Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :478.98Promethazine
CAS :Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .Formule :C17H20N2SDegré de pureté :99.76%Couleur et forme :CrystalsMasse moléculaire :284.42Trilostane
CAS :Trilostane (Win 24540) is a synthetic derivative of androstane with adrenocortical suppressive properties.Formule :C20H27NO3Degré de pureté :99.46% - >99.99%Couleur et forme :Tan CrystalsMasse moléculaire :329.43

