Apoptosi
Gli inibitori dell'apoptosi sono composti che prevengono o ritardano il processo di morte cellulare programmata, noto come apoptosi. Questi inibitori sono fondamentali per lo studio dei meccanismi di sopravvivenza cellulare e vengono utilizzati per indagare sulle malattie in cui l'apoptosi è disregolata, come il cancro, i disturbi neurodegenerativi e le malattie autoimmuni. Modulando l'apoptosi, questi inibitori possono aiutare nello sviluppo di terapie mirate a controllare la morte cellulare. Presso CymitQuimica, offriamo una vasta selezione di inibitori dell'apoptosi di alta qualità per supportare le tue ricerche in biologia cellulare, oncologia e campi correlati.
Sottocategorie di "Apoptosi"
- ASK(6 prodotti)
- BCL(11 prodotti)
- Caspasi(125 prodotti)
- FOXO1(3 prodotti)
- IAP(66 prodotti)
- Mdm2(12 prodotti)
- PD-1/PD-L1(125 prodotti)
- PDK(9 prodotti)
- PERK(25 prodotti)
- Chinasi di serina/treonina(15 prodotti)
- Survivin(13 prodotti)
- TNF(92 prodotti)
- c-RET(51 prodotti)
- p53(62 prodotti)
Mostrare 6 più sottocategorie
Trovati 5598 prodotti di "Apoptosi"
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TASIN-1 Hydrochloride
CAS:<p>TASIN-1 Hydrochloride (TASIN-1 HCl) is a selective inhibitor of truncated APC that acts by selectively killing colorectal cancer cells that express truncated</p>Formula:C18H29ClN2O3SPurezza:99.94%Colore e forma:SolidPeso molecolare:388.95BI-6C9
CAS:<p>BI-6C9 is an inhibitor of tBid (Kd = 20 μM).BI-6c9 prevented MOMP and mitochondrial fission, and protected the cells from cell death.</p>Formula:C23H25N3O4S2Purezza:98.39%Colore e forma:SolidPeso molecolare:471.59Palomid 529
CAS:<p>Palomid 529 (SG 00529) has been used in trials studying the treatment of Age-Related Macular Degeneration.</p>Formula:C24H22O6Purezza:98.40% - 98.59%Colore e forma:SolidPeso molecolare:406.43Paroxetine
CAS:<p>Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.</p>Formula:C19H20FNO3Purezza:98.89% - 99.45%Colore e forma:White To Off-White PowderPeso molecolare:329.37Romidepsin
CAS:<p>Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.</p>Formula:C24H36N4O6S2Purezza:99.4% - 99.94%Colore e forma:SolidPeso molecolare:540.7TrxR1-IN-B19
CAS:<p>TrxR1-IN-B19 (TrxR1 IN B19), a TrxR1 inhibitor, selectively kills gastric cancer cells by a small molecule via targeting TrxR1 and ROS-mediated ER stress</p>Formula:C21H22O5Purezza:98.6%Colore e forma:SolidPeso molecolare:354.4PX-12
CAS:<p>PX-12, a Trx-1 inhibitor, promotes apoptosis, reduces HIF-1α/VEGF, and inhibits tumor growth, suggesting use in advanced cancer therapy.</p>Formula:C7H12N2S2Purezza:98% - 99.21%Colore e forma:SolidPeso molecolare:188.31PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36ASTX660
CAS:<p>Tolinapant (ASTX660) is an orally bioavailable cIAP1/2 and XIAP antagonist.Cost-effective and quality-assured.</p>Formula:C30H42FN5O3Purezza:98.33% - 99.85%Colore e forma:SolidPeso molecolare:539.68Lenalidomide hemihydrate
CAS:<p>Lenalidomide hemihydrate inhibits TNF-α (IC50=13nM) and binds CRBN/DDB1 complexes.</p>Formula:C13H13N3O3H2OPurezza:96.22%Colore e forma:SolidPeso molecolare:268.28Fluazinam
CAS:<p>Fluazinam: a pyridinamine fungicide, broad-spectrum, strongly inhibits S. sclerotiorum mycelial growth.</p>Formula:C13H4Cl2F6N4O4Purezza:98% - 99.7%Colore e forma:Light Yellow CrystalsPeso molecolare:465.09NSC348884
CAS:<p>NSC348884, a nucleophosmin inhibitor, disrupts oligomers, induces apoptosis, and inhibits cancer cell growth (IC50: 1.7-4.0 μM).</p>Formula:C38H40N10Purezza:98.69% - 99.91%Colore e forma:SolidPeso molecolare:636.79Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formula:C38H50N6O5Purezza:99.50% - >99.99%Colore e forma:SolidPeso molecolare:670.84Fimasartan
CAS:<p>Fimasartan (BR-A-657), an ARB, treats hypertension and heart failure; safe with hydrochlorothiazide.</p>Formula:C27H31N7OSPurezza:98.96%Colore e forma:SolidPeso molecolare:501.65PCNA-I1
CAS:<p>PCNA-I1 is an inhibitor targeting PCNA chromatin association in prostate cancer.</p>Formula:C17H14N2O2SPurezza:97.64%Colore e forma:SolidPeso molecolare:310.37L-685458
CAS:<p>L-685458 (L-685,458) is a specific and potent inhibitor of A beta PP gamma-secretase activity with Ki of 17 nM.</p>Formula:C39H52N4O6Purezza:99.62% - 99.80%Colore e forma:SolidPeso molecolare:672.85Benzarone
CAS:<p>Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum.</p>Formula:C17H14O3Purezza:99.77%Colore e forma:SolidPeso molecolare:266.29Scoulerine
CAS:<p>Scoulerine is an inhibitor of ß-site amyloid precursor protein cleaving enzyme 1(BACE1).</p>Formula:C19H21NO4Purezza:98.62%Colore e forma:SolidPeso molecolare:327.37KYP-2047
CAS:<p>KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor.</p>Formula:C20H25N3O2Purezza:99.71%Colore e forma:SolidPeso molecolare:339.433-hydroxy-3-phenylpentanamide
CAS:<p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>Formula:C11H15NO2Purezza:98.42%Colore e forma:SolidPeso molecolare:193.24Angelicin
CAS:<p>Angelicin (Isopsoralen), is a furanocoumarin with anti-Y, antiviral, anti-inflammatory activity.</p>Formula:C11H6O3Purezza:99.86% - 99.89%Colore e forma:White SolidPeso molecolare:186.16SP-141
CAS:<p>SP 141 is a MDM2 inhibitor.SP-141 promotes MDM2 auto-ubiquitination and degradation, with anticancer activity.</p>Formula:C22H16N2OPurezza:98.01%Colore e forma:SolidPeso molecolare:324.38MG-101
CAS:<p>MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.</p>Formula:C20H37N3O4Purezza:98% - ≥98%Colore e forma:SolidPeso molecolare:383.53Ceftiofur
CAS:<p>Ceftiofur is a semisynthetic antibiotic, with activity against various gram-positive/negative, anaerobic and aerobic bacteria encountered by domestic animals.</p>Formula:C19H17N5O7S3Purezza:98.26%Colore e forma:SolidPeso molecolare:523.56N-Ethylmaleimide
CAS:<p>N-Ethylmaleimide (NEM) is a reagent for alkylation of free sulfhydryl groups, a cysteine protease inhibitor. Cost-effective and quality-assured.</p>Formula:C6H7NO2Purezza:99.50%Colore e forma:White SolidPeso molecolare:125.13GSK-J4
CAS:<p>GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.</p>Formula:C24H27N5O2Purezza:98.24% - 99.98%Colore e forma:SolidPeso molecolare:417.5NSC 3852
CAS:<p>NSC 3852 is a potent inhibitor of histone deacetylase.</p>Formula:C9H6N2O2Purezza:99.64%Colore e forma:Slightly Yellow To Yellow-Green PowderPeso molecolare:174.163,4 Dichloroisocoumarin
CAS:<p>3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitor</p>Formula:C9H4Cl2O2Purezza:97.94%Colore e forma:SolidPeso molecolare:215.03Thalidomide-NH-CH2-COOH TFA
CAS:<p>2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) is mainly used in compounds Synthesis.</p>Formula:C17H14F3N3O8Purezza:95.00%Colore e forma:SolidPeso molecolare:445.3036BIO-acetoxime
CAS:<p>BIO-acetoxime (GSK-3 Inhibitor X) is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fold selectivity over CDK5/p25, CDK2/cyclin A and CDK1/cyclin B.</p>Formula:C18H12BrN3O3Purezza:97.15%Colore e forma:SolidPeso molecolare:398.21NS-3-008 hydrochloride
CAS:<p>NS-3-008 hydrochloride (NS-3-008 HCl) is a transcriptional G0/G1 switch 2 (G0s2) inhibitor( IC50 of 2.25 μM).</p>Formula:C14H24ClN3Purezza:99.56%Colore e forma:SolidPeso molecolare:269.81Diallyl Trisulfide
CAS:<p>Diallyl Trisulfide is an organic polysulfide compound found in garlic that acts as an H2S donor.</p>Formula:C6H10S3Purezza:95% - ≥98%Colore e forma:LiquidPeso molecolare:178.34KEA1-97
CAS:<p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>Formula:C15H9Cl2FN4Purezza:97.07%Colore e forma:SolidPeso molecolare:335.16Dehydroeffusol
CAS:<p>Dehydroeffusol: anti-cancer, anxiolytic, sedative; halts gastric cancer growth via ER stress and apoptosis.</p>Formula:C17H14O2Purezza:99.35%Colore e forma:SolidPeso molecolare:250.29BMS-202
CAS:<p>BMS-202 (PD1-PDL1 inhibitor 2) is an inhibitor of the PD-1 (Programmed death- 1) /PD-Ll (Programmed death-ligand 1) protein/protein interaction.</p>Formula:C25H29N3O3Purezza:97.92% - 99.66%Colore e forma:SolidPeso molecolare:419.52Spautin-1
CAS:<p>Spautin-1 is an autophagy inhibitor that can suppress the deubiquitination activity of ubiquitin-specific peptidase USP10 and USP13. Cost-effective and quality-assured.</p>Formula:C15H11F2N3Purezza:97.69% - 98.99%Colore e forma:SolidPeso molecolare:271.26LY2409881 trihydrochloride
CAS:<p>LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher.</p>Formula:C24H32Cl4N6OSPurezza:≥95%Colore e forma:SolidPeso molecolare:594.43Valinomycin
CAS:<p>Valinomycin (NSC-122023) is a cyclic depsipeptide antibiotic and a potassium-specific ionophore.Valinomycin induces PINK1 activation and promotes Parkin</p>Formula:C54H90N6O18Purezza:95.37% - 97.16%Colore e forma:White SolidPeso molecolare:1111.32Taurochenodeoxycholic acid sodium
CAS:<p>Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).</p>Formula:C26H44NNaO6SPurezza:98.23% - 99.45%Colore e forma:White To Off-White PowderPeso molecolare:521.68Z-VAD-FMK
CAS:<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formula:C21H28FN3O7Purezza:98.24% - 99.79%Colore e forma:SolidPeso molecolare:453.46PD184161
CAS:<p>PD184161 is a novel, orally-active MEK inhibitor. PD184161 inhibited MEK activity (IC50 = 10-100 nM) in a time- and concentration-dependent manner[1].</p>Formula:C17H13BrClF2IN2O2Purezza:99.40%Colore e forma:SolidPeso molecolare:557.56Rhapontin
CAS:<p>Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.</p>Formula:C21H24O9Purezza:99% - 99.91%Colore e forma:Light YellowPeso molecolare:420.41Perillyl alcohol
CAS:<p>Perillyl Alcohol, a monoterpene with antitumor properties, inhibits protein activation blocking cancer cell growth.</p>Formula:C10H16OPurezza:97.36%Colore e forma:SolidPeso molecolare:152.23Z-DEVD-FMK
CAS:<p>Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,</p>Formula:C30H41FN4O12Purezza:96.19% - 99.69%Colore e forma:SolidPeso molecolare:668.66Caudatin
CAS:<p>Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.</p>Formula:C28H42O7Purezza:98.83% - 99.9%Colore e forma:SolidPeso molecolare:490.63MGCD-265 analog
CAS:<p>Glesatinib, an oral tyrosine kinase inhibitor, targets c-Met and VEGFR2 with IC50s of 29 nM and 10 nM, may treat cancer.</p>Formula:C26H20FN5O2S2Purezza:98.06% - 98.68%Colore e forma:SolidPeso molecolare:517.6Rebastinib
CAS:<p>DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,</p>Formula:C30H28FN7O3Purezza:99.53% - 99.79%Colore e forma:SolidPeso molecolare:553.59SBE13 Hydrochloride
CAS:<p>SBE13 Hydrochloride (SBE 13 HCl) is an effective and specific PLK1 inhibitor (IC50: 0.2 nM); no inhibition om Aurora A kinase, Plk2/3.</p>Formula:C24H28Cl2N2O4Purezza:99.00% - ≥95%Colore e forma:SolidPeso molecolare:479.4ZM 336372
CAS:<p>ZM 336372 is a potent and selective c-Raf inhibitor.</p>Formula:C23H23N3O3Purezza:97.24% - 97.51%Colore e forma:SolidPeso molecolare:389.45TG101209
CAS:<p>TG101209 is a selective JAK2 inhibitor with IC50 of 6 nM.</p>Formula:C26H35N7O2SPurezza:99% - >99.99%Colore e forma:SolidPeso molecolare:509.67Notoginsenoside R1
CAS:<p>Notoginsenoside R1 (Sanchinoside R1) has been shown to exhibit antioxidant, antiapoptotic, anti-inflammatory, and immune-stimulatory properties.</p>Formula:C47H80O18Purezza:99.57% - >99.99%Colore e forma:SolidPeso molecolare:933.13Geranylgeraniol
CAS:<p>Geranylgeraniol (FT0626663) is an isoprenoid found in fruits, vegetables, and grains, including rice.</p>Formula:C20H34OPurezza:99.17% - ≥98%Colore e forma:SolidPeso molecolare:290.48Quizartinib
CAS:<p>Quizartinib (AC220) is an inhibitor of FLT3 (Kd: 1.6 nM) and demonstrates high selectivity for FLT3 when tested against a panel of 227 additional kinases.</p>Formula:C29H32N6O4SPurezza:98% - 99.42%Colore e forma:SolidPeso molecolare:560.67Tamibarotene
CAS:<p>Tamibarotene (Amnolake) is an orally active, synthetic retinoid, developed to overcome all-trans retinoic acid (ATRA) resistance, with potential antineoplastic</p>Formula:C22H25NO3Purezza:98.55% - 99.73%Colore e forma:Crystalline SolidPeso molecolare:351.44(S)-10-Hydroxycamptothecin
CAS:<p>(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma.</p>Formula:C20H16N2O5Purezza:99.09% - 99.81%Colore e forma:SolidPeso molecolare:364.35Midostaurin
CAS:<p>PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.</p>Formula:C35H30N4O4Purezza:97.61% - >99.99%Colore e forma:SolidPeso molecolare:570.64Barasertib-HQPA
CAS:<p>Barasertib-HQPA (AZD2811) is a highly selective Aurora B inhibitor (IC50: 0.37 nM) and demonstrates ~3,700-fold greater selectivity than Aurora A.</p>Formula:C26H30FN7O3Purezza:98.43% - 99.29%Colore e forma:SolidPeso molecolare:507.56All-trans-retinal
CAS:<p>All-trans-retinal (Vitamin A aldehyde) is a one of the major vitamin A metabolites in the retina.</p>Formula:C20H28OPurezza:98.56% - 98.70%Colore e forma:SolidPeso molecolare:284.44Tomatine
CAS:<p>Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.</p>Formula:C50H83NO21Purezza:98.42% - 99.94%Colore e forma:White To Light YellowPeso molecolare:1034.19SSE15206
CAS:<p>SSE15206 is a microtubule polymerization inhibitor that overcomes multidrug resistance.</p>Formula:C19H21N3O3SPurezza:98.81%Colore e forma:SolidPeso molecolare:371.45Ac-DEVD-CHO acetate
<p>Caspase-3 Inhibitor I (N-acetyl-asp-glu-val-asp-al) is a specific inhibitor of Caspase-3.</p>Formula:C22H34N4O13Purezza:98.54%Colore e forma:SolidPeso molecolare:562.52Niraparib tosylate
CAS:<p>Niraparib tosylate (MK-4827 (tosylate))(with IC50 of 3.8 nM/2.1 nM) is a selective PARP1/PARP2 inhibitor.</p>Formula:C19H20N4O·C7H8O3SPurezza:99.34% - 99.87%Colore e forma:SolidPeso molecolare:492.59Tenovin-1
CAS:<p>Tenovin-1 inhibits protein-deacetylating activities of SirT1 and SirT2 and protects against MDM2-mediated p53 degradation, which involves ubiquitination.</p>Formula:C20H23N3O2SPurezza:99.33%Colore e forma:SolidPeso molecolare:369.48CA-5f
CAS:<p>CA-5f is a potent late-stage macroautophagy/autophagy inhibitor via inhibiting autophagosome-lysosome fusion.</p>Formula:C24H24N2O3Purezza:99.69%Colore e forma:SolidPeso molecolare:388.462-tert-Butyl-1,4-benzoquinone
CAS:<p>TBQ, a BHA metabolite, activates Nrf2 and S-arylates Keap1 in RAW264.7 cells.</p>Formula:C10H12O2Purezza:97.19%Colore e forma:SolidPeso molecolare:164.2SBI-0206965
CAS:<p>SBI-0206965 is a potent, selective and cell-permeable autophagy kinase ULK1 inhibitor with IC50 of 108 nM for ULK1 kinase activity and 711 nM for ULK2.</p>Formula:C21H21BrN4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:489.32Copanlisib
CAS:<p>Copanlisib (BAY 80-6946), a PI3K inhibitor, may block tumor growth and improve cancer treatment efficacy.</p>Formula:C23H28N8O4Purezza:99% - 99.88%Colore e forma:SolidPeso molecolare:480.52Tanespimycin
CAS:<p>Tanespimycin (KOS 953) is an Hsp90 inhibitor (IC50=5 nM) and is selective. Tanespimycin depletes intracellular STK38/NDR1. High-Quality, Low-Cost!</p>Formula:C31H43N3O8Purezza:99.07% - 99.83%Colore e forma:Dark Purple SolidPeso molecolare:585.69Palmatine
CAS:<p>Palmatine, also known as Burasaine, inhibits dopamine production and may treat flavivirus, jaundice, dysentery, hypertension, and liver issues.</p>Formula:C21H22NO4Purezza:96.28% - 99.49%Colore e forma:SolidPeso molecolare:352.4D-Pantothenic acid hemicalcium salt
CAS:<p>D-Pantothenic acid hemicalcium salt (Calcium pantothenate), a kind of water soluble vitamin, can reduce the patulin content of the apple juice.</p>Formula:C9H17NO5CaPurezza:98% - 99.89%Colore e forma:White Crystalline PowderPeso molecolare:239.28Niraparib hydrochloride
CAS:<p>Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.</p>Formula:C19H21ClN4OPurezza:99.26%Colore e forma:SolidPeso molecolare:356.85Propylparaben
CAS:<p>Propylparaben (Propyl parahydroxybenzoate) is an antimicrobial agent, preservative, flavouring agent</p>Formula:C10H12O3Purezza:99.84%Colore e forma:White Solid CrystallinePeso molecolare:180.20Navitoclax
CAS:<p>View and buy Navitoclax from TargetMol.Navitoclax (ABT-263) is a potent, orally bioavailable Bcl-2 family protein inhibitor that avidly binds Bcl-2.Cited in 4 publications.</p>Formula:C47H55ClF3N5O6S3Purezza:95.82% - >99.99%Colore e forma:Pale Yellow SolidPeso molecolare:974.61Tivantinib
CAS:<p>Tivantinib (ARQ 197) is an orally bioavailable small molecule inhibitor of c-Met with potential antineoplastic activity.</p>Formula:C23H19N3O2Purezza:98% - 99.41%Colore e forma:SolidPeso molecolare:369.42NSC 66811
CAS:<p>NSC 66811 inhibits MDM2-p53 interaction with 120 nM affinity, activating p53 in cancer cells.</p>Formula:C23H20N2OPurezza:96.94%Colore e forma:SolidPeso molecolare:340.42SKF-96365 hydrochloride
CAS:<p>SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y</p>Formula:C22H27ClN2O3Purezza:99.47% - 99.92%Colore e forma:SolidPeso molecolare:402.91(-)-Epipodophyllotoxin
CAS:<p>(-)-Epipodophyllotoxin: anticancer, GI50=0.36μM (HeLa), 0.24μM (MCF-7), inhibits spindle assembly.</p>Formula:C22H22O8Purezza:99.97%Colore e forma:SolidPeso molecolare:414.41JNJ-7706621
CAS:<p>JNJ-7706621 is a potent aurora kinase inhibitor, and also inhibits CDK1 and CDK2.</p>Formula:C15H12F2N6O3SPurezza:99.1% - 99.85%Colore e forma:SolidPeso molecolare:394.36Mycophenolic acid sodium
CAS:<p>Mycophenolic acid sodium inhibits IMPDH with EC50 of 0.24 μM, has antiviral, immunosuppressive, antiangiogenic, and antitumor properties.</p>Formula:C17H19NaO6Colore e forma:SolidPeso molecolare:342.323TVB-3166
CAS:<p>TVB-3166: reversible, selective FASN inhibitor, induces apoptosis, hinders xenograft growth (IC50: 42 nM FASN, 81 nM palmitate synthesis).</p>Formula:C24H24N4OPurezza:99.53% - 99.57%Colore e forma:SolidPeso molecolare:384.47Liproxstatin-1 hydrochloride
CAS:<p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>Formula:C19H22Cl2N4Colore e forma:SolidPeso molecolare:377.31Alisertib
CAS:<p>Alisertib (MLN 8237) is a specific Aurora A inhibitor (IC50: 1.2 nM). The selectivity of Alisertib(MLN 8237) is >200-fold higher for Aurora A than Aurora B.</p>Formula:C27H20ClFN4O4Purezza:98.31% - >99.99%Colore e forma:SolidPeso molecolare:518.92CVT-11127
CAS:<p>CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.</p>Formula:C25H23Cl2N5O3Purezza:98.32%Colore e forma:SolidPeso molecolare:512.39EPI-001
CAS:<p>EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.</p>Formula:C21H27ClO5Purezza:99% - 99.67%Colore e forma:SolidPeso molecolare:394.89Sirtinol
CAS:<p>Sirtinol is a selective SIRT1/2 inhibitor (IC50: 131/38 μM).</p>Formula:C26H22N2O2Purezza:97.12% - 99.96%Colore e forma:SolidPeso molecolare:394.47DAPK Substrate Peptide acetate
<p>DAPK Substrate Peptide acetate is a death-associated protein kinase (DAPK, Km = 9 μM) peptide substrate.</p>Formula:C70H115N25O17Purezza:98.12%Colore e forma:SolidPeso molecolare:1578.82Atezolizumab
CAS:<p>Atezolizumab is an antibody inhibitor, a humanized monoclonal antibody, IgG1, which targets PD-L1. Atezolizumab has antitumor effect. Cost-effective and quality-assured.</p>Purezza:95.10% - 99.3% （SEC-HPLC）Colore e forma:LiquidPeso molecolare:145 kDaEmbelin
CAS:<p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>Formula:C17H26O4Purezza:97.07% - 99.88%Colore e forma:SolidPeso molecolare:294.39Tubastatin A
CAS:<p>Tubastatin A: Selective HDAC6 inhibitor, IC50 of 15 nM, 1000x less effective on other isozymes except HDAC8.</p>Formula:C20H21N3O2Purezza:97.22% - 99.51%Colore e forma:SolidPeso molecolare:335.47,8-Dihydroxyflavone
CAS:<p>7,8-Dihydroxyflavone (7,8-DHF) is a naturally-occurring flavone and exist in Tridax procumbens, Godmania aesculifolia, and primula tree leaves.</p>Formula:C15H10O4Purezza:98.48% - 99.81%Colore e forma:SolidPeso molecolare:254.24VER-50589
CAS:<p>VER-50589 is a potent HSP90 inhibitor.</p>Formula:C19H17ClN2O5Purezza:99.96% - >99.99%Colore e forma:SolidPeso molecolare:388.8R406 free base
CAS:<p>R406 free base (R406 (free base)) is a potent Syk inhibitor.</p>Formula:C22H23FN6O5Purezza:97.64% - 99.11%Colore e forma:SolidPeso molecolare:470.45Concanavalin A
CAS:<p>Concanavalin A is a natural product, a phytoalexin. Concanavalin A has antitumor activity and can also induce acute liver injury. Cost effective and quality assured.</p>Formula:C23H32N6O8SPurezza:98%Colore e forma:SolidPeso molecolare:104-112 kDaPuromycin aminonucleoside
CAS:<p>Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner.</p>Formula:C12H18N6O3Purezza:99.85% - 99.9%Colore e forma:SolidPeso molecolare:294.31R406
CAS:<p>R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.</p>Formula:C22H23FN6O5·C6H6O3SPurezza:97.67% - 98.82%Colore e forma:SolidPeso molecolare:628.63Niraparib
CAS:<p>Niraparib (MK-4827) inhibits PARP1/PARP2 (IC50: 3.8/2.1 nM), effective on BRCA mutant cancers, 330x less effective on PARP3, V-PARP, Tank1.</p>Formula:C19H20N4OPurezza:98% - 99.91%Colore e forma:SolidPeso molecolare:320.39GSK 3 Inhibitor IX
CAS:<p>GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex.</p>Formula:C16H10BrN3O2Purezza:98% - 99.72%Colore e forma:SolidPeso molecolare:356.17MG 149
CAS:<p>MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).</p>Formula:C22H28O3Purezza:98.69% - 99.86%Colore e forma:SolidPeso molecolare:340.46FR 180204
CAS:<p>FR 180204 is a potent and selective ATP-competitive inhibitor of ERK1 and ERK2.</p>Formula:C18H13N7Purezza:98% - 99.74%Colore e forma:SolidPeso molecolare:327.34Selonsertib
CAS:<p>Selonsertib (GS-4997), an oral ASK1 inhibitor, may have anti-inflammatory, anti-fibrotic, and anti-cancer effects.</p>Formula:C24H24FN7OPurezza:95.04% - 99.53%Colore e forma:SolidPeso molecolare:445.49Bruceine D
CAS:<p>1.</p>Formula:C20H26O9Purezza:95% - 99.99%Colore e forma:SolidPeso molecolare:410.42Salermide
CAS:<p>Salermide is an inhibitor of Sirt1 and Sirt2, causing strong cancer-specific apoptotic cell death.</p>Formula:C26H22N2O2Purezza:97.09% - 99.55%Colore e forma:SolidPeso molecolare:394.47Trametinib
CAS:<p>Trametinib (GSK1120212), an ATP-noncompetitive MEK 1/2 inhibitor (IC50: 0.7/0.9 nM), weakly inhibits >180 kinases.</p>Formula:C26H23FIN5O4Purezza:98% - 99.96%Colore e forma:SolidPeso molecolare:615.39Wogonin
CAS:<p>Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.</p>Formula:C16H12O5Purezza:98% - 99.8%Colore e forma:Yellow CrystalPeso molecolare:284.26Dubermatinib
CAS:<p>Dubermatinib (TP0903) is a potent and selective Axl kinase inhibitor.</p>Formula:C24H30ClN7O2SPurezza:98.65% - 99.58%Colore e forma:SolidPeso molecolare:516.06Formosanin C
CAS:<p>Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity.</p>Formula:C51H82O20Purezza:99.75% - >99.99%Colore e forma:SolidPeso molecolare:1015.18WYC-209
CAS:<p>WYC-209 inhibits proliferation of malignant murine melanoma tumor-repopulating cells (TRCs, IC50: 0.19 uM). It targets the retinoic acid receptor (RAR).</p>Formula:C20H20N2O3SPurezza:99.77%Colore e forma:SolidPeso molecolare:368.45KW-2449
CAS:<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Formula:C20H20N4OPurezza:98.43% - 99.69%Colore e forma:SolidPeso molecolare:332.4Kevetrin hydrochloride
CAS:<p>Kevetrin hydrochloride (4-Isothioureidobutyronitrile hydrochloride) is a small molecule and activator of the tumor suppressor protein p53, with potential</p>Formula:C5H10ClN3SPurezza:99.32% - 99.93%Colore e forma:SolidPeso molecolare:179.67Nafamostat mesylate
CAS:<p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>Formula:C19H17N5O2·2CH4O3SPurezza:97.36% - 99.76%Colore e forma:Tan To Pale Orange SolidPeso molecolare:539.58Osthole
CAS:<p>Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.</p>Formula:C15H16O3Purezza:99.93% - 99.96%Colore e forma:Fine White PowderPeso molecolare:244.298-Prenylnaringenin
CAS:<p>8-Prenylnaringenin is a phytoestrogen with high estrogenic activity,</p>Formula:C20H20O5Purezza:98.26% - 99.46%Colore e forma:SolidPeso molecolare:340.37Tauroursodeoxycholate dihydrate
CAS:<p>Tauroursodeoxycholate (TUDCA ,Taurolite) dihydrate is a bile acid that reduces Caspase-3, Caspase-12, ERK, reducing endoplasmic reticulum stress mediated death.</p>Formula:C26H49NO8SPurezza:99.82%Colore e forma:SolidPeso molecolare:535.73Astragalin
CAS:<p>Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid.</p>Formula:C21H20O11Purezza:98.8% - ≥95%Colore e forma:SolidPeso molecolare:448.38Phellamurin
CAS:<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Formula:C26H30O11Purezza:97.91%Colore e forma:SolidPeso molecolare:518.51Cyasterone
CAS:<p>Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via regulating EGFR signaling pathway, it may be a promising</p>Formula:C29H44O8Purezza:99.32% - 99.70%Colore e forma:SolidPeso molecolare:520.65Bomedemstat
CAS:<p>Bomedemstat (IMG-7289),Irreversible LSD1 inhibitor. Active in MPN models. Antineoplastic effects. Used in AML and myelofibrosis research.</p>Formula:C28H34FN7O2Purezza:99.00%Colore e forma:SolidPeso molecolare:519.61Pracinostat
CAS:<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Formula:C20H30N4O2Purezza:99.15% - 99.67%Colore e forma:SolidPeso molecolare:358.48MK-2206 dihydrochloride
CAS:<p>MK-2206 dihydrochloride (MK-2206 2HCl) is a variant Akt inhibitor that inhibits Akt1, Akt2, and Akt3 (IC50=8/12/65 nM) with orally active, highly potent and</p>Formula:C25H23Cl2N5OPurezza:99.228% - 99.94%Colore e forma:SolidPeso molecolare:480.39UAMC-3203 hydrochloride
CAS:<p>UAMC-3203 hydrochloride is a potent and selective Ferroptosis inhibitor with an IC50 of 12 nM.</p>Formula:C25H38ClN5O2SPurezza:99.62%Colore e forma:SolidPeso molecolare:508.12Asiaticoside
CAS:<p>Asiaticoside, in Centella asiatica, may treat wounds/burns.</p>Formula:C48H78O19Purezza:98% - 99.96%Colore e forma:PowderPeso molecolare:959.12STF-118804
CAS:<p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 <10 nM.</p>Formula:C25H23N3O4SPurezza:98.66%Colore e forma:SolidPeso molecolare:461.53SKI II
CAS:<p>SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.</p>Formula:C15H11ClN2OSPurezza:99.34% - 99.93%Colore e forma:SolidPeso molecolare:302.78NSC 95397
CAS:<p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>Formula:C14H14O4S2Purezza:98.66%Colore e forma:SolidPeso molecolare:310.39S-trityl-L-Cysteine
CAS:<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Formula:C22H21NO2SPurezza:97.02%Colore e forma:Almost White To Light Yellow Granular PowderPeso molecolare:363.47LRRK2-IN-1
CAS:<p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>Formula:C31H38N8O3Purezza:98% - 98.82%Colore e forma:SolidPeso molecolare:570.69Glyphosate
CAS:<p>Glyphosate (Atila) is an herbicide. It also is a possible carcinogen to humans.</p>Formula:C3H8NO5PPurezza:99.12% - 99.91%Colore e forma:White Crystals (Darkens) Ph (1% Solution In Water) 2 5 (Ntp 1992)Peso molecolare:169.07HO-3867
CAS:<p>HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.</p>Formula:C28H30F2N2O2Purezza:91.18% - 99.21%Colore e forma:SolidPeso molecolare:464.55WT-161
CAS:<p>WT161 is a potent and selective inhibitor of HDAC6 (IC50:0.40 nM).</p>Formula:C27H30N4O3Purezza:95.98% - 98.34%Colore e forma:SolidPeso molecolare:458.55JX06
CAS:<p>JX06, a potent, selective and covalent PDK inhibitor, inhibits PDK1, PDK2 and PDK3 with IC50 of 49 nM, 101 nM and 313 nM respectively.</p>Formula:C10H16N2O2S4Purezza:99.4%Colore e forma:SolidPeso molecolare:324.51Dictamine
CAS:<p>Dictamine (Dectamine) shows anticholinesterase, anti-inflammatory, mutagenic, and has antimicrobial activity against bacteria and fungi.</p>Formula:C12H9NO2Purezza:99.72% - 99.889%Colore e forma:SolidPeso molecolare:199.21Baicalein monohydrate
CAS:<p>Baicalein monohydrate blocks 12-lipoxygenase, curbs leukotrienes, lysosomal enzymes, Ca2+ dynamics, and fights arthritis.</p>Formula:C15H12O6Colore e forma:SolidPeso molecolare:288.25Quisinostat
CAS:<p>Quisinostat (JNJ-26481585), a second-gen HDAC inhibitor, is most potent for HDAC1 (IC50 0.11 nM) and selectively affects HDACs 2, 4, 10, and 11.</p>Formula:C21H26N6O2Purezza:96.01% - ≥98%Colore e forma:SolidPeso molecolare:394.47Elesclomol
CAS:<p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>Formula:C19H20N4O2S2Purezza:97.17% - 99.51%Colore e forma:SolidPeso molecolare:400.52LCL161
CAS:<p>LCL161 is a SMAC mimetic, an IAP antagonist with oral activity that inhibits XIAP and cIAP1. LCL161 has potential antitumor activity. Cost-effective and quality-assured.</p>Formula:C26H33FN4O3SPurezza:99.13% - 99.87%Colore e forma:SolidPeso molecolare:500.63α-Hederin
CAS:<p>Alpha-Hederin (Tauroside E) is a water-soluble pentacyclic triterpenoid saponin found in the seeds of Nigella sativa, with hemolytic and apoptotic properties.</p>Formula:C41H66O12Purezza:99.44% - 99.89%Colore e forma:SolidPeso molecolare:750.96A-1331852
CAS:<p>A-1331852 is a potent and selectiveBCL-XL inhibitor and may be useful in the treatment of cancer, immune and autoimmune diseases.</p>Formula:C38H38N6O3SPurezza:98.15% - >99.99%Colore e forma:SolidPeso molecolare:658.81Guggulsterone
CAS:<p>Guggulsterone (Guggulsterone E&Z) E&Z is a 3-hydroxy steroid. It has a role as an androgen.</p>Formula:C21H28O2Purezza:99.4% - 99.8%Colore e forma:Light Yellow PowderPeso molecolare:312.45SGI-1776
CAS:<p>SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.</p>Formula:C20H22F3N5OPurezza:99.3% - >99.99%Colore e forma:SolidPeso molecolare:405.42L-Asparaginase
CAS:<p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>Formula:NAPurezza:97%Colore e forma:SolidPeso molecolare:N/ABV6
CAS:<p>BV6 is an antagonist of c-IAP1 and XIAP, members of the inhibitors of apoptosis (IAP) family.</p>Formula:C70H96N10O8Purezza:97.46% - 99.82%Colore e forma:SolidPeso molecolare:1205.57O6-Benzylguanine
CAS:<p>O6-Benzylguanine is a guanine analog with antineoplastic activity,and is a potent O6-alkylguanine DNA alkyltransferase (AGT) inactivator.</p>Formula:C12H11N5OPurezza:98.9%Colore e forma:Solid CrystallinePeso molecolare:241.25CCT128930 hydrochloride
CAS:<p>CCT128930 hydrochloride: Potent AKT inhibitor (IC50=6 nM), 28x selective over PKA, 20x over p70S6K, induces cell cycle arrest & DNA damage.</p>Formula:C18H21Cl2N5Purezza:98.55%Colore e forma:SolidPeso molecolare:378.3BMS-536924
CAS:<p>BMS-536924 (BMS 536924) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for</p>Formula:C25H26ClN5O3Purezza:99.02%Colore e forma:SolidPeso molecolare:479.96Genistein
CAS:<p>Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has antitumor effects. Cost effective and quality assured.</p>Formula:C15H10O5Purezza:98.22% - 99.64%Colore e forma:Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether SolidPeso molecolare:270.24(1E,6E)-Bis(demethoxy)curcumin
CAS:<p>(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) is a natural demethoxy derivative of curcumin,with anti-inflammatory and anti-cancer activities.</p>Formula:C19H16O4Purezza:97.45%Colore e forma:SolidPeso molecolare:308.33GDC-0152
CAS:<p>GDC-0152 is a potent inhibitor of IAPs.</p>Formula:C25H34N6O3SPurezza:97.18% - 99.32%Colore e forma:SolidPeso molecolare:498.64Avitinib
CAS:<p>Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor,</p>Formula:C26H26FN7O2Purezza:99.81% - >99.99%Colore e forma:SolidPeso molecolare:487.53AZ 628
CAS:<p>AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM, 34 nM and 29 nM, also inhibits VEGFR2, DDR2, Lyn, Flt1, FMS, etc.</p>Formula:C27H25N5O2Purezza:99.50%Colore e forma:SolidPeso molecolare:451.52SGI-1027
CAS:<p>SGI-1027 (DNA Methyltransferase Inhibitor II) is an effective and selective inhibitor of DNA methyltransferase (DNMT).</p>Formula:C27H23N7OPurezza:99.45% - 99.78%Colore e forma:SolidPeso molecolare:461.52RO8994
CAS:<p>RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).</p>Formula:C31H31Cl2FN4O4Purezza:99.31% - 99.44%Colore e forma:SolidPeso molecolare:613.51Rotenone
CAS:<p>Rotenone, a plant-derived insecticide, inhibits mitochondrial electron transport, found in Leguminosae.</p>Formula:C23H22O6Purezza:89.58% - 99.88%Colore e forma:Less To Brownish Crystals Or A White To Brownish-White Crystalline Powder Has Neither Odor Nor Taste (Ntp 1992)Peso molecolare:394.42LY2857785
CAS:<p>LY2857785 is a type I competitive and reversible ATP kinase inhibitor against CDK7/CDK8/CDK9 (IC50s: 246 nM/16 nM/11 nM).</p>Formula:C26H36N6OPurezza:99.68%Colore e forma:Solid PowderPeso molecolare:448.6Supinoxin
CAS:<p>Supinoxin (RX-5902) is an oral anti-cancer drug targeting p68 RNA helicase, inducing apoptosis in TNBC cells (IC50: 10-20nM).</p>Formula:C22H24FN5O4Purezza:99.83% - 99.95%Colore e forma:SolidPeso molecolare:441.462-Deoxy-D-glucose
CAS:<p>2-Deoxy-D-glucose (2-DG) is an analog of glucose, an inhibitor of glycolysis.</p>Formula:C6H12O5Purezza:99.31% - ≥98%Colore e forma:White PowderPeso molecolare:164.16Apomine
CAS:<p>Apomine (SR-9223i) 是一种 HMG-CoA-还原酶抑制剂，可在体外促进骨髓瘤细胞的凋亡，并与体内骨髓瘤的调节有关。 Apomine 加速 3-羟基-3-甲基戊二酰-CoA 还原酶的降解并刺激低密度脂蛋白受体活性。 Apomine 通过下调 3-羟基-3-甲基戊二酰-CoA 还原酶来增强洛伐他汀对骨髓瘤细胞的抗肿瘤作用。</p>Formula:C28H52O7P2Purezza:>99.99%Colore e forma:SolidPeso molecolare:562.661-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea
CAS:<p>SC-1 is a a derivative of the multiple tyrosine kinase inhibitor sorafenib.</p>Formula:C21H13ClF3N3O2Purezza:99.41%Colore e forma:SolidPeso molecolare:431.8PF-4989216
CAS:<p>PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.</p>Formula:C18H13FN6OSPurezza:99.85%Colore e forma:SolidPeso molecolare:380.4Epibrassinolide
CAS:<p>Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator with</p>Formula:C28H48O6Purezza:97.57% - 98.11%Colore e forma:SolidPeso molecolare:480.68Purvalanol A
CAS:<p>Purvalanol A (NG-60) is an effective and cell-permeable CDK inhibitor with IC50 of 70/4/35/850 nM for cdk2-cyclin A/B/E, and cdk4-cyclin D1, respectively.</p>Formula:C19H25ClN6OPurezza:98.13% - 99.68%Colore e forma:PowderPeso molecolare:388.89Temsirolimus
CAS:<p>Temsirolimus (CCI-779) is a specific mTOR inhibitor ( IC50: 1.76 μM), used in the treatment of advanced renal cell cancer.</p>Formula:C56H87NO16Purezza:97.76% - >99.99%Colore e forma:White Crystalline PowderPeso molecolare:1030.29Licochalcone D
CAS:<p>Licochalcone D may treat melanoma and heart injury, halt cell spread, and reduce inflammation and allergies.</p>Formula:C21H22O5Purezza:99.03% - 99.9%Colore e forma:SolidPeso molecolare:354.4GSK1324726A
CAS:<p>GSK1324726A (I-BET726) is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM).</p>Formula:C25H23ClN2O3Purezza:98.34% - 99.85%Colore e forma:SolidPeso molecolare:434.91MPI-0479605
CAS:<p>MPI-0479605 is an ATP competitive and selective inhibitor.</p>Formula:C22H29N7OPurezza:97.59% - >99.99%Colore e forma:SolidPeso molecolare:407.51TCS-PIM-1-4a
CAS:<p>SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).</p>Formula:C11H6F3NO2SPurezza:99.89%Colore e forma:SolidPeso molecolare:273.23Dihydrorotenone
CAS:<p>Dihydrorotenone is a potent mitochondrial inhibitor and probably induces Parkinsonian syndrome.</p>Formula:C23H24O6Purezza:98.98% - 99.58%Colore e forma:SolidPeso molecolare:396.43GSK778 hydrochloride
CAS:<p>GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to 143 nM, effective in cancer models.</p>Formula:C30H34ClN5O3Purezza:97.26% - 98.35%Colore e forma:SolidPeso molecolare:548.08GSK2334470
CAS:<p>GSK2334470 is a novel PDK1 inhibitor (IC50: ~10 nM, in a cell-free assay), with no inhibitory at other close related AGC-kinases.</p>Formula:C25H34N8OPurezza:99.57% - 99.87%Colore e forma:SolidPeso molecolare:462.59Methyl protodioscin
CAS:<p>Methyl protodioscin boosts HDL, lowers LDL and triglycerides, has anti-cancer effects, and promotes apoptosis via mitochondrial pathways.</p>Formula:C52H86O22Purezza:99.308% - 99.73%Colore e forma:SolidPeso molecolare:1063.23Scriptaid
CAS:<p>Scriptaid (GCK1026) is an inhibitor of HDAC, and has a greater effect on acetylated H4 than H3.</p>Formula:C18H18N2O4Purezza:96.74% - 99.45%Colore e forma:SolidPeso molecolare:326.35Pyroxamide
CAS:<p>Pyroxamide is an histone deacetylases (HDACs) inhibitor with antineoplastic properties ( HDAC1;IC50: 0.1-0.2 μM).</p>Formula:C13H19N3O3Purezza:98.46%Colore e forma:SolidPeso molecolare:265.31Ginsenoside Rg6
CAS:<p>Ginsenoside Rg6 inhibits the proliferation and induces apoptosis of human lymphoma JK cells</p>Formula:C42H70O12Purezza:97.34%Colore e forma:SolidPeso molecolare:767Teneligliptin hydrobromide
CAS:<p>Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.</p>Formula:C22H30N6OSBrHPurezza:97.83% - 99.92%Colore e forma:SolidPeso molecolare:628.86Flurbiprofen Axetil
CAS:<p>Flurbiprofen Axetil (Lipfen) is an anti-inflammatory used as an analgesic.</p>Formula:C19H19FO4Purezza:97.58% - 98%Colore e forma:SolidPeso molecolare:330.35Asperosaponin VI
CAS:<p>Asperosaponin VI, from Dipsacus asper rhizome, treats back pain, hematoma, and fractures.</p>Formula:C47H76O18Purezza:97.15% - 99.79%Colore e forma:SolidPeso molecolare:929.1Radotinib
CAS:<p>Radotinib (IY-5511), and sometimes referred to by its investigational name IY5511, is a drug for the treatment of different types of Y, most notably</p>Formula:C27H21F3N8OPurezza:99.13% - 99.97%Colore e forma:SolidPeso molecolare:530.5NSC 73150
CAS:<p>6-Methyl-1H-pyrimidin-4-one (NSC 73150) shows antitumor effects, impeding growth in breast, lung, liver cancer, and inducing apoptosis.</p>Formula:C12H12N4O2Purezza:99.84%Colore e forma:SolidPeso molecolare:244.25Phthalazinone pyrazole
CAS:<p>Phthalazinone pyrazole: a potent, selective oral Aurora-A kinase inhibitor, overexpressed in tumors with oncogenic activity.</p>Formula:C18H15N5OPurezza:97.03%Colore e forma:SolidPeso molecolare:317.34TAS6417
CAS:<p>Zipalertinib (TAS6417, CLN-081) is a novel, highly potent, orally active covalent EGFR tyrosine kinase inhibitor.Cost-effective and quality-assured.</p>Formula:C23H20N6OPurezza:99.71%Colore e forma:SolidPeso molecolare:396.44BMS-833923
CAS:<p>BMS-833923 (XL-139), an orally bioavailable Smoothened antagonist, inhibits BODIPY cyclopamine binding to SMO in a dose-dependent manner (IC50: 21 nM).</p>Formula:C30H27N5OPurezza:99.47% - 99.76%Colore e forma:SolidPeso molecolare:473.57EI1
CAS:<p>EI1 (Ezh2 inhibitor) is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively.</p>Formula:C23H26N4O2Purezza:99.93%Colore e forma:SolidPeso molecolare:390.48KRIBB11
CAS:<p>KRIBB11 is an inhibitor of Heat shock factor (HSF) inhibitor.</p>Formula:C13H12N6O2Purezza:97.25% - 99.91%Colore e forma:SolidPeso molecolare:284.27pimpinellin
CAS:<p>Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity.</p>Formula:C13H10O5Purezza:99.85% - ≥95%Colore e forma:SolidPeso molecolare:246.22β-Lapachone
CAS:<p>β-Lapachone (ARQ-501) is a specific DNA topoisomerase I inhibitor, and no inhibitory activities against DNA topoisomerase II or ligase.</p>Formula:C15H14O3Purezza:99.76% - 99.88%Colore e forma:SolidPeso molecolare:242.27MX69
CAS:<p>MX69 is the MDM2/XIAP inhibitor, blocking the MDM2 protein-XIAP RNA interaction, leading to MDM2 degradation.</p>Formula:C27H26N2O4SPurezza:97.27% - 99.57%Colore e forma:SolidPeso molecolare:474.57Isatin
CAS:<p>Isatin (2,3-Indolinedione) is an endogenous MAO inhibitor.</p>Formula:C8H5NO2Purezza:98.92%Colore e forma:Yellow To Reddish Crystalline SolidPeso molecolare:147.13BDA-366
CAS:<p>BDA-366, a potent Bcl2 antagonist, selectively binds the Bcl2-BH4 domain with high affinity (Ki = 3.3 nM), inducing a conformational change that nullifies its</p>Formula:C24H29N3O4Purezza:98.61%Colore e forma:SoildPeso molecolare:423.5Glaucocalyxin A
CAS:<p>Glaucocalyxin A improves drug delivery, activates apoptosis, inhibits cell growth, with potential as an antiplatelet agent.</p>Formula:C20H28O4Purezza:99.55% - 99.80%Colore e forma:SolidPeso molecolare:332.433BDO
CAS:<p>3BDO is a new mTOR activator. 3BDO inhibits autophagy.</p>Formula:C18H17NO5Purezza:97.76%Colore e forma:SolidPeso molecolare:327.33UNC1215
CAS:<p>UNC1215, a potent MBT antagonist, targets L3MBTL3 with high selectivity (IC50: 40 nM, Kd: 120 nM, 50x versus MBT family).</p>Formula:C32H43N5O2Purezza:98% - 99.04%Colore e forma:SolidPeso molecolare:529.72Sodium dichloroacetate
CAS:<p>Sodium dichloroacetate (BCA) inhibits PDK (IC50: 183 μM PDK2, 80 μM PDK4), triggers cancer cell apoptosis, and impedes tumor growth.</p>Formula:C2HCl2NaO2Purezza:99.32% - 99.87%Colore e forma:White PowderPeso molecolare:150.92Lupeol
CAS:<p>Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.</p>Formula:C30H50OPurezza:98% - 99.96%Colore e forma:Needles From Alcohol Acetone White PowderPeso molecolare:426.72Suberoyl bis-hydroxamic acid
CAS:<p>SBHA is an HDAC inhibitor, an enzyme key to transcription, cell cycle, and development.</p>Formula:C8H16N2O4Purezza:99.88%Colore e forma:SolidPeso molecolare:204.22Aminopurvalanol A
CAS:<p>Aminopurvalanol A is a competitive, selective and cell-permeable inhibitor of cyclin-dependent kinase (CDK) that potently inhibits Cyclin A/cdk2, Cyclin B/cdk1</p>Formula:C19H26ClN7OPurezza:99.73%Colore e forma:SolidPeso molecolare:403.91Ganetespib
CAS:<p>Ganetespib (STA-9090) is a synthetic small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity.</p>Formula:C20H20N4O3Purezza:98% - 99.95%Colore e forma:SolidPeso molecolare:364.4FLLL32
CAS:<p>FLLL32 is an effective JAK2/STAT3 inhibitor (IC50 of <5 μM).</p>Formula:C28H32O6Purezza:97% - 97.90%Colore e forma:SolidPeso molecolare:464.55Nur77 modulator 1
CAS:<p>Nur77 modulator 1: binds at 3.58 μM, boosts expression, alters location, triggers ER stress/autophagy, induces apoptosis, and fights hepatoma.</p>Formula:C28H25N5O2SPurezza:99.62%Colore e forma:SolidPeso molecolare:495.6Polyporenic acid C
CAS:<p>Polyporenic acid C shows inhibitory activity against human collagenase.</p>Formula:C31H46O4Purezza:96.84% - 99.71%Colore e forma:SolidPeso molecolare:482.69PD-1/PD-L1-IN-10
CAS:<p>PD-1/PD-L1-IN-10 is an orally available PD-1/PD-L1 inhibitor (IC50 value of 2.7 nM) that shows anti-tumor activity.Cost-effective and quality-assured.</p>Formula:C33H31N3O7Purezza:99.63%Colore e forma:SolidPeso molecolare:581.62
