
Ciclo cellulare/Checkpoint
Gli inibitori del ciclo cellulare/dei checkpoint sono composti che interrompono la normale progressione del ciclo cellulare, in particolare nei principali punti di controllo regolatori. Questi inibitori sono fondamentali per studiare la divisione cellulare, comprendere la proliferazione delle cellule cancerose e sviluppare terapie antitumorali. Mirando a fasi specifiche del ciclo cellulare, questi inibitori possono indurre l'arresto del ciclo cellulare, portando all'apoptosi o alla senescenza nelle cellule che si dividono rapidamente. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità del ciclo cellulare/dei checkpoint per supportare le tue ricerche in biologia del cancro, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Ciclo cellulare/Checkpoint"
- Chinasi aurora(114 prodotti)
- CDK(545 prodotti)
- Arresto del ciclo cellulare(5 prodotti)
- Chk(48 prodotti)
- DYRK(47 prodotti)
- Dynamin(27 prodotti)
- Ferroptosi(226 prodotti)
- HSP(179 prodotti)
- Integrina(249 prodotti)
- Chinesina(87 prodotti)
- LIM chinasi(20 prodotti)
- Microtubulo associato(274 prodotti)
- PKC(124 prodotti)
- PLK(25 prodotti)
- ROCK(62 prodotti)
- Rho(6 prodotti)
- Wee1(14 prodotti)
- c-Myc(76 prodotti)
Mostrare 10 più sottocategorie
Trovati 3859 prodotti di "Ciclo cellulare/Checkpoint"
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Benzamidine hydrochloride
CAS:Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.Formula:C7H9ClN2Purezza:99.25% - 99.97%Colore e forma:White To Off-White PowderPeso molecolare:156.61Peldesine dihydrochloride
CAS:Peldesine (BCX 34) dihydrochloride is an inhibitor of PNP in humans, rats, and mice, also hindering T-cell proliferation, used in lymphoma and HIV research.Formula:C12H13Cl2N5OColore e forma:SolidPeso molecolare:314.17TH5427 hydrochloride
CAS:TH5427 HCl inhibits NUDT5 with 29 nM IC50; 690x more selective over MTH1; blocks ATP in breast cancer cells, hindering growth.Formula:C20H21Cl3N8O3Colore e forma:SolidPeso molecolare:527.79Emvistegrast
CAS:Emvistegrast is a quinolone derivative that acts as an antagonist for the α4β7 integrin.Formula:C35H32F4N6O6Colore e forma:SolidPeso molecolare:708.66Datelliptium chloride hydrochloride
CAS:Datelliptium chloride hydrochloride is a DNA-intercalating agent derived from ellipticine. with anti-tumor activities.
Formula:C23H29Cl2N3OPurezza:99.46%Colore e forma:SolidPeso molecolare:434.4CCT 137690
CAS:CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).Formula:C26H31BrN8OPurezza:98.51% - 99.89%Colore e forma:SolidPeso molecolare:551.48Ref: TM-T2611
1mg39,00€5mg74,00€10mg96,00€25mgPrezzo su richiesta50mgPrezzo su richiesta1mL*10mM (DMSO)90,00€Dasabuvir
CAS:Dasabuvir (ABT-333) blocks HCV replication by inhibiting the essential NS5B RNA polymerase.Formula:C26H27N3O5SPurezza:99.54% - 99.62%Colore e forma:SolidPeso molecolare:493.57Favipiravir sodium
CAS:Favipiravir sodium inhibits viral RNA polymerases, effective against flu, West Nile, yellow fever, and more RNA viruses.Formula:C5H4FN3NaO2Colore e forma:SolidPeso molecolare:180.09MLS000532223
CAS:MLS000532223 is a selectiveRho family GTPases inhibitor(EC50 : 16 μM to 120 μM).Formula:C15H9NO3Purezza:98.6%Colore e forma:SolidPeso molecolare:251.24Ref: TM-T8473
1mg105,00€5mg250,00€10mg401,00€25mg685,00€50mg982,00€100mg1.341,00€1mL*10mM (DMSO)301,00€Hesperadin
CAS:Hesperadin(IC50=250 nM) effectively inhibits Aurora B.Formula:C29H32N4O3SPurezza:98.04% - 99.44%Colore e forma:SolidPeso molecolare:516.65Reversine
CAS:Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).Formula:C21H27N7OPurezza:98% - 99.45%Colore e forma:SolidPeso molecolare:393.49Ref: TM-T1825
1mg35,00€2mg50,00€5mg66,00€10mg84,00€25mg156,00€50mg212,00€100mg371,00€1mL*10mM (DMSO)66,00€SB-743921 hydrochloride
CAS:SB-743921 hydrochloride (SB743921 HCl) is an effective inhibitor of kinesin spindle protein, KSP, (Ki =0.1 nM).Formula:C31H34Cl2N2O3Purezza:95.58% - 99.70%Colore e forma:SolidPeso molecolare:553.52Ref: TM-T2255
1mg39,00€5mg101,00€10mg155,00€25mg263,00€50mg406,00€100mg622,00€500mg1.423,00€1mL*10mM (DMSO)123,00€RNase L-IN-2
CAS:RNase L-IN-2 activates RNase L at 22 uM, has antiviral effects on various RNA viruses, non-toxic at effective levels.Formula:C16H14N2O2SPurezza:98.81%Colore e forma:SolidPeso molecolare:298.36Ref: TM-T8591
1mg120,00€5mg264,00€10mg395,00€25mg627,00€50mg890,00€100mg1.198,00€200mg1.603,00€1mL*10mM (DMSO)243,00€Alovudine
CAS:3'-Fluoro-3'-deoxythymidine (3'-Deoxy-3'-fluorothymidine) is a marker of DNA synthesis,which is less susceptible to inflammatory changes than FDG.Formula:C10H13FN2O4Purezza:99.41%Colore e forma:Less Solid Colourless SolidPeso molecolare:244.22TAK-960 dihydrochloride
TAK-960 dihydrochloride: oral PLK1 inhibitor, IC50 0.8 nM; also Hinders PLK2 and PLK3 (IC50s 16.9/50.2 nM); curbs cancer cell growth.Formula:C27H36Cl2F3N7O3Colore e forma:SolidPeso molecolare:634.52H-Gly-Arg-Gly-Asp-Asn-Pro-OH
CAS:RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.Formula:C23H38N10O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:614.61STAMBP-IN-1
CAS:STAMBP-IN-1 is a novel selective antagonist of deubiquitinase STAM-binding protein (STAMBP), decreasing NALP7 protein levels and suppressing IL-1β release afterFormula:C27H28N4O4SPurezza:99.64%Colore e forma:SolidPeso molecolare:504.6Ref: TM-T8706
1mg67,00€5mg152,00€10mg236,00€25mg507,00€50mg730,00€100mg1.018,00€1mL*10mM (DMSO)192,00€LP-935509
CAS:LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1).Cost-effective and quality-assured.Formula:C20H24N6O3Purezza:98.34% - 99.64%Colore e forma:SolidPeso molecolare:396.44Ref: TM-T15781
1mg39,00€2mg51,00€5mg84,00€10mg131,00€25mg251,00€50mg469,00€100mg683,00€1mL*10mM (DMSO)92,00€BCH001
CAS:BCH001 is a specific small-molecule inhibitor of PAPD5.Formula:C20H15F3N2O5Purezza:99.06%Colore e forma:SolidPeso molecolare:420.34P005091
CAS:P005091 (P5091) is a selective and potent inhibitor of ubiquitin-specific protease 7 (USP7) with EC50 of 4.2 μM.Formula:C12H7Cl2NO3S2Purezza:99.53% - 99.87%Colore e forma:SolidPeso molecolare:348.22
