CymitQuimica logo
Ciclo cellulare/Checkpoint

Ciclo cellulare/Checkpoint

Gli inibitori del ciclo cellulare/dei checkpoint sono composti che interrompono la normale progressione del ciclo cellulare, in particolare nei principali punti di controllo regolatori. Questi inibitori sono fondamentali per studiare la divisione cellulare, comprendere la proliferazione delle cellule cancerose e sviluppare terapie antitumorali. Mirando a fasi specifiche del ciclo cellulare, questi inibitori possono indurre l'arresto del ciclo cellulare, portando all'apoptosi o alla senescenza nelle cellule che si dividono rapidamente. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità del ciclo cellulare/dei checkpoint per supportare le tue ricerche in biologia del cancro, biologia cellulare e sviluppo di farmaci.

Sottocategorie di "Ciclo cellulare/Checkpoint"

Mostrare 10 più sottocategorie

Trovati 3730 prodotti di "Ciclo cellulare/Checkpoint"

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Efalizumab

    CAS:
    Efalizumab: humanized monoclonal antibody CD11a; modulates T cell activation/adhesion; for plaque psoriasis, psoriatic arthritis research.
    Purezza:SDS-PAGE:95% SEC-HPLC:98.77%
    Colore e forma:Liquid
    Peso molecolare:146.14 kDa
  • Upamostat

    CAS:
    Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
    Formula:C32H47N5O6S
    Purezza:99.41%
    Colore e forma:Solid
    Peso molecolare:629.81
  • GSK-1520489A

    CAS:
    <p>GSK-1520489A is an active PKMYT1 inhibitor.</p>
    Formula:C21H23N5O3S
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:425.5
  • Ceftriaxone sodium hydrate

    CAS:
    Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.
    Formula:C18H16N8Na2O7S3·5H2O
    Purezza:99.77% - 99.78%
    Colore e forma:White Or Almost White Crystalline Powder Odorless
    Peso molecolare:661.6
  • Cyclin K degrader 1


    Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.
    Formula:C23H17Cl2N5O2
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:466.32
  • Cibisatamab

    CAS:
    Cibisatamab, a T-cell bispecific antibody, targets CEA on cancer cells and CD3 on T-cells, inducing T-cell-mediated tumor cell killing.
    Purezza:SDS-PAGE:99.1%;SEC-HPLC:96.5%
    Colore e forma:Liquid
    Peso molecolare:191.1 kDa
  • Butylparaben

    CAS:
    Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.
    Formula:C11H14O3
    Purezza:98.15%
    Colore e forma:Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)
    Peso molecolare:194.23
  • hSMG-1 inhibitor 11j

    CAS:
    <p>hSMG-1 inhibitor 11j: pyrimidine, IC50=0.11 nM, &gt;455x selective vs. mTOR/PI3Kα/γ/CDK1/CDK2; cancer research use.</p>
    Formula:C27H28ClN7O3S
    Purezza:99.22% - 99.65%
    Colore e forma:Solid
    Peso molecolare:566.07
  • XPW1

    CAS:
    <p>XPW1 is a CDK9 inhibitor with antitumor activity, inhibits DNA repair procedures, and can be used for the research of clear cell renal cell carcinoma.</p>
    Formula:C36H39ClFN7O2
    Purezza:98.08%
    Colore e forma:Soild
    Peso molecolare:656.19
  • HLM006474

    CAS:
    HLM006474 is a pan inhibitor of E2F. This inhibits E2F4 DNA-binding (IC50: 29.8 μM in A375 cells).
    Formula:C25H25N3O2
    Purezza:99.04% - 99.20%
    Colore e forma:Solid
    Peso molecolare:399.48
  • R-10015

    CAS:
    R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.
    Formula:C20H19ClN6O2
    Purezza:98.68%
    Colore e forma:Solid
    Peso molecolare:410.86
  • TAO Kinase inhibitor 2

    CAS:
    <p>TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.</p>
    Formula:C25H24N2O3
    Purezza:98.58%
    Colore e forma:Soild
    Peso molecolare:400.47
  • 6-Mercaptopurine

    CAS:
    6-Mercaptopurine (6-MP) is an antimetabolite antineoplastic agent with immunosuppressant properties.
    Formula:C5H4N4S
    Purezza:99.53% - 99.63%
    Colore e forma:Yellow Crystalline Powder Solid
    Peso molecolare:152.18
  • Metarrestin

    CAS:
    <p>Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis.</p>
    Formula:C31H30N4O
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:474.6
  • Lerociclib dihydrochloride

    CAS:
    Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/
    Formula:C26H36Cl2N8O
    Purezza:97.4%
    Colore e forma:Solid
    Peso molecolare:547.52
  • ATN-161 trifluoroacetate salt

    CAS:
    <p>ATN-161 TFA salt, a new integrin α5β1 inhibitor, curbs angiogenesis, liver metastases growth, enhances survival in mice.</p>
    Formula:C25H36F3N9O10S
    Purezza:98% - 99.98%
    Colore e forma:Solid
    Peso molecolare:711.67
  • Hycanthone

    CAS:
    <p>Hycanthone (Etrenol(mesylate)) is a potent drug of antischistosomal.</p>
    Formula:C20H24N2O2S
    Purezza:98.78%
    Colore e forma:Yellow-Orange Powder (Ntp 1992)
    Peso molecolare:356.48
  • Vitamin D2

    CAS:
    Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.
    Formula:C28H44O
    Purezza:98.73% - 99.89%
    Colore e forma:Prisms From Acetone 1998)
    Peso molecolare:396.65
  • Enrofloxacin

    CAS:
    <p>Enrofloxacin (BAY-Vp2674) is a veterinary antibacterial agent, used in poultry.</p>
    Formula:C19H22FN3O3
    Purezza:99.43% - >99.99%
    Colore e forma:Pale Yellow Crystals
    Peso molecolare:359.39
  • Doxifluridine

    CAS:
    <p>Doxifluridine (AMC 0101) is a fluoropyrimidine derivative and oral prodrug of the antineoplastic agent 5-fluorouracil (5-FU) with antitumor activity.</p>
    Formula:C9H11FN2O5
    Purezza:99.47% - 99.86%
    Colore e forma:White Solid
    Peso molecolare:246.19