Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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BQU57
CAS:<p>BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.</p>Formula:C16H13F3N4OPurezza:97.45% - 98.72%Colore e forma:SolidPeso molecolare:334.3[D-Phe12]-Bombesin acetate
<p>[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Formula:C76H116N22O20SPurezza:99.81%Colore e forma:SolidPeso molecolare:1689.94Tecadenoson
CAS:<p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>Formula:C14H19N5O5Purezza:98.83%Colore e forma:SolidPeso molecolare:337.332-Methoxyidazoxan monohydrochloride
CAS:<p>L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.</p>Formula:C12H14N2O3·HClPurezza:98.99%Colore e forma:SolidPeso molecolare:270.72Urantide acetate(669089-53-6 free base)
<p>Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in Ca²⁺ assay.</p>Formula:C53H70N10O14S2Purezza:99.22%Colore e forma:SolidPeso molecolare:1135.31Cinacalcet
CAS:<p>Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .</p>Formula:C22H22F3NPurezza:99.48%Colore e forma:Yellow OilPeso molecolare:357.41Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Formula:C25H33Cl2N5O2Purezza:99% - 99.86%Colore e forma:White SolidPeso molecolare:506.47RO 46-8443
CAS:<p>RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.</p>Formula:C31H35N3O8SPurezza:98.77% - 99.77%Colore e forma:SolidPeso molecolare:609.69Mizagliflozin
CAS:<p>Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.</p>Formula:C28H44N4O8Purezza:98.66% - 99.67%Colore e forma:SolidPeso molecolare:564.67Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Formula:C17H25N3O2S·HClPurezza:99.17% - 99.93%Colore e forma:Beige SolidPeso molecolare:371.93Lofexidine
CAS:<p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>Formula:C11H12Cl2N2OPurezza:98.78%Colore e forma:SolidPeso molecolare:259.13Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Formula:C21H25ClN2O3·C6H6O3SPurezza:99.83% - 99.9%Colore e forma:Brown Viscous LiquidPeso molecolare:547.06CYM5442
CAS:<p>CYM5442 is an S1P agonist, targeting to Sphingosine.</p>Formula:C23H27N3O4Purezza:98.02% - 99.48%Colore e forma:SolidPeso molecolare:409.48SBI-553
CAS:<p>SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).</p>Formula:C26H31FN4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:450.55Bremelanotide Acetate
CAS:<p>Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .</p>Formula:C52H72N14O12Purezza:96.72% - >99.99%Colore e forma:SolidPeso molecolare:1085.22α-MSH, amide Acetate
<p>a-MSH, amide Acetate as an endogenous neuropeptide.</p>Formula:C79H113N21O21SPurezza:98.67%Colore e forma:SolidPeso molecolare:1724.94RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.Formula:C69H105N19O16SPurezza:96.84%Colore e forma:SolidPeso molecolare:1488.77Norfluoxetine Hydrochloride
CAS:<p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>Formula:C16H17ClF3NOPurezza:99.71%Colore e forma:SolidPeso molecolare:331.76Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purezza:97.84% - 99.90%Colore e forma:SolidPeso molecolare:575.61HJC0350
CAS:HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.Formula:C15H19NO2SPurezza:99.27% - 99.65%Colore e forma:SolidPeso molecolare:277.38RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Formula:C14H16N2OPurezza:97.38%Colore e forma:SolidPeso molecolare:228.29Neuropeptide FF acetate(99566-27-5 free base)
<p>Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family.</p>Formula:C56H80N14O12Purezza:98.03%Colore e forma:SolidPeso molecolare:1141.32Ro 46-2005
CAS:<p>Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).</p>Formula:C23H27N3O6SPurezza:98.02% - 98.8%Colore e forma:SolidPeso molecolare:473.54SORT-PGRN interaction inhibitor 1
CAS:<p>SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).</p>Formula:C15H18N2O2Purezza:98.72%Colore e forma:SolidPeso molecolare:258.32MDL 100009
CAS:<p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>Formula:C22H28FNO3Purezza:98.96%Colore e forma:SolidPeso molecolare:373.46Albiglutide TFA (782500-75-8 free base)
<p>Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C150H225F3N40O47Purezza:>99.99%Colore e forma:SolidPeso molecolare:3397.63Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.Formula:C169H256N42O57Purezza:98.28%Colore e forma:SolidPeso molecolare:3788.14Bosentan
CAS:<p>Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.</p>Formula:C27H29N5O6SPurezza:99.74% - 99.84%Colore e forma:Pale Yellow To Off-White SolidPeso molecolare:551.614CJC-1295 acetate(863288-34-0 free base)
<p>CJC-1295 acetate is a synthetic GHRH analogue and GHS.</p>Formula:C154H256N44O44Purezza:97.29%Colore e forma:SolidPeso molecolare:3428.01Substance P 1-9 aceate
<p>Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.</p>Formula:C54H81N15O14Purezza:99.01%Colore e forma:SolidPeso molecolare:1164.31Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.Formula:C37H62N10O11Purezza:98.1800%Colore e forma:SolidPeso molecolare:822.95Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purezza:95.00%Colore e forma:SolidPeso molecolare:261.7Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurezza:97.71% - 99.78%Colore e forma:SolidPeso molecolare:4186.57Galanin (1-16), mouse, porcine, rat
CAS:<p>Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.</p>Formula:C78H116N20O21Purezza:98.65%Colore e forma:White PowderPeso molecolare:1669.88Montelukast sodium
CAS:<p>Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.</p>Formula:C35H35ClNNaO3SPurezza:99.14% - 99.89%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:608.17RFRP3(human) acetate(311309-27-0 free base)
<p>RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.</p>Formula:C47H76N14O12Purezza:97.09%Colore e forma:SolidPeso molecolare:1029.19Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purezza:99.24%Colore e forma:SolidPeso molecolare:485.96AM211
CAS:<p>AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)</p>Formula:C27H27F3N2O4Purezza:≥95%Colore e forma:SolidPeso molecolare:500.51nifenalol.HCl
CAS:<p>Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.</p>Formula:C11H17ClN2O3Purezza:99.96%Colore e forma:SolidPeso molecolare:260.72Flibanserin
CAS:<p>Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.</p>Formula:C20H21F3N4OPurezza:99.37% - 99.93%Colore e forma:White PowderPeso molecolare:390.41-Oleoyl lysophosphatidic acid sodium
CAS:<p>1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2</p>Formula:C21H40O7P·NaPurezza:98.75% - 99.24%Colore e forma:SolidPeso molecolare:458.51BAY 41-2272
CAS:<p>BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.</p>Formula:C20H17FN6Purezza:99.54%Colore e forma:SolidPeso molecolare:360.39Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Formula:C21H28N2O2·2ClHPurezza:99.73%Colore e forma:SolidPeso molecolare:413.39ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Formula:C17H11N3O6SPurezza:97.74%Colore e forma:SolidPeso molecolare:385.35Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formula:C24H30N2O2SPurezza:99.9% - 99.92%Colore e forma:SolidPeso molecolare:410.57Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C13H16N2·HClPurezza:99.94% - 99.94%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:236.74Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurezza:98.64% - 99.97%Colore e forma:SolidPeso molecolare:623.63Obestatin (rat) acetate
<p>Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).</p>Formula:C114H174N34O31Purezza:99.05%Colore e forma:SolidPeso molecolare:2516.81Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Formula:C21H35ClN2O5Purezza:99.33%Colore e forma:SolidPeso molecolare:430.97AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Formula:C23H31ClN2O2Purezza:99.71%Colore e forma:SolidPeso molecolare:402.96Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:1024.18FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Formula:C23H25Cl2N3OSPurezza:99.62%Colore e forma:SolidPeso molecolare:462.44Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Formula:C19H26N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:406.5Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurezza:97.25% - 97.36%Colore e forma:SolidPeso molecolare:321.34VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Formula:C13H15ClN4Purezza:99.66%Colore e forma:SolidPeso molecolare:262.74Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68Ramosetron
CAS:<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Formula:C17H17N3OPurezza:98.84%Colore e forma:SolidPeso molecolare:279.34SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Formula:C10H14ClN3·HClPurezza:99.89%Colore e forma:SolidPeso molecolare:248.15Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formula:C10H6N4O2Purezza:99.75%Colore e forma:SolidPeso molecolare:214.18Droxidopa
CAS:Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formula:C9H11NO5Purezza:97.27% - 99.88%Colore e forma:SolidPeso molecolare:213.19TC-G-1008
CAS:<p>TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).</p>Formula:C18H19ClN6O2SPurezza:97.37% - 99%Colore e forma:SolidPeso molecolare:418.9NPS-2143 hydrochloride
CAS:<p>NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.</p>Formula:C24H25ClN2O2·HClPurezza:99.38% - 99.67%Colore e forma:SolidPeso molecolare:445.38Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Levobetaxolol hydrochloride
CAS:<p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>Formula:C18H29NO3·HClPurezza:98.80% - 99.69%Colore e forma:SolidPeso molecolare:343.89Eptapirone
CAS:<p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>Formula:C16H23N7O2Purezza:99.39% - 99.65%Colore e forma:SolidPeso molecolare:345.4Loxiglumide
CAS:<p>Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.</p>Formula:C21H30Cl2N2O5Purezza:97.55% - 99.81%Colore e forma:SolidPeso molecolare:461.38Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Formula:C23H25ClN2OPurezza:98.86% - 99.85%Colore e forma:SolidPeso molecolare:380.91BETP
CAS:<p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>Formula:C20H17F3N2O2SPurezza:98.51%Colore e forma:SolidPeso molecolare:406.42Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1035.15Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purezza:98.02% - 99.68%Colore e forma:SolidPeso molecolare:503.56SB-649868
CAS:<p>SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).</p>Formula:C26H24FN3O3SPurezza:99.53%Colore e forma:SolidPeso molecolare:477.55Ponesimod
CAS:<p>Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.</p>Formula:C23H25ClN2O4SPurezza:99.42% - 99.96%Colore e forma:SolidPeso molecolare:460.97HCGRP-(8-37) acetate
<p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>Formula:C141H234N44O40Purezza:99.29%Colore e forma:SolidPeso molecolare:3185.64Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formula:C17H25N3O2SPurezza:99.85%Colore e forma:Light Yellow Or White PowerPeso molecolare:335.46S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formula:C31H34N2O4Purezza:99.77%Colore e forma:SolidPeso molecolare:498.61PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurezza:99.35%Colore e forma:SolidPeso molecolare:292.36MIPS521
CAS:<p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>Formula:C19H10ClF6NOSPurezza:99.76%Colore e forma:SolidPeso molecolare:449.8Eformoterol Hemifumarate
CAS:<p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>Formula:C19H24N2O4C4H4O4Purezza:99.86% - >99.99%Colore e forma:White PowderPeso molecolare:402.4Protease-Activated Receptor-2, amide
CAS:<p>Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)</p>Formula:C28H54N8O7Purezza:>99.99%Colore e forma:SolidPeso molecolare:614.78ML-178
CAS:<p>ML-178: selective S1PR4 agonist, EC50 of 46 nM; inactive on other S1P receptors at 25 μM.</p>Formula:C13H9Br2Cl2NO2Purezza:95.92%Colore e forma:SolidPeso molecolare:441.93Rizatriptan benzoate
CAS:<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Formula:C22H25N5O2Purezza:99% - 99.79%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:391.47SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurezza:99.83%Colore e forma:SolidPeso molecolare:286.35Istradefylline
CAS:<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Formula:C20H24N4O4Purezza:98.18% - 99.95%Colore e forma:SolidPeso molecolare:384.43H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurezza:98.81%Colore e forma:SolidPeso molecolare:316.79Cinaciguat
CAS:<p>Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.</p>Formula:C36H39NO5Purezza:98% - 99.18%Colore e forma:SolidPeso molecolare:565.71-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Formula:C13H13NO5Purezza:99.55%Colore e forma:SolidPeso molecolare:263.25RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Formula:C67H109N19O19Purezza:99.87%Colore e forma:SolidPeso molecolare:1484.71BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Formula:C59H83N13O14S2Purezza:99.7%Colore e forma:SolidPeso molecolare:1262.5Trazodone
CAS:<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Formula:C19H22ClN5OPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:371.86LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Formula:C30H34N4OPurezza:98.65%Colore e forma:SolidPeso molecolare:466.62JD-5037
CAS:<p>JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.</p>Formula:C27H27Cl2N5O3SPurezza:99.54% - 99.84%Colore e forma:SolidPeso molecolare:572.51Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Purezza:97.26%Colore e forma:LiquidPeso molecolare:N/ARamosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formula:C17H18ClN3OPurezza:99.95%Colore e forma:SolidPeso molecolare:315.8(R)-Propranolol hydrochloride
CAS:(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.Formula:C16H22ClNO2Purezza:98.63% - 99.01%Colore e forma:SolidPeso molecolare:295.8Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Formula:C32H41N5O10Purezza:97.69%Colore e forma:SolidPeso molecolare:655.7Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Purezza:98.42%Colore e forma:LiquidPeso molecolare:N/APancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.Purezza:97.53%Colore e forma:SolidPeso molecolare:N/AVanoxerine dihydrochloride
CAS:<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Formula:C28H34Cl2F2N2OPurezza:98.16% - 98.35%Colore e forma:White SolidPeso molecolare:523.49Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Formula:C10H17N3S·2HCl·H2OPurezza:99.68%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:302.26Sultopride hydrochloride
CAS:<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Formula:C17H27ClN2O4SPurezza:≥95%Colore e forma:White Or Yellowish PowderPeso molecolare:390.93
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