
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.523 prodotti)
- Apoptosi(5.792 prodotti)
- Ciclo cellulare/Checkpoint(4.449 prodotti)
- Cromatina/Epigenetica(2.238 prodotti)
- Segnalazione citoscheletrica(1.383 prodotti)
- Danno al DNA/Riparazione del DNA(2.825 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.526 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.202 prodotti)
- Trasportatore di membrana/canale ionico(2.790 prodotti)
- Metabolismo(9.448 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.926 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.016 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66641 prodotti di "Inibitori"
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ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Formula:C13H16ClN3O3Purezza:98.15%Colore e forma:SolidPeso molecolare:297.74trans-4-Hydroxycyclohexanecarboxylic Acid
CAS:<p>trans-4-Hydroxycyclohexanecarboxylic Acid is an organic intermediate.</p>Formula:C7H12O3Purezza:96.24%Colore e forma:SolidPeso molecolare:144.17DL-Laudanosine
CAS:<p>DL-Laudanosine (Laudanosine) is a recognized metabolite of atracurium and cisatracurium.</p>Formula:C21H27NO4Purezza:98.45% - 99.79%Colore e forma:SolidPeso molecolare:357.44Squalene
CAS:<p>Squalene (AddaVax) is an intermediate in cholesterol synthesis. Squalene has a variety of pharmacological properties. High-Quality, Low-Cost!</p>Formula:C30H50Purezza:99.33%Colore e forma:Pale Yellow Translucent Liquid Liquid ViscousPeso molecolare:410.72Triptorelin acetate(57773-63-4 free base)
CAS:<p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>Formula:C66H86N18O15Purezza:99.90%Colore e forma:White PowderPeso molecolare:1371.53Dimethyl Trisulfide
CAS:<p>Dimethyl trisulfide is the simplest organic trisulfide found in garlic, onion, broccoli, and similar plants. Dimethyl trisulfide is a cyanide antidote.</p>Formula:C2H6S3Purezza:98%Colore e forma:LiquidPeso molecolare:126.26Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Formula:C22H28BrNPurezza:97.99%Colore e forma:SolidPeso molecolare:386.37NSC59984
CAS:<p>NSC59984, a p53 pathway activator, induces mutant p53 protein degradation and p73 activation.</p>Formula:C12H15N3O4Purezza:99.33% - 99.59%Colore e forma:SolidPeso molecolare:265.27ODQ
CAS:<p>ODQ is an effective and selective soluble guanylyl cyclase (sGC) inhibitor.</p>Formula:C9H5N3O2Purezza:98.98%Colore e forma:Off-White To Light Yellow PowderPeso molecolare:187.15SC66
CAS:<p>SC66 is a AKT inhibitor in HepG2, HA22T/VGH, and PLC/PRF/5 cells (IC50: about 0.75 μg/ml, at 72 h).</p>Formula:C18H16N2OPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:276.33PF-562271 besylate
CAS:<p>PF-562271 besylate: potent, ATP-competitive FAK inhibitor, IC50 1.5 nM, 10x less effective on Pyk2, highly selective vs other kinases.</p>Formula:C21H20F3N7O3S·C6H6O3SPurezza:97.65% - 99.01%Colore e forma:SolidPeso molecolare:665.66Acetyl-L-lysine
CAS:<p>Acetyl-L-lysine: N-acetylated amino acid, normally found in trace urine amounts, elevated in aminoacylase I deficiency.</p>Formula:C8H16N2O3Purezza:99.40% - 99.83%Colore e forma:SolidPeso molecolare:188.22BCIP
CAS:<p>BCIP (BCIP p-toluidine salt) (BCIP p-toluidine salt) is an artificial chromogenic substrate.</p>Formula:C15H15BrClN2O4PPurezza:99.31% - ≥98%Colore e forma:CrystalsPeso molecolare:433.62β-Sitosterol
CAS:<p>Beta-Sitosterol induces G2/M arrest, endoreduplication, and apoptosis, possibly affecting cancer therapy, cholesterol metabolism, and inflammation.</p>Formula:C29H50OPurezza:98.54% - 99.95%Colore e forma:White SolidPeso molecolare:414.71AG-1478
CAS:<p>AG-1478 (NSC-693255) (Tyrphostin AG-1478) is a selective EGFR inhibitor.</p>Formula:C16H14ClN3O2Purezza:99.03% - 99.71%Colore e forma:SolidPeso molecolare:315.75Fenoxycarb
CAS:<p>Fenoxycarb (Insegar) is an insecticide against mosquitoes.</p>Formula:C17H19NO4Purezza:97.01%Colore e forma:Colorless To White Crystals SolidPeso molecolare:301.34Palmitic acid
CAS:<p>Palmitic acid (Cetylic acid) is a natural product, a common saturated fatty acid found in animals, plants and microorganisms.</p>Formula:C16H32O2Purezza:99.17% - 99.67%Colore e forma:White Crystalline Scales SolidPeso molecolare:256.42Indole-3-butyric acid
CAS:<p>Indole-3-butyric acid (IBA) is a plant hormone in the auxin family and is an ingredient in many commercial plant rooting horticultural products.</p>Formula:C12H13NO2Purezza:99.29% - 99.92%Colore e forma:White To Slightly Yellow Crystals SolidPeso molecolare:203.24PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Formula:C19H17ClFN5SPurezza:97.79% - 98.07%Colore e forma:SolidPeso molecolare:401.89D-Galacturonic acid hydrate
CAS:<p>D-Galacturonic acid hydrate is used in the synthesis of N-(D-galacturonoyl) amino acids and dipeptides.</p>Formula:C6H12O8Purezza:97% - 99.97%Colore e forma:White To Light Beige Fine PowderPeso molecolare:212.15MK2-IN-3
CAS:<p>MK2-IN-3 is a potent MK-2 inhibitor, cell-permeable, for rheumatoid arthritis treatment.</p>Formula:C21H16N4OPurezza:99.01%Colore e forma:SolidPeso molecolare:340.38Carnostatine hydrochloride
<p>Carnostatine HCl (SAN9812 HCl) is a potent, selective CN1 inhibitor, with Ki 11 nM, potential DN treatment.</p>Formula:C10H17ClN4O4Purezza:98%Colore e forma:SolidPeso molecolare:292.72[D-Phe12,Leu14]-Bombesin acetate
<p>[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Formula:C77H118N22O20Purezza:98.41% - 99.14%Colore e forma:SolidPeso molecolare:1671.9Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Formula:C18H19N3O·HClPurezza:99.78%Colore e forma:White PowderPeso molecolare:329.82Methyl heptadecanoate
CAS:<p>Methyl heptadecanoate is a natural product.</p>Formula:C18H36O2Purezza:97.72%Colore e forma:SolidPeso molecolare:284.48Zofenopril calcium
CAS:<p>Zofenopril calcium (SQ26991) is an antioxidant that acts as an angiotensin-converting enzyme inhibitor.</p>Formula:C44H44CaN2O8S4Purezza:98.37%Colore e forma:White Or Whitish Crystalline PowderPeso molecolare:897.17Pirozadil
CAS:<p>Pirozadil shows hypolipidemic activity.</p>Formula:C27H29NO10Purezza:97.54% - 98.31%Colore e forma:SolidPeso molecolare:527.52MNS
CAS:<p>MNS is a tyrosine kinases inhibitor, inhibits Syk, Src, p97 with IC50 of 2.5 μM, 29.3 μM and 1.7 μM, respectively.</p>Formula:C9H7NO4Purezza:98.53%Colore e forma:Yellow PowderPeso molecolare:193.16Ibiglustat hydrochloride
CAS:<p>Ibiglustat hydrochloride is a potent and selective Glucosylceramide synthase inhibitor and ceramide glucosyltransferase inhibitor.</p>Formula:C20H25ClFN3O2SColore e forma:SolidPeso molecolare:425.95N4-Benzoyl-2′-deoxycytidine
CAS:<p>N4-Benzoyl-2′-deoxycytidine is a synthetic nucleoside analog of the natural nucleoside deoxycytidine (dC), a competitive inhibitor of DNA polymerase.</p>Formula:C16H17N3O5Purezza:99.41%Colore e forma:SolidPeso molecolare:331.32Tipifarnib (S enantiomer)
CAS:<p>Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).</p>Formula:C27H22Cl2N4OPurezza:99.05%Colore e forma:SolidPeso molecolare:489.4Acebilustat
CAS:<p>Acebilustat (CTX-4430) (ZK322) is an effective and specific leukotriene B4 hydrolase inhibitor.</p>Formula:C29H27N3O4Purezza:99.59% - 99.88%Colore e forma:SolidPeso molecolare:481.54Hoechst 33258 trihydrochloride
CAS:<p>Hoechst 33258 trihydrochloride (Bisbenzimide) is a benzimidazole anti-filarial agent. Hoechst 33258 is fluorescent when it binds to certain nucleotides in DNA.</p>Formula:C25H24N6O·3HClPurezza:95.68% - 99.47%Colore e forma:Yellow-Green PowderPeso molecolare:533.9GDC0575 monohydrochloride
CAS:<p>GDC0575 (ARRY575), a potent Chk1 inhibitor, IC50 1.2nM, disrupts cell cycle arrest, allowing DNA repair before mitosis.</p>Formula:C16H21BrClN5OPurezza:97.85%Colore e forma:SolidPeso molecolare:414.731,3,6-Tri-O-galloyl-β-D-glucose
CAS:<p>1,3,6-Tri-O-galloyl-beta-D-glucose (1,3,6-Tri-O-galloylglucose) is a phenolic compound in Black Walnut Kernels. It shows anti-inflammatory activity.</p>Formula:C27H24O18Purezza:98.94% - 99.47%Colore e forma:SolidPeso molecolare:636.475-Acetylsalicylic acid
CAS:<p>5-Acetylsalicylic acid treats inflammatory bowel diseases and maintains Crohn's remission.</p>Formula:C9H8O4Purezza:99.33% - 99.53%Colore e forma:SolidPeso molecolare:180.16Mycophenolate Mofetil
CAS:<p>Mycophenolate Mofetil (TM-MMF), is an immunosuppressive agent, 2-morpholinoethyl ester of MPA, and an inhibitor of inosine monophosphate dehydrogenase (IMPDH).</p>Formula:C23H31NO7Purezza:98.27% - 99.85%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:433.49Spermidine
CAS:<p>Spermidine inhibits nNOS, precipitates DNA for protein purification, activates PNK & NMDA, and boosts NMDA currents.</p>Formula:C7H19N3Purezza:99.21% - ≥98%Colore e forma:LiquidPeso molecolare:145.257-Ketocholesterol
CAS:<p>7-Ketocholesterol is a metabolite of Cholesterol</p>Formula:C27H44O2Purezza:97.59% - 98.84%Colore e forma:SolidPeso molecolare:400.65Keratin hydrolyzed
CAS:<p>Keratin hydrolyzed is a processed form of keratin that allows it to penetrate the hair cuticle.</p>Formula:C2H2BrClO2Purezza:80%Colore e forma:SolidPeso molecolare:173.393CCT196969
CAS:<p>CCT196969 is a novel orally available, pan-RAF inhibitor with anti-SRC activity. It also inhibits SRC, LCK, and the p38 MAPKs.</p>Formula:C27H24FN7O3Purezza:98.93% - 99.65%Colore e forma:SolidPeso molecolare:513.526-ethenylquinoline
CAS:<p>6-ethenylquinoline: aromatic, used in drugs, inhibits enzymes like cytochrome P450.</p>Formula:C11H9NPurezza:97.09%Colore e forma:SolidPeso molecolare:155.2N-Nitrosodiethylamine
CAS:<p>N-Nitrosodiethylamine (NDEA) is a potent hepatocarcinogenic dialkylnitrosoamine.</p>Formula:C4H10N2OPurezza:99.26% - 99.88%Colore e forma:SolidPeso molecolare:102.146-Hydroxy-4-methylcoumarin
CAS:<p>6-Hydroxy-4-methylcoumarin (6-Hydroxy-4-Methyl-2H-Chromen-2-One) is a secondary metabolite of coumarin, which has anticancer effects.</p>Formula:C10H8O3Purezza:98.93%Colore e forma:SolidPeso molecolare:176.17Iclaprim
CAS:<p>Iclaprim (AR-100) is a novel specific bacterial Dihydrofolate inhibitor. It can inhibit the growth of S. aureus (MIC90: 0.06 μg/mL).</p>Formula:C19H22N4O3Purezza:99.66%Colore e forma:SolidPeso molecolare:354.4Deapioplatycodin D
CAS:<p>Deapioplatycodin D and platycodin D can regulate the production and secretion of airway mucin and, explains the use of aqueous extract of APG as expectorants.</p>Formula:C52H84O24Purezza:97.33% - 99.64%Colore e forma:SolidPeso molecolare:1093.21PNU 22394 hydrochloride
CAS:<p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>Formula:C13H17ClN2Purezza:97.83%Colore e forma:SolidPeso molecolare:236.74Valorphin TFA(144313-54-2(free base))
<p>Valorphin TFA(144313-54-2(free base)) is a semisynthetic derivative of dihydrovaltrate with opioid analgesic activity</p>Formula:C46H62F3N9O13Purezza:≥98%Colore e forma:SolidPeso molecolare:1006.03β-Tocopherol
CAS:<p>Beta-Tocopherol has effects on human erythroleukemia cell (HEL) adhesion induced by phorbol 12-myristate 13-acetate (PMA).Cost-effective and quality-assured.</p>Formula:C28H48O2Purezza:99.8% - 99.92%Colore e forma:SolidPeso molecolare:416.68SAG hydrochloride (912545-86-9(free base))
CAS:<p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>Formula:C28H29Cl2N3OSPurezza:99.19% - 99.77%Colore e forma:SolidPeso molecolare:526.52
