Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(36 produtos)
- Cisteína Protease(111 produtos)
- DPP-4(24 produtos)
- Glutaminase(44 produtos)
- HIV Protease(501 produtos)
- PAI-1(26 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(54 produtos)
- Proteassoma(89 produtos)
- Protease serina(54 produtos)
- p97(15 produtos)
Exibir 3 mais subcategorias
Foram encontrados 994 produtos de "Proteases/Proteassoma"
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Benzylsulfonyl Fluoride [for Biochemical Research]
CAS:Fórmula:C7H7FO2SPureza:>98.0%(GC)Cor e Forma:White to Almost white powder to crystalPeso molecular:174.19Disodium Dihydrogen Ethylenediaminetetraacetate Dihydrate [for Biochemical Research]
CAS:Fórmula:C10H14N2Na2O8·2H2OPureza:>99.0%(T)Cor e Forma:White powder to crystalinePeso molecular:372.24Nafamostat Mesylate
CAS:Fórmula:C19H17N5O2·2CH4O3SPureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:539.58Nelfinavir Mesylate
CAS:Fórmula:C32H45N3O4S·CH4O3SPureza:>97.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:663.89Atazanavir Sulfate
CAS:Fórmula:C38H52N6O7·H2SO4Pureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:802.94Camostat Mesylate
CAS:Fórmula:C20H22N4O5·CH4O3SPureza:>98.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:494.52Gabexate Mesylate
CAS:Fórmula:C16H23N3O4·CH4O3SPureza:>97.0%(N)Cor e Forma:White to Almost white powder to crystalPeso molecular:417.48Ethylene Glycol Bis(2-aminoethyl Ether)-N,N,N',N'-tetraacetic Acid [for Biochemical Research]
CAS:Fórmula:C14H24N2O10Pureza:>95.0%(T)Cor e Forma:White to Almost white powder to crystalPeso molecular:380.35Benzamidine Hydrochloride [for Biochemical Research]
CAS:Fórmula:C7H8N2·HClPureza:>95.0%(T)(N)Cor e Forma:White to Almost white powder to crystalPeso molecular:156.611,10-Phenanthroline Monohydrate [for Biochemical Research]
CAS:Fórmula:C12H8N2·H2OPureza:>99.0%(T)Cor e Forma:White powder to crystalPeso molecular:198.23Limonin
CAS:Fórmula:C26H30O8Pureza:>95.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:470.524-(2-Aminoethyl)benzenesulfonyl Fluoride Hydrochloride [for Biochemical Research]
CAS:Fórmula:C8H10FNO2S·HClPureza:>99.0%(HPLC)Cor e Forma:White to Almost white powder to crystalPeso molecular:239.692-Iodoacetamide [for Biochemical Research]
CAS:Fórmula:C2H4INOPureza:>98.0%(N)Cor e Forma:White to Light yellow powder to crystalPeso molecular:184.96Ritonavir
CAS:Fórmula:C37H48N6O5S2Pureza:>98.0%(HPLC)(N)Cor e Forma:White to Almost white powder to crystalinePeso molecular:720.95Atazanavir
CAS:Fórmula:C38H52N6O7Pureza:>95.0%(HPLC)Cor e Forma:White to Light yellow powder to crystalPeso molecular:704.87Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Fórmula:C19H17NO7Pureza:97.99%Cor e Forma:SolidPeso molecular:371.34Ref: TM-T15574
1mg84,00€2mg89,00€5mg113,00€10mg178,00€25mg371,00€50mg573,00€100mg802,00€200mg1.099,00€1mL*10mM (DMSO)90,00€3-Aminopropionitrile fumarate (2:1)
CAS:3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.Fórmula:C4H4O4·2C3H6N2Pureza:99.76% - 99.79%Cor e Forma:White Crystalline PowderPeso molecular:256.26RA190
CAS:RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.Fórmula:C28H23Cl5N2O2Pureza:97.7%Cor e Forma:SolidPeso molecular:596.76Ref: TM-T13858
1mg54,00€5mg109,00€10mg159,00€25mg233,00€50mg414,00€100mg608,00€1mL*10mM (DMSO)142,00€KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Fórmula:C29H31N5O5SPureza:99.28%Cor e Forma:SolidPeso molecular:561.65Ethylenediaminetetraacetic acid disodium salt dihydrate
CAS:Fórmula:C10H18N2Na2O10Pureza:97%Cor e Forma:SolidPeso molecular:372.2369(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
CAS:Fórmula:C16H24N2O4Pureza:98%Cor e Forma:SolidPeso molecular:308.3728Ref: IN-DA00370Q
1g132,00€5g223,00€10g532,00€25gA consultar50gA consultar100gA consultar10mg29,00€250gA consultar50mg34,00€100mg44,00€250mg68,00€Benzoic acid, 4-[(aminoiminomethyl)amino]-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate
CAS:Fórmula:C20H21N5O5SPureza:98%Cor e Forma:SolidPeso molecular:443.4762L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Fórmula:C26H41N3O5Pureza:98%Cor e Forma:SolidPeso molecular:475.6208Ref: IN-DA0072SK
1gA consultar5mg68,00€10mg90,00€25mg124,00€50mg168,00€100mg229,00€250mg500,00€500mgA consultarLevovirin
CAS:Levovirin (L-Ribavirin) is a guanosine nucleoside analog that has immunomodulatory activity and is used in the study of hepatitis C virus infection.Fórmula:C8H12N4O5Pureza:99.81% - >99.99%Cor e Forma:SolidPeso molecular:244.20Mecarbinate
CAS:Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.Fórmula:C13H15NO3Pureza:99.28%Cor e Forma:Off-White Crystalline PowderPeso molecular:233.26PMSF
CAS:PMSF (Phenylmethylsulfonyl fluoride) is an irreversible inhibitor of serine/cysteine protease , preparation of cell lysates. High-Quality, Low-Cost!Fórmula:C7H7FO2SPureza:97.75% - 99.88%Cor e Forma:White To Cream SolidPeso molecular:174.193-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-
CAS:Fórmula:C32H45N3O4SPureza:98%Cor e Forma:SolidPeso molecular:567.7824Benzoic acid, 4-[[6-[(aminoiminomethyl)amino]-1-oxohexyl]oxy]-, ethylester, monomethanesulfonate
CAS:Fórmula:C17H27N3O7SPureza:98%Cor e Forma:SolidPeso molecular:417.4772CL-82198
CAS:CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Fórmula:C17H22N2O3Pureza:95.91%Cor e Forma:SolidPeso molecular:302.37Ref: TM-T14978
5mg47,00€10mg73,00€25mg153,00€50mg243,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)50,00€Ref: IN-DA00BBLC
1g57,00€5g128,00€25g262,00€5mg30,00€100gA consultar10mg30,00€50mg30,00€100mg37,00€250mg44,00€4-(2-Aminoethyl)benzenesulfonyl fluoride, HCl
CAS:Fórmula:C8H11ClFNO2SPureza:98%Cor e Forma:SolidPeso molecular:239.6948Bivalirudin acetate
Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.Fórmula:C100H142N24O35Pureza:99.84%Cor e Forma:SolidPeso molecular:2240.34BAY-85-8501
CAS:BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Fórmula:C22H17F3N4O3SPureza:99.16%Cor e Forma:SolidPeso molecular:474.46Ref: TM-T12613L
1mg92,00€2mg122,00€5mg200,00€10mg298,00€25mg535,00€50mg750,00€100mg1.035,00€1mL*10mM (DMSO)208,00€Saxagliptin hydrate
CAS:Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).Fórmula:C18H25N3O2·H2OPureza:99.52%Cor e Forma:SolidPeso molecular:333.43GSK2838232
CAS:GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.
Fórmula:C48H73ClN2O6Pureza:97.97%Cor e Forma:SolidPeso molecular:809.56DPP-IV-IN-2
CAS:DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Fórmula:C18H26N4O5Pureza:99.08%Cor e Forma:SolidPeso molecular:378.42HCV-IN-29
CAS:HCV-IN-29 is a hepatitis C virus (HCV) inhibitor.Fórmula:C26H32Cl4N6Pureza:99.89%Cor e Forma:SolidPeso molecular:570.38(Rac)-Telinavir
CAS:N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.
Fórmula:C33H44N6O5Pureza:99.30%Cor e Forma:SolidPeso molecular:604.74Ethylene glycol bis(2-aminoethyl ether)-N,N,N',N'-tetraacetic acid
CAS:Fórmula:C14H24N2O10Pureza:97%Cor e Forma:SolidPeso molecular:380.3478Ref: IN-DA0034HK
5gA consultar10g21,00€1kg124,00€25g25,00€50g25,00€5kg563,00€100g34,00€250g60,00€500g75,00€50kgA consultarBenzenemethanesulfonyl fluoride
CAS:Fórmula:C7H7FO2SPureza:99%Cor e Forma:SolidPeso molecular:174.1927N-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Fórmula:C17H18ClNO3SPureza:97%Cor e Forma:SolidPeso molecular:351.8477Ref: IN-DA003O5U
1g542,00€5gA consultar10mg61,00€25mg94,00€50mg148,00€100mg191,00€250mg197,00€500mg333,00€Gly-Pro-pNA hydrochloride
CAS:Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidaseFórmula:C13H17ClN4O4Pureza:99.84%Cor e Forma:SolidPeso molecular:328.75Sofosbuvir impurity G
CAS:Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.Fórmula:C22H29FN3O9PPureza:98.04%Cor e Forma:SolidPeso molecular:529.45Ref: TM-T12962
1mg1.103,00€5mg2.547,00€10mg3.449,00€25mg5.120,00€50mg6.925,00€1mL*10mM (DMSO)3.202,00€2-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Fórmula:C17H30N2O5Pureza:98%Cor e Forma:SolidPeso molecular:342.4305Ref: IN-DA0032JK
5g22,00€10g26,00€1kg229,00€25g30,00€50g40,00€100g59,00€10kgA consultar250g114,00€500g164,00€Dabigatran ethyl ester hydrochloride
CAS:Dabigatran prevents blood clots, inhibiting NQO2 and thrombin with IC50 0.8 μM.Fórmula:C27H30ClN7O3Pureza:99.65%Cor e Forma:SolidPeso molecular:536.03Sofosbuvir impurity F
CAS:Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNAFórmula:C34H45FN4O13P2Pureza:98.05%Cor e Forma:SolidPeso molecular:798.69ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Fórmula:C17H20N2O5SPureza:97.18%Cor e Forma:SolidPeso molecular:364.423-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-, methanesulfonate (1:1)
CAS:Fórmula:C33H49N3O7S2Pureza:96%Cor e Forma:SolidPeso molecular:663.8881Dabigatran etexilate
CAS:Dabigatran etexilate (BIBR 1048) is a thrombin inhibitor, which acts by binding and blocking thrombogenic activity and the prevention of thrombus formation.Fórmula:C34H41N7O5Pureza:98.19% - 99.98%Cor e Forma:White PowderPeso molecular:627.73Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Pureza:> 95%Cor e Forma:LiquidPeso molecular:145.42 kDaDBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Fórmula:C16H25FN4O2Pureza:99.68%Cor e Forma:SolidPeso molecular:324.39Ref: TM-T15079
1mg48,00€5mg100,00€10mg133,00€25mg215,00€50mg306,00€100mg414,00€200mg573,00€1mL*10mM (DMSO)110,00€Anisindione
CAS:Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.Fórmula:C16H12O3Pureza:98.25%Cor e Forma:Pale Yellow Crystals From Acetic Acid Or Ethanol SolidPeso molecular:252.26Avoralstat
CAS:Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.Fórmula:C28H27N5O5Pureza:99.77%Cor e Forma:SolidPeso molecular:513.54ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Fórmula:C17H24BF3N2O4Pureza:97.06%Cor e Forma:SolidPeso molecular:388.19Ref: TM-T12079
1mg109,00€2mg158,00€5mg259,00€10mg409,00€25mg677,00€50mg954,00€100mg1.288,00€200mg1.728,00€1mL*10mM (DMSO)285,00€Salicylanilide
CAS:Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.
Fórmula:C13H11NO2Pureza:99.55%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:213.23Trelagliptin
CAS:Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.Fórmula:C18H20FN5O2Pureza:98.88%Cor e Forma:SolidPeso molecular:357.38Retagliptin Phosphate
CAS:Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Fórmula:C19H21F6N4O7PPureza:98.70%Cor e Forma:SolidPeso molecular:562.36Ref: TM-T12710
1mg34,00€2mg42,00€5mg60,00€10mg87,00€25mg161,00€50mg245,00€100mgA consultar1mL*10mM (DMSO)79,00€LSP-249
CAS:LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.Fórmula:C24H22ClN5OPureza:99.51%Cor e Forma:SolidPeso molecular:431.92BLT-1
CAS:BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.Fórmula:C12H23N3SPureza:97.97%Cor e Forma:SolidPeso molecular:241.4Ref: TM-T14667
1mg43,00€2mg56,00€5mg93,00€10mg152,00€25mg259,00€50mg409,00€100mg592,00€1mL*10mM (DMSO)90,00€Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Fórmula:C49H55FN10O7SPureza:96.87% - 99.93%Cor e Forma:SolidPeso molecular:947.09Dolutegravir intermediate-1
CAS:Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.Fórmula:C13H17NO8Pureza:99.52%Cor e Forma:SolidPeso molecular:315.28RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Fórmula:C19H13Cl4NOPureza:98.89% - 99.38%Cor e Forma:SolidPeso molecular:413.12LDN-27219
CAS:LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.Fórmula:C20H16N4O2S2Pureza:99.01% - 99.38%Cor e Forma:SolidPeso molecular:408.5Ref: TM-T11831
1mg35,00€5mg66,00€10mg92,00€25mg160,00€50mg234,00€100mg351,00€200mg515,00€1mL*10mM (DMSO)71,00€Probenecid
CAS:Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.Fórmula:C13H19NO4SPureza:98.95% - 99.84%Cor e Forma:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Peso molecular:285.36BJJF078
CAS:BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Fórmula:C27H29N3O6SPureza:99.56%Cor e Forma:SoildPeso molecular:523.6MK-0608
CAS:MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).Fórmula:C12H16N4O4Pureza:98.48%Cor e Forma:SolidPeso molecular:280.28Ref: TM-T16088
1mg46,00€2mg59,00€5mg96,00€10mg133,00€25mg250,00€50mg411,00€100mg660,00€1mL*10mM (DMSO)92,00€(Rac)-Telmesteine
CAS:(Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) is an inhibitor of protease and is thus a suitable enzyme stabilizer.Fórmula:C7H11NO4SPureza:99.91%Cor e Forma:SolidPeso molecular:205.23(ETHYLENEDINITRILO)TETRAACETIC ACID, TRISODIUM SALT HYDRATE
CAS:Fórmula:C10H18N2NaO9Pureza:97%Cor e Forma:SolidPeso molecular:333.2477Tyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Fórmula:C19H14BrClN4OCor e Forma:SolidPeso molecular:429.7STK33-IN-1
CAS:STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.Fórmula:C24H27N7O2Cor e Forma:SolidPeso molecular:445.527Talabostat
CAS:Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.Fórmula:C9H19BN2O3Cor e Forma:SolidPeso molecular:214.07Ichorcumab
CAS:Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.
Cor e Forma:LiquidPROTAC CG167
PROTAC CG167 is a potent and selective PROTAC degrader of CypA. It degrades CypA in a dose-dependent manner in Jurkat cells, with a DC50 of 123 nM. Additionally, PROTAC CG167 exhibits antiviral activity by inhibiting HIV-1 and HCV. (Pink: CypA Ligand; Black: Linker; Blue: E3LigaseLigand)Fórmula:C65H79N13O11SCor e Forma:SolidPeso molecular:1250.47Nitidanin
Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.Fórmula:C21H24O8Cor e Forma:SolidPeso molecular:404.4155-epi-Arvestonate A
CAS:5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.
Fórmula:C16H26O5Cor e Forma:SolidPeso molecular:298.37HCV-IN-7 hydrochloride
CAS:HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.Fórmula:C40H50Cl2N8O6SPureza:98%Cor e Forma:SolidPeso molecular:841.85RXP470
CAS:RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).Fórmula:C35H35BrClN4O10PCor e Forma:SolidPeso molecular:818RJS308
RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)Fórmula:C63H75N13O11SCor e Forma:SolidPeso molecular:1222.42Grazoprevir potassium salt
CAS:Grazoprevir, a drug for hepatitis C, is a second-gen NS3/4a protease inhibitor.
Fórmula:C38H49KN6O9SCor e Forma:SolidPeso molecular:805Relacatib
CAS:Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.Fórmula:C27H32N4O6SCor e Forma:SolidPeso molecular:540.64VD2173
CAS:VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.Fórmula:C31H45N9O6SCor e Forma:SolidPeso molecular:671.81Bortezomib analog
Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.Cor e Forma:Odour SolidHIV-1 Rev (34-50)
CAS:HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.Fórmula:C97H173N51O24Pureza:99.91%Cor e Forma:SolidPeso molecular:2437.746,6′-Dihydroxythiobinupharidine
CAS:6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-foldFórmula:C30H42N2O4SCor e Forma:SolidPeso molecular:526.73GCPII-IN-1
CAS:GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.
Fórmula:C12H21N3O7Cor e Forma:SolidPeso molecular:319.314PSI-7409
CAS:PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).
Fórmula:C10H16FN2O14P3Pureza:98%Cor e Forma:SolidPeso molecular:500.16Neutrophil elastase inhibitor 4
Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.Fórmula:C20H21N3O5Cor e Forma:SolidPeso molecular:383.4AP-C2
CAS:AP-C2 is a potent small molecule guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2 for cGKII.Fórmula:C18H16N4SPureza:99.99%Cor e Forma:SoildPeso molecular:320.4115,16-Dihydrotanshindiol C
15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.Fórmula:C18H18O5Cor e Forma:SolidPeso molecular:314.337
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