Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(35 produtos)
- Cisteína Protease(96 produtos)
- DPP-4(20 produtos)
- Glutaminase(40 produtos)
- HIV Protease(450 produtos)
- PAI-1(25 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(53 produtos)
- Proteassoma(94 produtos)
- Protease serina(50 produtos)
- p97(14 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1044 produtos de "Proteases/Proteassoma"
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HCV-IN-30
CAS:<p>HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).</p>Fórmula:C36H44N6O4Pureza:99.6%Cor e Forma:SolidPeso molecular:624.77Carboxypeptidase G2 (CPG2) Inhibitor
CAS:<p>Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.</p>Fórmula:C13H15NO6SPureza:99.96%Cor e Forma:SolidPeso molecular:313.33Cathepsin Inhibitor 1
CAS:<p>Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.</p>Fórmula:C20H24ClN5O2Pureza:99.78%Cor e Forma:SolidPeso molecular:401.89BAY-678 racemate
CAS:<p>BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.</p>Fórmula:C20H15F3N4O2Pureza:98%Cor e Forma:SolidPeso molecular:400.35Tyrosinase-IN-4
CAS:<p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>Fórmula:C15H9ClO3Cor e Forma:SolidPeso molecular:272.68WNK-IN-7
CAS:<p>WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.</p>Fórmula:C26H29N3OPureza:98%Cor e Forma:SolidPeso molecular:399.53BR351 precursor
CAS:<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C27H32N2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:576.68RS-104966
CAS:<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Fórmula:C19H21NO6SPureza:98%Cor e Forma:SolidPeso molecular:391.44Ono-3307 mesylate
CAS:<p>no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.</p>Fórmula:C15H18N4O7S2Pureza:97.60% - 98.16%Cor e Forma:SolidPeso molecular:430.46Thrombin inhibitor 6
CAS:<p>Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.</p>Fórmula:C18H19ClN4O2SCor e Forma:SolidPeso molecular:390.89MDK0734
CAS:<p>MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Fórmula:C15H17N3O2Pureza:98%Cor e Forma:SolidPeso molecular:271.31LY 135305
CAS:<p>LY 135305 is a inhibition of spontaneous metastasis.</p>Fórmula:C19H20ClNPureza:98%Cor e Forma:SolidPeso molecular:297.82Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Fórmula:C23H31N3NaO4S2Pureza:98%Cor e Forma:SolidPeso molecular:500.63HCV-IN-37
CAS:<p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>Fórmula:C31H35F2N5Cor e Forma:SolidPeso molecular:515.64RO-9187
CAS:<p>RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).</p>Fórmula:C9H12N6O5Pureza:98%Cor e Forma:SolidPeso molecular:284.23ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Fórmula:C15H16ClNO3S2Pureza:99.49%Cor e Forma:SolidPeso molecular:357.88Ro 09-1679
CAS:<p>Ro 09-1679 is a thrombin inhibitor.</p>Fórmula:C22H39N9O6Pureza:98%Cor e Forma:SolidPeso molecular:525.6SQ 32602
CAS:<p>SQ 32602 is a cathepsin E inhibitor.</p>Fórmula:C32H52N3O7PCor e Forma:SolidPeso molecular:621.74Tyrosinase-IN-8
<p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>Fórmula:C16H12O4Cor e Forma:SolidPeso molecular:268.26Cysteine protease inhibitor-2
CAS:<p>Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.</p>Fórmula:C13H5N5OPureza:98%Cor e Forma:SolidPeso molecular:247.21ZD8321
CAS:<p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>Fórmula:C18H28F3N3O5Pureza:98%Cor e Forma:SolidPeso molecular:423.43Proteasome-IN-1
CAS:<p>Proteasome-IN-1 is an inhibitor of proteasome.</p>Fórmula:C42H35N5O3Pureza:98%Cor e Forma:SolidPeso molecular:657.76DPP-4-IN-2
CAS:<p>DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.</p>Fórmula:C18H18N6OCor e Forma:SolidPeso molecular:334.38Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Fórmula:C32H30F3N5O7S2Pureza:98%Cor e Forma:SolidPeso molecular:717.73Cofrogliptin
CAS:<p>Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).</p>Fórmula:C18H19F5N4O3SCor e Forma:SolidPeso molecular:466.43Thrombin Inhibitor 2
CAS:<p>Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.</p>Fórmula:C19H16ClF3N6O2Pureza:98%Cor e Forma:SolidPeso molecular:452.82HCV-IN-3
CAS:<p>HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).</p>Fórmula:C13H11F2NOPureza:98%Cor e Forma:SolidPeso molecular:235.23PSI-7409 tetrasodium
CAS:<p>PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.</p>Fórmula:C10H16FN2Na4O14P3Pureza:98%Cor e Forma:SolidPeso molecular:592.117Levovirin valinate HCl
CAS:Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.Fórmula:C13H22ClN5O6Pureza:98%Cor e Forma:SolidPeso molecular:379.8TAPI-1
CAS:<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Fórmula:C26H37N5O5Pureza:≥95%Cor e Forma:SolidPeso molecular:499.6AGLME
CAS:<p>AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.</p>Fórmula:C11H21N3O4Cor e Forma:SolidPeso molecular:259.3Evogliptin HCl
CAS:<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Fórmula:C19H27ClF3N3O3Cor e Forma:SolidPeso molecular:437.88LY 806303
CAS:<p>LY 806303 is a highly selective thrombin inhibitor.</p>Fórmula:C16H14O5SPureza:98%Cor e Forma:SolidPeso molecular:318.34ZYZ-488
CAS:<p>ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.</p>Fórmula:C20H29N3O11Pureza:99.04%Cor e Forma:SolidPeso molecular:487.462-MPPA
CAS:<p>2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.</p>Fórmula:C8H14O4SPureza:99.81%Cor e Forma:SolidPeso molecular:206.26Nucleoside-Analog-2
CAS:<p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>Fórmula:C9H11N5O6Pureza:98%Cor e Forma:SolidPeso molecular:285.21Ici 186756
CAS:Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.Fórmula:C33H49N5O9Pureza:98%Cor e Forma:SolidPeso molecular:659.77GLS1 Inhibitor
CAS:<p>GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.</p>Fórmula:C19H21N7O2SCor e Forma:SolidPeso molecular:411.48MMP2-IN-2
CAS:<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Fórmula:C13H8N4O4Pureza:98.09%Cor e Forma:SolidPeso molecular:284.23NVP DPP 728 dihydrochloride
CAS:<p>NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.</p>Fórmula:C15H18N6OCor e Forma:SolidPeso molecular:298.34Bz-D-Arg-pNA hydrochloride
CAS:<p>Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.</p>Fórmula:C19H23ClN6O4Cor e Forma:SolidPeso molecular:434.88ND-336
CAS:<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Fórmula:C16H18ClNO3S2Cor e Forma:SolidPeso molecular:371.9YM-53601
CAS:<p>YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.</p>Fórmula:C21H22ClFN2OPureza:99.65%Cor e Forma:SolidPeso molecular:372.86Nucleoside-Analog-1
CAS:Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.Fórmula:C9H9N5O5Pureza:98%Cor e Forma:SolidPeso molecular:267.2Chymase-IN-2
CAS:<p>Chymase-IN-2 is a modulator of chymase.</p>Fórmula:C19H15ClF2NO3PSPureza:98%Cor e Forma:SolidPeso molecular:441.82GS-9256
CAS:<p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>Fórmula:C46H56ClF2N6O8PSPureza:98%Cor e Forma:SolidPeso molecular:957.46A-953227
CAS:<p>A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.</p>Fórmula:C25H20FN5O3Pureza:98%Cor e Forma:SolidPeso molecular:457.46L 658758
CAS:<p>L 658758 is an inhibitor of serine proteinase.</p>Fórmula:C16H20N2O9SCor e Forma:SolidPeso molecular:416.4Z-LLF-CHO
CAS:<p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>Fórmula:C29H39N3O5Pureza:98%Cor e Forma:SolidPeso molecular:509.64WAY-151693
CAS:<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Fórmula:C21H22ClN3O5SCor e Forma:SolidPeso molecular:463.93Duazomycin
CAS:<p>Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.</p>Fórmula:C8H11N3O4Cor e Forma:SolidPeso molecular:213.19Moxicoumone
CAS:<p>Moxicoumone is an anticoagulant agent.</p>Fórmula:C22H30N2O6Pureza:98%Cor e Forma:SolidPeso molecular:418.48MMP13-IN-4
CAS:<p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>Fórmula:C21H17BrN4O5Pureza:98%Cor e Forma:SolidPeso molecular:485.29Tyrosinase-IN-11
CAS:<p>Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.</p>Fórmula:C15H14O5Cor e Forma:SolidPeso molecular:274.27Epostatin
CAS:<p>Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.</p>Fórmula:C23H33N3O5Pureza:98%Cor e Forma:SolidPeso molecular:431.53GSK-2793660
CAS:GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.Fórmula:C20H27N3O3Pureza:98%Cor e Forma:SolidPeso molecular:357.45Cathepsin L/S-IN-1
<p>Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.</p>Fórmula:C29H33BrN4O4SCor e Forma:SolidPeso molecular:613.57TNK2-IN-1
CAS:<p>TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.</p>Fórmula:C23H24N6O2Cor e Forma:SolidPeso molecular:416.48Tyrphostin A46
CAS:<p>Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.</p>Fórmula:C10H8N2O3Pureza:98%Cor e Forma:Off-White SolidPeso molecular:204.18K 579
CAS:<p>K 579 is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C17H24N6OPureza:98%Cor e Forma:SolidPeso molecular:328.41PTIQ
CAS:<p>MMP-3 expression inhibitor</p>Fórmula:C13H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:235.28Flovagatran
CAS:Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.Fórmula:C27H36BN3O7Pureza:99.56%Cor e Forma:SolidPeso molecular:525.4N-Phenylthiourea
CAS:<p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>Fórmula:C7H8N2SPureza:99.71%Cor e Forma:SolidPeso molecular:152.22Glutaminase-IN-4
CAS:<p>Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).</p>Fórmula:C23H22N6O2S2Cor e Forma:SolidPeso molecular:478.59JPM-OEt
CAS:<p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>Fórmula:C20H28N2O6Pureza:98%Cor e Forma:SolidPeso molecular:392.45KIN1400
CAS:<p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>Fórmula:C24H17F2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:449.47Grazoprevir sodium salt
CAS:Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.Fórmula:C38H50N6NaO9SPureza:98%Cor e Forma:SolidPeso molecular:789.9Prodipine hydrochloride
CAS:<p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>Fórmula:C20H26ClNPureza:98%Cor e Forma:SolidPeso molecular:315.88ZM223 hydrochloride (2031177-48-5 free base)
<p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>Fórmula:C23H18ClF3N4O2S2Pureza:98%Cor e Forma:SolidPeso molecular:538.99FK-448 Free base
CAS:<p>FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.</p>Fórmula:C25H30N2O3Pureza:98%Cor e Forma:SolidPeso molecular:406.52(S)-BI-1001
CAS:<p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>Fórmula:C19H15BrClNO3Pureza:98%Cor e Forma:SolidPeso molecular:420.68BC-23
CAS:<p>BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.</p>Fórmula:C21H14ClN3O4SPureza:98%Cor e Forma:SolidPeso molecular:439.87BMS-986094
CAS:<p>INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.</p>Fórmula:C30H39N6O9PCor e Forma:SolidPeso molecular:658.64Navuridine
CAS:<p>Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.</p>Fórmula:C9H11N5O4Pureza:99.83%Cor e Forma:SolidPeso molecular:253.22p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Fórmula:C7H11Cl2N3Pureza:99.00% - 99.56%Cor e Forma:SolidPeso molecular:208.088LB-30057
CAS:<p>LB-30057 is used as an oral thrombin inhibitor.</p>Fórmula:C26H31N5O3SPureza:98%Cor e Forma:SolidPeso molecular:493.62U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Cor e Forma:SolidPeso molecular:448.56MDL-101146, (S)-
CAS:<p>MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.</p>Fórmula:C29H37F5N4O6Pureza:98%Cor e Forma:SolidPeso molecular:632.62PMPA sodium
CAS:<p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>Fórmula:C6H11Na4O7PPureza:98%Cor e Forma:SolidPeso molecular:318.08IMB-26
CAS:<p>IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.</p>Fórmula:C20H23BrN2O6Cor e Forma:SolidPeso molecular:467.31Diprotin B
CAS:<p>Diprotin B is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C16H29N3O4Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:327.42Desethyl KBT-3022
CAS:<p>Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.</p>Fórmula:C23H20N2O4SPureza:98%Cor e Forma:SolidPeso molecular:420.48PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Cor e Forma:SolidPeso molecular:464.96DTS
CAS:<p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>Fórmula:C14H14S3Pureza:98%Cor e Forma:SolidPeso molecular:278.46ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Fórmula:C24H32F3N3O5Pureza:95% - 99.53%Cor e Forma:SolidPeso molecular:499.52STOCK2S-26016
CAS:<p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>Fórmula:C20H19N3O2Cor e Forma:SolidPeso molecular:333.38FQ
CAS:<p>FQ is a novel reversible inhibitor of mixed-type tyrosinase.</p>Fórmula:C14H9FN2OCor e Forma:SolidPeso molecular:240.23NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Fórmula:C13H20N2O5SPureza:98.41%Cor e Forma:SolidPeso molecular:316.37AA9 TG2 inhibitor
CAS:<p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>Fórmula:C32H36N4O5Cor e Forma:SolidPeso molecular:556.65Desirudin
CAS:<p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>Cor e Forma:SolidCyclophilin inhibitor 3
CAS:<p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>Fórmula:C34H38N4O6Cor e Forma:SolidPeso molecular:598.69SLK/STK10-IN-1
CAS:<p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>Fórmula:C17H13ClN2O3Pureza:99.34%Cor e Forma:SolidPeso molecular:328.75ADAMTS-5 Inhibitor
CAS:<p>ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.</p>Fórmula:C16H11ClF3N3OS3Pureza:99.66%Cor e Forma:SolidPeso molecular:449.92AL-9
CAS:<p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>Fórmula:C23H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:402.45TNIK-IN-1
CAS:<p>TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).</p>Fórmula:C19H17N5O3SPureza:98%Cor e Forma:SolidPeso molecular:395.43Diethyl pyimDC
CAS:<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Fórmula:C14H15N3O4Cor e Forma:SolidPeso molecular:289.29Aldumastat
CAS:Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.Fórmula:C20H24F2N4O3Pureza:99.87%Cor e Forma:SolidPeso molecular:406.43RID-F
CAS:<p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>Fórmula:C38H50N2O2Pureza:98%Cor e Forma:SolidPeso molecular:566.82Efegatran sulfate
CAS:<p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>Fórmula:C21H34N6O7SPureza:≥98% - ≥98%Cor e Forma:SolidPeso molecular:514.6MK-4882
CAS:<p>MK-4882 is an effective inhibitor of HCV NS5A.</p>Fórmula:C42H50N8O7Pureza:98%Cor e Forma:SolidPeso molecular:778.9
