Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(34 produtos)
- Cisteína Protease(96 produtos)
- DPP-4(20 produtos)
- Glutaminase(40 produtos)
- HIV Protease(449 produtos)
- PAI-1(25 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(53 produtos)
- Proteassoma(94 produtos)
- Protease serina(50 produtos)
- p97(14 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1044 produtos de "Proteases/Proteassoma"
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Zampilimab
CAS:<p>Zampilimab (UCB-7858) is a humanised monoclonal antibody targeting TGM2, inhibits the cross-linking transamidase activity of TG2, renal fibrosis.</p>Pureza:95%Cor e Forma:LiquidHCV-IN-30
CAS:<p>HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).</p>Fórmula:C36H44N6O4Pureza:99.6%Cor e Forma:SolidPeso molecular:624.77Carboxypeptidase G2 (CPG2) Inhibitor
CAS:<p>Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.</p>Fórmula:C13H15NO6SPureza:99.96%Cor e Forma:SolidPeso molecular:313.33Cathepsin Inhibitor 1
CAS:<p>Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.</p>Fórmula:C20H24ClN5O2Pureza:99.78%Cor e Forma:SolidPeso molecular:401.89A-933548
CAS:<p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>Fórmula:C25H21N5O3Pureza:98%Cor e Forma:SolidPeso molecular:439.47Cysteine Protease inhibitor hydrochloride
CAS:<p>Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.</p>Fórmula:C18H15ClN4OPureza:98%Cor e Forma:SolidPeso molecular:338.79Tec-IN-21
CAS:<p>Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).</p>Fórmula:C16H15ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:362.83Sheng Gelieting
CAS:<p>CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.</p>Fórmula:C17H16F6N4OCor e Forma:SolidPeso molecular:406.33CP-471474
CAS:<p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>Fórmula:C16H17FN2O5SPureza:98%Cor e Forma:SolidPeso molecular:368.38AGLME
CAS:<p>AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.</p>Fórmula:C11H21N3O4Cor e Forma:SolidPeso molecular:259.3SJA6017
CAS:<p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>Fórmula:C17H25FN2O4SPureza:98%Cor e Forma:SolidPeso molecular:372.45SQ 32602
CAS:<p>SQ 32602 is a cathepsin E inhibitor.</p>Fórmula:C32H52N3O7PCor e Forma:SolidPeso molecular:621.74Tyrosinase-IN-8
<p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>Fórmula:C16H12O4Cor e Forma:SolidPeso molecular:268.26DPP-4-IN-2
CAS:<p>DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.</p>Fórmula:C18H18N6OCor e Forma:SolidPeso molecular:334.38Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Fórmula:C32H30F3N5O7S2Pureza:98%Cor e Forma:SolidPeso molecular:717.73Thrombin Inhibitor 2
CAS:<p>Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.</p>Fórmula:C19H16ClF3N6O2Pureza:98%Cor e Forma:SolidPeso molecular:452.82(Rac)-Tanomastat
CAS:<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Fórmula:C23H19ClO3SCor e Forma:SolidPeso molecular:410.91PSI-7409 tetrasodium
CAS:<p>PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.</p>Fórmula:C10H16FN2Na4O14P3Pureza:98%Cor e Forma:SolidPeso molecular:592.117Evogliptin HCl
CAS:<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Fórmula:C19H27ClF3N3O3Cor e Forma:SolidPeso molecular:437.88LY 806303
CAS:<p>LY 806303 is a highly selective thrombin inhibitor.</p>Fórmula:C16H14O5SPureza:98%Cor e Forma:SolidPeso molecular:318.34Nucleoside-Analog-2
CAS:<p>Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.</p>Fórmula:C9H11N5O6Pureza:98%Cor e Forma:SolidPeso molecular:285.21BI-L 45XX
CAS:<p>BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.</p>Fórmula:C10H9F3N2O2SCor e Forma:SolidPeso molecular:278.25Tyrphostin 47
CAS:<p>Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.</p>Fórmula:C10H8N2O2SCor e Forma:SolidPeso molecular:220.25Levovirin valinate HCl
CAS:<p>Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.</p>Fórmula:C13H22ClN5O6Pureza:98%Cor e Forma:SolidPeso molecular:379.8Ici 186756
CAS:<p>Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.</p>Fórmula:C33H49N5O9Pureza:98%Cor e Forma:SolidPeso molecular:659.77Chymase-IN-2
CAS:<p>Chymase-IN-2 is a modulator of chymase.</p>Fórmula:C19H15ClF2NO3PSPureza:98%Cor e Forma:SolidPeso molecular:441.82A-953227
CAS:<p>A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.</p>Fórmula:C25H20FN5O3Pureza:98%Cor e Forma:SolidPeso molecular:457.46Duazomycin
CAS:<p>Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.</p>Fórmula:C8H11N3O4Cor e Forma:SolidPeso molecular:213.19Moxicoumone
CAS:<p>Moxicoumone is an anticoagulant agent.</p>Fórmula:C22H30N2O6Pureza:98%Cor e Forma:SolidPeso molecular:418.48GLS1 Inhibitor
CAS:<p>GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.</p>Fórmula:C19H21N7O2SCor e Forma:SolidPeso molecular:411.48Tyrphostin A46
CAS:<p>Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.</p>Fórmula:C10H8N2O3Pureza:98%Cor e Forma:Off-White SolidPeso molecular:204.18NVP DPP 728 dihydrochloride
CAS:<p>NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.</p>Fórmula:C15H18N6OCor e Forma:SolidPeso molecular:298.34MDK0734
CAS:<p>MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Fórmula:C15H17N3O2Pureza:98%Cor e Forma:SolidPeso molecular:271.31Bz-D-Arg-pNA hydrochloride
CAS:<p>Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.</p>Fórmula:C19H23ClN6O4Cor e Forma:SolidPeso molecular:434.88FQ
CAS:<p>FQ is a novel reversible inhibitor of mixed-type tyrosinase.</p>Fórmula:C14H9FN2OCor e Forma:SolidPeso molecular:240.23ND-336
CAS:<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Fórmula:C16H18ClNO3S2Cor e Forma:SolidPeso molecular:371.9ADAMTS-5 Inhibitor
CAS:<p>ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.</p>Fórmula:C16H11ClF3N3OS3Pureza:99.66%Cor e Forma:SolidPeso molecular:449.92DPP-IV-IN-1
CAS:<p>DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).</p>Fórmula:C11H18FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:243.28TNIK-IN-1
CAS:<p>TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).</p>Fórmula:C19H17N5O3SPureza:98%Cor e Forma:SolidPeso molecular:395.43Diethyl pyimDC
CAS:<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Fórmula:C14H15N3O4Cor e Forma:SolidPeso molecular:289.29Aldumastat
CAS:<p>Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.</p>Fórmula:C20H24F2N4O3Pureza:99.87%Cor e Forma:SolidPeso molecular:406.43YM-53601
CAS:<p>YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.</p>Fórmula:C21H22ClFN2OPureza:99.65%Cor e Forma:SolidPeso molecular:372.86MK-4882
CAS:<p>MK-4882 is an effective inhibitor of HCV NS5A.</p>Fórmula:C42H50N8O7Pureza:98%Cor e Forma:SolidPeso molecular:778.9Gosogliptin
CAS:<p>Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.</p>Fórmula:C17H24F2N6OPureza:99.74%Cor e Forma:SolidPeso molecular:366.41Nucleoside-Analog-1
CAS:<p>Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.</p>Fórmula:C9H9N5O5Pureza:98%Cor e Forma:SolidPeso molecular:267.2Sortin1
CAS:<p>Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.</p>Fórmula:C26H19NO6Pureza:98%Cor e Forma:SolidPeso molecular:441.43MDK7677
CAS:<p>MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>Fórmula:C12H10N4O3Cor e Forma:SolidPeso molecular:258.23Furaprofen
CAS:<p>Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.</p>Fórmula:C17H14O3Pureza:98.49% - 99.52%Cor e Forma:SolidPeso molecular:266.29GEMSA
CAS:<p>GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].</p>Fórmula:C7H13N3O4SCor e Forma:SolidPeso molecular:235.26WAY-151693
CAS:<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Fórmula:C21H22ClN3O5SCor e Forma:SolidPeso molecular:463.93AK 275
CAS:<p>AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.</p>Fórmula:C20H31N3O4Cor e Forma:SolidPeso molecular:377.48AZD-9684
CAS:<p>AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.</p>Fórmula:C10H14N2O2SCor e Forma:SolidPeso molecular:226.3ITX-4520
CAS:<p>ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.</p>Fórmula:C24H23F2N3OSCor e Forma:SolidPeso molecular:439.52Epostatin
CAS:<p>Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.</p>Fórmula:C23H33N3O5Pureza:98%Cor e Forma:SolidPeso molecular:431.53L 722151
CAS:<p>L 722151 is an FXIIIa inhibitor.</p>Fórmula:C8H9ClN2O5S3Pureza:98%Cor e Forma:SolidPeso molecular:344.82Chymase-IN-1
CAS:<p>Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).</p>Fórmula:C20H15ClNO4PSPureza:99.17%Cor e Forma:SolidPeso molecular:431.83GSK-2793660
CAS:<p>GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.</p>Fórmula:C20H27N3O3Pureza:98%Cor e Forma:SolidPeso molecular:357.45ADAMTS-5-IN-2
CAS:<p>ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.</p>Fórmula:C17H15N3OSCor e Forma:SolidPeso molecular:309.39Safironil
CAS:<p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>Fórmula:C15H23N3O4Pureza:99.83%Cor e Forma:SolidPeso molecular:309.36TNK2-IN-1
CAS:<p>TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.</p>Fórmula:C23H24N6O2Cor e Forma:SolidPeso molecular:416.48SP-Chymostatin B
CAS:<p>SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.</p>Fórmula:C30H41N7O6Pureza:98%Cor e Forma:SolidPeso molecular:595.69K 579
CAS:<p>K 579 is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C17H24N6OPureza:98%Cor e Forma:SolidPeso molecular:328.41Antiviral agent 30
CAS:<p>Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].</p>Fórmula:C21H32N2O3SCor e Forma:SolidPeso molecular:392.56PTIQ
CAS:<p>MMP-3 expression inhibitor</p>Fórmula:C13H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:235.28BAY-678 racemate
CAS:<p>BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.</p>Fórmula:C20H15F3N4O2Pureza:98%Cor e Forma:SolidPeso molecular:400.35WNK-IN-7
CAS:<p>WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.</p>Fórmula:C26H29N3OPureza:98%Cor e Forma:SolidPeso molecular:399.53ABT-770
CAS:<p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>Fórmula:C22H22F3N3O6Cor e Forma:SolidPeso molecular:481.42BR351 precursor
CAS:<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C27H32N2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:576.68CA 074
CAS:<p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>Fórmula:C18H29N3O6Pureza:97.80%Cor e Forma:SolidPeso molecular:383.44XMU-MP-2
CAS:<p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>Fórmula:C32H33F3N8O2Pureza:99.29%Cor e Forma:SolidPeso molecular:618.65RS-104966
CAS:<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Fórmula:C19H21NO6SPureza:98%Cor e Forma:SolidPeso molecular:391.44Ono-3307 mesylate
CAS:<p>no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.</p>Fórmula:C15H18N4O7S2Pureza:97.60% - 98.16%Cor e Forma:SolidPeso molecular:430.46Thrombin inhibitor 6
CAS:<p>Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.</p>Fórmula:C18H19ClN4O2SCor e Forma:SolidPeso molecular:390.892',5-Difluoro-2'-deoxycytidine
CAS:<p>2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.</p>Fórmula:C9H11F2N3O4Pureza:98%Cor e Forma:SolidPeso molecular:263.2Gü1303
CAS:<p>Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).</p>Fórmula:C20H22N4O3Cor e Forma:SolidPeso molecular:366.41LY 135305
CAS:<p>LY 135305 is a inhibition of spontaneous metastasis.</p>Fórmula:C19H20ClNPureza:98%Cor e Forma:SolidPeso molecular:297.82Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Fórmula:C23H31N3NaO4S2Pureza:98%Cor e Forma:SolidPeso molecular:500.63HCV-IN-37
CAS:<p>HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.</p>Fórmula:C31H35F2N5Cor e Forma:SolidPeso molecular:515.64BrBzGCp2
CAS:<p>BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.</p>Fórmula:C27H38BrN3O6SPureza:98.68% - 98.68%Cor e Forma:SolidPeso molecular:612.58ACH-806
CAS:<p>ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.</p>Fórmula:C19H20F3N3O2SPureza:98%Cor e Forma:SolidPeso molecular:411.44Tyrosinase-IN-1
CAS:<p>Tyrosinase-IN-1: potent inhibitor for skin-whitening & food preservation with uses in cosmetics & medicine.</p>Fórmula:C10H9N3O2S2Cor e Forma:SolidPeso molecular:267.33KIN1400
CAS:<p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>Fórmula:C24H17F2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:449.47MK-2048
CAS:<p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>Fórmula:C21H21ClFN5O4Pureza:98%Cor e Forma:SolidPeso molecular:461.87OM-189
CAS:<p>OM-189 is a selective inhibitor of synthetic thrombin.</p>Fórmula:C24H36N6O3SPureza:98%Cor e Forma:SolidPeso molecular:488.65Adafosbuvir PM
CAS:<p>Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.</p>Fórmula:C10H13FN2O6Pureza:97.08%Cor e Forma:SolidPeso molecular:276.22FK-448 Free base
CAS:<p>FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.</p>Fórmula:C25H30N2O3Pureza:98%Cor e Forma:SolidPeso molecular:406.52BMS-986094
CAS:<p>INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.</p>Fórmula:C30H39N6O9PCor e Forma:SolidPeso molecular:658.64BR351
CAS:<p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C20H25FN2O5SPureza:98%Cor e Forma:SolidPeso molecular:424.49LB-30057
CAS:<p>LB-30057 is used as an oral thrombin inhibitor.</p>Fórmula:C26H31N5O3SPureza:98%Cor e Forma:SolidPeso molecular:493.62U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Cor e Forma:SolidPeso molecular:448.56MDL-101146, (S)-
CAS:<p>MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.</p>Fórmula:C29H37F5N4O6Pureza:98%Cor e Forma:SolidPeso molecular:632.62Gemigliptin Tartrate(911637-19-9 free base)
CAS:<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Fórmula:C22H25F8N5O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:639.45Cysteine protease inhibitor-2
CAS:<p>Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.</p>Fórmula:C13H5N5OPureza:98%Cor e Forma:SolidPeso molecular:247.21ZD8321
CAS:<p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>Fórmula:C18H28F3N3O5Pureza:98%Cor e Forma:SolidPeso molecular:423.43Proteasome-IN-1
CAS:<p>Proteasome-IN-1 is an inhibitor of proteasome.</p>Fórmula:C42H35N5O3Pureza:98%Cor e Forma:SolidPeso molecular:657.76Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Fórmula:C23H19ClO3SPureza:98%Cor e Forma:SolidPeso molecular:410.91IMB-26
CAS:<p>IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.</p>Fórmula:C20H23BrN2O6Cor e Forma:SolidPeso molecular:467.31TAPI-1
CAS:<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Fórmula:C26H37N5O5Pureza:≥95%Cor e Forma:SolidPeso molecular:499.6Desethyl KBT-3022
CAS:<p>Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.</p>Fórmula:C23H20N2O4SPureza:98%Cor e Forma:SolidPeso molecular:420.48ZYZ-488
CAS:<p>ZYZ-488 is an Apoptosis protease activating factor-1 (Apaf-1) inhibitor, which suppresses the activation of procaspase-9 and procaspase-3.</p>Fórmula:C20H29N3O11Pureza:99.04%Cor e Forma:SolidPeso molecular:487.46STOCK2S-26016
CAS:<p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>Fórmula:C20H19N3O2Cor e Forma:SolidPeso molecular:333.38Efegatran sulfate
CAS:<p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>Fórmula:C21H34N6O7SPureza:≥98% - ≥98%Cor e Forma:SolidPeso molecular:514.6AA9 TG2 inhibitor
CAS:<p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>Fórmula:C32H36N4O5Cor e Forma:SolidPeso molecular:556.65Desirudin
CAS:<p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>Cor e Forma:SolidGS-9256
CAS:<p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>Fórmula:C46H56ClF2N6O8PSPureza:98%Cor e Forma:SolidPeso molecular:957.46Z-LLF-CHO
CAS:<p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>Fórmula:C29H39N3O5Pureza:98%Cor e Forma:SolidPeso molecular:509.64MMP13-IN-4
CAS:<p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>Fórmula:C21H17BrN4O5Pureza:98%Cor e Forma:SolidPeso molecular:485.29Cyclophilin inhibitor 3
CAS:<p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>Fórmula:C34H38N4O6Cor e Forma:SolidPeso molecular:598.69ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Fórmula:C15H16ClNO3S2Pureza:99.49%Cor e Forma:SolidPeso molecular:357.88DTS
CAS:<p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>Fórmula:C14H14S3Pureza:98%Cor e Forma:SolidPeso molecular:278.46Prodipine hydrochloride
CAS:<p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>Fórmula:C20H26ClNPureza:98%Cor e Forma:SolidPeso molecular:315.88SLK/STK10-IN-1
CAS:<p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>Fórmula:C17H13ClN2O3Pureza:99.34%Cor e Forma:SolidPeso molecular:328.75ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Fórmula:C24H32F3N3O5Pureza:95% - 99.53%Cor e Forma:SolidPeso molecular:499.52Grazoprevir sodium salt
CAS:<p>Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.</p>Fórmula:C38H50N6NaO9SPureza:98%Cor e Forma:SolidPeso molecular:789.9Tyrosinase-IN-4
CAS:<p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>Fórmula:C15H9ClO3Cor e Forma:SolidPeso molecular:272.68JPM-OEt
CAS:<p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>Fórmula:C20H28N2O6Pureza:98%Cor e Forma:SolidPeso molecular:392.45N-Phenylthiourea
CAS:<p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>Fórmula:C7H8N2SPureza:99.71%Cor e Forma:SolidPeso molecular:152.22(S)-BI-1001
CAS:<p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>Fórmula:C19H15BrClNO3Pureza:98%Cor e Forma:SolidPeso molecular:420.68p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Fórmula:C7H11Cl2N3Pureza:99.00% - 99.56%Cor e Forma:SolidPeso molecular:208.088PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Cor e Forma:SolidPeso molecular:464.96Ro 09-1679
CAS:<p>Ro 09-1679 is a thrombin inhibitor.</p>Fórmula:C22H39N9O6Pureza:98%Cor e Forma:SolidPeso molecular:525.6Cathepsin L/S-IN-1
<p>Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.</p>Fórmula:C29H33BrN4O4SCor e Forma:SolidPeso molecular:613.57NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Fórmula:C13H20N2O5SPureza:98.41%Cor e Forma:SolidPeso molecular:316.37Navuridine
CAS:<p>Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.</p>Fórmula:C9H11N5O4Pureza:99.83%Cor e Forma:SolidPeso molecular:253.22ZM223 hydrochloride (2031177-48-5 free base)
<p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>Fórmula:C23H18ClF3N4O2S2Pureza:98%Cor e Forma:SolidPeso molecular:538.99Diprotin B
CAS:<p>Diprotin B is a dipeptidyl peptidase IV inhibitor.</p>Fórmula:C16H29N3O4Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:327.42HCV-IN-3
CAS:<p>HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).</p>Fórmula:C13H11F2NOPureza:98%Cor e Forma:SolidPeso molecular:235.23Calpain Inhibitor XII
CAS:<p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>Fórmula:C26H34N4O5Cor e Forma:SolidPeso molecular:482.57Flovagatran
CAS:<p>Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.</p>Fórmula:C27H36BN3O7Pureza:99.56%Cor e Forma:SolidPeso molecular:525.4RO-9187
CAS:<p>RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).</p>Fórmula:C9H12N6O5Pureza:98%Cor e Forma:SolidPeso molecular:284.23Plasma kallikrein-IN-3
CAS:<p>Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.</p>Fórmula:C20H23N5O2Cor e Forma:SolidPeso molecular:365.432-MPPA
CAS:<p>2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.</p>Fórmula:C8H14O4SPureza:99.81%Cor e Forma:SolidPeso molecular:206.26Calpain-2-IN-1
CAS:<p>Calpain-2-IN-1 is a selective calpain-2 inhibitor that prolongs ERK activation and thus enhances learning and memory.</p>Fórmula:C28H37N3O7Cor e Forma:SolidPeso molecular:527.61Tyrosinase-IN-10
CAS:<p>Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'</p>Fórmula:C16H12O4Cor e Forma:SolidPeso molecular:268.26TAPI-0
CAS:<p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>Fórmula:C24H32N4O5Cor e Forma:SolidPeso molecular:456.53NAAA-IN-2
CAS:<p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>Fórmula:C11H13N3O2SCor e Forma:SolidPeso molecular:251.3HCV-IN-35
CAS:<p>HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.</p>Fórmula:C30H36ClN5Cor e Forma:SolidPeso molecular:502.09MMP-1-IN-1
<p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>Fórmula:C14H17ClN2O3Cor e Forma:SolidPeso molecular:296.75Calpain Inhibitor XI
CAS:<p>Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.</p>Fórmula:C26H40N4O6Cor e Forma:SolidPeso molecular:504.62(3S,4S)-A2-32-01
<p>(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .</p>Fórmula:C19H27NO2Cor e Forma:SolidPeso molecular:301.42Azo-Resveratrol
CAS:<p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>Fórmula:C12H10N2O3Cor e Forma:SolidPeso molecular:230.22AM 4299 B
CAS:<p>AM 4299 B is a novel inhibitor of a thiol protease.</p>Fórmula:C16H27N3O7Pureza:98%Cor e Forma:SolidPeso molecular:373.4HCV-IN-34
CAS:<p>HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.</p>Fórmula:C31H36ClN5Cor e Forma:SolidPeso molecular:514.1MDL 27399
CAS:<p>MDL 27399 suppresses human neutrophil cathepsin G.</p>Fórmula:C26H36N4O8Cor e Forma:SolidPeso molecular:532.59Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Fórmula:C15H10O5Pureza:99%Cor e Forma:SolidPeso molecular:270.24CAA0225
CAS:<p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>Fórmula:C28H29N3O5Cor e Forma:SolidPeso molecular:487.55BC-05
CAS:<p>BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for</p>Fórmula:C21H29BN2O9Pureza:98%Cor e Forma:SolidPeso molecular:464.27RID-F
CAS:<p>RID-F is an inhibitor of the nonpeptidic proteasome.</p>Fórmula:C38H50N2O2Pureza:98%Cor e Forma:SolidPeso molecular:566.82AL-9
CAS:<p>AL-9 is a GT-1b and GT-2a replication inhibitor.</p>Fórmula:C23H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:402.45Immunoproteasome inhibitor 1
CAS:<p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>Fórmula:C20H26N2O4Cor e Forma:SolidPeso molecular:358.43PMPA sodium
CAS:<p>PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.</p>Fórmula:C6H11Na4O7PPureza:98%Cor e Forma:SolidPeso molecular:318.08JO146
CAS:<p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂，其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM，可应用于细菌感染的抑制。</p>Fórmula:C31H44N3O7PCor e Forma:SolidPeso molecular:601.67L-873724
CAS:<p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>Fórmula:C23H26F3N3O3SPureza:98%Cor e Forma:SolidPeso molecular:481.53(R)-ND-336
CAS:<p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>Fórmula:C16H18ClNO3S2Cor e Forma:SolidPeso molecular:371.89Tyrosinase-IN-11
CAS:<p>Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.</p>Fórmula:C15H14O5Cor e Forma:SolidPeso molecular:274.27Kallikrein 5-IN-2
CAS:<p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.</p>Fórmula:C23H22N6OCor e Forma:SolidPeso molecular:398.46VA4 TG2 inhibitor
CAS:<p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>Fórmula:C33H41N5O6SCor e Forma:SolidPeso molecular:635.77AZD5248
CAS:<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Fórmula:C22H22N4O2Cor e Forma:SolidPeso molecular:374.44MMP-2/9-IN-1
CAS:<p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>Fórmula:C14H16IN7SCor e Forma:SolidPeso molecular:441.29GLS1 Inhibitor-3
CAS:<p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>Fórmula:C30H32N10O2SCor e Forma:SolidPeso molecular:596.71Elastase-IN-1
CAS:<p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>Fórmula:C17H12N4O3Cor e Forma:SolidPeso molecular:320.3HCV-IN-36
CAS:<p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>Fórmula:C30H36ClN5Cor e Forma:SolidPeso molecular:502.09BRD-8899
CAS:<p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>Fórmula:C17H22N4O3SCor e Forma:SolidPeso molecular:362.45Tyrosinase-IN-5
CAS:<p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>Fórmula:C18H13N3O6Cor e Forma:SolidPeso molecular:367.31BMS-363131
CAS:<p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.</p>Fórmula:C28H40N6O5Pureza:97.99%Cor e Forma:SolidPeso molecular:540.65α-Glucosidase-IN-5
CAS:<p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>Fórmula:C15H13NO3Cor e Forma:SolidPeso molecular:255.27SAP2-IN-1
CAS:<p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>Fórmula:C34H29NO7Cor e Forma:SolidPeso molecular:563.6Elasnin
CAS:<p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>Fórmula:C24H40O4Cor e Forma:SolidPeso molecular:392.57MMP2-IN-2
CAS:<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Fórmula:C13H8N4O4Pureza:98.09%Cor e Forma:SolidPeso molecular:284.23Glutaminase-IN-4
CAS:<p>Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).</p>Fórmula:C23H22N6O2S2Cor e Forma:SolidPeso molecular:478.59L 658758
CAS:<p>L 658758 is an inhibitor of serine proteinase.</p>Fórmula:C16H20N2O9SCor e Forma:SolidPeso molecular:416.4ASPER-29
CAS:<p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>Fórmula:C31H29BrN2O5SCor e Forma:SolidPeso molecular:621.54CAY10704
CAS:<p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>Fórmula:C18H20Cl2N2Cor e Forma:SolidPeso molecular:335.27DPP-4-IN-1
CAS:<p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>Fórmula:C19H19ClN6Cor e Forma:SolidPeso molecular:366.85AA10 TG2 inhibitor
CAS:<p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>Fórmula:C32H36N4O5Cor e Forma:SolidPeso molecular:556.65BAY8040
CAS:<p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>Fórmula:C21H16F3N5O2Cor e Forma:SolidPeso molecular:427.38PK44 phosphate
CAS:<p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>Fórmula:C17H19F5N7O5PCor e Forma:SolidPeso molecular:527.349VEL-0230
CAS:<p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>Fórmula:C14H24NNaO5Cor e Forma:SolidPeso molecular:309.33Alicapistat
CAS:<p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>Fórmula:C25H27N3O4Pureza:98%Cor e Forma:SolidPeso molecular:433.5Tyrosinase-IN-6
CAS:<p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>Fórmula:C24H31N3O2Cor e Forma:SolidPeso molecular:393.52Cysteine Protease inhibitor
CAS:<p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>Fórmula:C18H14N4OPureza:98%Cor e Forma:SolidPeso molecular:302.33Anticancer agent 82
CAS:<p>Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.</p>Fórmula:C19H18Cl2N4OCor e Forma:SolidPeso molecular:389.28Tyrosinase-IN-3
CAS:<p>Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.</p>Fórmula:C21H23NO5Cor e Forma:SolidPeso molecular:369.41BC-23
CAS:<p>BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.</p>Fórmula:C21H14ClN3O4SPureza:98%Cor e Forma:SolidPeso molecular:439.87Gü2602
CAS:<p>Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for mature</p>Fórmula:C16H22N4O3Cor e Forma:SolidPeso molecular:318.37Cofrogliptin
CAS:<p>Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).</p>Fórmula:C18H19F5N4O3SCor e Forma:SolidPeso molecular:466.43GSK2793660 HCl
CAS:<p>GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.</p>Fórmula:C22H32ClN3O3Cor e Forma:SolidPeso molecular:421.96HCV-IN-33
CAS:<p>HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.</p>Fórmula:C31H36ClN5Cor e Forma:SolidPeso molecular:514.1JNJ-10329670
CAS:<p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>Fórmula:C30H34ClF3N6O3SCor e Forma:SolidPeso molecular:651.14Setrobuvir
CAS:<p>Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension with</p>Fórmula:C25H25FN4O6S2Pureza:98.92% - >99.99%Cor e Forma:SolidPeso molecular:560.62KM-023
CAS:<p>KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.</p>Fórmula:C18H19N3O3Pureza:99.47% - >99.99%Cor e Forma:SolidPeso molecular:325.36AGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Fórmula:C18H17F2N3O2Pureza:98.92%Cor e Forma:SolidPeso molecular:345.34TS-021
CAS:<p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>Fórmula:C17H24FN3O5SPureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:401.4520S Proteasome activator 1
CAS:<p>20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.</p>Fórmula:C27H19ClF2N2OSPureza:99.82%Cor e Forma:SolidPeso molecular:492.97CPA inhibitor
CAS:<p>CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.</p>Fórmula:C18H19NO4Pureza:99.94%Cor e Forma:SolidPeso molecular:313.35Uprifosbuvir
CAS:<p>Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.</p>Fórmula:C22H29ClN3O9PPureza:99.73% - >99.99%Cor e Forma:SolidPeso molecular:545.91Atevirdine
CAS:<p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>Fórmula:C21H25N5O2Pureza:98.20%Cor e Forma:SolidPeso molecular:379.46CZL55
CAS:<p>CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).</p>Fórmula:C20H22N2O6Pureza:98.19%Cor e Forma:SolidPeso molecular:386.4Granotapide
CAS:<p>Granotapide is a microsomal triglyceride transfer protein (MTP) inhibitor that treats and rather prevents atherosclerosis, coronary artery disease, metabolic</p>Fórmula:C39H37F3N2O8Pureza:99.70% - 99.79%Cor e Forma:SolidPeso molecular:718.71BAY-43-9695
CAS:<p>BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.</p>Fórmula:C22H25N3O4SPureza:99.50% - 99.65%Cor e Forma:SolidPeso molecular:427.52
