Proteases/Proteassoma
Os inibidores de proteases e proteassomas são compostos que bloqueiam a atividade das proteases e do proteassoma, que estão envolvidos na degradação e renovação de proteínas. Esses inibidores são vitais para estudar a regulação da homeostase de proteínas, controle do ciclo celular e apoptose. Inibidores de proteases e proteassomas também são utilizados no tratamento de doenças como o câncer, onde a degradação anormal de proteínas desempenha um papel na progressão da doença. Ao inibir proteases ou o proteassoma, esses compostos podem induzir a morte celular em células cancerígenas e são ferramentas essenciais tanto na pesquisa básica quanto no desenvolvimento terapêutico. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteases e proteassomas de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Proteases/Proteassoma"
- Acetil- CoA Carboxilase(36 produtos)
- Cisteína Protease(110 produtos)
- DPP-4(20 produtos)
- Glutaminase(44 produtos)
- HIV Protease(506 produtos)
- PAI-1(26 produtos)
- Inibidores de Protease(50 produtos)
- Receptor activado por protease(54 produtos)
- Proteassoma(95 produtos)
- Protease serina(55 produtos)
- p97(15 produtos)
Exibir 3 mais subcategorias
Foram encontrados 1093 produtos de "Proteases/Proteassoma"
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KGP94
CAS:KGP94 is a potent, selective, and competitive inhibitor of the lysosomal endopeptidase enzyme.Fórmula:C14H12BrN3OSPureza:99.6%Cor e Forma:SolidPeso molecular:350.23Ref: TM-T27730
1mg69,00€5mg145,00€10mg226,00€25mg379,00€50mg538,00€100mg730,00€200mg979,00€1mL*10mM (DMSO)160,00€Camostat free base
CAS:Camostat (FOY 305) inhibits serine protease, treats cancer, viral infections, fibrosis, and blocks SARS-CoV, Coronavirus, and SARS-CoV-2 in studies.Fórmula:C20H22N4O5Cor e Forma:SolidPeso molecular:398.41ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Fórmula:C22H19N3O2SPureza:99.12% - 99.87%Cor e Forma:SolidPeso molecular:389.47Ref: TM-T3423
1mg35,00€5mg80,00€10mg97,00€25mg188,00€50mg311,00€100mg500,00€500mg1.093,00€1mL*10mM (DMSO)88,00€HZ-1157
CAS:HZ-1157 (DHFR-inhibitor) is a hepatitis C virus (HCV) inhibitor with inhibitory activities toward HCV NS3/4A protease.Fórmula:C12H16N4OPureza:98.23%Cor e Forma:SolidPeso molecular:232.28Asunaprevir
CAS:Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.Fórmula:C35H46ClN5O9SPureza:99.34% - 99.8%Cor e Forma:SolidPeso molecular:748.29Ref: TM-T4474
1mg52,00€5mg111,00€10mg180,00€25mg354,00€50mg540,00€100mg778,00€500mg1.605,00€1mL*10mM (DMSO)173,00€Histatin 5 acetate
Histatin 5 acetate inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM, respectively.Fórmula:C135H199N51O35Pureza:98.72%Cor e Forma:SolidPeso molecular:3096.35PSI-6130
CAS:PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.Fórmula:C10H14FN3O4Pureza:98.63% - 99.79%Cor e Forma:SolidPeso molecular:259.23Ref: TM-T7607
1mg40,00€5mg89,00€10mg129,00€25mg224,00€50mg329,00€100mg482,00€200mg652,00€1mL*10mM (DMSO)78,00€Z-Gly-Gly-Arg-AMC TFA (66216-78-2 free base)
CAS:Z-Gly-Gly-Arg-AMC TFA (66216-78-2 free base) is a thrombin-specific fluorogenic substrate for testing thrombin generation in PRP and platelet-poor plasma (PPP).Fórmula:C30H34F3N7O9Pureza:99.77%Cor e Forma:SolidPeso molecular:693.63Ref: TM-T8556
1mg88,00€5mg170,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)251,00€3-O-Ethyl-L-ascorbic acid
CAS:3-O-Ethyl-L-ascorbic acid is a cosmetic tyrosinase inhibitor with whitening ability and is a stabilized vitamin C derivative.Fórmula:C8H12O6Pureza:97.35% - 99.99%Cor e Forma:White To Very Pale Yellow Crystalline Powder Solid PowderPeso molecular:204.18Fulacimstat
CAS:Fulacimstat (BAY1142524) (BAY1142524) is a chymase inhibitor, with IC50s of 3, 4 nM for hamster and human chymase enzyme, respectively.Fórmula:C23H16F3N3O6Pureza:99.77%Cor e Forma:SolidPeso molecular:487.38Ref: TM-TQ0035
1mg106,00€5mg227,00€10mg329,00€25mg540,00€50mg777,00€100mg1.026,00€1mL*10mM (DMSO)244,00€Elbasvir
CAS:<p>Elbasvir (MK-8742) is an NS5A inhibitor developed for chronic HCV treatment.</p>Fórmula:C49H55N9O7Pureza:98.95% - 99.85%Cor e Forma:SolidPeso molecular:882.02PSI-6206
CAS:PSI-6206 (RO 2433) (RO2433) is a selective HCV RNA polymerase inhibitor.Fórmula:C10H13FN2O5Pureza:98% - 99.79%Cor e Forma:SolidPeso molecular:260.22(S,S)-TAPI-1
CAS:"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."Fórmula:C26H37N5O5Cor e Forma:SolidPeso molecular:499.6Ilomastat
CAS:<p>Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C20H28N4O4Pureza:97.04% - 99.51%Cor e Forma:SolidPeso molecular:388.46Trelagliptin succinate
CAS:Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Fórmula:C22H26FN5O6Pureza:99.27% - 99.92%Cor e Forma:SolidPeso molecular:475.47Tenofovir alafenamide hemifumarate
CAS:<p>Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.</p>Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Cor e Forma:SolidPeso molecular:534.51Odanacatib
CAS:Odanacatib is an inhibitor of cathepsin K with potential anti-osteoporotic activity.Fórmula:C25H27F4N3O3SPureza:98.53% - 99.53%Cor e Forma:SolidPeso molecular:525.56Ref: TM-T6035
2mg35,00€5mg52,00€10mg80,00€25mg120,00€50mg188,00€100mg354,00€200mgA consultar1mL*10mM (DMSO)60,00€VCH-916 free acid(1200133-34-1 free base)
CAS:VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Fórmula:C26H37NO4SPureza:98.45%Cor e Forma:SolidPeso molecular:459.64Ledipasvir (acetone)
CAS:Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.Fórmula:C52H60F2N8O7Pureza:99.72%Cor e Forma:SolidPeso molecular:947.08Ref: TM-T4203
1mg35,00€2mg48,00€5mg70,00€10mg93,00€25mg153,00€50mg235,00€100mg359,00€200mgA consultar1mL*10mM (DMSO)96,00€S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFórmula:C13H16O3SPureza:97.33%Cor e Forma:SolidPeso molecular:252.33Ref: TM-T4282
1mg88,00€5mg210,00€10mg338,00€25mg625,00€50mg938,00€100mg1.264,00€1mL*10mM (DMSO)188,00€
