GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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Luseogliflozin
CAS:<p>Luseogliflozin inhibits SGLT2 for glucose uptake with 1.10 nM potency.</p>Fórmula:C23H30O6SCor e Forma:SolidPeso molecular:434.55LRGILS-NH2
CAS:<p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>Fórmula:C29H56N10O7Pureza:98%Cor e Forma:SolidPeso molecular:656.82Alverine hydrochloride
CAS:<p>Alverine hydrochloride is a parasympatholytic.</p>Fórmula:C20H28ClNCor e Forma:SolidPeso molecular:317.9NPC 567
CAS:<p>NPC 567 is an antagonist of the bradykinin receptor.</p>Fórmula:C60H87N19O13Pureza:98%Cor e Forma:SolidPeso molecular:1282.48L-770644 dihydrochloride
CAS:<p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>Fórmula:C30H38ClN7O4SCor e Forma:SolidPeso molecular:628.19M40
CAS:<p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>Fórmula:C94H145N23O24Pureza:98%Cor e Forma:SolidPeso molecular:1981.33FR190997
CAS:<p>FR190997 is an agonist of bradykinin B2 receptor.</p>Fórmula:C37H33Cl2N5O5Cor e Forma:SolidPeso molecular:698.59Etelcalcetide
CAS:<p>Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.</p>Fórmula:C38H73N21O10S2Pureza:98%Cor e Forma:SolidPeso molecular:1048.26ADTN
CAS:<p>ADTN is an agonist of the dopamine receptor.</p>Fórmula:C10H13NO2Pureza:98%Cor e Forma:SolidPeso molecular:179.22AC-178335
CAS:<p>AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.</p>Fórmula:C49H63N13O7Cor e Forma:SolidPeso molecular:946.11NI-0701
<p>NI-0701 is a humanized antibody targeting CCL5/RANTES.</p>Pureza:95.4% (SDS-PAGE); 99.4% (SEC-HPLC) - 95.4% (SDS-PAGE); 99.4% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:145.5kDaApelin-17(human, bovine)
CAS:<p>Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).</p>Fórmula:C96H156N34O20SPureza:98%Cor e Forma:SolidPeso molecular:2138.565-HT2C agonist-4
CAS:<p>Compound 3i, a 5-HT2C agonist-4, acts as an agonist for the 5-HT2C receptor with an EC50 of 5.7 nM. It is capable of reducing locomotor activity in zebrafish larvae.</p>Fórmula:C24H25N5OCor e Forma:SolidPeso molecular:399.49Lobeline sulfate
CAS:<p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>Fórmula:C22H29NO6SPureza:98%Cor e Forma:White PowderPeso molecular:435.54Pneumadin, rat
CAS:<p>Rat Pneumadin (PNM), a decapeptide, stimulates AVP release, exerting strong antidiuretic effects in animals with an active AVP system.</p>Fórmula:C47H74N12O15Pureza:98%Cor e Forma:SolidPeso molecular:1047.17817-phenyl trinor Prostaglandin E2 ethyl amide
CAS:<p>17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.</p>Fórmula:C25H35NO4Cor e Forma:SolidPeso molecular:413.55L 366811
CAS:<p>L 366811 is a potent oxytocin antagonist.</p>Fórmula:C43H56N8O6Cor e Forma:SolidPeso molecular:780.951,8-Cineole
CAS:<p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>Fórmula:C10H18OPureza:97.44% - 97.44%Cor e Forma:SolidPeso molecular:154.25HAEGTFTSDVS acetate
<p>HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.</p>Fórmula:C50H75N13O22Pureza:97.47%Cor e Forma:SolidPeso molecular:1210.2Acrinor
CAS:<p>Acrinor is a adrenergic beta receptor agonist.</p>Fórmula:C35H46Cl2N10O8Pureza:98%Cor e Forma:SolidPeso molecular:805.72L-779976
CAS:<p>L-779,976 is an agonist of somatostatin receptor.</p>Fórmula:C33H43N7O3Cor e Forma:SolidPeso molecular:585.74TLX agonist 2
<p>TLX agonist 2 (compound 31) is a TLX agonist with an EC50 of 0.1 μM and a Kd of 0.16 μM. This compound enhances transcriptional activity by binding to TLX, thereby boosting the expression of TLX target genes. TLX agonist 2 is utilized in research on neurodegenerative diseases.</p>Cor e Forma:Odour SolidDOAM
CAS:<p>DOAM is an antagonist of the 5-HT2 receptor.</p>Fórmula:C16H27NO2Cor e Forma:SolidPeso molecular:265.39Preclamol hydrochloride
CAS:<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Fórmula:C14H22ClNOCor e Forma:SolidPeso molecular:255.78Khusimol
CAS:Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Fórmula:C15H24OPureza:98%Cor e Forma:SolidPeso molecular:220.35TGR5 agonist 6
CAS:<p>Compound 22b, also known as TGR5 agonist 6, is a non-systemic, intestine-targeted TGR5 agonist that demonstrates significant and sustained blood glucose-lowering effects with an acceptable safety profile.</p>Fórmula:C42H48Cl2N6O6Cor e Forma:SolidPeso molecular:803.77TRPV1/CB2 agonist 1
<p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>Cor e Forma:Odour SolidMisoprostol acid
CAS:<p>Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.</p>Fórmula:C21H36O5Pureza:98%Cor e Forma:SolidPeso molecular:368.51Metaraminol
CAS:<p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Fórmula:C9H13NO2Cor e Forma:SolidPeso molecular:167.21RGS2-Galpha-q interaction-IN-1
RGS2–Galpha-q interaction-IN-1 (Compound AJ-3) is an inhibitor of the RGS2-Galpha-q interaction. It inhibits the growth of cancer cell lines that express RGS2 and has anti-cell migration properties.Fórmula:C30H30ClN7O3Cor e Forma:SolidPeso molecular:572.06Tamuzimod
CAS:<p>Tamuzimod, an effective immunomodulator, exhibits modulatory activity on S1P Receptors with EC50 values below 1 μM [1] [2].</p>Fórmula:C21H13Cl3F3N5O3Cor e Forma:SolidPeso molecular:546.71Vapiprost hydrochloride
CAS:<p>Vapiprost hydrochloride is a biochemicla.</p>Fórmula:C30H40ClNO4Cor e Forma:SolidPeso molecular:514.1(+)-Oxypeucedanin methanolate
CAS:<p>(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].</p>Fórmula:C17H18O6Cor e Forma:SolidPeso molecular:318.32CAY10597
CAS:<p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>Fórmula:C20H14ClFN2O5Cor e Forma:SolidPeso molecular:416.79Serazapine
CAS:<p>Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.</p>Fórmula:C22H23N3O2Pureza:98.71% - 99.57%Cor e Forma:SolidPeso molecular:361.44O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Fórmula:C14H16Cl2O2Cor e Forma:SolidPeso molecular:287.18Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Cor e Forma:SolidPeso molecular:926.09Alcaftadine carboxylic acid
CAS:<p>Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.</p>Fórmula:C19H21N3O2Cor e Forma:SolidPeso molecular:323.39Vapiprost
CAS:<p>Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.</p>Fórmula:C30H39NO4Pureza:98%Cor e Forma:SolidPeso molecular:477.64LY-53857 free base
CAS:<p>LY-53857 free base is a bioactive chemical.</p>Fórmula:C23H32N2O3Cor e Forma:SolidPeso molecular:384.51IRAK inhibitor 4 trans
<p>IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.</p>Fórmula:C33H35F3N6O3Pureza:98%Cor e Forma:SolidPeso molecular:620.66Alprostadil ethyl ester
CAS:<p>Alprostadil ethyl ester is a biochemical used in the treatment of scleroderma.</p>Fórmula:C22H38O5Cor e Forma:SolidPeso molecular:382.53(S)-Azelastine hydrochloride
CAS:<p>(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Fórmula:C22H25Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:418.36Apelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Fórmula:C185H304N68O43SPureza:98%Cor e Forma:SolidPeso molecular:4200.93JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23Succinate/succinate receptor antagonist 1
CAS:<p>Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.</p>Fórmula:C17H15N3OPureza:99.53%Cor e Forma:SoildPeso molecular:277.32Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Fórmula:C26H47N7O9SPureza:98%Cor e Forma:SolidPeso molecular:633.76Ici 216140
CAS:<p>ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.</p>Fórmula:C45H65N13O8Cor e Forma:SolidPeso molecular:916.08(+)-Cloprostenol
CAS:<p>(+)-Cloprostenol is a analogue of prostaglandin F2α (PGF2α), and is selective prostaglandin receptor agonistic.</p>Fórmula:C22H29ClO6Pureza:98%Cor e Forma:SolidPeso molecular:424.92Pancreatic polypeptide TFA
<p>Pancreatic polypeptide TFA acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.</p>Cor e Forma:Odour SolidMK-7246 S enantiomer
MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.Fórmula:C21H21FN2O4SPureza:98%Cor e Forma:SolidPeso molecular:416.47Thiothixene
CAS:<p>Thiothixene has a wide range of applications in life science related research.</p>Fórmula:C23H29N3O2S2Cor e Forma:SolidPeso molecular:443.62Dulaglutide
CAS:<p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>Cor e Forma:SolidP2Y6R antagonist 1
<p>P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.</p>Cor e Forma:Odour SolidHAEGTFTSDVS
CAS:HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Fórmula:C48H71N13O20Pureza:98%Cor e Forma:SolidPeso molecular:1150.18HDAC6-IN-49
<p>HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.</p>Cor e Forma:Odour Solid4-fluoro MBZP
CAS:<p>4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.</p>Fórmula:C12H17FN2Cor e Forma:SolidPeso molecular:208.28Proglumide hemicalcium
CAS:Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.Fórmula:C18H28CaN2O4Pureza:98%Cor e Forma:SolidPeso molecular:376.51RS 18286
CAS:<p>RS 18286 is a LHRH antagonist.</p>Fórmula:C74H101Cl2N17O14Cor e Forma:SolidPeso molecular:1523.6Urocortin, rat
CAS:<p>Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.</p>Fórmula:C206H338N62O64Pureza:98%Cor e Forma:SolidPeso molecular:4707.26CB1R agonist 1
<p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>Fórmula:C20H18F3N3O3SCor e Forma:SolidPeso molecular:437.435Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFórmula:C80H112N18O19S2Pureza:97.86%Cor e Forma:SolidPeso molecular:1693.98CAY10606
CAS:<p>CAY10606 has a wide range of applications in life science related research.</p>Fórmula:C22H18ClNO3Cor e Forma:SolidPeso molecular:379.84NPS ALX Compound 4a hydrochloride(1:1)
<p>NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.</p>Fórmula:C25H26ClN3O2SPureza:99.84%Cor e Forma:SoildPeso molecular:468.011a,1b-dihomo Prostaglandin E1
CAS:<p>1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.</p>Fórmula:C22H38O5Cor e Forma:SolidPeso molecular:382.541PEN (human)
CAS:<p>PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.</p>Fórmula:C97H159N27O32Pureza:98%Cor e Forma:SolidPeso molecular:2215.49Nebokitug
<p>Nebokitug is a humanized IgG1κ antibody targeting CCL24, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.</p>Cor e Forma:Odour LiquidMRS 4062 triethylammonium salt
CAS:<p>MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).</p>Fórmula:C42H86N7O15P3Cor e Forma:SolidPeso molecular:1022.105DOTA-LM3 TFA
<p>DOTA-LM3 TFA is a somatostatin receptor (SSTR) antagonist with the molecular structure p-Cl-Phe-cyclo(D-Cys-Tyr-D-4-amino-Phe(carbamoyl)-Lys-Thr-Cys)D-Tyr-NH2.</p>Fórmula:C71H94ClF3N16O21S2Cor e Forma:SolidPeso molecular:1664.18GRL018-21
<p>GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].</p>Cor e Forma:Odour Solidβ2AR/M-receptor agonist-1
CAS:<p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>Fórmula:C43H56BrN3O7Cor e Forma:SolidPeso molecular:806.82INCB 3284 dimesylate
CAS:INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Fórmula:C28H39F3N4O10S2Pureza:98%Cor e Forma:SolidPeso molecular:712.765-Bromoimidazo[1,2-A]Pyrazine
CAS:<p>5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.</p>Fórmula:C6H4BrN3Pureza:97.04%Cor e Forma:SolidPeso molecular:198.02Kisspeptin-10, human
CAS:<p>Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.</p>Fórmula:C63H83N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1302.462Cannabidiolic acid methyl ester
CAS:<p>Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.</p>Fórmula:C23H32O4Cor e Forma:SolidPeso molecular:372.5Pasireotide
CAS:Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).Fórmula:C58H66N10O9Pureza:98%Cor e Forma:SolidPeso molecular:1047.2112(S)-HpEPE
CAS:<p>12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456Poly-D-lysine hydrobromide (MW 1000-5000)
<p>Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.</p>Cor e Forma:Odour SolidCafelkibart
<p>Cafelkibart is a chimeric IgG1κ monoclonal antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.</p>Cor e Forma:Odour LiquidD5R agonist 1
<p>D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.</p>Cor e Forma:Odour SolidEfranarelaxin alfa
CAS:<p>Efranarelaxin alfa is an agonist of the relaxin receptor. It shows potential for research in cardiovascular diseases and tissue repair.</p>Cor e Forma:LiquidGuanylate cyclase-IN-1
CAS:<p>Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.</p>Fórmula:C20H17FN8OCor e Forma:SolidPeso molecular:404.409Wy 43657
CAS:<p>Wy 43657 is a gonadorelin antagonist.</p>Fórmula:C71H86N14O13Pureza:98%Cor e Forma:SolidPeso molecular:1343.554FR 113680
CAS:FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.Fórmula:C35H39N5O6Pureza:98%Cor e Forma:SolidPeso molecular:625.726CAY10580
CAS:<p>CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).</p>Fórmula:C19H35NO4Cor e Forma:SolidPeso molecular:341.49Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Fórmula:C191H330N64O53S3Pureza:98%Cor e Forma:SolidPeso molecular:4467.29Bombinakinin M acetate
<p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>Fórmula:C102H163N31O26Pureza:99.80%Cor e Forma:SolidPeso molecular:2239.589-deoxy-9-methylene Prostaglandin E2
CAS:<p>9-deoxy-9-methylene PGE2: stable PGE2 analog with similar effects, less side effects, equal potency in rats, gerbils, primates.</p>Fórmula:C21H34O4Cor e Forma:SolidPeso molecular:350.4994-Chloromethamphetamine hydrochloride
CAS:<p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>Fórmula:C10H15Cl2NCor e Forma:SolidPeso molecular:220.14Protease-Activated Receptor-1 antagonist 2
CAS:<p>Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.</p>Fórmula:C24H23F2N3O2Cor e Forma:SolidPeso molecular:423.46NTRC-824
CAS:<p>NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.</p>Fórmula:C25H26F3N3O6SPureza:98%Cor e Forma:SolidPeso molecular:553.55Pal-Glu(OSu)-OH
CAS:<p>Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.</p>Fórmula:C25H42N2O7Cor e Forma:SolidPeso molecular:482.618Pasireotide ditrifluoroacetate
<p>Pasireotide is a stable cyclohexapeptide somatostatin mimic.</p>Fórmula:C62H68F6N10O13Pureza:98%Cor e Forma:SolidPeso molecular:1275.25SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Fórmula:C54H71N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1074.258APTAA-LHRH
CAS:<p>APTAA-LHRH is a gonadorelin antagonist.</p>Fórmula:C69H91Cl2N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1453.47R 50595
CAS:<p>R 50595 is a selective non-competitive cisapride antagonist.</p>Fórmula:C30H35Cl2F2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:594.52Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Fórmula:C215H358N72O66SPureza:98%Cor e Forma:SolidPeso molecular:5039.65[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS:<p>High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.</p>Fórmula:C189H284N54O56SPureza:98%Cor e Forma:SolidPeso molecular:4241LY83583
CAS:<p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>Fórmula:C15H10N2O2Pureza:99.54% - 99.80%Cor e Forma:SolidPeso molecular:250.25
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