GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(985 produtos)
- Receptor de adenosina(244 produtos)
- Receptor adrenérgico(2.991 produtos)
- Receptor de Bombesina(32 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(153 produtos)
- CaSR(33 produtos)
- Receptor de Canabinóides(209 produtos)
- Receptor de Dopamina(433 produtos)
- Receptor Endotelina(79 produtos)
- Receptor GNRH(77 produtos)
- GPCR19(32 produtos)
- GRK(33 produtos)
- GTPase(22 produtos)
- Receptor Glucagon(181 produtos)
- Hedgehog/Smoothened(46 produtos)
- Receptor de Histamina(380 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(26 produtos)
- Receptor OX(41 produtos)
- Receptor opioide(309 produtos)
- PAFR(12 produtos)
- PKA(51 produtos)
- Receptor S1P(18 produtos)
- SGLT(31 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5696 produtos de "GPCR/Proteína-G"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ilatreotide
CAS:<p>Ilatreotide is a Amadori compound of octreotide.</p>Fórmula:C61H86N10O20S2Pureza:98%Cor e Forma:SolidPeso molecular:1343.53Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Cor e Forma:SolidPeso molecular:926.09(3R,5R,6S)-Atogepant
<p>(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.</p>Fórmula:C29H23F6N5O3Cor e Forma:SolidPeso molecular:603.52[Ala17]-MCH acetate
<p>[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled).</p>Fórmula:C99H159N29O28S4Pureza:98.92%Cor e Forma:SolidPeso molecular:2331.76PAF C-16 Carboxylic Acid
CAS:PAF C-16, a natural phospholipid, triggers neutrophil migration, ROS, IL-6 production, and is linked to necrotizing enterocolitis.Fórmula:C26H52NO9PCor e Forma:SolidPeso molecular:553.67INCB 3284 dimesylate
CAS:INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Fórmula:C28H39F3N4O10S2Pureza:98%Cor e Forma:SolidPeso molecular:712.76[Ala1,3,11,15]-Endothelin
CAS:<p>Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).</p>Fórmula:C109H163N25O32SPureza:98%Cor e Forma:SolidPeso molecular:2368Imelciment
CAS:<p>Imelciment (REGN-9035) is a humanised monoclonal antibody targeting NPR1, which can be used for research into heart failure.</p>Pureza:95%Cor e Forma:SoildCetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Fórmula:C21H27Cl3N2O3Cor e Forma:SolidPeso molecular:461.81Osanetant
CAS:Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Fórmula:C35H41Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:606.62Protease-Activated Receptor-1 antagonist 2
CAS:<p>Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.</p>Fórmula:C24H23F2N3O2Cor e Forma:SolidPeso molecular:423.46Lisuride maleate
CAS:<p>Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.</p>Fórmula:C24H30N4O5Pureza:99.85%Cor e Forma:SolidPeso molecular:454.52Urocortin II, human TFA
<p>hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.</p>Fórmula:C196H340F3N63O56SPureza:98%Cor e Forma:SolidPeso molecular:4564.3PSB 0777 ammonium salt
CAS:<p>adenosine A2A receptor full agonist</p>Fórmula:C18H24N6O7S2Pureza:98%Cor e Forma:SolidPeso molecular:500.55(2R,2R)-PF-07258669
CAS:<p>(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.</p>Fórmula:C25H27FN6O2Cor e Forma:SolidPeso molecular:462.52CB2R probe 1
CAS:<p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>Fórmula:C36H42N4O4Cor e Forma:SolidPeso molecular:594.7412(S)-HpEPE
CAS:<p>12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456L-threo Lysosphingomyelin (d18:1)
CAS:L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).Fórmula:C23H49N2O5PCor e Forma:SolidPeso molecular:464.62Poly-D-lysine hydrobromide (MW 1000-5000)
<p>Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.</p>Cor e Forma:Odour SolidSB 201146
CAS:<p>SB 201146 is a leukotriene B4 antagonist with high affinity.</p>Fórmula:C30H35LiN2O5SCor e Forma:SolidPeso molecular:542.61JKC363 TFA
<p>JKC363 TFA is an MC4 receptor antagonist with 90x more affinity than MC3 (IC50: 0.5 nM vs 44.9 nM), blocks α-MSH's effect on TRH, and is anti-hyperalgesic.</p>Fórmula:C71H93F3N19O18S2Cor e Forma:SolidPeso molecular:1620.73D5R agonist 1
<p>D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.</p>Cor e Forma:Odour SolidTGR5 agonist 1
<p>Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].</p>Fórmula:C28H48NNaO6SCor e Forma:SolidPeso molecular:549.74Pal-Glu(OSu)-OH
CAS:<p>Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.</p>Fórmula:C25H42N2O7Cor e Forma:SolidPeso molecular:482.618Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Fórmula:C21H23ClFNO2Pureza:98%Cor e Forma:SolidPeso molecular:379.89Galcanezumab
CAS:Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.Pureza:> 95%Cor e Forma:LiquidPeso molecular:144.08 kDaDesmethyl Mirtazapine (hydrochloride)
CAS:<p>Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.</p>Fórmula:C16H18ClN3Cor e Forma:SolidPeso molecular:287.79Prepro-ANF (56-92), human
CAS:<p>Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.</p>Fórmula:C173H270N44O57Cor e Forma:SolidPeso molecular:3878.26S1P2 antagonist 1
CAS:S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.Fórmula:C23H21ClN4O4Cor e Forma:SolidPeso molecular:452.9FR 113680
CAS:FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.Fórmula:C35H39N5O6Pureza:98%Cor e Forma:SolidPeso molecular:625.726Tezusomant
CAS:Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Fórmula:C120H171N23O32SCor e Forma:SolidPeso molecular:2479.84Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Fórmula:C16H28N6O4Pureza:98%Cor e Forma:SolidPeso molecular:368.43GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Fórmula:C165H254N44O55SPureza:98%Cor e Forma:SolidPeso molecular:3766.19ACTH (1-17)
CAS:<p>ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.</p>Fórmula:C95H145N29O23SPureza:98%Cor e Forma:SolidPeso molecular:2093.41Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Fórmula:C85H139N29O21Pureza:98%Cor e Forma:SolidPeso molecular:1903.19Sarafotoxin S6c
CAS:<p>Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).</p>Fórmula:C103H147N27O37S5Pureza:98%Cor e Forma:SolidPeso molecular:2516Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:99.77% - 99.86%Cor e Forma:SoildPeso molecular:296.37GS-2278
CAS:<p>GS-2278 is an antagonist of LPAR1 (lysophosphatidic acid receptor 1) with potential applications in the study of idiopathic pulmonary fibrosis (IPF).</p>Fórmula:C22H16F5N9O3Cor e Forma:SolidPeso molecular:549.41Motilin, canine
CAS:<p>Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.</p>Fórmula:C120H194N36O34Pureza:98%Cor e Forma:SolidPeso molecular:2685.05d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.Fórmula:C49H71N11O13S2Pureza:98.86%Cor e Forma:SolidPeso molecular:1086.28[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Fórmula:C48H68N14O12Cor e Forma:SolidPeso molecular:1033.14PACAP (1-27), human, ovine, rat TFA
PACAP (1-27) TFA is a pacap-38 fragment and PACAP receptor antagonist with IC50s: 3nm (rat PAC1), 2nm (rat VPAC1), 5nm (human VPAC2).Fórmula:C144H225F3N40O41SPureza:98%Cor e Forma:SolidPeso molecular:3261.68Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Fórmula:C17H30ClN5O2SCor e Forma:SolidPeso molecular:403.97Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Fórmula:C61H94N18O13SCor e Forma:SolidPeso molecular:1319.58CB2 receptor antagonist 2
Compound 39, also known as CB2 receptor antagonist 2, is a potent CB2 antagonist exhibiting an IC50 of 0.33 μM.Cor e Forma:Odour Solid4-Butyl-α-agarofuran
CAS:4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.Fórmula:C18H30OCor e Forma:SolidPeso molecular:262.43MrgprX2 antagonist-2
CAS:<p>MrgprX2 antagonist-2, from patent WO2021092262A1 E163, is potent for skin inflammation studies.</p>Fórmula:C17H16F5N3O3Cor e Forma:SolidPeso molecular:405.325Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2
CAS:<p>Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2 is a biologically active peptide functioning as a selective agonist for Protease Activated Receptor 1 (PAR-1), a subtype</p>Fórmula:C42H63FN12O8Cor e Forma:SolidPeso molecular:883.02Neuropeptide Y (human)
CAS:<p>Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.</p>Fórmula:C189H285N55O57SPureza:98%Cor e Forma:SolidPeso molecular:4271.68Bamosiran
CAS:Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.Cor e Forma:SolidCetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Fórmula:C30H28Cl2N2Cor e Forma:SolidPeso molecular:487.46Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe andFórmula:C58H77N14O21S2Pureza:98.47% - 98.54%Cor e Forma:SoildPeso molecular:1370.44ELA-21 (human)
CAS:<p>Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.</p>Fórmula:C112H184N40O25S3Pureza:98%Cor e Forma:SolidPeso molecular:2587.12α-MSH TFA
CAS:<p>α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in the</p>Fórmula:C79H110F3N21O21SCor e Forma:SolidPeso molecular:1778.93PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44B-Raf IN 14
CAS:B-Raf IN 14 is a BRAF inhibitor.Fórmula:C15H14BrN5O3SPureza:98.38%Cor e Forma:SolidPeso molecular:424.27JKC363
CAS:<p>MC4 receptor antagonist; IC50: 0.5 nM (MC4), 44.9 nM (MC3). Blocks α-MSH, reduces TRH, food intake, and pain.</p>Fórmula:C69H91N19O16S2Pureza:98%Cor e Forma:SolidPeso molecular:1506.72GLP-1 moiety from Dulaglutide
<p>GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.</p>Fórmula:C149H221N37O49Pureza:98%Cor e Forma:SolidPeso molecular:3314.62J-115814
CAS:<p>J-115814 is a potent feeding stimulant.</p>Fórmula:C29H38ClN5O3SCor e Forma:SolidPeso molecular:572.16[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS:<p>High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.</p>Fórmula:C189H284N54O56SPureza:98%Cor e Forma:SolidPeso molecular:4241MRS 2365
CAS:Highly potent, selective P2Y1 receptor agonistFórmula:C13H19N5O9P2SPureza:98%Cor e Forma:SolidPeso molecular:483.33LY83583
CAS:<p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>Fórmula:C15H10N2O2Pureza:99.54% - 99.80%Cor e Forma:SolidPeso molecular:250.25Sarafotoxin S6a
CAS:Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo.Fórmula:C105H156N28O34S5Pureza:98%Cor e Forma:SolidPeso molecular:2514.85Anti-TSHR Antibody (M22)
Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.Cor e Forma:Odour LiquidHemopressin (human, mouse)
CAS:<p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>Fórmula:C50H79N13O12Pureza:98%Cor e Forma:SolidPeso molecular:1054.26α1A-AR Degrader 9c
CAS:α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Fórmula:C38H43N11O11Pureza:98%Cor e Forma:SolidPeso molecular:829.82Fabesetron
CAS:<p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>Fórmula:C18H19N3OCor e Forma:SolidPeso molecular:293.37Dipivefrin
CAS:<p>Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.</p>Fórmula:C19H29NO5Cor e Forma:SolidPeso molecular:351.44NI-203
<p>NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.</p>Cor e Forma:Odour LiquidAmylin (IAPP), feline
<p>Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.</p>Fórmula:C165H270N52O54S2Pureza:98%Cor e Forma:SolidPeso molecular:3910.45Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Fórmula:C24H21N5O5SCor e Forma:SolidPeso molecular:491.525-MeO-pyr-T
CAS:<p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>Fórmula:C15H20N2OCor e Forma:SolidPeso molecular:244.33Alosetron-d3
CAS:<p>Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Fórmula:C17H18N4OPureza:98%Cor e Forma:SolidPeso molecular:297.37MGV354
MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].Fórmula:C35H37N5O3Pureza:98%Cor e Forma:SolidPeso molecular:575.715(S)-HpEPE
CAS:15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456sGnRH-A
CAS:<p>sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.</p>Fórmula:C64H83N17O12Cor e Forma:SolidPeso molecular:1282.45Israpafant
CAS:Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Fórmula:C28H29ClN4SCor e Forma:SolidPeso molecular:489.07Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Fórmula:C225H349N48O68ClPureza:98%Cor e Forma:SolidPeso molecular:4849.91RXFP3/4 agonist 1
CAS:<p>RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).</p>Fórmula:C20H22ClN5OPureza:98%Cor e Forma:SolidPeso molecular:383.885-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Fórmula:C13H18N2OPureza:98.25%Cor e Forma:SolidPeso molecular:218.29LAS190792
CAS:LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.Fórmula:C39H43ClN4O9S2Cor e Forma:SolidPeso molecular:811.36Flunarizine
CAS:<p>Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.</p>Fórmula:C26H26F2N2Pureza:99.9%Cor e Forma:SolidPeso molecular:404.505-trans Latanoprost (free acid)
CAS:<p>Latanoprost, a prodrug eye drop, turns into active acid inside the body and treats high eye pressure. Its trans isomer also likely reduces eye pressure.</p>Fórmula:C23H34O5Cor e Forma:SolidPeso molecular:390.52CKLF1-C27 TFA
<p>CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.</p>Fórmula:C153H244F3N39O39Cor e Forma:SolidPeso molecular:3310.8Adrenomedullin (AM) (22-52), human TFA
<p>Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.</p>Fórmula:C161H253N46F3O50Pureza:98%Cor e Forma:SolidPeso molecular:3690.06ABT 724 trihydrochloride
CAS:<p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>Fórmula:C17H22Cl3N5Pureza:99.91%Cor e Forma:SolidPeso molecular:402.75Hemokinin 1 (mouse)
CAS:<p>Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.</p>Fórmula:C61H100N22O15SPureza:98%Cor e Forma:White PowderPeso molecular:1413.65(p-Iodo-Phe7)-ACTH (4-10)
CAS:<p>(p-Iodo-Phe7)-ACTH (4-10), an ACTH derivative and MC receptor antagonist, inhibits α-MSH-induced grooming in rats.</p>Fórmula:C44H58IN13O10SCor e Forma:SolidPeso molecular:1087.98Navafenterol
CAS:AZD-8871, a potential COPD and asthma treatment, may work well with ICS.Fórmula:C38H42N6O6S2Cor e Forma:SolidPeso molecular:742.91CB2R/FAAH modulator-3
CAS:<p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>Fórmula:C22H31NO2Pureza:99.81%Cor e Forma:SoildPeso molecular:341.49VVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Cor e Forma:SolidPicumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist.Fórmula:C22H31Cl2N3O4Pureza:99.8%Cor e Forma:SoildPeso molecular:472.4Naratriptan D3 Hydrochloride
CAS:Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.Fórmula:C17H26ClN3O2SPureza:98%Cor e Forma:SolidPeso molecular:374.94AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211(Rac)-Norcisapride
CAS:Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.Fórmula:C14H20ClN3O3Pureza:99.32%Cor e Forma:SoildPeso molecular:313.78ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
CAS:<p>ACTH (3-24) is the fragment 3-24 of ACTH, used in disease research including cancer and immune disorders.</p>Fórmula:C124H196N38O27SCor e Forma:SolidPeso molecular:2683.19Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Fórmula:C18H20ClNO4Cor e Forma:SolidPeso molecular:349.81Atrial natriuretic factor (1-28) (rat) TFA
ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.Fórmula:C130H206N45F3O41S2Pureza:98%Cor e Forma:SolidPeso molecular:3176.43PF-07062119
PF-07062119 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody designed to target and inhibit GUCY2C.Cor e Forma:Odour LiquidRp-UTP-α-S tetrasodium
Rp-UTP-α-S (tetrasodium) is a nucleotide agonist of the purinergic P2Y2 and P2Y4 receptors. It can induce the accumulation of inositol phosphate in 1321N1 cells expressing P2Y2 or P2Y4, with EC50 values of 5.4 and 27 μM, respectively.Cor e Forma:Odour Solid
![[Ala17]-MCH acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1997L.webp&w=3840&q=75)
![[Ala1,3,11,15]-Endothelin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2099.webp&w=3840&q=75)
![d[Leu4,Lys8]-VP acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1927L1.webp&w=3840&q=75)
![[Asu1,6-Arg8]Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76510.webp&w=3840&q=75)
![[Leu31,Pro34]-Neuropeptide Y(human,rat)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1985.webp&w=3840&q=75)
