GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Fórmula:C20H22BrFN2OPureza:99.81%Cor e Forma:White Crystalline PowderPeso molecular:405.304PF-5190457
CAS:<p>PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).</p>Fórmula:C29H32N6OSPureza:99.34%Cor e Forma:SolidPeso molecular:512.67Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Cor e Forma:SolidPeso molecular:395.43Indusatumab
CAS:<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Pureza:> 95% - > 95%Cor e Forma:LiquidPeso molecular:145.18 kDaAnamorelin
CAS:<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Fórmula:C31H42N6O3Pureza:99.35% - 99.94%Cor e Forma:SolidPeso molecular:546.7Tripelennamine hydrochloride
CAS:<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Fórmula:C16H21N3·HClPureza:99.54% - 99.81%Cor e Forma:White SolidPeso molecular:291.82PF-06882961
CAS:<p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Fórmula:C31H30FN5O4Pureza:98.06% - 99.54%Cor e Forma:SolidPeso molecular:555.62-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Fórmula:C11H9BrOPureza:98.51%Cor e Forma:White To Off-White PowderPeso molecular:237.09Cisapride
CAS:<p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>Fórmula:C23H29ClFN3O4Pureza:99.77%Cor e Forma:White To Slightly Biege Powder SolidPeso molecular:465.95Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Fórmula:C19H21N·HClPureza:98.54% - 99.98%Cor e Forma:SolidPeso molecular:299.84Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Pureza:97.76%Cor e Forma:SoildNylidrin hydrochloride
CAS:<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Fórmula:C19H26ClNO2Pureza:99.35%Cor e Forma:SolidPeso molecular:335.87Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Cor e Forma:SolidPeso molecular:1347.5Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Pureza:SDS-PAGE:95% SEC-HPLC:98.90%Cor e Forma:LiquidPeso molecular:146.43 kDaLafutidine
CAS:<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Fórmula:C22H29N3O4SPureza:98.55%Cor e Forma:Yellowish White Crystalline PowderPeso molecular:431.55Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Fórmula:C18H26ClN3O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:367.87Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Cor e Forma:White Crystalline PowderPeso molecular:313.86Erenumab
CAS:<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Pureza:99.43% (SEC-HPLC) - > 95%Cor e Forma:LiquidPeso molecular:146.2 kDaTalastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Fórmula:C19H21N3OPureza:98.50% - 99.44%Cor e Forma:SolidPeso molecular:307.39Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Fórmula:C10H13NO4Pureza:98.95% - 99.86%Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecular:211.21Desipramine hydrochloride
CAS:<p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>Fórmula:C18H23ClN2Pureza:99.58% - 99.94%Cor e Forma:White To Off-White PowderPeso molecular:302.842Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Fórmula:C21H22ClNPureza:98.75% - 99.84%Cor e Forma:SolidPeso molecular:323.86Fluoxetine hydrochloride
CAS:<p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Cor e Forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Cor e Forma:SolidPeso molecular:266.55Sergliflozin A
CAS:<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Fórmula:C20H24O7Pureza:99.43%Cor e Forma:SolidPeso molecular:376.4Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:463.79Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Fórmula:C28H32N2O7Pureza:99.03% - 99.67%Cor e Forma:SolidPeso molecular:508.56ML-180
CAS:<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Fórmula:C20H25ClN4O2Pureza:99.74%Cor e Forma:SolidPeso molecular:388.89CD80-IN-3
CAS:<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Fórmula:C17H10FN3O3Pureza:98.08%Cor e Forma:SolidPeso molecular:323.28CYM 50769
CAS:<p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>Fórmula:C24H17ClN2O3Pureza:98% - 99.08%Cor e Forma:SolidPeso molecular:416.86Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Fórmula:C19H25F3N2O6Pureza:99.92% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:434.41Silodosin
CAS:<p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>Fórmula:C25H32F3N3O4Pureza:99.282% - 99.76%Cor e Forma:Colorless To Pink SolidPeso molecular:495.53Metaproterenol hemisulfate
CAS:<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Fórmula:C11H17NO3·5H2O4SPureza:98.53% - 99.74%Cor e Forma:SolidPeso molecular:260.3Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Fórmula:C21H24ClNOPureza:99.77% - >99.99%Cor e Forma:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Urapidil hydrochloride
CAS:<p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3·HClPureza:99.58%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:423.94Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:383.51JNJ-18038683
CAS:<p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>Fórmula:C26H28ClN3O7Pureza:97.29%Cor e Forma:SolidPeso molecular:529.97PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Fórmula:C25H37Cl2N3O2Pureza:99.68%Cor e Forma:SolidPeso molecular:482.49Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Fórmula:C31H37N3O10SPureza:99.39% - 99.48%Cor e Forma:SolidPeso molecular:643.71Naftopidil
CAS:<p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>Fórmula:C24H28N2O3Pureza:99.60% - 99.97%Cor e Forma:White Crystalline PowderPeso molecular:392.49Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Fórmula:C21H27NO2Pureza:99.58%Cor e Forma:White Crystalline PowderPeso molecular:325.44Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Fórmula:C18H25ClN4OPureza:99.88% - 99.93%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:348.87Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H11ClFNO2Pureza:99.98%Cor e Forma:SoildPeso molecular:231.65Blonanserin
CAS:<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Fórmula:C23H30FN3Pureza:99.85%Cor e Forma:SolidPeso molecular:367.5Fosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Fórmula:C9H15ClNO5PPureza:99.84%Cor e Forma:SolidPeso molecular:283.65NF-56-EJ40 hydrochloride
CAS:<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Fórmula:C27H31Cl2N3O3Pureza:99.33%Cor e Forma:SoildPeso molecular:516.46Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White Crystalline PowderPeso molecular:341.43Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Fórmula:C17H18F3NOPureza:99.07% - 99.28%Cor e Forma:SolidPeso molecular:309.33Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Fórmula:C163H273N49O44Pureza:96.87%Cor e Forma:SolidPeso molecular:3623.21Diphenylpyraline hydrochloride
CAS:<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Fórmula:C19H23NO·HClPureza:98.72%Cor e Forma:SolidPeso molecular:317.85Chlorprothixene hydrochloride
CAS:<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Fórmula:C18H18ClNS·HClPureza:99.76%Cor e Forma:White PowderPeso molecular:352.32Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Fórmula:C17H20N4SPureza:99.86% - ≥95%Cor e Forma:Yellowish Crystalline PowderPeso molecular:312.43CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Fórmula:C15H18Cl2N4OPureza:99.5%Cor e Forma:SolidPeso molecular:341.24Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Cor e Forma:SolidPeso molecular:408.33MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Fórmula:C24H26F3N3O4Pureza:99.98%Cor e Forma:SolidPeso molecular:477.48Antazoline hydrochloride
CAS:<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Fórmula:C17H19N3·HClPureza:98% - 99.53%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:301.82Brefonalol HCl
<p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>Fórmula:C22H29ClN2O2Pureza:99.45%Cor e Forma:SolidPeso molecular:388.93Aripiprazole
CAS:<p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Cor e Forma:Colourless Flake Crystalline SolidPeso molecular:448.39YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Fórmula:C33H37N5O5SPureza:99.67%Cor e Forma:SolidPeso molecular:615.74Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Fórmula:C26H35NO7Pureza:98.53% - 99.43%Cor e Forma:CoaPeso molecular:473.57KGA-2727
CAS:<p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>Fórmula:C26H40N4O8Pureza:98.46%Cor e Forma:SolidPeso molecular:536.62(3aR,9aR)-Fluparoxan
CAS:<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Fórmula:C10H10FNO2Pureza:97.82%Cor e Forma:SoildPeso molecular:195.19Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Fórmula:C14H15Cl2NSPureza:99.85% - >99.99%Cor e Forma:White PowderPeso molecular:300.25Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Cor e Forma:White Or Kind Of White PowderPeso molecular:287.36Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:99.32% - >99.99%Cor e Forma:White Crystalline SolidPeso molecular:883.09AH 6809
CAS:<p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>Fórmula:C17H14O5Pureza:97.59%Cor e Forma:SolidPeso molecular:298.29Phenothiazine
CAS:<p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>Fórmula:C12H9NSPureza:99.95%Cor e Forma:Yellow Solid PelletsPeso molecular:199.27Noradrenaline bitartrate
CAS:<p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>Fórmula:C12H19NO10Pureza:99.53% - >99.99%Cor e Forma:SolidPeso molecular:337.28ESI-05
CAS:<p>ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.</p>Fórmula:C16H18O2SPureza:97.22%Cor e Forma:SolidPeso molecular:274.38Talipexole dihydrochloride
CAS:<p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>Fórmula:C10H17Cl2N3SPureza:99.89%Cor e Forma:Light Yellow SolidPeso molecular:282.23Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Fórmula:C21H21ClN4OSPureza:99.55%Cor e Forma:Tan SolidPeso molecular:412.94Levocetirizine
CAS:<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98% - 99.9%Cor e Forma:White PowderPeso molecular:388.89LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Fórmula:C30H58ClN7O8SPureza:98.02% - 99.31%Cor e Forma:SolidPeso molecular:712.34(R)-Elagolix
CAS:<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Fórmula:C32H30F5N3O5Pureza:99.08%Cor e Forma:SolidPeso molecular:631.59Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Fórmula:C31H38N2OPureza:97.49%Cor e Forma:SolidPeso molecular:454.65Azasetron hydrochloride
CAS:<p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>Fórmula:C17H20ClN3O3·HClPureza:99.50%Cor e Forma:SolidPeso molecular:386.27Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Fórmula:C18H25N3O6Pureza:99.66%Cor e Forma:SolidPeso molecular:379.41Filorexant
CAS:<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Fórmula:C24H25FN4O2Pureza:98.88%Cor e Forma:SolidPeso molecular:420.48Levodropropizine
CAS:<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Fórmula:C13H20N2O2Pureza:99.87% - 99.93%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.31Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Fórmula:C19H24N2O·HClPureza:99.84% - 99.92%Cor e Forma:White SolidPeso molecular:332.87Ro 10-5824 dihydrochloride
CAS:<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Fórmula:C17H22Cl2N4Pureza:99.79%Cor e Forma:SolidPeso molecular:353.29Moxisylyte hydrochloride
CAS:<p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>Fórmula:C16H26ClNO3Pureza:99.93% - ≥95%Cor e Forma:SolidPeso molecular:315.84Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Fórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Cor e Forma:SolidPeso molecular:449.4Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Fórmula:C26H27N5O2Pureza:99.61%Cor e Forma:Light Yellow SolidPeso molecular:441.52Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Fórmula:C22H34Cl2N2O2Pureza:98.55%Cor e Forma:SolidPeso molecular:429.42Dimenhydrinate
CAS:<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Adrenalone hydrochloride
CAS:<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Fórmula:C9H11NO3·HClPureza:99.94%Cor e Forma:SolidPeso molecular:217.65SBI-477
CAS:<p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>Fórmula:C24H25N3O6SPureza:99.3%Cor e Forma:SolidPeso molecular:483.54Promazine hydrochloride
CAS:<p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>Fórmula:C17H21ClN2SPureza:99.90%Cor e Forma:SolidPeso molecular:320.88Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Fórmula:C18H29ClN2O4Pureza:99.92% - >99.99%Cor e Forma:White Or Slightly Off-White Crystalline Powder SolidPeso molecular:372.89Pizotifen
CAS:<p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>Fórmula:C19H21NSPureza:99.93%Cor e Forma:SolidPeso molecular:295.44Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Fórmula:C59H79N15O21S6Pureza:97.93% - 98.71%Cor e Forma:SolidPeso molecular:1526.74MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Fórmula:C27H25N3O4S2Pureza:97.44%Cor e Forma:SolidPeso molecular:519.64Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Cor e Forma:SolidPeso molecular:296.79Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Fórmula:C16H15FN6OSPureza:98.62% - 99.7%Cor e Forma:SolidPeso molecular:358.39Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Cor e Forma:SolidPeso molecular:461.81Olinciguat
CAS:<p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>Fórmula:C21H16F5N7O3Pureza:99.33% - 99.71%Cor e Forma:SolidPeso molecular:509.39Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Fórmula:C19H29ClN2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:384.9Ciliobrevin D
CAS:<p>Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.</p>Fórmula:C17H8Cl3N3O2Pureza:98.09%Cor e Forma:SolidPeso molecular:392.62
