GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Fórmula:C23H24FN3O3Pureza:99.07% - 99.9%Cor e Forma:SolidPeso molecular:409.45Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Fórmula:C19H23NO3·CH4O3SPureza:99.18% - 99.87%Cor e Forma:Tan Or Off-White Cyrstalline SolidPeso molecular:409.5CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Fórmula:C16H11N3OPureza:99.81%Cor e Forma:SolidPeso molecular:261.28SSR240612
CAS:<p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>Fórmula:C42H53ClN4O7SPureza:98.59% - 99.16%Cor e Forma:SolidPeso molecular:793.41CYM-5541
CAS:<p>CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.</p>Fórmula:C19H28N2O2Pureza:99.74% - 99.76%Cor e Forma:SolidPeso molecular:316.44Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97Tandospirone hydrochloride
CAS:<p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>Fórmula:C21H30ClN5O2Cor e Forma:SolidPeso molecular:419.95LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Cor e Forma:SolidPeso molecular:226.53BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Fórmula:C59H80N14O13Pureza:95.3%Cor e Forma:SolidPeso molecular:1193.35Guanabenz Acetate
CAS:<p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>Fórmula:C8H8Cl2N4·C2H4O2Pureza:99% - 99.66%Cor e Forma:White Solid From Acetonitrile White SolidPeso molecular:291.13SB-222200
CAS:<p>SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).</p>Fórmula:C26H24N2OPureza:97.13%Cor e Forma:SolidPeso molecular:380.48BQU57
CAS:<p>BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.</p>Fórmula:C16H13F3N4OPureza:97.45% - 98.72%Cor e Forma:SolidPeso molecular:334.3Talinolol
CAS:<p>(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.</p>Fórmula:C20H33N3O3Pureza:98.8%Cor e Forma:SolidPeso molecular:363.49Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Fórmula:C20H22ClF3N4OCor e Forma:SolidPeso molecular:426.87Eprazinone dihydrochloride
CAS:<p>Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.</p>Fórmula:C24H32N2O2·2HClPureza:99.25%Cor e Forma:A White Or Almost White CrysPeso molecular:453.44Ibutamoren
CAS:<p>Ibutamoren (MK-677) is a drug which acts as a potent, orally active growth hormone secretagogue, mimicking the GH stimulating action of the endogenous hormone ghrelin. It also alters the metabolism of body fat and so may have an application in the treatment of obesity.</p>Fórmula:C27H36N4O5SPureza:97.59%Cor e Forma:SolidPeso molecular:528.66HS024
CAS:<p>HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.</p>Fórmula:C58H79N19O10S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1266.5Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Fórmula:C15H24N2O4SCor e Forma:SolidPeso molecular:328.43[D-Phe12]-Bombesin acetate
<p>[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Fórmula:C76H116N22O20SPureza:99.81%Cor e Forma:SolidPeso molecular:1689.94Ganirelix Acetate
CAS:<p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>Fórmula:C82H117ClN18O15Pureza:96.05%Cor e Forma:SolidPeso molecular:1630.4Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Fórmula:C23H29Cl2N3O3Cor e Forma:SolidPeso molecular:466.4PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:301.21Decynium 22
CAS:<p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>Fórmula:C23H23IN2Pureza:99.92%Cor e Forma:Dark Red CrystalsPeso molecular:454.35Poloxamer 407
CAS:<p>Poloxamer 407 is a nonionic surfactant.</p>Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:7700(Average)PD 117519
CAS:<p>PD 117519 (CI947) is an agonist of adenosine receptor</p>Fórmula:C19H21N5O4Pureza:99.98%Cor e Forma:SolidPeso molecular:383.4Takeda103A
CAS:<p>Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.</p>Fórmula:C24H23F2N7OPureza:97.17%Cor e Forma:SolidPeso molecular:463.48PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Fórmula:C26H32O4Pureza:98.53%Cor e Forma:SolidPeso molecular:408.53Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Fórmula:C20H22N2O6Pureza:99.39%Cor e Forma:SolidPeso molecular:386.49-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Fórmula:C7H9N5Pureza:99.35% - 99.41%Cor e Forma:SolidPeso molecular:163.18Talnetant hydrochloride
CAS:<p>Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.</p>Fórmula:C25H23ClN2O2Cor e Forma:SolidPeso molecular:418.92Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Cor e Forma:White Crystalline PowderPeso molecular:546.053-CPMT
CAS:<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Fórmula:C21H25Cl2NOPureza:99.03%Cor e Forma:SolidPeso molecular:378.33Fosaprepitant dimeglumine
CAS:<p>Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.</p>Fórmula:C37H56F7N6O16PPureza:98% - 99.03%Cor e Forma:SolidPeso molecular:1004.83Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Fórmula:C20H20FNO3S·HClPureza:99.39% - 99.79%Cor e Forma:SolidPeso molecular:409.9Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Fórmula:C17H25N7O4Pureza:99.74%Cor e Forma:SolidPeso molecular:391.425-HT1A modulator 2 hydrochloride
CAS:<p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>Fórmula:C11H16ClNOPureza:98.5%Cor e Forma:SolidPeso molecular:213.7Metadoxine
CAS:<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Cor e Forma:Off-White PowderPeso molecular:298.29Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Fórmula:C18H15BrF2N4O2Pureza:98.42% - 99.88%Cor e Forma:SolidPeso molecular:437.24SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Cor e Forma:SolidPeso molecular:324.245-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Fórmula:C18H20N2OPureza:99.13%Cor e Forma:SolidPeso molecular:280.36Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Fórmula:C32H34N4O5SPureza:98.26% - 99.43%Cor e Forma:SolidPeso molecular:586.7C14TKL-1 acetate
<p>C14TKL-1 acetate is a NK1 receptor agonist.</p>Fórmula:C65H102N20O15S2Pureza:98.56%Cor e Forma:SolidPeso molecular:1467.75Cangrelor free acid
CAS:<p>Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.</p>Fórmula:C17H25Cl2F3N5O12P3S2Cor e Forma:SolidPeso molecular:776.36Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Fórmula:C21H25ClN2O3·C6H6O3SPureza:99.83% - 99.9%Cor e Forma:Brown Viscous LiquidPeso molecular:547.06RO 46-8443
CAS:<p>RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.</p>Fórmula:C31H35N3O8SPureza:98.77% - 99.77%Cor e Forma:SolidPeso molecular:609.69Asapiprant
CAS:<p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>Fórmula:C24H27N3O7SPureza:99.64%Cor e Forma:SolidPeso molecular:501.55MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C23H21N5O3SPureza:97.69% - 98.15%Cor e Forma:SolidPeso molecular:447.51Fabomotizole
CAS:<p>Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.</p>Fórmula:C15H21N3O2SPureza:99.4%Cor e Forma:SolidPeso molecular:307.41[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Fórmula:C46H62F3N11O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1018.05Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Fórmula:C172H265N43O51Pureza:97.65% - 99.04%Cor e Forma:SolidPeso molecular:3751.25D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Fórmula:C20H23N5Pureza:98.82%Cor e Forma:SolidPeso molecular:333.43LY310762
CAS:<p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>Fórmula:C24H27FN2O2·HClPureza:99.8%Cor e Forma:SolidPeso molecular:430.94[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
<p>Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.</p>Fórmula:C81H113N19O14Pureza:97.68%Cor e Forma:SolidPeso molecular:1576.91Neurokinin A
CAS:<p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>Fórmula:C50H80N14O14SPureza:>99.99%Cor e Forma:White To Off-White Lyophilized SolidPeso molecular:1133.32Ropinirole hydrochloride
CAS:<p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>Fórmula:C16H24N2O·HClPureza:99.87% - 99.98%Cor e Forma:Off-White SolidPeso molecular:296.84NPS2390
CAS:<p>NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)</p>Fórmula:C19H21N3OPureza:97.13%Cor e Forma:SolidPeso molecular:307.39Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Fórmula:C52H77N13O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1092.27M617 acetate
<p>M617 acetate is a selective agonist of galanin receptor 1 (GAL1).</p>Fórmula:C112H161N29O28Pureza:96.02%Cor e Forma:SolidPeso molecular:2361.65Fluoroclebopride
CAS:<p>Fluoroclebopride is a dopamine (DA) D2 receptor ligand.</p>Fórmula:C20H23ClFN3O2Pureza:99.68% - 99.91%Cor e Forma:SolidPeso molecular:391.87Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Cor e Forma:White To Tan Powder SolidPeso molecular:383.4GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Fórmula:C20H20N4O4Pureza:99.92%Cor e Forma:SolidPeso molecular:380.4Darusentan
CAS:<p>Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteries</p>Fórmula:C22H22N2O6Pureza:98.72%Cor e Forma:SolidPeso molecular:410.43GBR 12935
CAS:<p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>Fórmula:C28H34N2OCor e Forma:SolidPeso molecular:414.58Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:440.94Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Fórmula:C16H24N4O2Pureza:99.23% - 99.93%Cor e Forma:White SolidPeso molecular:304.39Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Fórmula:C16H19ClN2Cor e Forma:SolidPeso molecular:274.79Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Fórmula:C22H15F3N2O7SPureza:99.33%Cor e Forma:SolidPeso molecular:508.42A-836339
CAS:<p>A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.</p>Fórmula:C16H26N2O2SPureza:99.94%Cor e Forma:SolidPeso molecular:310.45Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Fórmula:C19H20ClN3Pureza:98% - 99.65%Cor e Forma:SolidPeso molecular:325.84AM281
CAS:<p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>Fórmula:C21H19Cl2IN4O2Pureza:98.6% - >99.99%Cor e Forma:White To Off-White SolidPeso molecular:557.21Zuclopenthixol dihydrochloride
CAS:<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Fórmula:C22H27Cl3N2OSPureza:98%Cor e Forma:SolidPeso molecular:473.89GLPG2938
CAS:<p>GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and</p>Fórmula:C20H19F6N7O2Pureza:98.25%Cor e Forma:SolidPeso molecular:503.4RBC8
CAS:<p>RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.</p>Fórmula:C25H20N4O3Pureza:98.44% - 99.81%Cor e Forma:SolidPeso molecular:424.45HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C35H51N9O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:821.84Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Fórmula:C28H37N3O3Pureza:99.86% - >99.99%Cor e Forma:SolidPeso molecular:463.61E7046
CAS:<p>E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.</p>Fórmula:C22H18F5N3O4Pureza:99.86%Cor e Forma:SolidPeso molecular:483.4ML 154
CAS:<p>ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.</p>Fórmula:C29H26BrN2PSPureza:99.53%Cor e Forma:SolidPeso molecular:545.47Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Fórmula:C35H47FN10O8Pureza:97.97%Cor e Forma:SolidPeso molecular:754.85Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Cor e Forma:Appearance White Crystalline PowderPeso molecular:264.19VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Fórmula:C16H14O2Pureza:98.15%Cor e Forma:SolidPeso molecular:238.2812PF-06882961 Tris
CAS:<p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Fórmula:C35H41FN6O7Pureza:98.74% - 99.79%Cor e Forma:SolidPeso molecular:676.7Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Fórmula:C26H24F4N6OPureza:98.75% - >99.99%Cor e Forma:SolidPeso molecular:512.5LY2828360
CAS:<p>LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.</p>Fórmula:C22H27ClN6OPureza:98.45% - 99.51%Cor e Forma:SolidPeso molecular:426.94EST64454 hydrochloride
CAS:<p>EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.</p>Fórmula:C18H23ClF2N4O2Pureza:99.15%Cor e Forma:SolidPeso molecular:400.85Urantide acetate(669089-53-6 free base)
<p>Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in Ca²⁺ assay.</p>Fórmula:C53H70N10O14S2Pureza:99.22%Cor e Forma:SolidPeso molecular:1135.31CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Fórmula:C20H21N7O3Pureza:98.78%Cor e Forma:SolidPeso molecular:407.43Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Fórmula:C27H36N6O4Pureza:99.62%Cor e Forma:SolidPeso molecular:508.61Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Fórmula:C17H20BrNOCor e Forma:SolidPeso molecular:334.25Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Fórmula:C17H20N2O2S·HClPureza:99.58%Cor e Forma:SolidPeso molecular:352.88Carazolol
CAS:<p>Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.</p>Fórmula:C18H22N2O2Pureza:99% - 99.53%Cor e Forma:Yellowish SolidPeso molecular:298.38Darbufelone mesylate
CAS:<p>Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).</p>Fórmula:C19H28N2O5S2Pureza:96.81% - 99.92%Cor e Forma:SolidPeso molecular:428.57Albiglutide TFA (782500-75-8 free base)
<p>Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C150H225F3N40O47Pureza:>99.99%Cor e Forma:SolidPeso molecular:3397.63LUN42518 HCl 47142-51-8(free base)
<p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>Fórmula:C17H20ClN3OPureza:99.96%Cor e Forma:SolidPeso molecular:317.81Atrasentan
CAS:<p>Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.</p>Fórmula:C29H38N2O6Pureza:97.65% - 99.08%Cor e Forma:SolidPeso molecular:510.62CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Fórmula:C25H19N3O4Pureza:99.03%Cor e Forma:SolidPeso molecular:425.441-Oleoyl lysophosphatidic acid sodium
CAS:<p>1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2</p>Fórmula:C21H40O7P·NaPureza:98.75% - 99.24%Cor e Forma:SolidPeso molecular:458.51
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