GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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CCG215022
CAS:<p>CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.</p>Fórmula:C26H22FN7O3Pureza:97.63% - 99.69%Cor e Forma:SolidPeso molecular:499.5Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Fórmula:C19H21Cl2N3Pureza:>99.99%Cor e Forma:SolidPeso molecular:362.3Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Fórmula:C9H10Cl2N4Cor e Forma:SolidPeso molecular:245.11PGS-IN-1
CAS:<p>PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).</p>Fórmula:C19H26O3Pureza:99.39%Cor e Forma:SolidPeso molecular:302.41BAR 501 impurity
CAS:<p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>Fórmula:C26H46O3Pureza:98.78%Cor e Forma:SolidPeso molecular:406.64Cinaciguat hydrochloride
CAS:<p>Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.</p>Fórmula:C36H40ClNO5Cor e Forma:SolidPeso molecular:602.17HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Fórmula:C24H23ClN4O3Pureza:95.73%Cor e Forma:SolidPeso molecular:450.92PD-168077 maleate
CAS:<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Fórmula:C24H26N4O5Pureza:99.13%Cor e Forma:SolidPeso molecular:450.49Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Fórmula:C21H25ClN2O3Pureza:99.75%Cor e Forma:SolidPeso molecular:388.89SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Fórmula:C28H28ClN3OSPureza:97.37% - 98.88%Cor e Forma:SolidPeso molecular:490.06Ciliobrevin A
CAS:<p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.</p>Fórmula:C17H9Cl2N3O2Pureza:98.54% - 99.57%Cor e Forma:SolidPeso molecular:358.18Harmine hydrochloride
CAS:<p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>Fórmula:C13H13ClN2OPureza:99.61% - >99.99%Cor e Forma:Yellow To Slightly Green Crystalline PowderPeso molecular:248.71JNJ-5207852
CAS:<p>JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.</p>Fórmula:C20H32N2OPureza:97.19%Cor e Forma:SolidPeso molecular:316.48Empagliflozin
CAS:<p>Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.</p>Fórmula:C23H27ClO7Pureza:98% - 99.98%Cor e Forma:SolidPeso molecular:450.91Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:463SANT-1
CAS:<p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>Fórmula:C23H27N5Pureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:373.49Alizapride
CAS:<p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>Fórmula:C16H21N5O2Cor e Forma:SolidPeso molecular:315.37Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Fórmula:C46H65N13O11S2Pureza:99.65%Cor e Forma:SolidPeso molecular:1040.22Geissoschizine methyl ether
CAS:<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Fórmula:C22H26N2O3Pureza:99.24% - 99.68%Cor e Forma:SolidPeso molecular:366.45VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Fórmula:C15H19N5Pureza:99.44% - 99.57%Cor e Forma:SolidPeso molecular:269.34Treprostinil
CAS:<p>Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).</p>Fórmula:C23H34O5Pureza:99.29%Cor e Forma:SolidPeso molecular:390.51Lys-[Des-Arg9]Bradykinin,TFA
<p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2</p>Fórmula:C54H75F6N13O15Pureza:97.35%Cor e Forma:SolidPeso molecular:1260.24Asapiprant
CAS:<p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>Fórmula:C24H27N3O7SPureza:99.64%Cor e Forma:SolidPeso molecular:501.55Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Fórmula:C17H20BrNOCor e Forma:SolidPeso molecular:334.25NIBR-0213
CAS:<p>NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H29ClN2O3Pureza:98.36% - 99.34%Cor e Forma:SolidPeso molecular:464.98Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Fórmula:C25H34FN3O2Pureza:97.84% - 99.69%Cor e Forma:Pale Yellow To Pale Orange SolidPeso molecular:427.55Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38Ticagrelor metabolite M5
CAS:<p>Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.</p>Fórmula:C14H22N6O4SPureza:99.35%Cor e Forma:SolidPeso molecular:370.43Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Fórmula:C18H18ClIN6O4Pureza:98.97%Cor e Forma:SolidPeso molecular:544.73Ozanimod
CAS:<p>Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.</p>Fórmula:C23H24N4O3Pureza:98.68% - 99.58%Cor e Forma:SolidPeso molecular:404.46Eledoisin Related Peptide 2TFA
<p>Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.</p>Fórmula:C38H60F6N8O10SPureza:99%Cor e Forma:SolidPeso molecular:934.99GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Cor e Forma:SolidPeso molecular:487.5GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Fórmula:C149H226N40O45Pureza:99.85%Cor e Forma:White PowderPeso molecular:3297.63Paltusotine
CAS:<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Fórmula:C27H22F2N4OPureza:99.91%Cor e Forma:SolidPeso molecular:456.49MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Fórmula:C8H11ClN4·HClPureza:99.88%Cor e Forma:SolidPeso molecular:235.12β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Fórmula:C120H178N34O37SPureza:99.64%Cor e Forma:SolidPeso molecular:2720.97RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Fórmula:C17H16FN3Pureza:99.32%Cor e Forma:SolidPeso molecular:281.33Tripelennamine
CAS:<p>Tripelennamine: ethylenediamine derivative, H1-receptor blocker, reduces allergic reactions, treats rhinitis and conjunctivitis.</p>Fórmula:C16H21N3Cor e Forma:SolidPeso molecular:255.361-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Fórmula:C6H9N3O2Pureza:99.29%Cor e Forma:SolidPeso molecular:155.15Jatrorrhizine
CAS:<p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>Fórmula:C20H20NO4Pureza:97.18% - 99.06%Cor e Forma:SolidPeso molecular:338.38Emorfazone
CAS:<p>Emorfazone (PH011085) has an anti-nociceptive effect.</p>Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Fórmula:C14H21Cl2F3N6O3Cor e Forma:SolidPeso molecular:449.26Fenoprofen Calcium
CAS:<p>Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.</p>Fórmula:C30H26CaO6Pureza:99.24% - 99.66%Cor e Forma:SolidPeso molecular:522.6Org 27569
CAS:<p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>Fórmula:C24H28ClN3OPureza:>99.99% - ≥95%Cor e Forma:SolidPeso molecular:409.955-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Fórmula:C18H20N2OPureza:99.13%Cor e Forma:SolidPeso molecular:280.36Galanin Receptor Ligand M35 TFA
<p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>Fórmula:C109H154N27F3O28Pureza:99.45%Cor e Forma:SolidPeso molecular:2347.62CYM-5541
CAS:<p>CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.</p>Fórmula:C19H28N2O2Pureza:99.74% - 99.76%Cor e Forma:SolidPeso molecular:316.44Betazole
CAS:<p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>Fórmula:C5H9N3Cor e Forma:SolidPeso molecular:111.15Detomidine hydrochloride
CAS:<p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71[Pyr1]-Apelin-13
CAS:<p>[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.</p>Fórmula:C69H108N22O16SPureza:99.71%Cor e Forma:SolidPeso molecular:1533.8VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35Mequitazine
CAS:<p>Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.</p>Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.47ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Fórmula:C24H29N3O3Cor e Forma:SolidPeso molecular:407.51Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C215H347N61O65S·6C2H4O2Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:5218.88MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Fórmula:C27H21F3N2O3Pureza:99.54% - 99.59%Cor e Forma:SolidPeso molecular:478.46Chlorcyclizine
CAS:<p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>Fórmula:C18H21ClN2Pureza:98.75%Cor e Forma:SolidPeso molecular:300.83GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Fórmula:C18H17Cl2F3N4O2Pureza:99.47%Cor e Forma:SolidPeso molecular:449.25Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Cor e Forma:SolidPeso molecular:403.52Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Cor e Forma:SolidPeso molecular:301.81Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Fórmula:C48H68N14O14S2Pureza:98.84% - >99.99%Cor e Forma:SolidPeso molecular:1129.26SCH 58261
CAS:<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Fórmula:C18H15N7OPureza:99.07% - 99.75%Cor e Forma:SolidPeso molecular:345.36Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Fórmula:C32H51F3N8O9Pureza:99.88%Cor e Forma:SolidPeso molecular:748.79Sumatriptan hydrochloride
CAS:<p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>Fórmula:C14H22ClN3O2SCor e Forma:SolidPeso molecular:331.86BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Fórmula:C25H28Cl2N2OCor e Forma:SolidPeso molecular:443.41NPY 5RA972
CAS:<p>NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist</p>Fórmula:C21H25N3O2Pureza:99.02% - 99.56%Cor e Forma:SolidPeso molecular:351.44Cetirizine Impurity B dihydrochloride
CAS:<p>Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.</p>Fórmula:C19H23Cl3N2O2Pureza:99.24%Cor e Forma:SolidPeso molecular:417.76Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Fórmula:C26H31N3O4Pureza:98.13% - 99.66%Cor e Forma:SolidPeso molecular:449.54Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Fórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Fórmula:C16H17NO2·HClPureza:99.1% - 99.51%Cor e Forma:SolidPeso molecular:291.77S 38093 HCl
CAS:<p>S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.</p>Fórmula:C17H25ClN2O2Pureza:97.91%Cor e Forma:SolidPeso molecular:324.85D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Fórmula:C20H23N5Pureza:98.82%Cor e Forma:SolidPeso molecular:333.43Droxidopa hydrochloride
CAS:<p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>Fórmula:C9H12ClNO5Cor e Forma:SolidPeso molecular:249.65Eprazinone dihydrochloride
CAS:<p>Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.</p>Fórmula:C24H32N2O2·2HClPureza:99.25%Cor e Forma:A White Or Almost White CrysPeso molecular:453.44Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4Melanin Concentrating Hormone, salmon acetate
<p>Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.</p>Fórmula:C91H143N27O26S4Pureza:99.41%Cor e Forma:SolidPeso molecular:2157Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Fórmula:C27H36N6O4Pureza:99.62%Cor e Forma:SolidPeso molecular:508.61Ropinirole hydrochloride
CAS:<p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>Fórmula:C16H24N2O·HClPureza:99.87% - 99.98%Cor e Forma:Off-White SolidPeso molecular:296.84Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Cor e Forma:SolidPeso molecular:241.33DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Cor e Forma:SolidPeso molecular:424.44Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:452.652-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
<p>2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.</p>Fórmula:C38H64F3N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:891.98Dazoxiben
CAS:<p>Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase</p>Fórmula:C12H13ClN2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:268.7Metiamide
CAS:<p>Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .</p>Fórmula:C9H16N4S2Pureza:97.41%Cor e Forma:SolidPeso molecular:244.38Atrasentan
CAS:<p>Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.</p>Fórmula:C29H38N2O6Pureza:97.65% - 99.08%Cor e Forma:SolidPeso molecular:510.62Darbufelone mesylate
CAS:<p>Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).</p>Fórmula:C19H28N2O5S2Pureza:96.81% - 99.92%Cor e Forma:SolidPeso molecular:428.57Tolnapersine
CAS:<p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>Fórmula:C21H26N2OPureza:98%Cor e Forma:SolidPeso molecular:322.44Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Fórmula:C19H22ClN3OPureza:98%Cor e Forma:SolidPeso molecular:343.86Urotensin I acetate (83930-33-0 Free base)
<p>Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.</p>Pureza:95.44% - 96.09%Cor e Forma:SolidPeso molecular:N/AOtenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Fórmula:C25H25Cl2N7OPureza:99.43%Cor e Forma:SolidPeso molecular:510.42DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Fórmula:C16H24N4O2Pureza:99.23% - 99.93%Cor e Forma:White SolidPeso molecular:304.39PACAP 1-38 acetate
<p>PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), not VIP1.</p>Pureza:98.16%Cor e Forma:LiquidPeso molecular:N/ATCS-OX2-29
CAS:<p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.</p>Fórmula:C23H31N3O3Pureza:99.81%Cor e Forma:SolidPeso molecular:397.51Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Cor e Forma:SolidPeso molecular:224.26Elinzanetant
CAS:<p>Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.</p>Fórmula:C33H35F7N4O3Pureza:98% - 99.13%Cor e Forma:SolidPeso molecular:668.64Pardoprunox hydrochloride
CAS:<p>Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)</p>Fórmula:C12H16ClN3O2Pureza:98.95% - 99.13%Cor e Forma:SolidPeso molecular:269.73JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Fórmula:C20H34Cl2N2OPureza:99.51%Cor e Forma:SolidPeso molecular:389.4Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55Velneperit
CAS:<p>Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.</p>Fórmula:C17H24F3N3O3SPureza:99.70%Cor e Forma:SolidPeso molecular:407.45BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Cor e Forma:SolidPeso molecular:458.42Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95
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