GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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3-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Fórmula:C149H234N40O47SPureza:98% - 99.65%Cor e Forma:SolidPeso molecular:3369.76Canagliflozin
CAS:<p>Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.</p>Fórmula:C24H25FO5SPureza:98.01% - >99.99%Cor e Forma:SolidPeso molecular:444.52Veralipride
CAS:<p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>Fórmula:C17H25N3O5SPureza:99.65%Cor e Forma:SolidPeso molecular:383.46NAN-190 hydrobromide
CAS:<p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>Fórmula:C23H28BrN3O3Pureza:95.20%Cor e Forma:SolidPeso molecular:474.39Medetomidine hydrochloride
CAS:<p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>Fórmula:C13H16N2·HClPureza:99.96%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.74GLP-1 receptor agonist 9
CAS:<p>1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.</p>Fórmula:C32H31ClFN3O5Pureza:98%Cor e Forma:SolidPeso molecular:592.06Betaxolol
CAS:<p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>Fórmula:C18H29NO3Pureza:99.01%Cor e Forma:White Crystalline SolidPeso molecular:307.43OXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Fórmula:C79H125N23O22Pureza:98.52%Cor e Forma:SolidPeso molecular:1748.98MK-0557
CAS:<p>MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).</p>Fórmula:C22H19FN4O3Pureza:99.88%Cor e Forma:SolidPeso molecular:406.41Ditolylguanidine
CAS:<p>Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).</p>Fórmula:C15H17N3Pureza:98.42%Cor e Forma:White To Pinkish Solid PowderPeso molecular:239.32Midodrine
CAS:<p>Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.</p>Fórmula:C12H18N2O4Pureza:99.89%Cor e Forma:SolidPeso molecular:254.28CGS 21680 Hydrochloride
CAS:<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Fórmula:C23H29N7O6·HClPureza:96.74% - 99.53%Cor e Forma:SolidPeso molecular:535.98DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Cor e Forma:SolidPeso molecular:424.44AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Fórmula:C30H27BrN4O3Pureza:98.12%Cor e Forma:SolidPeso molecular:571.46Peptide YY (PYY) (3-36), human
CAS:<p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>Fórmula:C176H272N52O54Pureza:97.76%Cor e Forma:SolidPeso molecular:3980.42Doxazosin
CAS:<p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>Fórmula:C23H25N5O5Pureza:99.47% - 99.87%Cor e Forma:SolidPeso molecular:451.48Ropinirole hydrochloride
CAS:<p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>Fórmula:C16H24N2O·HClPureza:99.87% - 99.98%Cor e Forma:Off-White SolidPeso molecular:296.84D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Fórmula:C20H23N5Pureza:98.82%Cor e Forma:SolidPeso molecular:333.43Anisotropine Methylbromide
CAS:<p>Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.</p>Fórmula:C17H32BrNO2Pureza:99.73%Cor e Forma:Crystals From Acetone SolidPeso molecular:362.35ABT-702 dihydrochloride
CAS:<p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>Fórmula:C22H21BrCl2N6OPureza:98.42% - 98.98%Cor e Forma:SolidPeso molecular:536.25A-381393
CAS:<p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>Fórmula:C20H24N4Pureza:99.00%Cor e Forma:SolidPeso molecular:320.43Diquafosol tetrasodium
CAS:<p>Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear film</p>Fórmula:C18H22N4Na4O23P4Pureza:98.25% - 99.97%Cor e Forma:SolidPeso molecular:878.23Velneperit
CAS:<p>Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.</p>Fórmula:C17H24F3N3O3SPureza:99.70%Cor e Forma:SolidPeso molecular:407.45SCH442416
CAS:<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Fórmula:C20H19N7O2Pureza:99.58%Cor e Forma:SolidPeso molecular:389.41Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38Galanin Receptor Ligand M35 TFA
<p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>Fórmula:C109H154N27F3O28Pureza:99.45%Cor e Forma:SolidPeso molecular:2347.62TY-52156
CAS:<p>TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).</p>Fórmula:C18H19Cl2N3OPureza:99.91% - 99.91%Cor e Forma:SolidPeso molecular:364.27HT-2157
CAS:<p>HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.</p>Fórmula:C21H13F3N2OPureza:98.33%Cor e Forma:SolidPeso molecular:366.34Phenelzine
CAS:<p>Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.</p>Fórmula:C8H12N2Pureza:98%Cor e Forma:LiquidPeso molecular:136.19MK-1064
CAS:<p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>Fórmula:C24H20ClN5O3Pureza:99.19% - 99.82%Cor e Forma:SolidPeso molecular:461.9Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.36Zatebradine
CAS:<p>Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).</p>Fórmula:C26H36N2O5Pureza:98%Cor e Forma:SolidPeso molecular:456.57RS-67333
CAS:<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Fórmula:C19H29ClN2O2Pureza:99.24%Cor e Forma:SolidPeso molecular:352.9Tolnapersine
CAS:<p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>Fórmula:C21H26N2OPureza:98%Cor e Forma:SolidPeso molecular:322.44[D-Phe12,Leu14]-Bombesin acetate
<p>[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>Fórmula:C77H118N22O20Pureza:98.41% - 99.14%Cor e Forma:SolidPeso molecular:1671.9Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Cor e Forma:White SolidPeso molecular:238.24Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Fórmula:C43H77N17O12S2Pureza:99.79%Cor e Forma:SolidPeso molecular:1088.32AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89Betahistine dihydrochloride
CAS:<p>Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.</p>Fórmula:C8H14Cl2N2Pureza:99.34% - 99.88%Cor e Forma:White To Light Yellow Crystalline PowderPeso molecular:209.12Mosapride
CAS:<p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>Fórmula:C21H25ClFN3O3Pureza:99.56%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:421.89KH7
CAS:<p>KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.</p>Fórmula:C17H15BrN4O2SPureza:98.43%Cor e Forma:SolidPeso molecular:419.3Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Fórmula:C32H51F3N8O9Pureza:99.88%Cor e Forma:SolidPeso molecular:748.79Zuclopenthixol dihydrochloride
CAS:<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Fórmula:C22H27Cl3N2OSPureza:98%Cor e Forma:SolidPeso molecular:473.89GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Fórmula:C18H17Cl2F3N4O2Pureza:99.47%Cor e Forma:SolidPeso molecular:449.25SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:319.32ACTH 1-14 acetate(25696-21-3 free base)
<p>ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.</p>Fórmula:C79H113N21O22SPureza:>99.99%Cor e Forma:SolidPeso molecular:1740.96L-765314
CAS:<p>L-765314: potent α1B adrenergic receptor antagonist, used for blood pressure research.</p>Fórmula:C27H34N6O5Pureza:99.73%Cor e Forma:SolidPeso molecular:522.6Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Fórmula:C19H20N2O3Pureza:99.84% - 99.86%Cor e Forma:White PowderPeso molecular:324.37Netupitant
CAS:<p>Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C30H32F6N4OPureza:99.43%Cor e Forma:SolidPeso molecular:578.59SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Cor e Forma:SolidPeso molecular:394.85CS 2100
CAS:<p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>Fórmula:C25H23N3O4SPureza:99.19%Cor e Forma:SolidPeso molecular:461.53RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Fórmula:C17H16FN3Pureza:99.32%Cor e Forma:SolidPeso molecular:281.33Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.419-FLUORENOL
CAS:<p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>Fórmula:C13H10OPureza:99.98%Cor e Forma:Off-White Crystalline PowderPeso molecular:182.22ELA-14(human) acetate
<p>ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.</p>Fórmula:C77H123N25O19S2Pureza:97.2%Cor e Forma:SolidPeso molecular:1767.09Neuropeptide Y (29-64), amide, human acetate
<p>Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.</p>Pureza:98.42%Cor e Forma:LiquidPeso molecular:N/APancreatic Polypeptide (human) acetate
<p>Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.</p>Pureza:97.26%Cor e Forma:LiquidPeso molecular:N/ANaratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Cor e Forma:SolidPeso molecular:335.47Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Cor e Forma:SolidPeso molecular:241.33NAV-2729
CAS:<p>NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.</p>Fórmula:C25H17ClN4O3Pureza:98.83% - 98.91%Cor e Forma:SolidPeso molecular:456.88Praliciguat
CAS:<p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>Fórmula:C21H14F8N6O2Pureza:98.82%Cor e Forma:SolidPeso molecular:534.36Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Fórmula:C24H40NaO4Pureza:99.66% - 99.96%Cor e Forma:SolidPeso molecular:415.56BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Cor e Forma:SolidPeso molecular:458.42Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Fórmula:C23H30N2O10Pureza:99.98%Cor e Forma:SolidPeso molecular:494.495-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Fórmula:C18H20N2OPureza:99.13%Cor e Forma:SolidPeso molecular:280.36Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Cor e Forma:White Crystalline PowderPeso molecular:546.05S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Fórmula:C23H24FN3O3Pureza:99.07% - 99.9%Cor e Forma:SolidPeso molecular:409.45WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Cor e Forma:SolidPeso molecular:538.64Detomidine hydrochloride
CAS:<p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71MCL0020
CAS:<p>MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.</p>Fórmula:C34H39N7O4Pureza:99.18%Cor e Forma:SolidPeso molecular:609.72[Pyr1]-Apelin-13
CAS:<p>[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.</p>Fórmula:C69H108N22O16SPureza:99.71%Cor e Forma:SolidPeso molecular:1533.8VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87Mequitazine
CAS:<p>Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.</p>Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.47Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C215H347N61O65S·6C2H4O2Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:5218.88MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Fórmula:C27H21F3N2O3Pureza:99.54% - 99.59%Cor e Forma:SolidPeso molecular:478.46Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Cor e Forma:SolidPeso molecular:403.52Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Fórmula:C20H22N2O6Pureza:99.39%Cor e Forma:SolidPeso molecular:386.4Epinastine hydrochloride
CAS:<p>Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.</p>Fórmula:C16H15N3·HClPureza:99.26% - 99.62%Cor e Forma:White SolidPeso molecular:285.77BWX 46 Acetate
<p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>Fórmula:C118H190N36O30S2Pureza:96.86%Cor e Forma:SolidPeso molecular:2657.12AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Fórmula:C21H24ClF2NOPureza:99.89%Cor e Forma:SolidPeso molecular:379.87Raclopride
CAS:<p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>Fórmula:C15H20Cl2N2O3Pureza:99.17%Cor e Forma:SolidPeso molecular:347.24SCH 58261
CAS:<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Fórmula:C18H15N7OPureza:99.07% - 99.75%Cor e Forma:SolidPeso molecular:345.36Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Cor e Forma:SolidPeso molecular:369.5JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Fórmula:C14H16ClN3OPureza:99.83% - 99.96%Cor e Forma:SolidPeso molecular:277.75Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Fórmula:C23H30N4O2SPureza:99.23%Cor e Forma:White PowderPeso molecular:426.57DAPTA
CAS:<p>DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.</p>Fórmula:C35H56N10O15Pureza:>99.99%Cor e Forma:SolidPeso molecular:856.88Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Fórmula:C36H55F3N8O12SPureza:>99.99%Cor e Forma:SolidPeso molecular:880.93NPY 5RA972
CAS:<p>NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist</p>Fórmula:C21H25N3O2Pureza:99.02% - 99.56%Cor e Forma:SolidPeso molecular:351.44RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Fórmula:C25H27N3O3Pureza:98.64% - 99.62%Cor e Forma:SolidPeso molecular:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Cor e Forma:SolidPeso molecular:240.69Ivabradine hydrochloride
CAS:<p>Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.</p>Fórmula:C27H37ClN2O5Pureza:99% - 99.73%Cor e Forma:SolidPeso molecular:505.05Chlorphenesin
CAS:<p>Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.</p>Fórmula:C9H11ClO3Pureza:99.59%Cor e Forma:SolidPeso molecular:202.63ZK 756326
CAS:<p>ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.</p>Fórmula:C21H28N2O3Pureza:99.43%Cor e Forma:SolidPeso molecular:356.46OXOMEMAZINE
CAS:<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Fórmula:C18H22N2O2SPureza:99.58%Cor e Forma:SolidPeso molecular:330.44Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Fórmula:C19H20ClN3Pureza:98% - 99.65%Cor e Forma:SolidPeso molecular:325.84AC-55541
CAS:<p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>Fórmula:C25H20BrN5O3Pureza:98% - 99.33%Cor e Forma:SolidPeso molecular:518.36Litorin acetate(55749-97-8 Free base)
<p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>Fórmula:C53H72N14O13SPureza:98.61%Cor e Forma:SolidPeso molecular:1145.29Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Cor e Forma:Off-White SolidPeso molecular:419.41
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