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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Fórmula:C17H18BrNO
    Pureza:95.00% - 99.82%
    Cor e Forma:Solid
    Peso molecular:332.23
  • AM095

    CAS:
    <p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>
    Fórmula:C27H23N2NaO5
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:478.47
  • ML401

    CAS:
    <p>ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .</p>
    Fórmula:C20H20BrClN2O
    Pureza:99.13%
    Cor e Forma:Solid
    Peso molecular:419.74
  • Sevoflurane

    CAS:
    <p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>
    Fórmula:C4H3F7O
    Pureza:98%
    Cor e Forma:Less Oil Colorless Oil
    Peso molecular:200.05
  • Binodenoson

    CAS:
    <p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>
    Fórmula:C17H25N7O4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:391.42
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Cor e Forma:Solid
    Peso molecular:403.52
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • Pizuglanstat

    CAS:
    <p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>
    Fórmula:C27H36N6O4
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:508.61
  • Bradykinin (acetate)

    CAS:
    <p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>
    Fórmula:C52H77N15O13
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1120.26
  • ACTH (1-39) human

    CAS:
    <p>Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.</p>
    Fórmula:C207H308N56O58S
    Pureza:99.6%
    Cor e Forma:White Lyophilised Solid
    Peso molecular:4541.14
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Cor e Forma:Solid
    Peso molecular:436.21
  • Azaphen

    CAS:
    <p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>
    Fórmula:C16H21Cl2N5O
    Pureza:97.62%
    Cor e Forma:Solid
    Peso molecular:370.28
  • BisfluoroModafinil

    CAS:
    <p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>
    Fórmula:C15H13F2NO2S
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:309.33
  • Harmine hydrochloride

    CAS:
    <p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>
    Fórmula:C13H13ClN2O
    Pureza:99.61% - >99.99%
    Cor e Forma:Yellow To Slightly Green Crystalline Powder
    Peso molecular:248.71
  • ACEPROMAZINE MALEATE

    CAS:
    <p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>
    Fórmula:C23H26N2O5S
    Pureza:98.87% - 99.51%
    Cor e Forma:Off White Or Yellow Crystalline Powder
    Peso molecular:442.53
  • ML-SI3

    CAS:
    <p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>
    Fórmula:C23H31N3O3S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:429.58
  • ML-097

    CAS:
    ML-097 (CID-2160985) is a pan activator of Ras-related GTPases
    Fórmula:C14H11BrO3
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:307.139
  • Taminadenant

    CAS:
    <p>Taminadenant is an adenosine receptor antagonist.</p>
    Fórmula:C10H8BrN7
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:306.12
  • Solabegron HCl

    CAS:
    <p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>
    Fórmula:C23H24Cl2N2O3
    Cor e Forma:Solid
    Peso molecular:447.35
  • Raclopride

    CAS:
    <p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>
    Fórmula:C15H20Cl2N2O3
    Pureza:99.17%
    Cor e Forma:Solid
    Peso molecular:347.24
  • Pimavanserin

    CAS:
    <p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>
    Fórmula:C25H34FN3O2
    Pureza:97.84% - 99.69%
    Cor e Forma:Pale Yellow To Pale Orange Solid
    Peso molecular:427.55
  • Betahistine EP Impurity C

    CAS:
    <p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>
    Fórmula:C15H19N3
    Pureza:≥95%
    Cor e Forma:Solid
    Peso molecular:241.33
  • Alprenolol hydrochloride

    CAS:
    <p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>
    Fórmula:C15H24ClNO2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:285.81
  • Eledoisin Related Peptide 2TFA


    <p>Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.</p>
    Fórmula:C38H60F6N8O10S
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:934.99
  • SAX-187

    CAS:
    <p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>
    Fórmula:C15H13ClN4O2S2
    Pureza:97.82% - 98%
    Cor e Forma:Solid
    Peso molecular:380.87
  • K 41498 aceate


    <p>K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for CRF1; blocks aSvg-30 effect on cAMP in cells.</p>
    Pureza:96.4%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • Human growth hormone-releasing factor acetate


    <p>Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on</p>
    Pureza:99.26%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • idalopirdine

    CAS:
    <p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>
    Fórmula:C20H19F5N2O
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:398.37
  • Carazolol

    CAS:
    <p>Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.</p>
    Fórmula:C18H22N2O2
    Pureza:99% - 99.53%
    Cor e Forma:Yellowish Solid
    Peso molecular:298.38
  • [Leu31,Pro34]-Neuropeptide Y (porcine)

    CAS:
    <p>[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.</p>
    Fórmula:C190H286N54O56
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:4223
  • Isocorynoxeine

    CAS:
    <p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>
    Fórmula:C22H26N2O4
    Pureza:98% - 99.9%
    Cor e Forma:Solid
    Peso molecular:382.45
  • Dasotraline

    CAS:
    <p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>
    Fórmula:C16H15Cl2N
    Cor e Forma:Solid
    Peso molecular:292.2
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:754.85
  • Desipramine

    CAS:
    <p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>
    Fórmula:C18H22N2
    Cor e Forma:Solid
    Peso molecular:266.38
  • Indacaterol

    CAS:
    <p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>
    Fórmula:C24H28N2O3
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:392.49
  • Detomidine hydrochloride

    CAS:
    <p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>
    Fórmula:C12H14N2·HCl
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:222.71
  • Thozalinone

    CAS:
    <p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>
    Fórmula:C11H12N2O2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:204.23
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:335.47
  • Org 27569

    CAS:
    <p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>
    Fórmula:C24H28ClN3O
    Pureza:>99.99% - ≥95%
    Cor e Forma:Solid
    Peso molecular:409.95
  • DORA-22

    CAS:
    <p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>
    Fórmula:C23H22F2N4O2
    Pureza:97.67%
    Cor e Forma:Solid
    Peso molecular:424.44
  • Galanin Receptor Ligand M35 TFA


    <p>Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).</p>
    Fórmula:C109H154N27F3O28
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:2347.62
  • CCG-50014

    CAS:
    <p>CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.</p>
    Fórmula:C16H13FN2O2S
    Pureza:98.53%
    Cor e Forma:Solid
    Peso molecular:316.35
  • β-CGRP, human acetate


    <p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>
    Fórmula:C164H271N51O50S3
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:3853.46
  • Batefenterol

    CAS:
    <p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>
    Fórmula:C40H42ClN5O7
    Pureza:97.94% - 98.4%
    Cor e Forma:Solid
    Peso molecular:740.24
  • 4i

    CAS:
    <p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>
    Fórmula:C16H12ClN3O
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:297.74
  • RS102895

    CAS:
    <p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>
    Fórmula:C21H21F3N2O2
    Pureza:97.64% - 99.80%
    Cor e Forma:Solid
    Peso molecular:390.4
  • BMS-813160

    CAS:
    <p>BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.</p>
    Fórmula:C25H40N8O2
    Pureza:99.66% - 99.79%
    Cor e Forma:Solid
    Peso molecular:484.64
  • H2L 5765834

    CAS:
    <p>H2L 5765834 is a lysophosphatidic acid receptors antagonist</p>
    Fórmula:C21H12N2O7
    Pureza:98.25% - 99.47%
    Cor e Forma:Solid
    Peso molecular:404.33
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:469.55
  • Namodenoson

    CAS:
    <p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>
    Fórmula:C18H18ClIN6O4
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:544.73
  • BI-6015

    CAS:
    <p>BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.</p>
    Fórmula:C15H13N3O4S
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:331.35
  • Clopidogrel thiolactone

    CAS:
    <p>Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.</p>
    Fórmula:C16H16ClNO3S
    Pureza:98.79%
    Cor e Forma:Solid
    Peso molecular:337.82
  • Dexpramipexole

    CAS:
    <p>Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.</p>
    Fórmula:C10H17N3S
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:211.33
  • Latrepirdine dihydrochloride

    CAS:
    <p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>
    Fórmula:C21H25N3·2HCl
    Pureza:98.45%
    Cor e Forma:Solid
    Peso molecular:392.37
  • Ketanserin tartrate

    CAS:
    <p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>
    Fórmula:C26H28FN3O9
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:545.51
  • LP-533401 hydrochloride

    CAS:
    <p>LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.</p>
    Fórmula:C27H23ClF4N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:562.94
  • Renzapride

    CAS:
    <p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>
    Fórmula:C16H22ClN3O2
    Pureza:98.97% - 99.09%
    Cor e Forma:Solid
    Peso molecular:323.82
  • Jatrorrhizine chloride

    CAS:
    <p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>
    Fórmula:C20H20ClNO4
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:373.8
  • Atipamezole

    CAS:
    <p>Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.</p>
    Fórmula:C14H16N2
    Pureza:99.88%
    Cor e Forma:Off-White To Light Yellow Crystal Powder
    Peso molecular:212.29
  • INCB 3284

    CAS:
    INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.
    Fórmula:C26H31F3N4O4
    Pureza:97.81% - 99.42%
    Cor e Forma:Solid
    Peso molecular:520.54
  • WAY-100635 maleate

    CAS:
    <p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>
    Fórmula:C25H34N4O2·xC4H4O4
    Pureza:>99.99%
    Cor e Forma:White Solid
    Peso molecular:538.645
  • SB 243213

    CAS:
    <p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>
    Fórmula:C22H19F3N4O2
    Pureza:98.78% - 99.86%
    Cor e Forma:Solid
    Peso molecular:428.41
  • CP-105696

    CAS:
    <p>CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.</p>
    Fórmula:C28H28O4
    Pureza:99.78%
    Cor e Forma:Solid
    Peso molecular:428.52
  • Canagliflozin hemihydrate

    CAS:
    <p>Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.</p>
    Fórmula:C48H52F2O11S2
    Pureza:99.42% - 99.96%
    Cor e Forma:Solid
    Peso molecular:907.05
  • S-Methoprene

    CAS:
    <p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>
    Fórmula:C19H34O3
    Pureza:97.05% - 98.55%
    Cor e Forma:Solid
    Peso molecular:310.47
  • Opipramol

    CAS:
    <p>Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.</p>
    Fórmula:C23H29N3O
    Pureza:99.84% - 99.98%
    Cor e Forma:Solid
    Peso molecular:363.5
  • WIN 51,708

    CAS:
    <p>WIN 51,708 is an antagonist of neurokinin-1 receptor.</p>
    Fórmula:C29H33N3O
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:439.59
  • Atogepant

    CAS:
    <p>Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.</p>
    Fórmula:C29H23F6N5O3
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:603.52
  • Fenoterol hydrobromide

    CAS:
    <p>Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.</p>
    Fórmula:C17H22BrNO4
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:384.27
  • CGP 20712 A

    CAS:
    <p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>
    Fórmula:C24H29F3N4O8S
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:590.57
  • (R)-Mirtazapine

    CAS:
    <p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>
    Fórmula:C17H19N3
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Rolofylline

    CAS:
    <p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>
    Fórmula:C20H28N4O2
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:356.46
  • Citalopram

    CAS:
    <p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>
    Fórmula:C20H21FN2O
    Pureza:99.78% - 99.89%
    Cor e Forma:Solid
    Peso molecular:324.39
  • Levocetirizine Dihydrochloride

    CAS:
    <p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>
    Fórmula:C21H27Cl3N2O3
    Pureza:99.89%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:461.81
  • (S)-Mirtazapine

    CAS:
    <p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>
    Fórmula:C17H19N3
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:265.35
  • GRK6-IN-2

    CAS:
    <p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>
    Fórmula:C21H21FN6
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:376.43
  • BMS-986278

    CAS:
    <p>BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,</p>
    Fórmula:C22H31N5O5
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:445.51
  • L-368,899 hydrochloride

    CAS:
    <p>L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.</p>
    Fórmula:C26H43ClN4O5S2
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:591.23
  • S1RA

    CAS:
    <p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>
    Fórmula:C20H23N3O2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:337.42
  • GAT211

    CAS:
    <p>GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.</p>
    Fórmula:C22H18N2O2
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:342.39
  • Nebentan potassium

    CAS:
    <p>Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.</p>
    Fórmula:C24H20KN5O5S
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:529.61
  • Maropitant citrate

    CAS:
    <p>Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.</p>
    Fórmula:C38H50N2O9
    Pureza:98.91%
    Cor e Forma:Solid
    Peso molecular:678.81
  • AF-710B

    CAS:
    <p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>
    Fórmula:C20H27N3OS
    Pureza:98.62% - 99.89%
    Cor e Forma:Solid
    Peso molecular:357.51
  • Rizatriptan

    CAS:
    <p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>
    Fórmula:C15H19N5
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:269.35
  • Rotigotine

    CAS:
    <p>Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.</p>
    Fórmula:C19H25NOS
    Pureza:99.04% - 99.88%
    Cor e Forma:Solid
    Peso molecular:315.47
  • Trabodenoson

    CAS:
    <p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>
    Fórmula:C15H20N6O6
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:380.36
  • Medetomidine

    CAS:
    <p>Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.</p>
    Fórmula:C13H16N2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:200.28
  • Ozanimod hydrochloride

    CAS:
    <p>Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.</p>
    Fórmula:C23H25ClN4O3
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:440.92
  • A2ti-1

    CAS:
    <p>A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.</p>
    Fórmula:C20H22N4O2S
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:382.48
  • CB1/2 agonist 3

    CAS:
    <p>CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.</p>
    Fórmula:C25H41NO2
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:387.6
  • Protein deglycase DJ-1 against-1

    CAS:
    <p>Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.</p>
    Fórmula:C24H23N3O4
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:417.46
  • SID 7969543

    CAS:
    <p>SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.</p>
    Fórmula:C24H24N2O7
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:452.46
  • Bucindolol

    CAS:
    <p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>
    Fórmula:C22H25N3O2
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:363.45
  • Fenoprofen

    CAS:
    <p>Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.</p>
    Fórmula:C15H14O3
    Pureza:98.4%
    Cor e Forma:Solid
    Peso molecular:242.27
  • ACT-462206

    CAS:
    <p>ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.</p>
    Fórmula:C20H24N2O4S
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:388.48
  • Setiptiline

    CAS:
    <p>Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.</p>
    Fórmula:C19H19N
    Pureza:98.05% - 98.07%
    Cor e Forma:Solid
    Peso molecular:261.36
  • Alfuzosin

    CAS:
    <p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>
    Fórmula:C19H27N5O4
    Pureza:99.64%
    Cor e Forma:White Crystaline Powder
    Peso molecular:389.45
  • Trazpiroben

    CAS:
    <p>Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.</p>
    Fórmula:C31H39N3O4
    Pureza:99.41% - >99.99%
    Cor e Forma:Solid
    Peso molecular:517.66
  • Tandospirone

    CAS:
    <p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>
    Fórmula:C21H29N5O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:383.49
  • UCM 608

    CAS:
    <p>UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.</p>
    Fórmula:C19H20N2O2
    Pureza:98.88%
    Cor e Forma:Solid
    Peso molecular:308.37