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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • Bambuterol hydrochloride

    CAS:
    <p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>
    Fórmula:C18H30ClN3O5
    Pureza:99.53% - 99.61%
    Cor e Forma:White Solid
    Peso molecular:403.91
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53
  • AM095 free acid

    CAS:
    <p>AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).</p>
    Fórmula:C27H24N2O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:456.49
  • Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>
    Fórmula:C28H30N2O8
    Pureza:99.7% - >99.99%
    Cor e Forma:Powder
    Peso molecular:522.55
  • YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:615.74
  • Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Fórmula:C20H22BrFN2O
    Pureza:99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:405.304
  • Urocortin (rat) acetate


    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Pureza:97.76%
    Cor e Forma:Soild
  • Blonanserin

    CAS:
    <p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>
    Fórmula:C23H30FN3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:367.5
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Fórmula:C18H29ClN2O4
    Pureza:99.92% - >99.99%
    Cor e Forma:White Or Slightly Off-White Crystalline Powder Solid
    Peso molecular:372.89
  • Olanzapine

    CAS:
    <p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>
    Fórmula:C17H20N4S
    Pureza:99.86% - ≥95%
    Cor e Forma:Yellowish Crystalline Powder
    Peso molecular:312.43
  • Salmeterol

    CAS:
    <p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Cor e Forma:Solid
    Peso molecular:415.57
  • Terfenadine

    CAS:
    <p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>
    Fórmula:C32H41NO2
    Pureza:98.76% - 99.75%
    Cor e Forma:Solid
    Peso molecular:471.67
  • MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Fórmula:C27H25N3O4S2
    Pureza:97.44%
    Cor e Forma:Solid
    Peso molecular:519.64
  • Diphenylpyraline hydrochloride

    CAS:
    <p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>
    Fórmula:C19H23NO·HCl
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:317.85
  • Hydroxyzine Pamoate

    CAS:
    <p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>
    Fórmula:C44H43ClN2O8
    Pureza:99.49%
    Cor e Forma:Solid
    Peso molecular:763.27
  • Levocetirizine

    CAS:
    <p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>
    Fórmula:C21H25ClN2O3
    Pureza:98% - 99.9%
    Cor e Forma:White Powder
    Peso molecular:388.89
  • Evocalcet

    CAS:
    <p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>
    Fórmula:C24H26N2O2
    Pureza:98.88% - 99.68%
    Cor e Forma:Solid
    Peso molecular:374.48
  • Ketotifen fumarate

    CAS:
    <p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>
    Fórmula:C23H23NO5S
    Pureza:99.25% - 99.73%
    Cor e Forma:Solid
    Peso molecular:425.50
  • MK-0812 Succinate

    CAS:
    <p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>
    Fórmula:C28H40F3N3O7
    Pureza:98.62% - 99.93%
    Cor e Forma:Solid
    Peso molecular:587.63
  • Promethazine hydrochloride

    CAS:
    <p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>
    Fórmula:C17H20N2S·HCl
    Pureza:99.85%
    Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Peso molecular:320.88
  • Capeserod

    CAS:
    <p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>
    Fórmula:C23H25ClN4O4
    Pureza:98.10% - 99.94%
    Cor e Forma:Solid
    Peso molecular:456.92
  • SEP-363856 hydrochloride

    CAS:
    <p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>
    Fórmula:C9H14ClNOS
    Pureza:99.86% - 99.99%
    Cor e Forma:Solid
    Peso molecular:219.73
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Fórmula:C15H24N2O4S·HCl
    Pureza:99.4% - 99.77%
    Cor e Forma:Solid
    Peso molecular:364.89
  • Brompheniramine maleate

    CAS:
    <p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>
    Fórmula:C16H19BrN2·C4H4O4
    Pureza:99.80%
    Cor e Forma:Crystal Powder
    Peso molecular:435.31
  • AC265347

    CAS:
    <p>AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity for the study of neuroblastoma.</p>
    Fórmula:C17H17NOS
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:283.39
  • Naftifine hydrochloride

    CAS:
    <p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>
    Fórmula:C21H22ClN
    Pureza:98.75% - 99.84%
    Cor e Forma:Solid
    Peso molecular:323.86
  • Bucumolol

    CAS:
    <p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>
    Fórmula:C17H23NO4
    Pureza:99.66%
    Cor e Forma:Soild
    Peso molecular:305.37
  • Iobenguane sulfate

    CAS:
    <p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>
    Fórmula:C8H10IN3H2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:324.12
  • Amitriptyline hydrochloride

    CAS:
    <p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>
    Fórmula:C20H24ClN
    Pureza:97% - 99.94%
    Cor e Forma:Crystals White To Off-White Powder
    Peso molecular:313.86
  • REV 5901A

    CAS:
    <p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>
    Fórmula:C22H26ClNO2
    Pureza:98.04%
    Cor e Forma:Soild
    Peso molecular:371.90
  • Balovaptan

    CAS:
    <p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>
    Fórmula:C22H24ClN5O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Nicergoline

    CAS:
    <p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>
    Fórmula:C24H26BrN3O3
    Pureza:98% - 99.80%
    Cor e Forma:Solid
    Peso molecular:484.39
  • Doxofylline

    CAS:
    <p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>
    Fórmula:C11H14N4O4
    Pureza:99.958% - >99.99%
    Cor e Forma:Solid
    Peso molecular:266.25
  • Naftidrofuryl oxalate

    CAS:
    <p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>
    Fórmula:C26H35NO7
    Pureza:97.12% - 98.38%
    Cor e Forma:Solid
    Peso molecular:473.56
  • [Leu15]-Gastrin I, human

    CAS:
    <p>[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.</p>
    Fórmula:C98H126N20O31
    Pureza:98.02% - 98.84%
    Cor e Forma:Solid
    Peso molecular:2080.16
  • Rebamipide

    CAS:
    <p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>
    Fórmula:C19H15ClN2O4
    Pureza:99.48% - 99.61%
    Cor e Forma:White Powder
    Peso molecular:370.79
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Fórmula:C21H23N3OS
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:365.49
  • Tolnapersine TFA


    <p>Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.</p>
    Fórmula:C23H27F3N2O3
    Pureza:99.14%
    Cor e Forma:Soild
    Peso molecular:436.47
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Fórmula:C21H25NO·CH4SO3
    Pureza:98.41% - 99.96%
    Cor e Forma:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecular:403.53
  • Iloperidone

    CAS:
    <p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>
    Fórmula:C24H27FN2O4
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:426.48
  • ONC206

    CAS:
    <p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>
    Fórmula:C23H22F2N4O
    Pureza:99.38% - 99.81%
    Cor e Forma:Solid
    Peso molecular:408.44
  • Mebhydrolin napadisylate

    CAS:
    <p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>
    Fórmula:C19H20N2C10H8O6S2
    Pureza:99.35% - 99.96%
    Cor e Forma:White Or Almost White Crystalline
    Peso molecular:420.52
  • Carebastine

    CAS:
    <p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>
    Fórmula:C32H37NO4
    Pureza:99.16%
    Cor e Forma:Off-White Solid
    Peso molecular:499.64
  • Phenoxybenzamine hydrochloride

    CAS:
    <p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>
    Fórmula:C18H23Cl2NO
    Pureza:98.04% - >99.99%
    Cor e Forma:Antihypertensive Drug
    Peso molecular:340.3
  • Tipepidine hydrochloride

    CAS:
    <p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>
    Fórmula:C15H18ClNS2
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:311.89
  • Paliperidone

    CAS:
    <p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>
    Fórmula:C23H27FN4O3
    Pureza:95% - 99.08%
    Cor e Forma:Off White To Light Orange Coloured Solid
    Peso molecular:426.48
  • Lesopitron HCl

    CAS:
    <p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>
    Fórmula:C15H22Cl2N6
    Pureza:97.05% - 99.89%
    Cor e Forma:Soild
    Peso molecular:357.28
  • Lintopride HCl

    CAS:
    <p>Lintopride HCl is a 5HT-4 antagonist.</p>
    Fórmula:C14H20Cl2N4O2
    Pureza:98.42% - 98.81%
    Cor e Forma:Soild
    Peso molecular:347.24
  • Ritodrine hydrochloride

    CAS:
    <p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>
    Fórmula:C17H21NO3·HCl
    Pureza:99% - 99.52%
    Cor e Forma:Solid
    Peso molecular:323.82
  • Avexitide acetate

    CAS:
    <p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>
    Fórmula:C155H246N40O53S
    Pureza:96.64% - 98.65%
    Cor e Forma:Solid
    Peso molecular:3549.91
  • 2',5'-Dideoxyadenosine

    CAS:
    <p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>
    Fórmula:C10H13N5O2
    Pureza:99.55%
    Cor e Forma:White Solid
    Peso molecular:235.24
  • Metoclopramide hydrochloride

    CAS:
    <p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>
    Fórmula:C14H22ClN3O2·HCl
    Pureza:99.99%
    Cor e Forma:White To Off-White Powder
    Peso molecular:336.26
  • Carbinoxamine Maleate Salt

    CAS:
    <p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>
    Fórmula:C20H23ClN2O5
    Pureza:99.97%
    Cor e Forma:Off-White Solid
    Peso molecular:406.86
  • Aniracetam

    CAS:
    <p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>
    Fórmula:C12H13NO3
    Pureza:99.88% - 99.89%
    Cor e Forma:White Crystalline Or Crystalline Powde
    Peso molecular:219.24
  • Frovatriptan succinate hydrate

    CAS:
    <p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>
    Fórmula:C18H25N3O6
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:379.41
  • Desvenlafaxine

    CAS:
    <p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>
    Fórmula:C16H25NO2
    Pureza:99.46% - 99.81%
    Cor e Forma:White Crystalline Powder
    Peso molecular:263.38
  • SBI-477

    CAS:
    <p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>
    Fórmula:C24H25N3O6S
    Pureza:99.3%
    Cor e Forma:Solid
    Peso molecular:483.54
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Fórmula:C25H28N2O5S
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:468.57
  • PF-04995274

    CAS:
    <p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>
    Fórmula:C23H32N2O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:432.51
  • Ozagrel

    CAS:
    <p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>
    Fórmula:C13H12N2O2
    Pureza:97.90% - 99.38%
    Cor e Forma:White Powder
    Peso molecular:228.25
  • Azacyclonol

    CAS:
    <p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>
    Fórmula:C18H21NO
    Pureza:99.46%
    Cor e Forma:Solid Powder
    Peso molecular:267.37
  • BP 897 hydrochloride

    CAS:
    <p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>
    Fórmula:C26H32ClN3O2
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:454
  • Enrasentan

    CAS:
    <p>Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure and protects myocardial function.</p>
    Fórmula:C29H30O8
    Pureza:97.9% - 98.39%
    Cor e Forma:Solid
    Peso molecular:506.54
  • YT 146

    CAS:
    <p>YT 146 is a biochemical.</p>
    Fórmula:C18H25N5O4
    Pureza:98.81% - 99.25%
    Cor e Forma:Solid
    Peso molecular:375.42
  • Midodrine hydrochloride

    CAS:
    <p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>
    Fórmula:C12H19ClN2O4
    Pureza:99.79% - >99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:290.74
  • HJC0197

    CAS:
    <p>HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.</p>
    Fórmula:C19H21N3OS
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:339.45
  • Azelastine hydrochloride

    CAS:
    <p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>
    Fórmula:C22H24ClN3O·HCl
    Pureza:98% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:418.36
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Fórmula:C10H16N6S
    Pureza:99.82%
    Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Peso molecular:252.34
  • Flunarizine dihydrochloride

    CAS:
    <p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>
    Fórmula:C26H28Cl2F2N2
    Pureza:99.53% - 99.89%
    Cor e Forma:White Crystalline Powder Odorless And Tasteless
    Peso molecular:477.42
  • Loxapine succinate

    CAS:
    <p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>
    Fórmula:C22H24ClN3O5
    Pureza:99.69%
    Cor e Forma:White To Of-White Solid
    Peso molecular:445.9
  • Quercetin-3'-o-phosphate TEA


    <p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>
    Fórmula:C21H26NO10P
    Pureza:95.63%
    Cor e Forma:Soild
    Peso molecular:483.41
  • Tropisetron hydrochloride

    CAS:
    <p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>
    Fórmula:C17H21ClN2O2
    Pureza:99.72% - 99.83%
    Cor e Forma:Solid
    Peso molecular:320.82
  • Fluphenazine dihydrochloride

    CAS:
    <p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>
    Fórmula:C22H28Cl2F3N3OS
    Pureza:99.23%
    Cor e Forma:Off-White Solid
    Peso molecular:510.44
  • Retatrutide sodium salt


    <p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>
    Pureza:99.97%
    Cor e Forma:Soild
  • Latozinemab


    <p>Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.</p>
    Pureza:> 95%
    Cor e Forma:Liquid
    Peso molecular:146.28 kDa
  • Ramelteon

    CAS:
    <p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>
    Fórmula:C16H21NO2
    Pureza:97.21% - 99.92%
    Cor e Forma:Crystalline Solid
    Peso molecular:259.34
  • Ranitidine Hydrochloride

    CAS:
    <p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>
    Fórmula:C13H23ClN4O3S
    Pureza:99.30% - 99.49%
    Cor e Forma:Solid
    Peso molecular:350.86
  • Cloperastine hydrochloride

    CAS:
    <p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>
    Fórmula:C20H25Cl2NO
    Pureza:97.74% - 99.42%
    Cor e Forma:Solid
    Peso molecular:366.33
  • Labetalol hydrochloride

    CAS:
    <p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>
    Fórmula:C19H25ClN2O3
    Pureza:99.54% - 99.85%
    Cor e Forma:Solid
    Peso molecular:364.87
  • Pimethixene

    CAS:
    <p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 &amp; muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>
    Fórmula:C19H19NS
    Pureza:97.50%
    Cor e Forma:Solid
    Peso molecular:293.43
  • Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Fórmula:C36H51Cl2N3O4
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:660.71
  • Carbazochrome sodium sulfonate

    CAS:
    <p>Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.</p>
    Fórmula:C10H11N4NaO5S
    Pureza:99.63%
    Cor e Forma:Orange Yellow Crystalline Powder
    Peso molecular:322.03
  • Retatrutide

    CAS:
    <p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>
    Fórmula:C221H342N46O68
    Pureza:98.31%
    Cor e Forma:Solid
    Peso molecular:4732.09
  • Nardeterol HCl


    <p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>
    Fórmula:C20H25ClFN3O2
    Pureza:97.72% - 98.65%
    Cor e Forma:Soild
    Peso molecular:393.88
  • 6-Iodopravadoline

    CAS:
    <p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>
    Fórmula:C23H25IN2O3
    Pureza:99.29%
    Cor e Forma:Off-White Solid
    Peso molecular:504.36
  • JHU 75528

    CAS:
    <p>JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.</p>
    Fórmula:C23H21Cl2N5O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:470.35
  • Dapoxetine hydrochloride

    CAS:
    <p>Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.</p>
    Fórmula:C21H23NO·HCl
    Pureza:99.70% - 99.91%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:341.87
  • Sulpiride

    CAS:
    <p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>
    Fórmula:C15H23N3O4S
    Pureza:99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid

    CAS:
    <p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>
    Fórmula:C20H29N3O8
    Pureza:99.72%
    Cor e Forma:Soild
    Peso molecular:439.46
  • Xylometazoline hydrochloride

    CAS:
    <p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>
    Fórmula:C16H24N2·HCl
    Pureza:99.77% - 99.87%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:280.84
  • Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Fórmula:C22H23ClN2O2
    Pureza:99.71% - 99.98%
    Cor e Forma:White Powder
    Peso molecular:382.88
  • PHM-27 (human) acetate


    <p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>
    Fórmula:C137H215F3N34O42S
    Pureza:99.20%
    Cor e Forma:Soild
    Peso molecular:3099.44
  • Benserazide hydrochloride

    CAS:
    <p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>
    Fórmula:C10H15N3O5·HCl
    Pureza:98.63% - 99.74%
    Cor e Forma:White Crystalline Solid
    Peso molecular:293.7
  • Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Fórmula:C17H22ClNO
    Pureza:99.86%
    Cor e Forma:White Solid
    Peso molecular:291.82
  • Pheniramine maleate

    CAS:
    <p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>
    Fórmula:C16H20N2·C4H4O4
    Pureza:99.85%
    Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
    Peso molecular:356.42
  • Timonacic

    CAS:
    <p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>
    Fórmula:C4H7NO2S
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:133.17
  • Tropanserin

    CAS:
    <p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>
    Fórmula:C17H23NO2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:273.37
  • Ifenprodil

    CAS:
    <p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 &amp; GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>
    Fórmula:C21H27NO2
    Pureza:99.58%
    Cor e Forma:White Crystalline Powder
    Peso molecular:325.44
  • Carteolol hydrochloride

    CAS:
    <p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>
    Fórmula:C16H24N2O3·HCl
    Pureza:99.84% - 99.91%
    Cor e Forma:Solid
    Peso molecular:328.83
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Fórmula:C21H27NO2C4H6O6
    Pureza:99.02% - 99.55%
    Cor e Forma:Solid
    Peso molecular:400.49