
GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Fórmula:C18H30ClN3O5Pureza:99.53% - 99.61%Cor e Forma:White SolidPeso molecular:403.91hGPR91 antagonist 1
CAS:<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Fórmula:C31H23F4N3OPureza:98.89%Cor e Forma:SolidPeso molecular:529.53AM095 free acid
CAS:<p>AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).</p>Fórmula:C27H24N2O5Pureza:99.88%Cor e Forma:SolidPeso molecular:456.49Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Fórmula:C33H37N5O5SPureza:99.67%Cor e Forma:SolidPeso molecular:615.74Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Fórmula:C20H22BrFN2OPureza:99.81%Cor e Forma:White Crystalline PowderPeso molecular:405.304Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Pureza:97.76%Cor e Forma:SoildBlonanserin
CAS:<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Fórmula:C23H30FN3Pureza:99.85%Cor e Forma:SolidPeso molecular:367.5Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Fórmula:C18H29ClN2O4Pureza:99.92% - >99.99%Cor e Forma:White Or Slightly Off-White Crystalline Powder SolidPeso molecular:372.89Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Fórmula:C17H20N4SPureza:99.86% - ≥95%Cor e Forma:Yellowish Crystalline PowderPeso molecular:312.43Salmeterol
CAS:<p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>Fórmula:C25H37NO4Pureza:99.2% - 99.9%Cor e Forma:SolidPeso molecular:415.57Terfenadine
CAS:<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Fórmula:C32H41NO2Pureza:98.76% - 99.75%Cor e Forma:SolidPeso molecular:471.67MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Fórmula:C27H25N3O4S2Pureza:97.44%Cor e Forma:SolidPeso molecular:519.64Diphenylpyraline hydrochloride
CAS:<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Fórmula:C19H23NO·HClPureza:98.72%Cor e Forma:SolidPeso molecular:317.85Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Fórmula:C44H43ClN2O8Pureza:99.49%Cor e Forma:SolidPeso molecular:763.27Levocetirizine
CAS:<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98% - 99.9%Cor e Forma:White PowderPeso molecular:388.89Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Fórmula:C24H26N2O2Pureza:98.88% - 99.68%Cor e Forma:SolidPeso molecular:374.48Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Fórmula:C23H23NO5SPureza:99.25% - 99.73%Cor e Forma:SolidPeso molecular:425.50MK-0812 Succinate
CAS:<p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>Fórmula:C28H40F3N3O7Pureza:98.62% - 99.93%Cor e Forma:SolidPeso molecular:587.63Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Capeserod
CAS:<p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>Fórmula:C23H25ClN4O4Pureza:98.10% - 99.94%Cor e Forma:SolidPeso molecular:456.92SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Fórmula:C9H14ClNOSPureza:99.86% - 99.99%Cor e Forma:SolidPeso molecular:219.73Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Fórmula:C15H24N2O4S·HClPureza:99.4% - 99.77%Cor e Forma:SolidPeso molecular:364.89Brompheniramine maleate
CAS:<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Cor e Forma:Crystal PowderPeso molecular:435.31AC265347
CAS:<p>AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity for the study of neuroblastoma.</p>Fórmula:C17H17NOSPureza:>99.99%Cor e Forma:SolidPeso molecular:283.39Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Fórmula:C21H22ClNPureza:98.75% - 99.84%Cor e Forma:SolidPeso molecular:323.86Bucumolol
CAS:<p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>Fórmula:C17H23NO4Pureza:99.66%Cor e Forma:SoildPeso molecular:305.37Iobenguane sulfate
CAS:<p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>Fórmula:C8H10IN3H2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:324.12Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Fórmula:C20H24ClNPureza:97% - 99.94%Cor e Forma:Crystals White To Off-White PowderPeso molecular:313.86REV 5901A
CAS:<p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>Fórmula:C22H26ClNO2Pureza:98.04%Cor e Forma:SoildPeso molecular:371.90Balovaptan
CAS:<p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>Fórmula:C22H24ClN5OPureza:99.88%Cor e Forma:SolidPeso molecular:409.91Nicergoline
CAS:<p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>Fórmula:C24H26BrN3O3Pureza:98% - 99.80%Cor e Forma:SolidPeso molecular:484.39Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Fórmula:C11H14N4O4Pureza:99.958% - >99.99%Cor e Forma:SolidPeso molecular:266.25Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Fórmula:C26H35NO7Pureza:97.12% - 98.38%Cor e Forma:SolidPeso molecular:473.56[Leu15]-Gastrin I, human
CAS:<p>[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.</p>Fórmula:C98H126N20O31Pureza:98.02% - 98.84%Cor e Forma:SolidPeso molecular:2080.16Rebamipide
CAS:<p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>Fórmula:C19H15ClN2O4Pureza:99.48% - 99.61%Cor e Forma:White PowderPeso molecular:370.79Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Fórmula:C21H23N3OSPureza:99.61%Cor e Forma:SolidPeso molecular:365.49Tolnapersine TFA
<p>Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.</p>Fórmula:C23H27F3N2O3Pureza:99.14%Cor e Forma:SoildPeso molecular:436.47Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Fórmula:C24H27FN2O4Pureza:99.42%Cor e Forma:SolidPeso molecular:426.48ONC206
CAS:<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Fórmula:C23H22F2N4OPureza:99.38% - 99.81%Cor e Forma:SolidPeso molecular:408.44Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Fórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.96%Cor e Forma:White Or Almost White CrystallinePeso molecular:420.52Carebastine
CAS:<p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>Fórmula:C32H37NO4Pureza:99.16%Cor e Forma:Off-White SolidPeso molecular:499.64Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Fórmula:C18H23Cl2NOPureza:98.04% - >99.99%Cor e Forma:Antihypertensive DrugPeso molecular:340.3Tipepidine hydrochloride
CAS:<p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>Fórmula:C15H18ClNS2Pureza:99.97%Cor e Forma:SolidPeso molecular:311.89Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Fórmula:C23H27FN4O3Pureza:95% - 99.08%Cor e Forma:Off White To Light Orange Coloured SolidPeso molecular:426.48Lesopitron HCl
CAS:<p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>Fórmula:C15H22Cl2N6Pureza:97.05% - 99.89%Cor e Forma:SoildPeso molecular:357.28Lintopride HCl
CAS:<p>Lintopride HCl is a 5HT-4 antagonist.</p>Fórmula:C14H20Cl2N4O2Pureza:98.42% - 98.81%Cor e Forma:SoildPeso molecular:347.24Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Fórmula:C17H21NO3·HClPureza:99% - 99.52%Cor e Forma:SolidPeso molecular:323.82Avexitide acetate
CAS:<p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>Fórmula:C155H246N40O53SPureza:96.64% - 98.65%Cor e Forma:SolidPeso molecular:3549.912',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Fórmula:C10H13N5O2Pureza:99.55%Cor e Forma:White SolidPeso molecular:235.24Metoclopramide hydrochloride
CAS:<p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>Fórmula:C14H22ClN3O2·HClPureza:99.99%Cor e Forma:White To Off-White PowderPeso molecular:336.26Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Cor e Forma:Off-White SolidPeso molecular:406.86Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Fórmula:C12H13NO3Pureza:99.88% - 99.89%Cor e Forma:White Crystalline Or Crystalline PowdePeso molecular:219.24Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Fórmula:C18H25N3O6Pureza:99.66%Cor e Forma:SolidPeso molecular:379.41Desvenlafaxine
CAS:<p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>Fórmula:C16H25NO2Pureza:99.46% - 99.81%Cor e Forma:White Crystalline PowderPeso molecular:263.38SBI-477
CAS:<p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>Fórmula:C24H25N3O6SPureza:99.3%Cor e Forma:SolidPeso molecular:483.54Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Fórmula:C25H28N2O5SPureza:97.09%Cor e Forma:SolidPeso molecular:468.57PF-04995274
CAS:<p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>Fórmula:C23H32N2O6Pureza:99.52%Cor e Forma:SolidPeso molecular:432.51Ozagrel
CAS:<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Fórmula:C13H12N2O2Pureza:97.90% - 99.38%Cor e Forma:White PowderPeso molecular:228.25Azacyclonol
CAS:<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Fórmula:C18H21NOPureza:99.46%Cor e Forma:Solid PowderPeso molecular:267.37BP 897 hydrochloride
CAS:<p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>Fórmula:C26H32ClN3O2Pureza:99.42%Cor e Forma:SolidPeso molecular:454Enrasentan
CAS:<p>Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure and protects myocardial function.</p>Fórmula:C29H30O8Pureza:97.9% - 98.39%Cor e Forma:SolidPeso molecular:506.54YT 146
CAS:<p>YT 146 is a biochemical.</p>Fórmula:C18H25N5O4Pureza:98.81% - 99.25%Cor e Forma:SolidPeso molecular:375.42Midodrine hydrochloride
CAS:<p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>Fórmula:C12H19ClN2O4Pureza:99.79% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:290.74HJC0197
CAS:<p>HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.</p>Fórmula:C19H21N3OSPureza:98.05%Cor e Forma:SolidPeso molecular:339.45Azelastine hydrochloride
CAS:<p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>Fórmula:C22H24ClN3O·HClPureza:98% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:418.36Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Fórmula:C10H16N6SPureza:99.82%Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecular:252.34Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Fórmula:C26H28Cl2F2N2Pureza:99.53% - 99.89%Cor e Forma:White Crystalline Powder Odorless And TastelessPeso molecular:477.42Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Fórmula:C22H24ClN3O5Pureza:99.69%Cor e Forma:White To Of-White SolidPeso molecular:445.9Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Fórmula:C21H26NO10PPureza:95.63%Cor e Forma:SoildPeso molecular:483.41Tropisetron hydrochloride
CAS:<p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>Fórmula:C17H21ClN2O2Pureza:99.72% - 99.83%Cor e Forma:SolidPeso molecular:320.82Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Fórmula:C22H28Cl2F3N3OSPureza:99.23%Cor e Forma:Off-White SolidPeso molecular:510.44Retatrutide sodium salt
<p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>Pureza:99.97%Cor e Forma:SoildLatozinemab
<p>Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:146.28 kDaRamelteon
CAS:<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Fórmula:C16H21NO2Pureza:97.21% - 99.92%Cor e Forma:Crystalline SolidPeso molecular:259.34Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Cloperastine hydrochloride
CAS:<p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>Fórmula:C20H25Cl2NOPureza:97.74% - 99.42%Cor e Forma:SolidPeso molecular:366.33Labetalol hydrochloride
CAS:<p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>Fórmula:C19H25ClN2O3Pureza:99.54% - 99.85%Cor e Forma:SolidPeso molecular:364.87Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Fórmula:C19H19NSPureza:97.50%Cor e Forma:SolidPeso molecular:293.43Aripiprazole Lauroxil
CAS:<p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>Fórmula:C36H51Cl2N3O4Pureza:99.64%Cor e Forma:SolidPeso molecular:660.71Carbazochrome sodium sulfonate
CAS:<p>Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.</p>Fórmula:C10H11N4NaO5SPureza:99.63%Cor e Forma:Orange Yellow Crystalline PowderPeso molecular:322.03Retatrutide
CAS:<p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>Fórmula:C221H342N46O68Pureza:98.31%Cor e Forma:SolidPeso molecular:4732.09Nardeterol HCl
<p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>Fórmula:C20H25ClFN3O2Pureza:97.72% - 98.65%Cor e Forma:SoildPeso molecular:393.886-Iodopravadoline
CAS:<p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>Fórmula:C23H25IN2O3Pureza:99.29%Cor e Forma:Off-White SolidPeso molecular:504.36JHU 75528
CAS:<p>JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.</p>Fórmula:C23H21Cl2N5O2Pureza:99.79%Cor e Forma:SolidPeso molecular:470.35Dapoxetine hydrochloride
CAS:<p>Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.</p>Fórmula:C21H23NO·HClPureza:99.70% - 99.91%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:341.87Sulpiride
CAS:<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Fórmula:C15H23N3O4SPureza:99.94%Cor e Forma:White Crystalline PowderPeso molecular:341.43(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Fórmula:C20H29N3O8Pureza:99.72%Cor e Forma:SoildPeso molecular:439.46Xylometazoline hydrochloride
CAS:<p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>Fórmula:C16H24N2·HClPureza:99.77% - 99.87%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:280.84Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Fórmula:C22H23ClN2O2Pureza:99.71% - 99.98%Cor e Forma:White PowderPeso molecular:382.88PHM-27 (human) acetate
<p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>Fórmula:C137H215F3N34O42SPureza:99.20%Cor e Forma:SoildPeso molecular:3099.44Benserazide hydrochloride
CAS:<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Fórmula:C10H15N3O5·HClPureza:98.63% - 99.74%Cor e Forma:White Crystalline SolidPeso molecular:293.7Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Fórmula:C17H22ClNOPureza:99.86%Cor e Forma:White SolidPeso molecular:291.82Pheniramine maleate
CAS:<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Fórmula:C16H20N2·C4H4O4Pureza:99.85%Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Fórmula:C4H7NO2SPureza:99.99%Cor e Forma:SolidPeso molecular:133.17Tropanserin
CAS:<p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>Fórmula:C17H23NO2Pureza:99.74%Cor e Forma:SolidPeso molecular:273.37Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Fórmula:C21H27NO2Pureza:99.58%Cor e Forma:White Crystalline PowderPeso molecular:325.44Carteolol hydrochloride
CAS:<p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>Fórmula:C16H24N2O3·HClPureza:99.84% - 99.91%Cor e Forma:SolidPeso molecular:328.83Ifenprodil Tartrate
CAS:<p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>Fórmula:C21H27NO2C4H6O6Pureza:99.02% - 99.55%Cor e Forma:SolidPeso molecular:400.49

