GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
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Romifidine
CAS:Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Fórmula:C9H9BrFN3Cor e Forma:SolidPeso molecular:258.09SC 51089
CAS:SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.Fórmula:C22H20Cl2N4O3Pureza:98%Cor e Forma:SolidPeso molecular:459.338-M-PDOT
CAS:<p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>Fórmula:C14H19NO2Pureza:99.54% - 99.54%Cor e Forma:SolidPeso molecular:233.31PAF-AN-1
CAS:<p>PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.</p>Fórmula:C28H28N2O3Pureza:98.06%Cor e Forma:SolidPeso molecular:440.53Masupirdine mesylate
CAS:<p>Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease</p>Fórmula:C23H32BrN3O9S3Pureza:99.57%Cor e Forma:SolidPeso molecular:670.61MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Fórmula:C23H24F3N3O2Pureza:99.90%Cor e Forma:SolidPeso molecular:431.45GW-876167
CAS:<p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>Fórmula:C16H21N5O2Pureza:98%Cor e Forma:SolidPeso molecular:315.37AZ-GHS-22
CAS:<p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>Fórmula:C27H33ClN6O5S2Cor e Forma:SolidPeso molecular:621.17WAY 629 hydrochloride
CAS:5-HT2C agonistFórmula:C15H19ClN2Pureza:98%Cor e Forma:SolidPeso molecular:262.78RP101988
<p>RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.</p>Fórmula:C23H22N4O4Cor e Forma:SolidPeso molecular:418.45OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Fórmula:C23H28ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:413.94Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Fórmula:C22H34ClN3O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:423.98RBI-257 Maleate
CAS:<p>RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.</p>Fórmula:C25H32IN3O5Cor e Forma:SolidPeso molecular:581.44Clenproperol
CAS:<p>Clenproperol is a β2-adrenergic agonist.</p>Fórmula:C11H16Cl2N2OCor e Forma:SolidPeso molecular:263.16BPIPP
CAS:<p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>Fórmula:C22H16BrN3O3Pureza:98%Cor e Forma:SolidPeso molecular:450.28MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Fórmula:C21H19ClN2O5SCor e Forma:SolidPeso molecular:446.9PF-04628935
CAS:<p>PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.</p>Fórmula:C24H26ClN7OSPureza:98%Cor e Forma:SolidPeso molecular:496.03KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81Ksg 504
CAS:<p>Ksg 504 has superior selectivity and affinity to CCK-A receptors and derived from proglumide.</p>Fórmula:C31H49N5O8SCor e Forma:SolidPeso molecular:651.81XCC
CAS:<p>XCC is an Adenosine receptor antagonist.</p>Fórmula:C19H22N4O5Pureza:98%Cor e Forma:SolidPeso molecular:386.4JHW 007 hydrochloride
CAS:<p>JHW 007 hydrochloride is a Dopamine uptake inhibitor.</p>Fórmula:C24H30ClF2NOPureza:98%Cor e Forma:SolidPeso molecular:421.95OUP-186
CAS:<p>OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.</p>Fórmula:C19H30ClN3SCor e Forma:SolidPeso molecular:367.98Isothipendyl
CAS:Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.Fórmula:C16H19N3SCor e Forma:SolidPeso molecular:285.41(S)-Carvedilol
CAS:<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47Sortilin antagonist 1
CAS:<p>Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.</p>Fórmula:C20H24N2O4Cor e Forma:SolidPeso molecular:356.42Antiplatelet agent 1
CAS:<p>Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.</p>Fórmula:C21H24F2N6O4SCor e Forma:SolidPeso molecular:494.51ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Fórmula:C16H23ClN2O4Pureza:99.26%Cor e Forma:SolidPeso molecular:342.82CP 59430
CAS:<p>CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.</p>Fórmula:C21H22N8O3Cor e Forma:SolidPeso molecular:434.45Ranitidine bismuth citrate
CAS:<p>Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.</p>Fórmula:C19H27BiN4O10SCor e Forma:SolidPeso molecular:712.48TBC3711
CAS:<p>TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.</p>Fórmula:C20H21N3O5S2Pureza:98%Cor e Forma:SolidPeso molecular:447.53Fulimetibant
CAS:<p>Fulimetibant is a bradykinin receptor antagonist.</p>Fórmula:C25H21F4N3O3Cor e Forma:SolidPeso molecular:487.45Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Fórmula:C25H25NO6Pureza:99.809%Cor e Forma:SolidPeso molecular:435.48SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Fórmula:C18H31ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:374.97TSHR antagonist S37a
CAS:TSHR antagonist S37a is a selective, orally bioavailable TSHR antagonist that inhibits TSH-induced cAMP in TSHR-expressing HEK 293 cells.Fórmula:C25H20N2O3S2Pureza:98%Cor e Forma:SolidPeso molecular:460.57ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Fórmula:C25H31BrCl2F3N5OCor e Forma:SolidPeso molecular:625.35Guanoxabenz
CAS:<p>Guanoxabenz is an α2 adrenergic receptor agonist.</p>Fórmula:C8H8Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:247.08(2R,3R)-E1R
CAS:(2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.Fórmula:C13H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:232.28CBK289001
CAS:<p>CBK289001 inhibits TRAP 5b MV, 5b OX & 5a OX with IC50s: 125μM, 4.21μM, 14.2μM.</p>Fórmula:C19H20N6O4Cor e Forma:SolidPeso molecular:396.4MRS1097
CAS:<p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>Fórmula:C26H27NO4Pureza:98%Cor e Forma:SolidPeso molecular:417.5Prostaglandin D2
CAS:<p>Prostaglandin D2 (PGD2) is one of the major PGs actively produced in the brain of various mammals,and is a potent endogenous sleep promoting substances.</p>Fórmula:C20H32O5Pureza:>99.99%Cor e Forma:SolidPeso molecular:352.47AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Fórmula:C17H20ClN5O2SPureza:>99.99%Cor e Forma:SolidPeso molecular:393.89Clencyclohexerol
CAS:<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Fórmula:C14H20Cl2N2O2Cor e Forma:SolidPeso molecular:319.23A1AR antagonist 5
CAS:<p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>Fórmula:C17H15ClN4OCor e Forma:SolidPeso molecular:326.78Zinterol
CAS:<p>Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).</p>Fórmula:C19H26N2O4SPureza:98%Cor e Forma:SolidPeso molecular:378.49SGS518 oxalate
CAS:<p>SGS518 oxalate is a 5-HT6 antagonist.</p>Fórmula:C23H24F2N2O7SPureza:98%Cor e Forma:SolidPeso molecular:510.51Roxindole hydrochloride
CAS:<p>Dopamine D2 autoreceptor agonist</p>Fórmula:C23H27ClN2OPureza:98%Cor e Forma:SolidPeso molecular:382.93Fluphenazine Decanoate Dihydrochloride
CAS:<p>Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.</p>Fórmula:C32H46Cl2F3N3O2SPureza:98%Cor e Forma:SolidPeso molecular:664.69GLP-1R agonist 1
CAS:<p>GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.</p>Fórmula:C32H29ClFN3O5Cor e Forma:SolidPeso molecular:590.04DR4485 hydrochloride
CAS:<p>5-HT7 antagonist</p>Fórmula:C26H29Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:491.88Nafadotride
CAS:<p>Nafadotride is a dopamine D3 receptor antagonist.</p>Fórmula:C22H27N3O2Cor e Forma:SolidPeso molecular:365.47Midodrine D6 hydrochloride
CAS:<p>Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.</p>Fórmula:C12H19ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:296.78JPC-211
CAS:<p>JPC-211 is an agonist of dopamine-receptor.</p>Fórmula:C17H27NO2Pureza:98%Cor e Forma:SolidPeso molecular:277.4A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Fórmula:C17H12N4OCor e Forma:SolidPeso molecular:288.3COR 170
CAS:<p>inverse agonist of CB2 receptors</p>Fórmula:C31H36N2O2Pureza:98%Cor e Forma:SolidPeso molecular:468.63U-101958 Maleate
CAS:<p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>Fórmula:C25H33N3O5Pureza:98%Cor e Forma:SolidPeso molecular:455.55Iloperidone hydrochloride
CAS:<p>Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.</p>Fórmula:C24H28ClFN2O4Pureza:98%Cor e Forma:SolidPeso molecular:462.95ML233
CAS:<p>"ML233: potent apelin receptor agonist, EC50=3.7 μM, 21-fold selective over AT1 receptor."</p>Fórmula:C19H21NO4SCor e Forma:SolidPeso molecular:359.44Ketotifen
CAS:<p>Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.</p>Fórmula:C19H19NOSCor e Forma:SolidPeso molecular:309.43CB1/2 agonist 2
CAS:<p>CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.</p>Fórmula:C26H43NO3Cor e Forma:SolidPeso molecular:417.62BMS-192364
CAS:<p>BMS-192364 is a bio-active chemical.</p>Fórmula:C15H9ClF3N3O2Cor e Forma:SolidPeso molecular:355.70AF40431
CAS:AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 μM; Kd: 0.7 μM). AF40431 is bound in the neurotensin-binding site of sortilin.Fórmula:C17H21NO5Cor e Forma:SolidPeso molecular:319.35GTS-21
CAS:<p>GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.</p>Fórmula:C19H20N2O2Pureza:98%Cor e Forma:SolidPeso molecular:308.37Pitolisant oxalate
CAS:<p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C19H28ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:385.88WAY 161503 hydrochloride
CAS:<p>WAY 161503 hydrochloride is a 5-HT2C receptor agonist.</p>Fórmula:C11H12Cl3N3OPureza:98%Cor e Forma:SolidPeso molecular:308.59UCM710
CAS:<p>UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).</p>Fórmula:C19H34O3Pureza:98%Cor e Forma:SolidPeso molecular:310.47SKF-83822
CAS:<p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>Fórmula:C20H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:343.85Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Fórmula:C31H56N2O8SPureza:98%Cor e Forma:SolidPeso molecular:616.85RWJ 52353
CAS:<p>α2D adrenergic receptor agonist</p>Fórmula:C11H10N2SPureza:98%Cor e Forma:SolidPeso molecular:202.28(Rac)-E1R
CAS:<p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>Fórmula:C13H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:232.28Fenmetozole HCl
CAS:<p>Fenmetozole HCl is an antagonist of the actions of ethanol. It attenuates the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate content.</p>Fórmula:C10H11Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:281.57GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Fórmula:C21H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:387.9Abanoquil
CAS:Abanoquil is an antagonist of alpha-1 adrenoceptor.Fórmula:C22H25N3O4Cor e Forma:SolidPeso molecular:395.45MRGPRX4 modulator-1
CAS:<p>MRGPRX4 modulator-1 (compound 31-2), potent MRGPR X4 antagonist, IC50 < 100nM, for itch, pain, autoimmune research.</p>Fórmula:C16H13ClF3NO3Cor e Forma:SolidPeso molecular:359.73Tiamenidine
CAS:<p>Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.</p>Fórmula:C8H10ClN3SPureza:98%Cor e Forma:SolidPeso molecular:215.7JMV3002
CAS:<p>JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.</p>Fórmula:C35H34N6O3Cor e Forma:SolidPeso molecular:586.68Resomelagon
CAS:<p>Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.</p>Fórmula:C14H14N6O2Cor e Forma:SolidPeso molecular:298.3ONO-2952
CAS:<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Fórmula:C22H20ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.86S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSCor e Forma:SolidPeso molecular:337.87Pirolate
CAS:<p>Pirolate is a receptor of histamine H1.</p>Fórmula:C16H15N3O5Pureza:98%Cor e Forma:SolidPeso molecular:329.31Panamesine
CAS:<p>Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.</p>Fórmula:C23H26N2O6Cor e Forma:SolidPeso molecular:426.46(-)-S-Timolol
CAS:<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Fórmula:C13H26N4O4SCor e Forma:SolidPeso molecular:334.44L-733060 hydrochloride
CAS:<p>Potent NK1 antagonist</p>Fórmula:C20H20ClF6NOPureza:98%Cor e Forma:SolidPeso molecular:439.82Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Fórmula:C25H26F2N8O4S2Cor e Forma:SolidPeso molecular:604.65A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Fórmula:C32H24N4O4SCor e Forma:SolidPeso molecular:560.62Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Fórmula:C20H21NO5Cor e Forma:SolidPeso molecular:355.38R 121919 hydrochloride
CAS:<p>CRF1 antagonist with Ki=3.5 nM, lowers stress-induced ACTH, has anxiolytic and antidepressant effects, orally bioavailable.</p>Fórmula:C22H33ClN6Cor e Forma:SolidPeso molecular:417.0L 760735
CAS:<p>L 760735 is a NK1 receptor antagonist.</p>Fórmula:C26H29ClF7N5O2Pureza:98%Cor e Forma:SolidPeso molecular:611.98TC-2153
CAS:<p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>Fórmula:C7H5ClF3NS5Cor e Forma:SolidPeso molecular:355.89FR 64822
CAS:<p>FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.</p>Fórmula:C11H14N4OCor e Forma:SolidPeso molecular:218.26LY 344864 hydrochloride
CAS:<p>LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor.</p>Fórmula:C21H23ClFN3OCor e Forma:SolidPeso molecular:387.88CM572
CAS:<p>CM572 is a selective putative sigma-2 antagonist.</p>Fórmula:C22H23FN4O2SCor e Forma:SolidPeso molecular:426.51IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SCor e Forma:SolidPeso molecular:373.51L 648051
CAS:<p>L 648051 is a leukotriene D4 receptor antagonist.</p>Fórmula:C24H28O8SPureza:98%Cor e Forma:SolidPeso molecular:476.54JNJ-28610244
CAS:<p>JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.</p>Fórmula:C16H21N3OPureza:98%Cor e Forma:SolidPeso molecular:271.36Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Cor e Forma:SolidPeso molecular:255.74A1AR antagonist 3
CAS:<p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>Fórmula:C25H20N2O3SCor e Forma:SolidPeso molecular:428.5EP1-antagonist-1
CAS:<p>EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).</p>Fórmula:C19H15BrCl2N2O3Pureza:97.06%Cor e Forma:SolidPeso molecular:470.14CAY10680
CAS:<p>CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.</p>Fórmula:C18H16N2O2SCor e Forma:SolidPeso molecular:324.4
