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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • N6-Ethyladenosine

    CAS:
    <p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>
    Fórmula:C12H17N5O4
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:295.29
  • Azelastine hydrochloride

    CAS:
    <p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>
    Fórmula:C22H24ClN3O·HCl
    Pureza:98% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:418.36
  • (S)-(-)-Atenolol

    CAS:
    <p>(S)-(-)-Atenolol has beta-adrenergic blocking effects.</p>
    Fórmula:C14H22N2O3
    Pureza:99.31% - 99.81%
    Cor e Forma:Solid
    Peso molecular:266.34
  • Lamotrigine

    CAS:
    <p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>
    Fórmula:C9H7Cl2N5
    Pureza:99.76% - 99.95%
    Cor e Forma:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Peso molecular:256.09
  • DREADD agonist 21

    CAS:
    <p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>
    Fórmula:C17H18N4
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:278.35
  • Centanafadine hydrochloride

    CAS:
    Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).
    Fórmula:C15H16ClN
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:245.75
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Fórmula:C25H28N2O5S
    Pureza:97.09%
    Cor e Forma:Solid
    Peso molecular:468.57
  • GANT 58

    CAS:
    <p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>
    Fórmula:C24H16N4S
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:392.48
  • PHM-27 (human) acetate


    <p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>
    Fórmula:C137H215F3N34O42S
    Pureza:99.20%
    Cor e Forma:Soild
    Peso molecular:3099.44
  • Molindone hydrochloride

    CAS:
    <p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>
    Fórmula:C16H24N2O2·HCl
    Pureza:99% - 99.99%
    Cor e Forma:Solid
    Peso molecular:312.84
  • Ogerin

    CAS:
    <p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>
    Fórmula:C17H17N5O
    Pureza:99.5% - 99.75%
    Cor e Forma:Solid
    Peso molecular:307.35
  • NS-2028

    CAS:
    <p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>
    Fórmula:C9H5BrN2O3
    Pureza:99.44%
    Cor e Forma:A Crystalline Solid
    Peso molecular:269.05
  • Vabicaserin hydrochloride

    CAS:
    <p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>
    Fórmula:C15H21ClN2
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:264.79
  • Iloperidone

    CAS:
    <p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>
    Fórmula:C24H27FN2O4
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:426.48
  • Isoprenaline hydrochloride

    CAS:
    <p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>
    Fórmula:C11H18ClNO3
    Pureza:98% - 99.65%
    Cor e Forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Peso molecular:247.719
  • Roluperidone

    CAS:
    <p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>
    Fórmula:C22H23FN2O2
    Pureza:96.46% - 97.77%
    Cor e Forma:Solid
    Peso molecular:366.43
  • Vibozilimod

    CAS:
    <p>Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .</p>
    Fórmula:C29H36ClN3O5
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:542.07
  • p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Fórmula:C25H28ClIN4O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:578.87
  • Isoxsuprine hydrochloride

    CAS:
    <p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>
    Fórmula:C18H24ClNO3
    Pureza:99.38%
    Cor e Forma:Crystals From Water Solid
    Peso molecular:337.84
  • Sertraline hydrochloride

    CAS:
    <p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>
    Fórmula:C17H18Cl3N
    Pureza:99.12% - 99.89%
    Cor e Forma:Solid Powder
    Peso molecular:342.691
  • Latanoprostene bunod

    CAS:
    <p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>
    Fórmula:C27H41NO8
    Pureza:99.33% - 99.69%
    Cor e Forma:Solid
    Peso molecular:507.62
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Fórmula:C11H16BrCl2N
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:313.06
  • Benserazide hydrochloride

    CAS:
    <p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>
    Fórmula:C10H15N3O5·HCl
    Pureza:98.63% - 99.74%
    Cor e Forma:White Crystalline Solid
    Peso molecular:293.7
  • Dipivefrin hydrochloride

    CAS:
    <p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>
    Fórmula:C19H27NO5·HCl
    Pureza:99.22% - 99.92%
    Cor e Forma:Less Gas With A Sweet Odor Colorless Gas With A Sweet Odor
    Peso molecular:387.9
  • AM095 free acid

    CAS:
    <p>AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).</p>
    Fórmula:C27H24N2O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:456.49
  • Ornidazole

    CAS:
    <p>Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.</p>
    Fórmula:C7H10ClN3O3
    Pureza:99.47%
    Cor e Forma:Crystalline Solid
    Peso molecular:219.63
  • Cimetidine

    CAS:
    <p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>
    Fórmula:C10H16N6S
    Pureza:99.82%
    Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Peso molecular:252.34
  • Mianserin hydrochloride

    CAS:
    <p>Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.</p>
    Fórmula:C18H21ClN2
    Pureza:99.63% - 99.82%
    Cor e Forma:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
    Peso molecular:300.83
  • PIT

    CAS:
    <p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>
    Fórmula:C20H16N2O5S
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:396.42
  • Promethazine

    CAS:
    <p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>
    Fórmula:C17H20N2S
    Pureza:99.76%
    Cor e Forma:Crystals
    Peso molecular:284.42
  • Cloperastine hydrochloride

    CAS:
    <p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>
    Fórmula:C20H25Cl2NO
    Pureza:97.74% - 99.42%
    Cor e Forma:Solid
    Peso molecular:366.33
  • Talipexole dihydrochloride

    CAS:
    <p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>
    Fórmula:C10H17Cl2N3S
    Pureza:99.89%
    Cor e Forma:Light Yellow Solid
    Peso molecular:282.23
  • Tipepidine hydrochloride

    CAS:
    <p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>
    Fórmula:C15H18ClNS2
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:311.89
  • Avexitide acetate

    CAS:
    <p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>
    Fórmula:C155H246N40O53S
    Pureza:96.64% - 98.65%
    Cor e Forma:Solid
    Peso molecular:3549.91
  • Rebamipide

    CAS:
    <p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>
    Fórmula:C19H15ClN2O4
    Pureza:99.48% - 99.61%
    Cor e Forma:White Powder
    Peso molecular:370.79
  • Tolnaftate

    CAS:
    <p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>
    Fórmula:C19H17NOS
    Pureza:98.85%
    Cor e Forma:White Powder
    Peso molecular:307.41
  • Midodrine hydrochloride

    CAS:
    <p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>
    Fórmula:C12H19ClN2O4
    Pureza:99.79% - >99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:290.74
  • Abarelix

    CAS:
    <p>Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.</p>
    Fórmula:C72H95ClN14O14
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1416.06
  • Pramipexole

    CAS:
    <p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>
    Fórmula:C10H17N3S
    Pureza:98% - 99.96%
    Cor e Forma:Solid
    Peso molecular:211.33
  • Clomipramine hydrochloride

    CAS:
    <p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>
    Fórmula:C19H23ClN2·HCl
    Pureza:99.04% - 99.47%
    Cor e Forma:White To Slightly Yellow Crystalline Powder
    Peso molecular:351.31
  • Mizolastine

    CAS:
    <p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>
    Fórmula:C24H25FN6O
    Pureza:98% - 99.75%
    Cor e Forma:Solid
    Peso molecular:432.49
  • Delequamine

    CAS:
    <p>Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.</p>
    Fórmula:C18H26N2O3S
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:350.48
  • Sulpiride

    CAS:
    <p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>
    Fórmula:C15H23N3O4S
    Pureza:99.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:341.43
  • Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.64% - 99.98%
    Cor e Forma:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Peso molecular:390.87
  • L-741626

    CAS:
    <p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>
    Fórmula:C20H21ClN2O
    Pureza:98.57%
    Cor e Forma:Solid
    Peso molecular:340.85
  • SBI-477

    CAS:
    <p>SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.</p>
    Fórmula:C24H25N3O6S
    Pureza:99.3%
    Cor e Forma:Solid
    Peso molecular:483.54
  • Amylin, amide, human

    CAS:
    <p>Amylin, amide, human(DAP Amide) is a 37-amino acid peptide hormone co-secreted with insulin to regulate postprandial glucose levels.</p>
    Fórmula:C165H261N51O55S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3903.28
  • ONC206

    CAS:
    <p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>
    Fórmula:C23H22F2N4O
    Pureza:99.38% - 99.81%
    Cor e Forma:Solid
    Peso molecular:408.44
  • CCX140

    CAS:
    <p>CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.</p>
    Fórmula:C20H13ClF3N5O3S
    Pureza:99.66% - 99.95%
    Cor e Forma:Solid
    Peso molecular:495.86
  • Azasetron hydrochloride

    CAS:
    <p>Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.</p>
    Fórmula:C17H20ClN3O3·HCl
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:386.27
  • Asenapine Maleate

    CAS:
    <p>Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.</p>
    Fórmula:C21H20ClNO5
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:401.84
  • Balovaptan

    CAS:
    <p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>
    Fórmula:C22H24ClN5O
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Betaxolol hydrochloride

    CAS:
    <p>Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.</p>
    Fórmula:C18H30ClNO3
    Pureza:99.48% - 99.56%
    Cor e Forma:Solid
    Peso molecular:343.89
  • ML-109

    CAS:
    <p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>
    Fórmula:C31H29N3O5
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:523.58
  • Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Fórmula:C36H51Cl2N3O4
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:660.71
  • CCR2-RA-[R]

    CAS:
    <p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>
    Fórmula:C18H19ClFNO3
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:351.8
  • PF-04995274

    CAS:
    <p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>
    Fórmula:C23H32N2O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:432.51
  • Tropisetron hydrochloride

    CAS:
    <p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>
    Fórmula:C17H21ClN2O2
    Pureza:99.72% - 99.83%
    Cor e Forma:Solid
    Peso molecular:320.82
  • Promethazine hydrochloride

    CAS:
    <p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>
    Fórmula:C17H20N2S·HCl
    Pureza:99.85%
    Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Peso molecular:320.88
  • Risperidone

    CAS:
    <p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>
    Fórmula:C23H27FN4O2
    Pureza:99.73%
    Cor e Forma:Crystalline Solid
    Peso molecular:410.48
  • Ethamsylate

    CAS:
    <p>Ethamsylate (Dicynene) 通常用作止血药,增加毛细血管内皮阻力和血小板粘附,抑制前列腺素的生物合成和作用。</p>
    Fórmula:C10H17NO5S
    Pureza:98.55%
    Cor e Forma:White Crystals Or Crystalline Powder
    Peso molecular:263.31
  • Ziprasidone hydrochloride monohydrate

    CAS:
    <p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>
    Fórmula:C21H21ClN4OS·HCl·H2O
    Pureza:98% - 99.83%
    Cor e Forma:Off-White Powder
    Peso molecular:467.12
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Fórmula:C21H27NO2C4H6O6
    Pureza:99.02% - 99.55%
    Cor e Forma:Solid
    Peso molecular:400.49
  • AB928

    CAS:
    <p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>
    Fórmula:C23H22N8O
    Pureza:98.09% - >99.99%
    Cor e Forma:Solid
    Peso molecular:426.47
  • Flunarizine dihydrochloride

    CAS:
    <p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>
    Fórmula:C26H28Cl2F2N2
    Pureza:99.53% - 99.89%
    Cor e Forma:White Crystalline Powder Odorless And Tasteless
    Peso molecular:477.42
  • Clopidogrel hydrogen sulfate

    CAS:
    <p>Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.</p>
    Fórmula:C16H16ClNO2S·H2SO4
    Pureza:99.57% - 99.79%
    Cor e Forma:Solid
    Peso molecular:419.9
  • Tetrabenazine

    CAS:
    <p>Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.</p>
    Fórmula:C19H27NO3
    Pureza:98% - 99.91%
    Cor e Forma:White To Off-White White To Off-White Solid
    Peso molecular:317.42
  • Levocetirizine

    CAS:
    <p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>
    Fórmula:C21H25ClN2O3
    Pureza:98% - 99.9%
    Cor e Forma:White Powder
    Peso molecular:388.89
  • Olopatadine hydrochloride

    CAS:
    <p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>
    Fórmula:C21H23NO3·HCl
    Pureza:99.62% - 99.64%
    Cor e Forma:White Solid
    Peso molecular:373.87
  • REV 5901A

    CAS:
    <p>REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in mice</p>
    Fórmula:C22H26ClNO2
    Pureza:98.04%
    Cor e Forma:Soild
    Peso molecular:371.90
  • Capeserod

    CAS:
    <p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>
    Fórmula:C23H25ClN4O4
    Pureza:98.10% - 99.94%
    Cor e Forma:Solid
    Peso molecular:456.92
  • Phenoxybenzamine hydrochloride

    CAS:
    <p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>
    Fórmula:C18H23Cl2NO
    Pureza:98.04% - >99.99%
    Cor e Forma:Antihypertensive Drug
    Peso molecular:340.3
  • Orphenadrine hydrochloride

    CAS:
    <p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>
    Fórmula:C18H23NO·HCl
    Pureza:99.88%
    Cor e Forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)
    Peso molecular:305.85
  • Ziprasidone

    CAS:
    <p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>
    Fórmula:C21H21ClN4OS
    Pureza:99.55%
    Cor e Forma:Tan Solid
    Peso molecular:412.94
  • Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Fórmula:C22H23ClN2O2
    Pureza:99.71% - 99.98%
    Cor e Forma:White Powder
    Peso molecular:382.88
  • Lintopride HCl

    CAS:
    <p>Lintopride HCl is a 5HT-4 antagonist.</p>
    Fórmula:C14H20Cl2N4O2
    Pureza:98.42% - 98.81%
    Cor e Forma:Soild
    Peso molecular:347.24
  • Carvedilol EP IMpurity E

    CAS:
    <p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>
    Fórmula:C9H14ClNO2
    Pureza:99.53%
    Cor e Forma:White To Almost White Solid Crystalline
    Peso molecular:203.666
  • Carbinoxamine Maleate Salt

    CAS:
    <p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>
    Fórmula:C20H23ClN2O5
    Pureza:99.97%
    Cor e Forma:Off-White Solid
    Peso molecular:406.86
  • INCB-9471

    CAS:
    <p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>
    Fórmula:C30H40F3N5O2
    Pureza:98.80%
    Cor e Forma:Solid
    Peso molecular:559.666
  • YT 146

    CAS:
    <p>YT 146 is a biochemical.</p>
    Fórmula:C18H25N5O4
    Pureza:98.81% - 99.25%
    Cor e Forma:Solid
    Peso molecular:375.42
  • Mirtazapine

    CAS:
    <p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>
    Fórmula:C17H19N3
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Evocalcet

    CAS:
    <p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>
    Fórmula:C24H26N2O2
    Pureza:98.88% - 99.68%
    Cor e Forma:Solid
    Peso molecular:374.48
  • J-113863

    CAS:
    <p>J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).</p>
    Fórmula:C30H37Cl2IN2O2
    Pureza:95.11%
    Cor e Forma:Solid
    Peso molecular:655.44
  • Ramelteon

    CAS:
    <p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>
    Fórmula:C16H21NO2
    Pureza:97.21% - 99.92%
    Cor e Forma:Crystalline Solid
    Peso molecular:259.34
  • Efloxate

    CAS:
    <p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>
    Fórmula:C19H16O5
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:324.33
  • Degarelix acetate(214766-78-6 free base)

    CAS:
    <p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>
    Fórmula:C84H107ClN18O18
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:1692.34
  • MK-0812 Succinate

    CAS:
    <p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>
    Fórmula:C28H40F3N3O7
    Pureza:98.62% - 99.93%
    Cor e Forma:Solid
    Peso molecular:587.63
  • S1P2 antagonist 1

    CAS:
    <p>S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.</p>
    Fórmula:C23H21ClN4O4
    Cor e Forma:Solid
    Peso molecular:452.9
  • (D-Trp6)-LHRH free acid

    CAS:
    (D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .
    Fórmula:C64H81N17O14
    Peso molecular:1312.43
  • NPFF2-R ligand 1


    <p>NPFF2-R ligand 1 (Compound 16a) is an NPFF2-R ligand with Ki values of 228 nM for NPFF1-R and 27 nM for NPFF2-R, and can be utilized in research on central nervous system-related disorders.</p>
    Fórmula:C32H41N3O
    Peso molecular:483.32496
  • Adrenomedullin (16-31), human TFA


    Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.
    Fórmula:C84H130F3N25O23S2
    Cor e Forma:Solid
    Peso molecular:1979.21
  • [D-Trp8,Tyr11] Somatostatin

    CAS:
    [D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,
    Fórmula:C76H104N18O20S2
    Peso molecular:1653.88
  • Anthramycin

    CAS:
    <p>Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.</p>
    Fórmula:C16H17N3O4
    Cor e Forma:Solid
    Peso molecular:315.32
  • [8-L-arginine] deaminovasopressin

    CAS:
    <p>[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .</p>
    Fórmula:C46H64N14O13S2
    Cor e Forma:Solid
    Peso molecular:1085.22
  • LysoPalloT-NH-amide-C3-ph-m-O-C11

    CAS:
    <p>LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.</p>
    Fórmula:C27H47N2O9P
    Cor e Forma:Solid
    Peso molecular:574.64
  • Calcitonin (8-32), salmon

    CAS:
    <p>Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.</p>
    Fórmula:C119H198N36O37
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2725.06
  • CB2R/FAAH modulator-2

    CAS:
    <p>CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.</p>
    Fórmula:C24H33NO2
    Pureza:99.15%
    Cor e Forma:Soild
    Peso molecular:367.52
  • LH-RH (7-10)

    CAS:
    LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.
    Fórmula:C19H36N8O4
    Cor e Forma:Solid
    Peso molecular:440.54
  • BIM-23190 hydrochloride


    <p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>
    Cor e Forma:Liquid
  • Galanin (1-29)(rat, mouse)

    CAS:
    <p>Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.</p>
    Fórmula:C141H211N43O41
    Pureza:98%
    Cor e Forma:White Lyophilized Powder
    Peso molecular:3164.499