GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Mapenterol hydrochloride
CAS:<p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>Fórmula:C14H21Cl2F3N2OPureza:98.11% - 99.98%Cor e Forma:SolidPeso molecular:361.23Cortistatin-8
CAS:<p>ghrelin receptor antagonist</p>Fórmula:C47H68N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1009.25L-796,778 acetate
<p>L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.</p>Fórmula:C31H44N6O9Pureza:98%Cor e Forma:SoildPeso molecular:644.72Vedaprofen
CAS:<p>Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.</p>Fórmula:C19H22O2Pureza:99.24% - 99.70%Cor e Forma:SolidPeso molecular:282.38PF-07062119
<p>PF-07062119 is a humanized immunoglobulin G1 (IgG1) monoclonal antibody designed to target and inhibit GUCY2C.</p>Cor e Forma:Odour LiquidPACAP (1-38) free acid
CAS:<p>PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.</p>Cor e Forma:SolidBAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Fórmula:C26H28BrCl2N3O3Cor e Forma:SolidPeso molecular:581.33Tafluprost acid
CAS:<p>Tafluprost acid is a selective agonist at the prostaglandin F receptor.</p>Fórmula:C22H28F2O5Cor e Forma:SolidPeso molecular:410.46Tafluprost ethyl amide
CAS:<p>Tafluprost ethyl amide is a prostaglandin derivative.</p>Fórmula:C24H33F2NO4Cor e Forma:SolidPeso molecular:437.52Neuropeptide Y (1-24) (human)
CAS:Neuropeptide Y (1-24) inhibits rat vas deferens twitch and activates NMDA-induced neurons in rat hippocampus.Fórmula:C116H170N30O40SPeso molecular:2656.83Preclamol hydrochloride
CAS:<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Fórmula:C14H22ClNOCor e Forma:SolidPeso molecular:255.78Suntinorexton
CAS:<p>Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.</p>Fórmula:C23H28F2N2O4SPureza:99.89%Cor e Forma:SolidPeso molecular:466.54Galanin (1-30), human
CAS:Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Fórmula:C139H210N42O43Pureza:98%Cor e Forma:SolidPeso molecular:3157.46CCR8 antagonist 1
CAS:<p>CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.</p>Fórmula:C26H29N3O5SPureza:99.51%Cor e Forma:SolidPeso molecular:495.59Desglymidodrine
CAS:<p>Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.</p>Fórmula:C10H15NO3Pureza:99.56%Cor e Forma:SolidPeso molecular:197.23Femoxetine
CAS:<p>Femoxetine: antidepressant, enhances morphine, inhibits MAO-A/B, boosts mice's exercise capacity.</p>Fórmula:C20H25NO2Pureza:99.1% - 99.35%Cor e Forma:SolidPeso molecular:311.42Israpafant
CAS:<p>Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.</p>Fórmula:C28H29ClN4SCor e Forma:SolidPeso molecular:489.07Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Fórmula:C22H27ClN2O3Cor e Forma:SolidPeso molecular:402.91Atrial natriuretic factor (1-28) (rat) TFA
<p>ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.</p>Fórmula:C130H206N45F3O41S2Pureza:98%Cor e Forma:SolidPeso molecular:3176.43Benzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Fórmula:C22H32N2O5Pureza:94.86%Cor e Forma:SolidPeso molecular:404.5Tryptamine hydrochloride
CAS:<p>Tryptamine hydrochloride is a monoamine alkaloid, metabolite of tryptophan and CNS active substance, agonist of 5-HT4 receptor, TAAR1, AHR.</p>Fórmula:C10H13ClN2Pureza:99.89%Cor e Forma:SolidPeso molecular:196.68Methicillin sodium hydrate
CAS:<p>Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.</p>Fórmula:C17H21N2NaO7SCor e Forma:SolidPeso molecular:420.41Substance P (4-11)
CAS:Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.Fórmula:C46H67N11O10SCor e Forma:SolidPeso molecular:966.16Propranolol hydrochloride
CAS:<p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>Fórmula:C16H22ClNO2Pureza:99.94% - >99.99%Cor e Forma:White Or Almost White Powder White PowderPeso molecular:295.80Utreglutide
CAS:<p>Utreglutide is a potent glucagon-like peptide 1 (GLP-1) receptor agonit [1] .</p>Fórmula:C191H298N46O58Cor e Forma:SolidPeso molecular:4166.67σ1 Receptor ligand 1
σ1 Receptor ligand 1 (compound 5I) is a σ1 receptor ligand with a Ki value of 3.9 nM. It demonstrates a high plasma protein binding rate (89%) and exhibits good metabolic stability in the presence of mouse liver microsomes and NADPH. σ1 Receptor ligand 1 is applicable in neuroscience and cancer research.Fórmula:C22H28N2O2Cor e Forma:SolidPeso molecular:352.47RFRP-3(human)
CAS:<p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>Fórmula:C45H72N14O10Pureza:98%Cor e Forma:SolidPeso molecular:969.15α1A-AR Degrader 9c
CAS:<p>α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.</p>Fórmula:C38H43N11O11Pureza:98%Cor e Forma:SolidPeso molecular:829.82Synephrine hemitartrate
CAS:<p>Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.</p>Fórmula:C9H13NO2C4H6O6Cor e Forma:SolidPeso molecular:242.26CB1R antagonist 2
<p>CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.</p>Fórmula:C24H26N4OCor e Forma:SolidPeso molecular:386.49d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Fórmula:C52H72F3N13O13S2Cor e Forma:SolidPeso molecular:1208.33Apraglutide
CAS:Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.Fórmula:C172H263N43O52Pureza:98%Cor e Forma:SolidPeso molecular:3765.25Kisspeptin-10, human
CAS:<p>Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.</p>Fórmula:C63H83N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1302.462JNJ-10181457 (hydrochloride)
CAS:<p>JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations</p>Fórmula:C20H30Cl2N2OCor e Forma:SolidPeso molecular:385.377-Hydroxy-PIPAT maleate
CAS:<p>7-Hydroxy-PIPAT maleate is a D3R agonist.</p>Fórmula:C16H22INOCor e Forma:SolidPeso molecular:371.262GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Fórmula:C165H254N44O55SPureza:98%Cor e Forma:SolidPeso molecular:3766.19Exendin-3/4 (59-86)
<p>Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.</p>Fórmula:NAPureza:98%Cor e Forma:SolidPeso molecular:3055.49β-CGRP (mouse)
<p>β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.</p>Fórmula:C165H265N49O55S2Cor e Forma:SolidPeso molecular:3879.29Endothelin 1 (swine, human), Alexa Fluor 488-labeled
<p>Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.</p>Cor e Forma:SolidPeso molecular:2848.4(Iso)-RJW100
CAS:<p>Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).</p>Fórmula:C28H34OPureza:99.79%Cor e Forma:SoildPeso molecular:386.57LP 12 hydrochloride
CAS:<p>LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).</p>Fórmula:C32H40ClN3OCor e Forma:SolidPeso molecular:518.14GLP-1 receptor agonist 8
CAS:<p>GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.</p>Fórmula:C34H36ClFN6O4Cor e Forma:SolidPeso molecular:647.14NESS 0327
CAS:<p>NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.</p>Fórmula:C24H23Cl3N4OPureza:99.78%Cor e Forma:SolidPeso molecular:489.82CCK Octapeptide, non-sulfated acetate
<p>CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.</p>Fórmula:C51H66N10O15S2Pureza:98.9700%Cor e Forma:SolidPeso molecular:1123.26Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Fórmula:C22H26O4Cor e Forma:SolidPeso molecular:354.446Minaprine
CAS:<p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>Fórmula:C17H22N4OPureza:98%Cor e Forma:SolidPeso molecular:298.388-iso Prostaglandin E1
CAS:<p>8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.</p>Fórmula:C20H34O5Cor e Forma:Light Yellow Crystalline SolidPeso molecular:354.48SGLT1/2-IN-2
CAS:<p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>Fórmula:C23H26F2O7Cor e Forma:SolidPeso molecular:452.451CRF(6-33)(human)
CAS:<p>CRFBP inhibitor peptide; blocks CRF, reduces weight gain, boosts activity in obese rats.</p>Fórmula:C141H231N41O43SPureza:98%Cor e Forma:SolidPeso molecular:3220.68Jmv 179
CAS:<p>Jmv 179 is an antagonist of the cholecystokinin receptor.</p>Fórmula:C51H67N7O15SCor e Forma:SolidPeso molecular:1050.19LysoPalloT-NH-amide-C3-ph-m-O-C11
CAS:<p>LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.</p>Fórmula:C27H47N2O9PCor e Forma:SolidPeso molecular:574.64Oxatomide
CAS:<p>Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).</p>Fórmula:C27H30N4OPureza:98.82% - 99.72%Cor e Forma:White PowderPeso molecular:426.55RS 56812
CAS:<p>RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.</p>Fórmula:C18H21N3O2Pureza:99.38%Cor e Forma:SoildPeso molecular:311.38Vazegepant
CAS:<p>Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.</p>Fórmula:C36H46N8O3Pureza:98.61%Cor e Forma:SolidPeso molecular:638.8020-Carboxy-Leukotriene B4
CAS:<p>20-COOH LTB4, a metabolite of LTB4, binds BLT1 receptor and inhibits LTB4-induced neutrophil responses.</p>Fórmula:C20H30O6Cor e Forma:SolidPeso molecular:366.45Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:<p>Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.</p>Fórmula:C25H26O13Cor e Forma:SolidPeso molecular:534.47Secretoneurin, rat
CAS:<p>Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).</p>Fórmula:C159H252N40O58Pureza:98%Cor e Forma:SolidPeso molecular:3651.95NSC380324
<p>NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.</p>Fórmula:C31H24N4O4Cor e Forma:SolidPeso molecular:516.55Glucagon (19-29), human
CAS:Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Fórmula:C61H89N15O18SPureza:98%Cor e Forma:SolidPeso molecular:1352.53Nα-Methylhistamine FA
<p>Nα-Methylhistamine FA is a histamine H3 receptor agonist</p>Fórmula:C7H13N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:171.2NXT-10796
<p>NXT-10796 is an orally active, intestinally restricted agonist of the EP4 receptor [1].</p>Fórmula:C23H31N3O6Pureza:98%Cor e Forma:SolidPeso molecular:445.51GLP-1 (9-36) amide
CAS:<p>GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.</p>Fórmula:C140H214N36O43Pureza:97%Cor e Forma:SolidPeso molecular:3089.41DETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Fórmula:C22H25Cl2NO3Cor e Forma:SolidPeso molecular:422.34BMS-193885
CAS:<p>BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.</p>Fórmula:C33H42N4O6Pureza:99.73%Cor e Forma:SolidPeso molecular:590.71γ-1-Melanocyte Stimulating Hormone (MSH), amide
<p>γ-1-Melanocyte Stimulating Hormone (MSH), amide, a peptide consisting of 11 amino acids, plays a critical role in regulating sodium (Na+) balance and blood</p>Fórmula:C72H97N21O14SCor e Forma:SolidPeso molecular:1512.9LHRH, Ala(6)-
CAS:<p>LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.</p>Fórmula:C56H77N17O13Cor e Forma:SolidPeso molecular:1196.32MRS7925
<p>MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosis</p>Fórmula:C20H26IN5O3Pureza:98%Cor e Forma:SolidPeso molecular:511.36[D-Pro2] Spantide I TFA
<p>[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].</p>Fórmula:C75H108N20O13·xC2HF3O2Pureza:98%Cor e Forma:SolidLHRH
CAS:<p>Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and has</p>Fórmula:C55H74N16O14Pureza:98%Cor e Forma:SolidPeso molecular:1183.27CB2R agonist 3
<p>CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [</p>Pureza:98%Cor e Forma:Odour SolidTetrapeptide-1
CAS:<p>Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].</p>Fórmula:C20H36N4O6Pureza:98%Cor e Forma:SolidPeso molecular:428.52Zoliprofen
CAS:<p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.29Neocarzinostatin
CAS:<p>Neocarzinostatin is an effective DNA-damaging, anti-tumor antibiotic.</p>Pureza:98%Cor e Forma:SolidPeso molecular:N/ATT 232
CAS:<p>sst1/sst4 somatostatin receptors agonist</p>Fórmula:C45H58N10O9S2Pureza:98%Cor e Forma:SolidPeso molecular:947.13α-CGRP (mouse, rat) TFA
<p>α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and</p>Fórmula:C162H262N50O52S2·C2HF3O2Pureza:98%Cor e Forma:SolidFFN246
CAS:<p>FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and</p>Fórmula:C15H13FN2OPureza:98%Cor e Forma:SolidPeso molecular:256.27Sigma-1 receptor antagonist 5
<p>Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors</p>Fórmula:C26H27N3OPureza:98%Cor e Forma:SolidPeso molecular:397.51Galanin-Like Peptide (rat)
CAS:<p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>Fórmula:C288H461N87O83SPureza:98%Cor e Forma:SolidPeso molecular:6502.34JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23Vapiprost
CAS:<p>Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.</p>Fórmula:C30H39NO4Pureza:98%Cor e Forma:SolidPeso molecular:477.64Rubraxanthone
CAS:<p>Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.</p>Fórmula:C24H26O6Cor e Forma:SolidPeso molecular:410.466FGH31
<p>FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].</p>Fórmula:C33H36N4O2Pureza:98%Cor e Forma:SolidPeso molecular:520.66A 76154
CAS:<p>A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).</p>Fórmula:C70H93FN12O12Cor e Forma:SolidPeso molecular:1313.584L-779976
CAS:<p>L-779,976 is an agonist of somatostatin receptor.</p>Fórmula:C33H43N7O3Cor e Forma:SolidPeso molecular:585.74Vapreotide
CAS:<p>Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).</p>Fórmula:C57H70N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1131.38MCL0129
CAS:<p>MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.</p>Fórmula:C34H47FN4OPureza:98%Cor e Forma:SolidPeso molecular:546.764-Methylhistamine
CAS:<p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>Fórmula:C6H11N3Pureza:98%Cor e Forma:SolidPeso molecular:125.17Conopeptide rho-TIA
CAS:<p>Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive</p>Fórmula:C105H160N36O21S4Pureza:98%Cor e Forma:SolidPeso molecular:2390.8811-deoxy Prostaglandin E1
CAS:<p>11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause</p>Fórmula:C20H34O4Cor e Forma:SolidPeso molecular:338.48Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Fórmula:C10H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:233.69Vapreotide diacetate
CAS:<p>Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.</p>Fórmula:C61H78N12O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1251.47Orexin B, rat, mouse
CAS:<p>Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.</p>Fórmula:C126H215N45O34SPureza:98%Cor e Forma:SolidPeso molecular:2936.451-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Fórmula:C207H308N56O58S·C2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:4655.16KB-5492 FA
<p>KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8</p>Fórmula:C24H32N2O8Pureza:98.12%Cor e Forma:SolidPeso molecular:476.52Pobilukast
CAS:<p>Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.</p>Fórmula:C26H34O5SPureza:99.65% - 99.84%Cor e Forma:SolidPeso molecular:458.61CAY10597
CAS:<p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>Fórmula:C20H14ClFN2O5Cor e Forma:SolidPeso molecular:416.79Cisapride hydrate
CAS:<p>Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.</p>Fórmula:C23H31ClFN3O5Pureza:98%Cor e Forma:SolidPeso molecular:483.965-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Fórmula:C13H18N2OPureza:98.25%Cor e Forma:SolidPeso molecular:218.2920-hydroxy Prostaglandin F2α
CAS:<p>20-hydroxy Prostaglandin F2α (20-hydroxy PGF2α) is the ω-oxidation product of PGF2α.</p>Fórmula:C20H34O6Cor e Forma:SolidPeso molecular:370.4861-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid
CAS:1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid (Compound 31) is a metabolite of AB-FUBINACA. It acts as an MRGPRX4 antagonist with an IC50 greater than 2.5 μM.Fórmula:C15H11FN2O2Cor e Forma:SolidPeso molecular:270.26
