GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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GI-560192
CAS:<p>GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.</p>Fórmula:C20H16N2O2Pureza:99.53%Cor e Forma:SoildPeso molecular:316.35TGR5 agonist 2
<p>TGR5 agonist 2 (compound 19) serves as a highly potent agonist of TGR5, demonstrating an EC50 value of 0.27 µM [1].</p>Fórmula:C29H50NNaO6SCor e Forma:SolidPeso molecular:563.77Tafluprost acid
CAS:<p>Tafluprost acid is a selective agonist at the prostaglandin F receptor.</p>Fórmula:C22H28F2O5Cor e Forma:SolidPeso molecular:410.46(S)-V-0219 hydrochloride
<p>(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.</p>Fórmula:C20H26ClF3N4O2Cor e Forma:SolidPeso molecular:446.89Picumeterol FA
<p>picumeterol FA is a potent and selective β2-adrenergic receptor agonist.</p>Fórmula:C22H31Cl2N3O4Pureza:99.8%Cor e Forma:SoildPeso molecular:472.4SR 142948 dihydrochloride
<p>SR 142948 dihydrochloride is a selective oral non-peptide NT antagonist, IC50 <4 nM, with brain penetration and potential for psychiatric research.</p>Fórmula:C39H53Cl2N5O6Cor e Forma:SolidPeso molecular:758.77APJ receptor agonist 1
CAS:<p>Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.</p>Fórmula:C31H26ClN3O3Cor e Forma:SolidPeso molecular:524.02MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Fórmula:C60H90N20O11SPureza:98%Cor e Forma:SolidPeso molecular:1299.56PAR-2 (1-6) (human)
CAS:<p>PAR-2 (1-6) (human) (SLIGKV), a peptide ligand, is a PAR-2 agonist [1] .</p>Fórmula:C28H53N7O8Cor e Forma:SolidPeso molecular:615.76RFRP-3(human)
CAS:<p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>Fórmula:C45H72N14O10Pureza:98%Cor e Forma:SolidPeso molecular:969.15GLP-1R agonist 19
CAS:<p>GLP-1R agonist 19 (M3190) is a potent, selective GLP-1 receptor agonist that demonstrates excellent plasma and liver microsomal stability, along with low hERG toxicity [1].</p>Fórmula:C94H136FN21O25Cor e Forma:SolidPeso molecular:1979.21[Nle13]-Motilin
CAS:<p>[Nle13]-Motilin, a motilin analogue, is a motilin receptor agonist [1] [2] .</p>Fórmula:C121H190N34O35Cor e Forma:SolidPeso molecular:2681.01GLI1-IN-3
<p>GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.</p>Cor e Forma:Odour SolidSeptide
CAS:<p>Septide is an NK1 receptor agonist acting at a site distinct from substance P.</p>Fórmula:C39H53N7O7SPureza:98%Cor e Forma:SolidPeso molecular:763.95MrgprX2 antagonist-5
CAS:<p>MrgprX2 antagonist-5 from patent WO2020223255A1 inhibits MrgprX2, useful for inflammatory skin disorder studies.</p>Fórmula:C19H13ClF2N4O2SCor e Forma:SolidPeso molecular:434.85HAEGT
CAS:<p>HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.</p>Fórmula:C20H31N7O9Pureza:98%Cor e Forma:SolidPeso molecular:513.5ACTH (1-17)
CAS:<p>ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.</p>Fórmula:C95H145N29O23SPureza:98%Cor e Forma:SolidPeso molecular:2093.41α1A-AR Degrader 9c
CAS:<p>α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.</p>Fórmula:C38H43N11O11Pureza:98%Cor e Forma:SolidPeso molecular:829.82Cetirizine Impurity D
CAS:<p>Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.</p>Fórmula:C30H28Cl2N2Cor e Forma:SolidPeso molecular:487.46Prostaglandin J2
CAS:<p>PGJ2, a PGD2 metabolite, is a DP agonist (Ki: 0.9 nM hDP, 6.6 nM hCRTH2), induces cAMP (EC50: 1.2 nM), oxidative stress, neuronal apoptosis, and neurotoxicity.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.4515(R)-17-phenyl trinor Prostaglandin F2α
CAS:<p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>Fórmula:C23H32O5Cor e Forma:SolidPeso molecular:388.5L-threo Lysosphingomyelin (d18:1)
CAS:<p>L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).</p>Fórmula:C23H49N2O5PCor e Forma:SolidPeso molecular:464.62ELA-11(human)
CAS:<p>Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.</p>Fórmula:C58H90N16O13S2Pureza:98%Cor e Forma:SolidPeso molecular:1283.57Spantide acetate
<p>Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.</p>Fórmula:C77H112N20O15Pureza:98.9200%Cor e Forma:SolidPeso molecular:1557.84GnRH Associated Peptide (1-24), human
CAS:<p>GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.</p>Fórmula:C117H190N32O43Cor e Forma:SolidPeso molecular:2732.95DSP-1053
CAS:<p>Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.</p>Fórmula:C26H32BrNO4Pureza:98%Cor e Forma:SolidPeso molecular:502.44GLP-1R agonist 14
CAS:<p>GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].</p>Fórmula:C45H42F2N10O5Cor e Forma:SolidPeso molecular:840.885-HT7R antagonist 1 free base
CAS:<p>5-HT7R antagonist 1 (free base) is a G protein-biased antagonist for the 5-HT 7 R receptor, with a dissociation constant (K i) of 6.5 nM.</p>Fórmula:C14H17ClN4Cor e Forma:SolidPeso molecular:276.77GLP-1 receptor agonist 9 citrate
<p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>Fórmula:C38H39ClFN3O12Pureza:98.76%Cor e Forma:SolidPeso molecular:784.18PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44Hemopressin (human, mouse)
CAS:<p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>Fórmula:C50H79N13O12Pureza:98%Cor e Forma:SolidPeso molecular:1054.26Antibiotic Sch 60057
CAS:<p>Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.</p>Fórmula:C45H84O6Cor e Forma:SolidPeso molecular:721.16113,14-dihydro-15-keto Prostaglandin F1α
CAS:<p>13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.</p>Fórmula:C20H36O5Cor e Forma:SolidPeso molecular:356.5Isobutyryl-L-carnitine
CAS:<p>Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.</p>Fórmula:C11H21NO4Pureza:98%Cor e Forma:SolidPeso molecular:231.29GLP-1 (9-36) amide
CAS:<p>GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.</p>Fórmula:C140H214N36O43Pureza:97%Cor e Forma:SolidPeso molecular:3089.41CB2R probe 1
CAS:<p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>Fórmula:C36H42N4O4Cor e Forma:SolidPeso molecular:594.74Jatrorrhizine hydroxide
CAS:<p>Jatrorrhizine hydroxide: alkaloid from Coptis chinensis; neuroprotective, antimicrobial, antiplasmodial, antioxidant; AChE inhibitor, affects 5-HT/NE uptake.</p>Fórmula:C20H21NO5Cor e Forma:SolidPeso molecular:355.38Adrenomedullin (16-31), human
CAS:<p>Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).</p>Fórmula:C82H129N25O21S2Pureza:98%Cor e Forma:SolidPeso molecular:1865.19Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Fórmula:C86H115FN16O21Cor e Forma:SolidPeso molecular:1727.93Chir 2279
CAS:<p>CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).</p>Fórmula:C34H36N4O4Cor e Forma:SolidPeso molecular:564.67SB656104
CAS:<p>SB656104 is a bioactive chemical.</p>Fórmula:C25H30ClN3O3SCor e Forma:SolidPeso molecular:488.04Benzomalvin B
CAS:<p>Benzomalvin B, a metabolite from Penicillium, blocks 24% NK1 receptor binding at 100 μg/ml.</p>Fórmula:C24H17N3O2Cor e Forma:SolidPeso molecular:379.419LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Fórmula:C39H43ClN4O9S2Cor e Forma:SolidPeso molecular:811.36Vortioxetine D8
CAS:<p>Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).</p>Fórmula:C18H22N2SPureza:98%Cor e Forma:SolidPeso molecular:306.5Brexpiprazole S-oxide D8
CAS:<p>Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.</p>Fórmula:C25H19D8N3O3SPureza:98%Cor e Forma:SolidPeso molecular:457.61Prolactin Releasing Peptide (1-31), human
CAS:<p>Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).</p>Fórmula:C160H252N56O42SPureza:98%Cor e Forma:SolidPeso molecular:3664.15Luseogliflozin hydrate
CAS:<p>Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.</p>Fórmula:C23H32O7SCor e Forma:SolidPeso molecular:452.56Guanylin TFA (mouse,rat)
<p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>Fórmula:C60H90N16O22S4·xC2HF3O2Cor e Forma:SolidPeso molecular:1515.71 (free base)PACAP (6-38), human, ovine, rat TFA
<p>PACAP (6-38) is a PACAP receptor blocker with IC50s of 30, 600, 40 nM for type I, VIP1, and VIP2 receptors.</p>Fórmula:C184H301N56FO47SPureza:98%Cor e Forma:SolidPeso molecular:4138.76Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Fórmula:C19H23N3Pureza:99.88%Cor e Forma:White/Pale Yellow Crystalline SolidPeso molecular:293.41Mosapride citrate dihydrate
CAS:<p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>Fórmula:C27H35ClFN3O11Pureza:98%Cor e Forma:SolidPeso molecular:632.04KwFwLL-NH2
CAS:<p>KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).</p>Fórmula:C49H66N10O6Cor e Forma:SolidPeso molecular:891.11Adrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Fórmula:C248H381N77O75S5Pureza:98%Cor e Forma:SolidPeso molecular:5729.5β-CGRP (mouse)
<p>β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.</p>Fórmula:C165H265N49O55S2Cor e Forma:SolidPeso molecular:3879.29SGLT1/2-IN-2
CAS:<p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>Fórmula:C23H26F2O7Cor e Forma:SolidPeso molecular:452.451Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Fórmula:C12H14ClN5O2SeCor e Forma:SolidPeso molecular:374.68Y1 receptor antagonist 1 formic
<p>H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.</p>Fórmula:C29H35N5O5Cor e Forma:SolidPeso molecular:533.62cAC 253 acetate
<p>cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.</p>Fórmula:C128H206N42O42S2Pureza:98.16% - 99.99%Cor e Forma:SoildPeso molecular:3069.39Pentagastrin meglumine
CAS:<p>Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.</p>Fórmula:C44H66N8O14SCor e Forma:SolidPeso molecular:963.11YM 09538
CAS:<p>YM 09538 is a biochemical.</p>Fórmula:C18H25ClN2O5SCor e Forma:SolidPeso molecular:416.92ONO-8711
CAS:<p>ONO-8711 is a potent and selective competitive antagonist of EP1 receptor with Kis of 0.6 nM and 1.7 nM for human and mouse EP1, respectively.</p>Fórmula:C22H30ClNO4SCor e Forma:SolidPeso molecular:440ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
CAS:<p>ACTH (3-24) is the fragment 3-24 of ACTH, used in disease research including cancer and immune disorders.</p>Fórmula:C124H196N38O27SCor e Forma:SolidPeso molecular:2683.192-Furoyl-LIGRLO-amide
CAS:<p>2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.</p>Fórmula:C36H63N11O8Pureza:98%Cor e Forma:SolidPeso molecular:777.95Senktide TFA
<p>Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.</p>Cor e Forma:Odour SolidMMC(TMZ)-TOC TFA
<p>MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.</p>Fórmula:C74H99F3N20O21S2Cor e Forma:SolidPeso molecular:1725.82Imipramine N-oxide
CAS:<p>Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.</p>Fórmula:C19H24N2OPureza:99.80%Cor e Forma:SolidPeso molecular:296.41Neuromedin N
CAS:<p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>Fórmula:C38H63N7O8Pureza:98%Cor e Forma:SolidPeso molecular:745.95Neuropeptide Y(29-64)
CAS:<p>Neuropeptide Y(29-64) is a 36 amino acid peptide, a fragment of Neuropeptide Y.</p>Fórmula:C189H284N54O58SPureza:98%Cor e Forma:SolidPeso molecular:4272.7Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:1583.78 (free base)Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Fórmula:C61H94N18O13SCor e Forma:SolidPeso molecular:1319.5819(R)-hydroxy Prostaglandin E1
CAS:<p>19(R)-hydroxy Prostaglandin E1 is an agonist of EP1 and EP3 receptor subtypes and exhibits contractile activity on smooth muscle and is the major prostaglandin</p>Fórmula:C20H34O6Cor e Forma:SolidPeso molecular:370.486Cyclosomatostatin Acetate
<p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>Fórmula:C46H61N7O8Pureza:98.83%Cor e Forma:SolidPeso molecular:840.02GLP-1(7-36), amide acetate
CAS:<p>GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.</p>Fórmula:C151H230N40O47Pureza:99.89%Cor e Forma:SolidPeso molecular:3357.68NSC380324
<p>NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.</p>Fórmula:C31H24N4O4Cor e Forma:SolidPeso molecular:516.55des-Gln14-Ghrelin
CAS:<p>Endogenous rat ghrelin gene variant binds GHS-R1a; strong Ca2+ release (EC50=2.4 nM); boosts GH secretion in vivo.</p>Fórmula:C142H237N43O40Pureza:98%Cor e Forma:SolidPeso molecular:3186.7S1PR1 modulator 1
CAS:<p>S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.</p>Fórmula:C23H24N2O3SPureza:99.69%Cor e Forma:SolidPeso molecular:408.51YM 16638
CAS:<p>YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.</p>Fórmula:C18H22N2O5S3Pureza:99.18%Cor e Forma:SolidPeso molecular:442.57Donetidine
CAS:<p>Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.</p>Fórmula:C20H25N5O3SPureza:99.32%Cor e Forma:SolidPeso molecular:415.51MM 07
CAS:<p>Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.</p>Fórmula:C67H106N22O14S3Pureza:98%Cor e Forma:SolidPeso molecular:1539.91-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Fórmula:C207H308N56O58S·C2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:4655.16Neuropeptide Y (22-36)
CAS:<p>Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.</p>Fórmula:C85H139N29O21Pureza:98%Cor e Forma:SolidPeso molecular:1903.19SR142948A
CAS:<p>SR142948A is a selective and reversible non-peptide neurotensin receptor antagonist blocking hypothermia and analgesic effects, NMDA-induced dopamine release.</p>Fórmula:C39H52ClN5O6Pureza:98%Cor e Forma:SolidPeso molecular:722.31Pexopiprant
CAS:<p>Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.</p>Fórmula:C21H17Cl2F2NO4Cor e Forma:SolidPeso molecular:456.27Tocrifluor T1117
CAS:<p>Fluorescent form of AM 251, CB1 receptor antagonist</p>Fórmula:C56H53Cl2N7O5Pureza:98%Cor e Forma:SolidPeso molecular:974.97Amylin, amide, rat
CAS:<p>Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.</p>Fórmula:C167H272N52O53S2Pureza:99.92%Cor e Forma:SolidPeso molecular:3920.44Kisspeptin-10, human
CAS:<p>Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.</p>Fórmula:C63H83N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1302.462Pancreatic Polypeptide, bovine
CAS:Agonist at Y4 neuropeptide Y receptors.Fórmula:C186H287N53O56S2Pureza:98%Cor e Forma:SolidPeso molecular:4225.78Urocortin II, human
Human urocortin (hUcn) II is a new member of the corticotropin-releasing-factor (CRF) family. It selectively binds to the CRF2 receptor.Fórmula:C194H339N63O54SPureza:98%Cor e Forma:SolidPeso molecular:4450.28Alosetron-d3
CAS:<p>Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Fórmula:C17H18N4OPureza:98%Cor e Forma:SolidPeso molecular:297.37Spantide I
CAS:<p>Spantide antagonizes both bombesin & substance P. It is also tachykinin receptor antagonist.</p>Fórmula:C75H108N20O13Pureza:98%Cor e Forma:SolidPeso molecular:1497.7915(S)-HpEPE
CAS:<p>15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456Cagrilintide acetate
<p>.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.</p>Fórmula:C196H316N54O61S2Pureza:99.88%Cor e Forma:SolidPeso molecular:4469.06GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Fórmula:C165H254N44O55SPureza:98%Cor e Forma:SolidPeso molecular:3766.19HAEGTFT
CAS:<p>HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C33H47N9O12Pureza:98%Cor e Forma:SolidPeso molecular:761.785-HT1AR/5-HT6R ligand-1
<p>5-HT1AR/5-HT6R ligand-1 (Compound PP13) functions as a ligand for the 5-HT receptor, demonstrating high affinity for 5-HT1AR, 5-HT6R, and 5-HT7R with Ki values of 19, 69, and 198 nM, respectively. In HEK293 cells, it inhibits cAMP production with EC50 values of 1535, 488, and 53 nM for these receptors. Additionally, 5-HT1AR/5-HT6R ligand-1 exhibits antiproliferative effects on several cancer cell lines, including 1321N1, U87MG, MCF7, and AsPC-1, with IC50 values of 9.6, 13.6, 19.3, and 14.6 μM, respectively. The compound also shows antagonistic activity towards the dopamine receptor D2R, with a Ki of 1903 nM.</p>Fórmula:C25H29ClN4O2SCor e Forma:SolidPeso molecular:485.04Sarafotoxin S6b
CAS:<p>non-selective endothelin receptor agonist</p>Fórmula:C110H163N27O34S5Pureza:98%Cor e Forma:SolidPeso molecular:2567.96Icatibant
CAS:<p>Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).</p>Fórmula:C59H89N19O13SPureza:98%Cor e Forma:White SolidPeso molecular:1304.52Kinetensin
CAS:Kinetensin is a neurotensin-like peptide.Fórmula:C56H85N17O11Pureza:98%Cor e Forma:White Lyophilised SolidPeso molecular:1172.38(D-Phe7)-α-MSH
CAS:<p>(D-Phe7)-α-MSH is an α-MSH analogue [1] .</p>Fórmula:C77H109N21O19SCor e Forma:SolidPeso molecular:1664.88LSN3160440
CAS:<p>LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.</p>Fórmula:C27H27Cl2N3OCor e Forma:SolidPeso molecular:480.43
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