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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5378 produtos de "GPCR/Proteína-G"

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  • RO1138452
    Targetmol
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    RO1138452

    CAS:
    <p>RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).</p>
    Fórmula:C19H23N3O
    Pureza:97.01% - 99.34%
    Cor e Forma:Solid
    Peso molecular:309.41

    Ref: TM-T4436

  • CYN 154806 TFA
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    CYN 154806 TFA

    CAS:
    <p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>
    Fórmula:C58H69F3N12O16S2
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:1311.36

    Ref: TM-TP1346

  • Olcegepant
    Targetmol
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    Olcegepant

    CAS:
    <p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>
    Fórmula:C38H47Br2N9O5
    Pureza:96.08% - 97.24%
    Cor e Forma:Solid
    Peso molecular:869.65

    Ref: TM-T12293L

  • Bepotastine
    Targetmol
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    Bepotastine

    CAS:
    <p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>
    Fórmula:C21H25ClN2O3
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:388.89

    Ref: TM-T7893

  • Substance P 1-9 aceate
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    Substance P 1-9 aceate

    <p>Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.</p>
    Fórmula:C54H81N15O14
    Pureza:99.01%
    Cor e Forma:Solid
    Peso molecular:1164.31

    Ref: TM-TP1819L

  • Ondansetron hydrochloride
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    Ondansetron hydrochloride

    CAS:
    <p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>
    Fórmula:C18H19N3O·HCl
    Pureza:99.78%
    Cor e Forma:White Powder
    Peso molecular:329.82

    Ref: TM-T6616

  • Brexpiprazole HCl
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    Brexpiprazole HCl

    CAS:
    <p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>
    Fórmula:C25H27N3O2S·xHCl
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:433.6

    Ref: TM-T8690

  • Sigma-LIGAND-1 hydrochloride
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    Sigma-LIGAND-1 hydrochloride

    CAS:
    <p>Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.</p>
    Fórmula:C27H34ClNO4
    Cor e Forma:Solid
    Peso molecular:472.02

    Ref: TM-T63048

  • Etrasimod
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    Etrasimod

    CAS:
    <p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>
    Fórmula:C26H26F3NO3
    Pureza:98.52% - 99.73%
    Cor e Forma:Solid
    Peso molecular:457.48

    Ref: TM-TQ0227

  • Litorin acetate(55749-97-8 Free base)
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    Litorin acetate(55749-97-8 Free base)

    <p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>
    Fórmula:C53H72N14O13S
    Pureza:98.61%
    Cor e Forma:Solid
    Peso molecular:1145.29

    Ref: TM-T20604L

  • Volinanserin
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    Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Fórmula:C22H28FNO3
    Pureza:98.94% - 99.95%
    Cor e Forma:Solid
    Peso molecular:373.46

    Ref: TM-T5389

  • BP 897
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    BP 897

    CAS:
    <p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>
    Fórmula:C26H31N3O2
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:417.54

    Ref: TM-T9100

  • L-745870 hydrochloride
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    L-745870 hydrochloride

    CAS:
    <p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>
    Fórmula:C18H20Cl2N4
    Pureza:97.36%
    Cor e Forma:Solid
    Peso molecular:363.28

    Ref: TM-T11799

  • Rimegepant
    Targetmol
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    Rimegepant

    CAS:
    <p>View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.</p>
    Fórmula:C28H28F2N6O3
    Pureza:99.1% - 99.99%
    Cor e Forma:Solid
    Peso molecular:534.56

    Ref: TM-T4610

  • Enprofylline
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    Enprofylline

    CAS:
    <p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>
    Fórmula:C8H10N4O2
    Pureza:98.37%
    Cor e Forma:Solid
    Peso molecular:194.19

    Ref: TM-T21389

  • Puerarin
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    Puerarin

    CAS:
    <p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>
    Fórmula:C21H20O9
    Pureza:98.90% - 99.21%
    Cor e Forma:Yellow Brown Fine Powder
    Peso molecular:416.38

    Ref: TM-T2815

  • Vericiguat
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    Vericiguat

    CAS:
    <p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>
    Fórmula:C19H16F2N8O2
    Pureza:98.86% - 99.93%
    Cor e Forma:Solid
    Peso molecular:426.38

    Ref: TM-T17226

  • Riociguat
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    Riociguat

    CAS:
    Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterial
    Fórmula:C20H19FN8O2
    Pureza:99.28% - 99.95%
    Cor e Forma:Solid
    Peso molecular:422.42

    Ref: TM-T6968

  • Protease-Activated Receptor-1, PAR-1 Agonist acetate
    Targetmol
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    Protease-Activated Receptor-1, PAR-1 Agonist acetate

    PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.
    Fórmula:C37H62N10O11
    Pureza:98.1800%
    Cor e Forma:Solid
    Peso molecular:822.95

    Ref: TM-T38836L

  • Mozavaptan
    Targetmol
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    Mozavaptan

    CAS:
    <p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>
    Fórmula:C27H29N3O2
    Pureza:98.98% - 99.12%
    Cor e Forma:Solid
    Peso molecular:427.54

    Ref: TM-T6288