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GPCR/Proteína-G

GPCR/Proteína-G

Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.

Subcategorias de "GPCR/Proteína-G"

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Foram encontrados 5352 produtos de "GPCR/Proteína-G"

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  • Adrenocorticotropic Hormone (ACTH) (4-10) TFA
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    Adrenocorticotropic Hormone (ACTH) (4-10) TFA

    <p>Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .</p>
    Fórmula:C46H60F3N13O12S
    Pureza:98.49%
    Cor e Forma:Solid
    Peso molecular:1076.12

    Ref: TM-T7627L

  • Pramlintide acetate(151126-32-8 free base)
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    Pramlintide acetate(151126-32-8 free base)

    CAS:
    <p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>
    Fórmula:C173H271N51O55S2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:4009

    Ref: TM-TP2320

  • Terazosin hydrochloride dihydrate
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    Terazosin hydrochloride dihydrate

    CAS:
    <p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>
    Fórmula:C19H25N5O4·HCl·2H2O
    Pureza:99.81%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:459.92

    Ref: TM-T6701

  • Relenopride hydrochloride
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    Relenopride hydrochloride

    CAS:
    <p>Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.</p>
    Fórmula:C24H31Cl2FN4O4
    Cor e Forma:Solid
    Peso molecular:529.43

    Ref: TM-T28512

  • Nafarelin acetate(76932-56-4 free base)
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    Nafarelin acetate(76932-56-4 free base)

    CAS:
    <p>Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.</p>
    Fórmula:C68H87N17O15
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:1382.55

    Ref: TM-T21309

  • BQ-788 sodium salt
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    BQ-788 sodium salt

    CAS:
    BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).
    Fórmula:C34H51N5NaO7
    Cor e Forma:Solid
    Peso molecular:664.8

    Ref: TM-T10595L

  • Naluzotan
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    Naluzotan

    CAS:
    <p>Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:450.64

    Ref: TM-T16265

  • ELA-11 (human) acetate(1784687-32-6 free base)
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    ELA-11 (human) acetate(1784687-32-6 free base)

    <p>ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.</p>
    Fórmula:C60H94N16O15S2
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:1343.61

    Ref: TM-TP1922L1

  • CB1 antagonist 4
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    CB1 antagonist 4

    CAS:
    <p>TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.</p>
    Fórmula:C30H25Cl2F3N4OS
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:617.51

    Ref: TM-T8511

  • Fenspiride
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    Fenspiride

    CAS:
    <p>Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.</p>
    Fórmula:C15H20N2O2
    Cor e Forma:Solid
    Peso molecular:260.33

    Ref: TM-T60417

  • Fluorogestone acetate
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    Fluorogestone acetate

    CAS:
    <p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>
    Fórmula:C23H31FO5
    Pureza:99.47%
    Cor e Forma:Coa
    Peso molecular:406.49

    Ref: TM-T21335

  • RTICBM-189
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    RTICBM-189

    CAS:
    <p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>
    Fórmula:C15H14Cl2N2O
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:309.19

    Ref: TM-T9466

  • Naftopidil hydrochloride
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    Naftopidil hydrochloride

    CAS:
    <p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>
    Fórmula:C24H29ClN2O3
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:428.95

    Ref: TM-T9220

  • Darusentan
    Targetmol
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    Darusentan

    CAS:
    <p>Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteries</p>
    Fórmula:C22H22N2O6
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:410.43

    Ref: TM-T5458

  • NPS2390
    Targetmol
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    NPS2390

    CAS:
    <p>NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)</p>
    Fórmula:C19H21N3O
    Pureza:97.13%
    Cor e Forma:Solid
    Peso molecular:307.39

    Ref: TM-T8457

  • LY310762
    Targetmol
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    LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Fórmula:C24H27FN2O2·HCl
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:430.94

    Ref: TM-T2688

  • Liraglutide
    Targetmol
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    Liraglutide

    CAS:
    <p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>
    Fórmula:C172H265N43O51
    Pureza:97.65% - 99.04%
    Cor e Forma:Solid
    Peso molecular:3751.25

    Ref: TM-T6876

  • [Des-Arg9]-Bradykinin TFA
    Targetmol
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    [Des-Arg9]-Bradykinin TFA

    CAS:
    <p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>
    Fórmula:C46H62F3N11O12
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1018.05

    Ref: TM-T8809

  • Orexin 2 Receptor Agonist
    Targetmol
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    Orexin 2 Receptor Agonist

    CAS:
    Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.
    Fórmula:C32H34N4O5S
    Pureza:98.26% - 99.43%
    Cor e Forma:Solid
    Peso molecular:586.7

    Ref: TM-T3177

  • Talnetant hydrochloride
    Targetmol
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    Talnetant hydrochloride

    CAS:
    <p>Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.</p>
    Fórmula:C25H23ClN2O2
    Cor e Forma:Solid
    Peso molecular:418.92

    Ref: TM-T62199