GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.949 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(410 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5378 produtos de "GPCR/Proteína-G"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Fórmula:C21H21FO5SPureza:99.38% - 99.70%Cor e Forma:SolidPeso molecular:404.45Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSCor e Forma:SolidPeso molecular:340.48Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Fórmula:C9H10Cl2N4Cor e Forma:SolidPeso molecular:245.11Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Fórmula:C23H29NO5SPureza:98%Cor e Forma:SolidPeso molecular:431.55S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Cor e Forma:SolidPeso molecular:407.48Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Fórmula:C15H20N8O6Pureza:98%Cor e Forma:SolidPeso molecular:408.37Siponimod hemifumarate
CAS:<p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>Fórmula:C62H74F6N4O10Cor e Forma:SolidPeso molecular:1149.282Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Fórmula:C18H22N2Cor e Forma:SolidPeso molecular:266.38BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Fórmula:C25H28Cl2N2OCor e Forma:SolidPeso molecular:443.41Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Fórmula:C19H23ClN2Cor e Forma:SolidPeso molecular:314.852RS 100329
CAS:<p>RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).</p>Fórmula:C20H25F3N4O3Cor e Forma:SolidPeso molecular:426.43Ajmalicine hydrochloride
CAS:<p>Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.</p>Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Fórmula:C24H29N3O3Cor e Forma:SolidPeso molecular:407.51PF3274167
CAS:PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Fórmula:C19H19ClFN5O3Pureza:99.67% - 99.88%Cor e Forma:SolidPeso molecular:419.84THIQ
CAS:<p>THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).</p>Fórmula:C33H41ClN6O2Pureza:98.93%Cor e Forma:SolidPeso molecular:589.17Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Cor e Forma:SolidPeso molecular:301.81Ornipressin Acetate(3397-23-7,free)
CAS:<p>Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent.</p>Fórmula:C47H67N13O124S2Pureza:>99.99%Cor e Forma:SolidPeso molecular:1102.25Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Fórmula:C16H14O2Pureza:98.15%Cor e Forma:SolidPeso molecular:238.2812Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Fórmula:C25H25Cl2N7OPureza:99.43%Cor e Forma:SolidPeso molecular:510.42Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95[Lys8, Lys9]-Neurotensin (8-13) acetate
<p>[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2</p>Fórmula:C40H68N8O10Pureza:99.31%Cor e Forma:SolidPeso molecular:821.02R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Fórmula:C41H55N9O12Pureza:99.52%Cor e Forma:SolidPeso molecular:865.93Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Fórmula:C14H16N2·HClPureza:99.74%Cor e Forma:SolidPeso molecular:248.75CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Fórmula:C20H21N7O3Pureza:98.78%Cor e Forma:SolidPeso molecular:407.43BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Fórmula:C23H22F3N3O3Pureza:99.37% - 99.89%Cor e Forma:SolidPeso molecular:445.437-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Fórmula:C5H11Cl2N3Pureza:99.12%Cor e Forma:SolidPeso molecular:184.067SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Fórmula:C16H17NO2·HClPureza:99.1% - 99.51%Cor e Forma:SolidPeso molecular:291.77Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Fórmula:C9H13NO2Pureza:99.5% - 99.89%Cor e Forma:SolidPeso molecular:167.21Piperoxan hydrochloride
CAS:<p>Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.</p>Fórmula:C14H20ClNO2Pureza:99.61%Cor e Forma:SolidPeso molecular:269.77Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Fórmula:C38H73N21O10S2HClPureza:>99.99%Cor e Forma:SolidPeso molecular:1353.33Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Fórmula:C17H18Cl3NOPureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:358.69Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Cor e Forma:White SolidPeso molecular:414.43Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Fórmula:C14H25NO6SPureza:99.35% - 99.75%Cor e Forma:SolidPeso molecular:335.42AC 187 Acetate
<p>AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.</p>Fórmula:C129H209N37O42Pureza:99.71%Cor e Forma:SolidPeso molecular:2950.26[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Fórmula:C69H108N22O16SPureza:99.71%Cor e Forma:SolidPeso molecular:1533.8VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Fórmula:C29H36F3N3O5Pureza:98.2% - 98.88%Cor e Forma:SolidPeso molecular:563.61Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.47Chlorcyclizine
CAS:<p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>Fórmula:C18H21ClN2Pureza:98.75%Cor e Forma:SolidPeso molecular:300.83Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Fórmula:C20H22N2O6Pureza:99.39%Cor e Forma:SolidPeso molecular:386.4BWX 46 Acetate
<p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>Fórmula:C118H190N36O30S2Pureza:96.86%Cor e Forma:SolidPeso molecular:2657.12AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Fórmula:C21H24ClF2NOPureza:99.89%Cor e Forma:SolidPeso molecular:379.87ACEPROMAZINE MALEATE
CAS:<p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>Fórmula:C23H26N2O5SPureza:98.87% - 99.51%Cor e Forma:Off White Or Yellow Crystalline PowderPeso molecular:442.53CGP71683 hydrochloride
CAS:<p>CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).</p>Fórmula:C26H30ClN5O2SPureza:99.92%Cor e Forma:SolidPeso molecular:512.07NPY 5RA972
CAS:<p>NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist</p>Fórmula:C21H25N3O2Pureza:99.02% - 99.56%Cor e Forma:SolidPeso molecular:351.44RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Fórmula:C25H27N3O3Pureza:98.64% - 99.62%Cor e Forma:SolidPeso molecular:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Cor e Forma:SolidPeso molecular:240.69N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Cor e Forma:Yellow Crystalline SolidPeso molecular:312.8OXOMEMAZINE
CAS:<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Fórmula:C18H22N2O2SPureza:99.58%Cor e Forma:SolidPeso molecular:330.44Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Fórmula:C19H20ClN3Pureza:98% - 99.65%Cor e Forma:SolidPeso molecular:325.84Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Fórmula:C26H24F4N6OPureza:98.75% - >99.99%Cor e Forma:SolidPeso molecular:512.5HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Fórmula:C24H23ClN4O3Pureza:95.73%Cor e Forma:SolidPeso molecular:450.92SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Fórmula:C28H28ClN3OSPureza:97.37% - 98.88%Cor e Forma:SolidPeso molecular:490.06Ciliobrevin A
CAS:<p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.</p>Fórmula:C17H9Cl2N3O2Pureza:98.54% - 99.57%Cor e Forma:SolidPeso molecular:358.18SANT-1
CAS:<p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>Fórmula:C23H27N5Pureza:99.98% - >99.99%Cor e Forma:SolidPeso molecular:373.49SB297006
CAS:<p>SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.</p>Fórmula:C18H18N2O5Pureza:99.59%Cor e Forma:SolidPeso molecular:342.35Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Fórmula:C59H80N14O13Pureza:95.3%Cor e Forma:SolidPeso molecular:1193.35Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Fórmula:C19H17FN8O2Pureza:99.19%Cor e Forma:SolidPeso molecular:408.39AR-M 1896 Acetate
<p>AR-M 1896 Acetate is the selective agonist of GalR2.</p>Fórmula:C56H85N13O16Pureza:99.76%Cor e Forma:SolidPeso molecular:1196.35Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Fórmula:C21H28N2O2Pureza:99.53%Cor e Forma:White Or Similar To White PowderPeso molecular:340.46PF-04418948
CAS:<p>PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.</p>Fórmula:C23H20FNO5Pureza:98.67% - 99.45%Cor e Forma:SolidPeso molecular:409.41Scyliorhinin II acetate
<p>Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.</p>Fórmula:C79H123N21O28S3Pureza:99.06%Cor e Forma:SolidPeso molecular:1911.14Tolazoline
CAS:<p>Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.</p>Fórmula:C10H12N2Pureza:99.52%Cor e Forma:SolidPeso molecular:160.22Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Fórmula:C23H23ClN2O5SPureza:97.6% - 97.78%Cor e Forma:SolidPeso molecular:474.96Levalbuterol tartrate
CAS:<p>Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.</p>Fórmula:C17H27NO9Pureza:98.97% - 99.79%Cor e Forma:SolidPeso molecular:389.393-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89ONO-7300243
CAS:<p>ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).</p>Fórmula:C28H31NO5Pureza:99.66%Cor e Forma:SolidPeso molecular:461.55HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C35H51N9O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:821.84Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Fórmula:C22H15F3N2O7SPureza:99.33%Cor e Forma:SolidPeso molecular:508.42ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Fórmula:C13H16ClN3O3Pureza:98.15%Cor e Forma:SolidPeso molecular:297.74GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Fórmula:C18H17Cl2F3N4O2Pureza:99.47%Cor e Forma:SolidPeso molecular:449.25OXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Fórmula:C79H125N23O22Pureza:98.52%Cor e Forma:SolidPeso molecular:1748.98MK-0557
CAS:<p>MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).</p>Fórmula:C22H19FN4O3Pureza:99.88%Cor e Forma:SolidPeso molecular:406.41Tetradecyl Phosphonate
CAS:<p>Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。</p>Fórmula:C14H31O3PPureza:99.95%Cor e Forma:White To Off-White PowderPeso molecular:278.37CGS 21680 Hydrochloride
CAS:<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Fórmula:C23H29N7O6·HClPureza:96.74% - 99.53%Cor e Forma:SolidPeso molecular:535.98AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Fórmula:C30H27BrN4O3Pureza:98.12%Cor e Forma:SolidPeso molecular:571.46Brimonidine
CAS:<p>Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.</p>Fórmula:C11H10BrN5Pureza:99.626%Cor e Forma:Yellow SolidPeso molecular:292.13Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Fórmula:C21H24ClN2NaO4SPureza:99.82%Cor e Forma:SolidPeso molecular:458.93PF-06291874
CAS:<p>PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.</p>Fórmula:C26H28F3N3O4Pureza:99.12% - 99.27%Cor e Forma:SolidPeso molecular:503.51Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Fórmula:C19H23NO3·CH4O3SPureza:99.18% - 99.87%Cor e Forma:Tan Or Off-White Cyrstalline SolidPeso molecular:409.5A-381393
CAS:<p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>Fórmula:C20H24N4Pureza:99.00%Cor e Forma:SolidPeso molecular:320.43Parmodulin 2
CAS:<p>ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).</p>Fórmula:C17H17BrN2O2Pureza:97.35% - 99.95%Cor e Forma:SolidPeso molecular:361.23Velneperit
CAS:<p>Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.</p>Fórmula:C17H24F3N3O3SPureza:99.70%Cor e Forma:SolidPeso molecular:407.45SCH442416
CAS:<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Fórmula:C20H19N7O2Pureza:99.58%Cor e Forma:SolidPeso molecular:389.41M871 acetate
<p>M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive</p>Fórmula:C110H167N27O30Pureza:99.84%Cor e Forma:SolidPeso molecular:2347.67Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Fórmula:C12H17ClN2O2Pureza:99.35%Cor e Forma:SolidPeso molecular:256.73Guanfacine hydrochloride
CAS:<p>Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.</p>Fórmula:C9H10Cl3N3OPureza:99.89% - 99.91%Cor e Forma:SolidPeso molecular:282.55L-732138
CAS:<p>L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)</p>Fórmula:C22H18F6N2O3Pureza:99.77%Cor e Forma:SolidPeso molecular:472.38Indophagolin
CAS:<p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>Fórmula:C19H15BrClF3N2O3SPureza:99.76%Cor e Forma:SolidPeso molecular:523.75Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Fórmula:C48H68N14O14S2Pureza:98.84% - >99.99%Cor e Forma:SolidPeso molecular:1129.26Azaphen dihydrochloride monohydrate
CAS:<p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C16H23Cl2N5O2Pureza:99.85%Cor e Forma:SolidPeso molecular:388.29ML382
CAS:<p>ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).</p>Fórmula:C18H20N2O4SPureza:99.79%Cor e Forma:SolidPeso molecular:360.43Asapiprant
CAS:<p>Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.</p>Fórmula:C24H27N3O7SPureza:99.64%Cor e Forma:SolidPeso molecular:501.55Dimaprit dihydrochloride
CAS:<p>Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.</p>Fórmula:C6H15N3S·2HClPureza:99.79%Cor e Forma:SolidPeso molecular:234.19GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Fórmula:C22H21ClN4O4Pureza:99.04%Cor e Forma:SolidPeso molecular:440.88Cloprostenol sodium salt
CAS:<p>Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.</p>Fórmula:C22H28ClNaO6Pureza:97.17% - 98.47%Cor e Forma:White To Almost White Hygroscopic PowderPeso molecular:446.9ZK 756326
CAS:<p>ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.</p>Fórmula:C21H28N2O3Pureza:99.43%Cor e Forma:SolidPeso molecular:356.46SLF1081851 TFA
CAS:<p>SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.</p>Fórmula:C23H34F3N3O3Cor e Forma:SolidPeso molecular:457.538AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Fórmula:C11H9Cl2N3O3SPureza:99.80% - >99.99%Cor e Forma:SolidPeso molecular:334.18AC-55541
CAS:<p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>Fórmula:C25H20BrN5O3Pureza:98% - 99.33%Cor e Forma:SolidPeso molecular:518.36Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Fórmula:C21H24Cl2FNO2Cor e Forma:SolidPeso molecular:412.33Ganirelix Acetate
CAS:<p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>Fórmula:C82H117ClN18O15Pureza:96.05%Cor e Forma:SolidPeso molecular:1630.4Litorin acetate(55749-97-8 Free base)
<p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>Fórmula:C53H72N14O13SPureza:98.61%Cor e Forma:SolidPeso molecular:1145.29Azaperone
CAS:Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4Eprazinone dihydrochloride
CAS:<p>Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.</p>Fórmula:C24H32N2O2·2HClPureza:99.25%Cor e Forma:A White Or Almost White CrysPeso molecular:453.44Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Fórmula:C22H26N2O4Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:382.45Vercirnon
CAS:<p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>Fórmula:C22H21ClN2O4SPureza:99.23%Cor e Forma:SolidPeso molecular:444.93Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Fórmula:C4H3F7OPureza:98%Cor e Forma:Less Oil Colorless OilPeso molecular:200.05ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Fórmula:C23H31N3O3SPureza:99.75%Cor e Forma:SolidPeso molecular:429.58Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Fórmula:C18H24ClNO3Pureza:97.15% - 99.94%Cor e Forma:SolidPeso molecular:337.84Vicriviroc maleate
CAS:<p>Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.</p>Fórmula:C32H42F3N5O6Pureza:98.16% - 98.37%Cor e Forma:SolidPeso molecular:649.7JK184
CAS:<p>JK184 is a potent Hedgehog (Hh) pathway inhibitor.</p>Fórmula:C19H18N4OSPureza:98.93% - 99.89%Cor e Forma:SolidPeso molecular:350.44Cenicriviroc
CAS:Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Fórmula:C41H52N4O4SPureza:97.87%Cor e Forma:SolidPeso molecular:696.94Maraviroc
CAS:<p>Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.</p>Fórmula:C29H41F2N5OPureza:97.13% - 99.59%Cor e Forma:Brown SolidPeso molecular:513.67AZD-4818
CAS:<p>AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Fórmula:C27H32Cl2N2O7Pureza:99.01%Cor e Forma:SolidPeso molecular:567.46Thrombin Receptor Activator for Peptide
<p>Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.</p>Fórmula:C32H51F3N8O9Pureza:99.88%Cor e Forma:SolidPeso molecular:748.79Dasotraline
CAS:<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Fórmula:C16H15Cl2NCor e Forma:SolidPeso molecular:292.2Vilazodone Hydrochloride
CAS:<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Fórmula:C26H27N5O2·HClPureza:99.56% - >99.99%Cor e Forma:SolidPeso molecular:477.99LUN42518 HCl 47142-51-8(free base)
<p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>Fórmula:C17H20ClN3OPureza:99.96%Cor e Forma:SolidPeso molecular:317.81Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Fórmula:C17H20BrNOCor e Forma:SolidPeso molecular:334.25Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Fórmula:C22H23N3O3SPureza:98.77%Cor e Forma:SolidPeso molecular:409.5ONO-AE3-208
CAS:<p>ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.</p>Fórmula:C24H21FN2O3Pureza:98.04% - 99.55%Cor e Forma:SolidPeso molecular:404.43Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Fórmula:C20H20NO4Pureza:97.18% - 99.06%Cor e Forma:SolidPeso molecular:338.38ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Fórmula:C16H15N7O2Pureza:97.02% - 99.69%Cor e Forma:SolidPeso molecular:337.34CYM2503
CAS:<p>CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.</p>Fórmula:C45H55N5O7Pureza:97.04%Cor e Forma:SolidPeso molecular:777.95Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Cor e Forma:White To Tan Powder SolidPeso molecular:383.4REV 5901
CAS:<p>REV 5901: oral leukotriene receptor antagonist and 5-lipoxygenase inhibitor with Ki of 0.7 μM, researched for asthma.</p>Fórmula:C22H25NO2Cor e Forma:SolidPeso molecular:335.44lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7Lidamidine Hydrochloride
CAS:Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Fórmula:C11H17ClN4OCor e Forma:SolidPeso molecular:256.73HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Fórmula:C27H33F3N4O9Pureza:99.51%Cor e Forma:SolidPeso molecular:614.57Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Fórmula:C25H29ClF6N2O3Cor e Forma:SolidPeso molecular:554.95d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Fórmula:C52H75N13O13S2Pureza:99.86%Cor e Forma:SolidPeso molecular:1154.37Brimonidine Tartrate
CAS:<p>Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).</p>Fórmula:C15H16BrN5O6Pureza:99.95%Cor e Forma:Off-White Crystalline SolidPeso molecular:442.22Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Fórmula:C27H29N3O2Pureza:98.98% - 99.12%Cor e Forma:SolidPeso molecular:427.54ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Fórmula:C29H29ClN4O2Pureza:99.88%Cor e Forma:SolidPeso molecular:501.02DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Cor e Forma:SolidPeso molecular:424.44Org 27569
CAS:<p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>Fórmula:C24H28ClN3OPureza:>99.99% - ≥95%Cor e Forma:SolidPeso molecular:409.952-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
<p>2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.</p>Fórmula:C38H64F3N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:891.98BAY 41-8543
CAS:<p>BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).</p>Fórmula:C21H21FN8OPureza:99.86%Cor e Forma:SolidPeso molecular:420.44Fenoprofen Calcium
CAS:<p>Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.</p>Fórmula:C30H26CaO6Pureza:99.24% - 99.66%Cor e Forma:SolidPeso molecular:522.6Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Cor e Forma:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Fórmula:C18H24ClN3O2Cor e Forma:SolidPeso molecular:349.86Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Fórmula:C18H19N3O·HClPureza:99.78%Cor e Forma:White PowderPeso molecular:329.82Gastrin I (1-14), human
CAS:Gastrin I (1-14), human: a short peptide from the hormone gastrin, which regulates gastric acid secretion.Fórmula:C79H100N16O27Pureza:98.19%Cor e Forma:SolidPeso molecular:1705.73Tolnapersine
CAS:<p>Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.</p>Fórmula:C21H26N2OPureza:98%Cor e Forma:SolidPeso molecular:322.44Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Fórmula:C19H22ClN3OPureza:98%Cor e Forma:SolidPeso molecular:343.86Ipsapirone hydrochloride
CAS:<p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>Fórmula:C19H24ClN5O3SCor e Forma:SolidPeso molecular:437.94Rimegepant
CAS:<p>View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.</p>Fórmula:C28H28F2N6O3Pureza:99.1% - 99.99%Cor e Forma:SolidPeso molecular:534.56Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Fórmula:C23H27ClFN3O2Pureza:98%Cor e Forma:SolidPeso molecular:431.93ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Fórmula:C19H20N2O3Pureza:99.21%Cor e Forma:SolidPeso molecular:324.37LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Cor e Forma:SolidPeso molecular:226.53PACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), not VIP1.Pureza:98.16%Cor e Forma:LiquidPeso molecular:N/ANeuropeptide W-23(human)
CAS:<p>Neuropeptide W-23(human) (NPW-23) is an endogenous ligand for NPBW1 and NPBW2.</p>Fórmula:C119H183N35O28SPureza:98.5%Cor e Forma:SolidPeso molecular:2584.019-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Fórmula:C7H9N5Pureza:99.35% - 99.41%Cor e Forma:SolidPeso molecular:163.18Montelukast dicyclohexylamine
CAS:<p>Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.</p>Fórmula:C47H59ClN2O3SCor e Forma:SolidPeso molecular:767.5Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Cor e Forma:Almost White To White Crystalline PowderPeso molecular:351.93SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:319.32Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Pureza:97.26%Cor e Forma:LiquidPeso molecular:N/AConopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Fórmula:C43H77N17O12S2Pureza:99.79%Cor e Forma:SolidPeso molecular:1088.32Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Cor e Forma:White SolidPeso molecular:238.24Bombesin acetate(31362-50-2 free base)
CAS:<p>Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).</p>Fórmula:C73H114N24O20SPureza:98.44%Cor e Forma:SolidPeso molecular:1679.92Verucerfont
CAS:<p>Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .</p>Fórmula:C22H26N6O2Pureza:99.90%Cor e Forma:SolidPeso molecular:406.48CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Fórmula:C33H31Cl2F3N6O3S2Pureza:99.08% - 99.76%Cor e Forma:SolidPeso molecular:751.67GUANABENZ
CAS:<p>GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.</p>Fórmula:C8H8Cl2N4Pureza:98.31%Cor e Forma:White Solid From Acetonitrile SolidPeso molecular:231.08Donitriptan Mesylate
CAS:<p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>Fórmula:C24H29N5O5SCor e Forma:SolidPeso molecular:499.58Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Fórmula:C21H27ClN2O2Pureza:99.54% - ≥95%Cor e Forma:Oil SolidPeso molecular:374.9Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Fórmula:C15H24N2O4SCor e Forma:SolidPeso molecular:328.43Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Fórmula:C19H25NOSPureza:98.08% - 99.59%Cor e Forma:SolidPeso molecular:315.47A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Fórmula:C16H26N2O2SPureza:99.94%Cor e Forma:SolidPeso molecular:310.45Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Fórmula:C28H37N3O3Pureza:99.86% - >99.99%Cor e Forma:SolidPeso molecular:463.61Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Fórmula:C149H234N40O47SPureza:98% - 99.65%Cor e Forma:SolidPeso molecular:3369.76Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Fórmula:C5H15ClNO4PPureza:99.481% - 99.85%Cor e Forma:SolidPeso molecular:219.6Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Pureza:98.42%Cor e Forma:LiquidPeso molecular:N/APranlukast hemihydrate
CAS:<p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>Fórmula:C27H23N5O40·5H2OPureza:99.28%Cor e Forma:SolidPeso molecular:490.52carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Fórmula:C24H31N3O2SPureza:98.06%Cor e Forma:SolidPeso molecular:425.59Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Cor e Forma:SolidPeso molecular:446.95Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Fórmula:C17H18ClN4OCor e Forma:SolidPeso molecular:329.11691Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Cor e Forma:SolidPeso molecular:224.26KB-5492 anhydrous
CAS:<p>KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.</p>Fórmula:C27H34N2O10Cor e Forma:SolidPeso molecular:546.57Bindarit
CAS:<p>Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.</p>Fórmula:C19H20N2O3Pureza:98.35% - 98.55%Cor e Forma:SolidPeso molecular:324.37Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Cor e Forma:SolidPeso molecular:369.5N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Fórmula:C9H15N3O3Pureza:98%Cor e Forma:SolidPeso molecular:213.23Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Fórmula:C23H30N2O10Pureza:99.98%Cor e Forma:SolidPeso molecular:494.49Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Cor e Forma:White Crystalline PowderPeso molecular:546.05GLP-1(7-36), amide
CAS:GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Fórmula:C149H226N40O45Pureza:99.85%Cor e Forma:White PowderPeso molecular:3297.63Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Fórmula:C12H14N2·HClPureza:99.97%Cor e Forma:SolidPeso molecular:222.71LIXIVAPTAN
CAS:<p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>Fórmula:C27H21ClFN3O2Pureza:98.36%Cor e Forma:SolidPeso molecular:473.93SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Fórmula:C15H13ClN4O2S2Pureza:97.82% - 98%Cor e Forma:SolidPeso molecular:380.87Calcitonin(salmon) Acetate(47931-85-1(free base))
<p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>Fórmula:C145H240N44O48S2Pureza:99.29%Cor e Forma:SolidPeso molecular:3431.85BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Fórmula:C18H22F3N3O4SPureza:98.05%Cor e Forma:SolidPeso molecular:433.45Motilin (26-47), human, porcine
CAS:<p>Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.</p>Fórmula:C120H188N34O35SPureza:98%Cor e Forma:SolidPeso molecular:2699.07AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Fórmula:C27H23ClN2O5Pureza:98.06% - 99.79%Cor e Forma:SolidPeso molecular:490.93Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Cor e Forma:SolidML-184
CAS:<p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>Fórmula:C25H34N4O3SPureza:99.45%Cor e Forma:SolidPeso molecular:470.63
![[Lys8, Lys9]-Neurotensin (8-13) acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT38807L.webp&w=3840&q=75)
![[Pyr1]-Apelin-13](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1260.webp&w=3840&q=75)
![d[Cha4]-AVP acetate(500170-27-4 free base)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2082L.webp&w=3840&q=75)
