GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Fórmula:C26H32N2O7Cor e Forma:SolidPeso molecular:484.549Sortilin antagonist 1
CAS:<p>Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.</p>Fórmula:C20H24N2O4Cor e Forma:SolidPeso molecular:356.42OX2R-IN-1
CAS:<p>OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.</p>Fórmula:C20H28ClN3O5SCor e Forma:SolidPeso molecular:457.97Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55MRS1097
CAS:<p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>Fórmula:C26H27NO4Pureza:98%Cor e Forma:SolidPeso molecular:417.5CBK289001
CAS:<p>CBK289001 inhibits TRAP 5b MV, 5b OX & 5a OX with IC50s: 125μM, 4.21μM, 14.2μM.</p>Fórmula:C19H20N6O4Cor e Forma:SolidPeso molecular:396.4GPR183-IN-2
CAS:<p>GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.</p>Fórmula:C19H23BrN2O3Cor e Forma:SolidPeso molecular:407.3SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Fórmula:C18H31ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:374.97Fulimetibant
CAS:<p>Fulimetibant is a bradykinin receptor antagonist.</p>Fórmula:C25H21F4N3O3Cor e Forma:SolidPeso molecular:487.45TBC3711
CAS:<p>TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.</p>Fórmula:C20H21N3O5S2Pureza:98%Cor e Forma:SolidPeso molecular:447.53Ranitidine bismuth citrate
CAS:<p>Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.</p>Fórmula:C19H27BiN4O10SCor e Forma:SolidPeso molecular:712.48Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Fórmula:C23H28ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:413.94LY320135
CAS:CB1 receptor antagonist/inverse agonistFórmula:C24H17NO4Pureza:98%Cor e Forma:SolidPeso molecular:383.4GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Fórmula:C21H19ClN2O5SCor e Forma:SolidPeso molecular:446.9(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SCor e Forma:SolidPeso molecular:322.47SDZ NKT 343
CAS:<p>human tachykinin NK1 receptor antagonist</p>Fórmula:C33H33N5O5Pureza:98%Cor e Forma:SolidPeso molecular:579.65Fenmetozole
CAS:<p>Fenmetozole is an antagonist of the actions of ethanol.</p>Fórmula:C10H10Cl2N2OCor e Forma:SolidPeso molecular:245.11Prasugrel (Maleic acid)
CAS:<p>Prasugrel Maleic acid: oral P2Y12 antagonist, thienopyridine prodrug, inhibits ADP-induced platelet aggregation.</p>Fórmula:C24H24FNO7SPureza:98%Cor e Forma:SolidPeso molecular:489.51KUL-7211 racemate
CAS:<p>KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.</p>Fórmula:C19H23NO5Pureza:98%Cor e Forma:SolidPeso molecular:345.39A-304121
CAS:<p>A-304121 is a histamine H(3) receptor.</p>Fórmula:C20H29N3O3Cor e Forma:SolidPeso molecular:359.46GSK466317A
CAS:GSK466317A is a GRK2 inhibitor.Fórmula:C21H16ClF3N4O2Pureza:98%Cor e Forma:SolidPeso molecular:448.83CB1R Allosteric modulator 4
CAS:<p>Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.</p>Fórmula:C20H17N3O2SCor e Forma:SolidPeso molecular:363.43AZ-GHS-22
CAS:<p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>Fórmula:C27H33ClN6O5S2Cor e Forma:SolidPeso molecular:621.17GP531
CAS:<p>GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.</p>Fórmula:C16H21N5O4Cor e Forma:SolidPeso molecular:347.37S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Fórmula:C21H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:336.43CGP 25454A
CAS:CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.Fórmula:C15H21Cl2N3O2Cor e Forma:SolidPeso molecular:346.25R-SKF-38393A HCl
CAS:R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.Fórmula:C16H18ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:291.775-Methylurapidil
CAS:<p>5-Methylurapidil is an alpha1A-adrenoceptor antagonist.</p>Fórmula:C21H31N5O3Pureza:98%Cor e Forma:SolidPeso molecular:401.5ER819762
CAS:<p>ER819762, an antagonist of the prostaglandin E2 EP4 receptor, inhibits Th1 differentiation and Th17 expansion.</p>Fórmula:C30H39N3O3Cor e Forma:SolidPeso molecular:489.65DR4485 hydrochloride
CAS:<p>5-HT7 antagonist</p>Fórmula:C26H29Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:491.88OSU 6162 hydrochloride
CAS:Dopamine stabilizerFórmula:C15H24ClNO2SPureza:98%Cor e Forma:SolidPeso molecular:317.88LG 82-4-01
CAS:LG 82-4-01 is an inhibitor of thromboxane (TX) synthetase.Fórmula:C10H10Cl2N2O3SPureza:98%Cor e Forma:SolidPeso molecular:309.17XCC
CAS:<p>XCC is an Adenosine receptor antagonist.</p>Fórmula:C19H22N4O5Pureza:98%Cor e Forma:SolidPeso molecular:386.4S1P1 Agonist III
CAS:<p>S1P1 Agonist III is an effective and orally active S1P1 agonist (EC50: 18 nM).</p>Fórmula:C21H16F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:415.37HEAT hydrochloride
CAS:<p>HEAT hydrochloride is an α1-adrenoceptor antagonist.</p>Fórmula:C19H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:331.84MK-212
CAS:<p>MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.</p>Fórmula:C8H11ClN4Cor e Forma:SolidPeso molecular:198.65MRS2179 tetrasodium
CAS:<p>competitive antagonist at P2Y1 receptors</p>Fórmula:C11H17N5Na4O9P2Pureza:98%Cor e Forma:SolidPeso molecular:517.19JTC-017
CAS:<p>JTC-017 is an antagonist of Corticotropin-releasing hormone receptor 1.</p>Fórmula:C20H25Cl2N3O5SCor e Forma:SolidPeso molecular:490.4ANEB-001
CAS:<p>ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.</p>Fórmula:C22H24ClF3N2O2Cor e Forma:SolidPeso molecular:440.89hBChE-IN-2
CAS:<p>hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.</p>Fórmula:C27H36N4O3Pureza:99.60% - 99.83%Cor e Forma:SoildPeso molecular:464.6Sulfisoxazole diethanolamine
CAS:<p>Sulfisoxazole diethanolamine: a sulfonamide antibacterial, endothelin receptors A and B antagonist, inhibits breast cancer exosomes.</p>Fórmula:C15H24N4O5SCor e Forma:SolidPeso molecular:372.44Zinterol hydrochloride
CAS:<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Fórmula:C19H27ClN2O4SCor e Forma:SolidPeso molecular:414.95Isoetharine
CAS:<p>Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.</p>Fórmula:C13H21NO3Cor e Forma:SolidPeso molecular:239.31Imnopitant
CAS:<p>Imnopitant is an antagonist of the NK1 receptor [1].</p>Fórmula:C28H28F6N4OCor e Forma:SolidPeso molecular:550.54R 75317
CAS:<p>R 75317 is a Platelet-activating factor (PAF) antagonist.</p>Fórmula:C29H50N3O8PSPureza:98%Cor e Forma:SolidPeso molecular:631.76E2508
CAS:<p>E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.</p>Fórmula:C36H47N3O7SPureza:98%Cor e Forma:SolidPeso molecular:665.84Trimipramine
CAS:<p>Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.</p>Fórmula:C20H26N2Pureza:98%Cor e Forma:SolidPeso molecular:294.43S-22153
CAS:<p>S22153 is an antagonist of melatonin receptor.</p>Fórmula:C14H17NOSCor e Forma:SolidPeso molecular:247.36GR 128107
CAS:<p>GR 128107 is an antagonist of melatonin receptor.</p>Fórmula:C16H20N2O2Cor e Forma:SolidPeso molecular:272.34EMD 386088 hydrochloride
CAS:<p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>Fórmula:C14H16Cl2N2Pureza:98%Cor e Forma:SolidPeso molecular:283.2HAMI 3379
CAS:<p>HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.</p>Fórmula:C34H45NO8Pureza:99.75%Cor e Forma:SolidPeso molecular:595.72Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Fórmula:C23H30N6O6Pureza:98%Cor e Forma:SolidPeso molecular:486.52Guanadrel
CAS:<p>Guanadrel is an antihypertensive agent.</p>Fórmula:C10H19N3O2Pureza:98%Cor e Forma:SolidPeso molecular:213.28PF-04628935
CAS:<p>PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.</p>Fórmula:C24H26ClN7OSPureza:98%Cor e Forma:SolidPeso molecular:496.03SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Fórmula:C15H13N3SPureza:98%Cor e Forma:SolidPeso molecular:267.35(2R,3R)-E1R
CAS:(2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.Fórmula:C13H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:232.28LEI 101 hydrochloride
CAS:<p>LEI 101 hydrochloride is potent and selective CB2 partial agonist.</p>Fórmula:C23H26ClFN4O4SCor e Forma:SolidPeso molecular:508.99Prostaglandin D2
CAS:<p>Prostaglandin D2 (PGD2) is one of the major PGs actively produced in the brain of various mammals,and is a potent endogenous sleep promoting substances.</p>Fórmula:C20H32O5Pureza:>99.99%Cor e Forma:SolidPeso molecular:352.47Arbutamine hydrochloride
CAS:<p>Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.</p>Fórmula:C18H24ClNO4Cor e Forma:SolidPeso molecular:353.84Zinterol
CAS:<p>Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).</p>Fórmula:C19H26N2O4SPureza:98%Cor e Forma:SolidPeso molecular:378.49Modipafant
CAS:<p>Modipaafant is a potent dihydropyridine PAF (platelet activating factor) antagonist.</p>Fórmula:C34H29ClN6O3Cor e Forma:SolidPeso molecular:605.09Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48GTS-21
CAS:<p>GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.</p>Fórmula:C19H20N2O2Pureza:98%Cor e Forma:SolidPeso molecular:308.37SKI 5C
CAS:SKI 5C is a selective inhibitor of Sphingosine Kinase 1.Fórmula:C26H45NO4Pureza:98%Cor e Forma:SolidPeso molecular:435.64IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SCor e Forma:SolidPeso molecular:373.51JNJ-40255293
CAS:<p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>Fórmula:C23H22N4O3Pureza:98%Cor e Forma:SolidPeso molecular:402.45Mabuterol hydrochloride
CAS:<p>Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.</p>Fórmula:C13H19Cl2F3N2OCor e Forma:SolidPeso molecular:347.20BMS-466442
CAS:<p>BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.</p>Fórmula:C31H30N4O5Cor e Forma:SolidPeso molecular:538.59DMP 696
CAS:<p>DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.</p>Fórmula:C18H21Cl2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:410.3Metrenperone
CAS:<p>Metrenperone is used as a S(2)-receptor blocker.</p>Fórmula:C24H26FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:407.48NPEC-caged-dopamine
CAS:<p>Dopamine receptor agonist</p>Fórmula:C17H18N2O6Pureza:98%Cor e Forma:SolidPeso molecular:346.33BI-L 239
CAS:BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.Fórmula:C16H15FOCor e Forma:SolidPeso molecular:242.29PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Fórmula:C21H25Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:438.35MS-0022
CAS:<p>MS-0022: SMO antagonist, inhibits Hh signaling in nM-µM ranges, curbs tumor cell growth, and delays tumor progression in vivo.</p>Fórmula:C21H16BrN3OCor e Forma:SolidPeso molecular:406.28Guanoxabenz hydrochloride
CAS:<p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>Fórmula:C8H9Cl3N4OCor e Forma:SolidPeso molecular:283.54Alprenolol tartrate, (S)-
CAS:<p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>Fórmula:C19H29NO8Pureza:98%Cor e Forma:SolidPeso molecular:399.44Etersalate
CAS:<p>Etersalate inhibits platelet function. It also reduces thromboxane A2 (TXA2) levels.</p>Fórmula:C19H19NO6Pureza:98%Cor e Forma:SolidPeso molecular:357.36Bufetolol
CAS:Bufetolol is an antagonist of beta-adrenoceptor.Fórmula:C18H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:323.43Deramciclane fumarate
CAS:<p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>Fórmula:C24H35NO5Cor e Forma:SolidPeso molecular:417.54Kadsurenone
CAS:<p>Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.</p>Fórmula:C21H24O5Cor e Forma:SolidPeso molecular:356.41Mosapramine
CAS:<p>Mosapramine is a dopamine D2-receptor antagonist.</p>Fórmula:C28H35ClN4OPureza:98%Cor e Forma:SolidPeso molecular:479.06Vestipitant
CAS:<p>Vestipitant (GW597599): a potent NK1 antagonist, may treat anxiety, depression, nausea, tinnitus, insomnia.</p>Fórmula:C23H24F7N3OCor e Forma:SolidPeso molecular:491.45SNT-207858 free base
CAS:<p>SNT-207858: selective MC-4 receptor antagonist, passes blood-brain barrier, orally active, IC50: 22 nM (binding), 11 nM (function).</p>Fórmula:C32H43Cl2N5O3Pureza:98%Cor e Forma:SolidPeso molecular:616.62Avosentan
CAS:<p>Avosentan（Ro 67-0565; SPP-301） is a potent endothelin receptor (ETA) antagonist.Cost-effective and quality-assured.</p>Fórmula:C23H21N5O5SPureza:98.31% - 99.47%Cor e Forma:SolidPeso molecular:479.515-HT6/5-HT2A receptor ligand-2
CAS:<p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>Fórmula:C20H18FN3O2Cor e Forma:SolidPeso molecular:351.37CCK-B Receptor Antagonist 2
CAS:<p>CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).</p>Fórmula:C27H28N6O3Cor e Forma:SolidPeso molecular:484.55CCG-224406
CAS:<p>CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.</p>Fórmula:C29H27FN6O5Cor e Forma:SolidPeso molecular:558.56I942
CAS:<p>I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilical</p>Fórmula:C20H19NO4SPureza:99.75%Cor e Forma:SolidPeso molecular:369.43Tetrahydrozoline nitrate
CAS:<p>Tetrahydrozoline, an imidazoline derivative, is an α-adrenergic agonist for nasal and eye congestion studies.</p>Fórmula:C13H17N3O3Cor e Forma:SolidPeso molecular:263.297Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Cor e Forma:SolidPeso molecular:369.29BMS-665053
CAS:<p>BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.</p>Fórmula:C16H14Cl3F2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:424.66CYM-5478
CAS:<p>CYM-5478, a strong S1P2 agonist, boosts C6 cell survival over 100nM under serum-starvation.</p>Fórmula:C21H19F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:388.38Talipexole
CAS:<p>Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.</p>Fórmula:C10H15N3SPureza:98%Cor e Forma:SolidPeso molecular:209.31Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Fórmula:C23H32Cl2FN3Pureza:98%Cor e Forma:SolidPeso molecular:440.42RXFP3/4 agonist 2
CAS:<p>RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.</p>Fórmula:C22H22N6O2Pureza:99.82%Cor e Forma:SolidPeso molecular:402.45Iso-SLR 080811
CAS:<p>Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).</p>Fórmula:C21H32ClN5OPureza:98.34%Cor e Forma:SolidPeso molecular:405.97JNJ-28610244
CAS:<p>JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.</p>Fórmula:C16H21N3OPureza:98%Cor e Forma:SolidPeso molecular:271.36Hedgehog IN-3
CAS:<p>Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].</p>Fórmula:C18H13ClF3N5OCor e Forma:SolidPeso molecular:407.78Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Cor e Forma:White To Pink PowderPeso molecular:291.39MK-4256
CAS:MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).Fórmula:C27H23FN8OCor e Forma:SolidPeso molecular:494.52RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:363.28CFM 1571 hydrochloride
CAS:<p>CFM 1571 hydrochloride stimulates sGC with EC50 of 5.49 μM; potential for cardiovascular research.</p>Fórmula:C23H29ClN4O3Cor e Forma:SolidPeso molecular:444.965-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45Isothipendyl hydrochloride
CAS:<p>Isothipendyl hydrochloride is a 1st generation H1 antagonist.</p>Fórmula:C16H20ClN3SCor e Forma:SolidPeso molecular:321.87CB1 inverse agonist 2
CAS:<p>CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.</p>Fórmula:C24H20ClFN2OSCor e Forma:SolidPeso molecular:438.94Acreozast
CAS:<p>Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.</p>Fórmula:C15H14ClN3O6Cor e Forma:SolidPeso molecular:367.74JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Cor e Forma:SolidPeso molecular:312.45FR-A 19
CAS:<p>FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.</p>Fórmula:C25H34Cl3F2N5Cor e Forma:SolidPeso molecular:548.93Methylcarbamyl PAF C-16
CAS:<p>Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.</p>Fórmula:C26H55N2O7PCor e Forma:SolidPeso molecular:538.7DW-1350
CAS:<p>DW-1350 is an antagonist of LTB4 receptor.</p>Fórmula:C25H31N3O3SPureza:98%Cor e Forma:SolidPeso molecular:453.6LY 344864 hydrochloride
CAS:<p>LY 344864 hydrochloride is a selective receptor agonist with an affinity of 6 nM (Ki) at the 5-HT1F receptor.</p>Fórmula:C21H23ClFN3OCor e Forma:SolidPeso molecular:387.88Phenindamine
CAS:<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Fórmula:C19H19NCor e Forma:SolidPeso molecular:261.36Eplivanserin hemifumarate
CAS:<p>Eplivanserin is an inverse agonist of 5-HT2A.</p>Fórmula:C23H25FN2O6Cor e Forma:SolidPeso molecular:444.45VUF-10497
CAS:<p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>Fórmula:C18H20ClN5SPureza:98%Cor e Forma:SolidPeso molecular:373.9BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Fórmula:C12H19N5O2S2Pureza:98%Cor e Forma:SolidPeso molecular:329.44A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Fórmula:C17H21N5Cor e Forma:SolidPeso molecular:295.38AM404
CAS:<p>AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.</p>Fórmula:C26H37NO2Cor e Forma:SolidPeso molecular:395.58(R)-V-0219
<p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>Fórmula:C20H25F3N4O2Cor e Forma:SolidPeso molecular:410.43L-733060 hydrochloride
CAS:<p>Potent NK1 antagonist</p>Fórmula:C20H20ClF6NOPureza:98%Cor e Forma:SolidPeso molecular:439.82S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFórmula:C6H11NO2SPureza:98%Cor e Forma:SolidPeso molecular:161.22Fenmetozole HCl
CAS:<p>Fenmetozole HCl is an antagonist of the actions of ethanol. It attenuates the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate content.</p>Fórmula:C10H11Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:281.57UCM710
CAS:<p>UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).</p>Fórmula:C19H34O3Pureza:98%Cor e Forma:SolidPeso molecular:310.47UNC9995
CAS:<p>UNC9995 is a β-Arrestin-Biased Dopamine D2 Receptor agonist (β-Arrestin, EC50 = 120 nM; Emax = 88%).</p>Fórmula:C20H21Cl2N3OSPureza:98%Cor e Forma:SolidPeso molecular:422.37SDZ 21009
CAS:<p>β-adrenoceptor and 5-HT1A/1B receptor antagonist</p>Fórmula:C19H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:348.44Adrenaline sulfate
CAS:<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Fórmula:C9H15NO7SCor e Forma:SolidPeso molecular:281.279PROTAC(H-PGDS)-7
CAS:<p>PROTAC(H-PGDS)-7, a potent H-PGDS degrader, inhibits PGD2 in KU812 cells; DC50 is 17.3 pM. Potential DMD treatment.</p>Fórmula:C40H38N8O7Cor e Forma:SolidPeso molecular:742.78hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Fórmula:C15H15N5OCor e Forma:SolidPeso molecular:281.31Anatibant
CAS:<p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>Fórmula:C34H36Cl2N6O5SPureza:98%Cor e Forma:SolidPeso molecular:711.66CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Fórmula:C19H28ClN5OPureza:99.72%Cor e Forma:SolidPeso molecular:377.91LUF 5834
CAS:A2A and A2B adenosine receptor partial agonistFórmula:C17H12N6OSPureza:98%Cor e Forma:SolidPeso molecular:348.38SF 11
CAS:<p>SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activity</p>Fórmula:C27H30N2O2SPureza:99.51%Cor e Forma:SolidPeso molecular:446.6ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Fórmula:C12H16N8OPureza:98%Cor e Forma:SolidPeso molecular:288.31AGI-41998
CAS:<p>AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.</p>Fórmula:C22H16BrF3N4O2Cor e Forma:SolidPeso molecular:505.29Palmitoyl serinol
CAS:<p>Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.</p>Fórmula:C19H39NO3Cor e Forma:SolidPeso molecular:329.52Eplivanserin
CAS:<p>Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.</p>Fórmula:C19H21FN2O2Pureza:97.04%Cor e Forma:SolidPeso molecular:328.38Pirolate
CAS:<p>Pirolate is a receptor of histamine H1.</p>Fórmula:C16H15N3O5Pureza:98%Cor e Forma:SolidPeso molecular:329.31SNT-207858
CAS:<p>SNT-207858: selective, BBB-penetrating, oral MC-4 receptor antagonist with 22 nM IC50 (binding), 11 nM (function).</p>Fórmula:C32H45Cl4N5O3Pureza:98%Cor e Forma:SolidPeso molecular:689.54Lu AA 47070
CAS:<p>adenosine A2A receptor antagonist</p>Fórmula:C17H20F2N3O6PSPureza:98%Cor e Forma:SolidPeso molecular:463.39BMS-192364
CAS:<p>BMS-192364 is a bio-active chemical.</p>Fórmula:C15H9ClF3N3O2Cor e Forma:SolidPeso molecular:355.70DOV-216,303 Free Base
CAS:<p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>Fórmula:C11H11Cl2NPureza:96.7%Cor e Forma:SolidPeso molecular:228.12EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Fórmula:C15H22N2OPureza:97.66% - 99.78%Cor e Forma:SolidPeso molecular:246.35Chlorazanil
CAS:<p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>Fórmula:C9H8ClN5Pureza:98.89%Cor e Forma:SolidPeso molecular:221.65CAY10590
CAS:<p>CAY10590 (GK115) inhibits sPLA2, used in chronic kidney inflammation research.</p>Fórmula:C21H33NO3Cor e Forma:SolidPeso molecular:347.49A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Fórmula:C17H12N4OCor e Forma:SolidPeso molecular:288.3Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34PRX933 hydrochloride
CAS:<p>PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.</p>Fórmula:C16H22ClN5O2Pureza:99.51% - 99.89%Cor e Forma:SolidPeso molecular:351.84Iferanserin
CAS:Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Fórmula:C23H28N2OCor e Forma:SolidPeso molecular:348.48RP101988
<p>RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.</p>Fórmula:C23H22N4O4Cor e Forma:SolidPeso molecular:418.45Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Fórmula:C20H31NOCor e Forma:SolidPeso molecular:301.47AS604872
CAS:<p>AS604872: Selective FP receptor antagonist, expedites cerebral/aorta degeneration, aids vascular disease models, inhibits uterine contraction.</p>Fórmula:C28H25N3O3S2Cor e Forma:SolidPeso molecular:515.65SKF83822 hydrobromide
CAS:<p>SKF83822 hydrobromide is a dopamine D1-like receptor agonist.</p>Fórmula:C20H23BrClNO2Pureza:98%Cor e Forma:SolidPeso molecular:424.76GRK5-IN-4
CAS:<p>GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.</p>Fórmula:C26H25N7O3Cor e Forma:SolidPeso molecular:483.52LY 306669
CAS:LY 306669 is an antagonist of leukotriene B4 receptor.Fórmula:C23H29FN4NaO2Cor e Forma:SolidPeso molecular:435.499JPC-211
CAS:<p>JPC-211 is an agonist of dopamine-receptor.</p>Fórmula:C17H27NO2Pureza:98%Cor e Forma:SolidPeso molecular:277.4PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Cor e Forma:SolidPeso molecular:315.24Gastrazole disodium
CAS:<p>Gastrazole, a CCK2 receptor antagonist, is used potentially for the treatment of pancreatic cancer.</p>Fórmula:C34H34FN5Na2O7Cor e Forma:SolidPeso molecular:689.652(±)-Tazifylline
CAS:<p>(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.</p>Fórmula:C23H32N6O3SPureza:99.54%Cor e Forma:SolidPeso molecular:472.6MRS2603
CAS:<p>MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.</p>Fórmula:C14H12ClN4O8PPureza:98%Cor e Forma:SolidPeso molecular:430.69Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Fórmula:C14H19ClN4O2Pureza:98%Cor e Forma:SolidPeso molecular:310.78Midodrine D6 hydrochloride
CAS:<p>Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.</p>Fórmula:C12H19ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:296.785-Carboxamidotryptamine maleate
CAS:<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31Mirisetron
CAS:<p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>Fórmula:C24H31N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:393.52TAS 205
CAS:<p>TAS 205 blocks H-PGDS (IC50= 55.8 nM), beats L-PGDS at 100 μM. Reduces PGD2 in human/rat basophils, dampens allergy in guinea pigs (30 mg/kg).</p>Fórmula:C27H38N6O5Cor e Forma:SolidPeso molecular:526.638ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Fórmula:C11H17F3N6OPureza:97.45%Cor e Forma:SolidPeso molecular:306.29Nafadotride
CAS:<p>Nafadotride is a dopamine D3 receptor antagonist.</p>Fórmula:C22H27N3O2Cor e Forma:SolidPeso molecular:365.472-CMDO
CAS:<p>2-CMDO is a Dopamine D2-like receptor antagonist.</p>Fórmula:C23H23ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:442.89Fluphenazine Decanoate Dihydrochloride
CAS:<p>Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.</p>Fórmula:C32H46Cl2F3N3O2SPureza:98%Cor e Forma:SolidPeso molecular:664.69PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Fórmula:C23H21ClFN5O4SPureza:97.59%Cor e Forma:SolidPeso molecular:517.96EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Cor e Forma:SolidPeso molecular:393.522Bemesetron
CAS:<p>Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.</p>Fórmula:C15H17Cl2NO2Pureza:99.77%Cor e Forma:SolidPeso molecular:314.21RXFP3 agonist 1
CAS:<p>RXFP3 agonist 1 is a nonpeptide RXFP3 agonist ( EC 50 =6937 nM) [1].</p>Fórmula:C18H18ClN5Cor e Forma:SolidPeso molecular:339.82YM-264
CAS:<p>YM-264 is a selective and orally active antagonist of platelet-activating factor (PAF) (pKi value of 8.85 for rabbit platelet membranes).</p>Fórmula:C28H36N4O5SPureza:98%Cor e Forma:SolidPeso molecular:540.67SK1-IN-1
CAS:SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be used to study cancer and neurodegenerative diseases.Fórmula:C22H30N4O3Pureza:98.72%Cor e Forma:SolidPeso molecular:398.5Fallypride
CAS:<p>Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.</p>Fórmula:C20H29FN2O3Pureza:98.97% - >99.99%Cor e Forma:SolidPeso molecular:364.45A2A/A1 AR antagonist-1
CAS:<p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>Fórmula:C15H12N6O2Cor e Forma:SolidPeso molecular:308.29Epanolol
CAS:<p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>Fórmula:C20H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:369.41Proglumide sodium
CAS:Non-selective cholecystokinin (CCK) antagonistFórmula:C18H26N2NaO4Pureza:98%Cor e Forma:SolidPeso molecular:357.4Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Fórmula:C18H22BrNSPureza:99.65%Cor e Forma:SolidPeso molecular:364.34Thioproperazine
CAS:<p>Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.</p>Fórmula:C22H30N4O2S2Pureza:99.45%Cor e Forma:SolidPeso molecular:446.63Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Fórmula:C31H35F6N4O5PPureza:98%Cor e Forma:SolidPeso molecular:688.6MS47134
<p>MS47134: potent MRGPRX4 agonist, EC50 = 149 nM, for pain/itch/hypersensitivity research.</p>Fórmula:C22H29NO3Cor e Forma:SolidPeso molecular:355.47MAT2A-IN-2
CAS:<p>MAT2A-IN-2 is a potent inhibitor of MAT2A. MAT2A-IN-2 has potential for cancer disease research.</p>Fórmula:C23H17F3N6O2Cor e Forma:SolidPeso molecular:466.42GT 2016
CAS:<p>GT 2016 is a H3 receptor antagonist.</p>Fórmula:C19H31N3OPureza:98%Cor e Forma:SolidPeso molecular:317.47A 987306
CAS:<p>A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.</p>Fórmula:C18H25N5OCor e Forma:SolidPeso molecular:327.42Bavisant dihydrochloride
CAS:<p>Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.</p>Fórmula:C19H29Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:402.36LY 125180
CAS:LY 125180 is a serotonin antagonist.Fórmula:C18H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:305.84B 4148
CAS:<p>B 4148 is a bradykinin inhibitor.</p>Fórmula:C62H95N19O14S2Cor e Forma:SolidPeso molecular:1394.67LUF6000
CAS:LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).Fórmula:C22H20Cl2N4Cor e Forma:SolidPeso molecular:411.33Guanoxabenz
CAS:<p>Guanoxabenz is an α2 adrenergic receptor agonist.</p>Fórmula:C8H8Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:247.08TSHR antagonist S37a
CAS:TSHR antagonist S37a is a selective, orally bioavailable TSHR antagonist that inhibits TSH-induced cAMP in TSHR-expressing HEK 293 cells.Fórmula:C25H20N2O3S2Pureza:98%Cor e Forma:SolidPeso molecular:460.57AB-MECA
CAS:<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Fórmula:C18H21N7O4Pureza:98%Cor e Forma:SolidPeso molecular:399.4A1/A3 AR antagonist 2
CAS:<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Fórmula:C22H16N2O3SCor e Forma:SolidPeso molecular:388.44BAY-27-9955
CAS:<p>BAY-27-9955 is a glucagon receptor antagonist.</p>Fórmula:C23H31FOCor e Forma:SolidPeso molecular:342.49YQA14
CAS:<p>YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.</p>Fórmula:C23H27ClN4O3Pureza:99.52%Cor e Forma:SolidPeso molecular:442.94LUF 6283
CAS:partial agonist of hydroxycarboxylic acid receptor 2 (HCA2)Fórmula:C8H12N2O2Cor e Forma:SolidPeso molecular:168.19CB1/2 agonist 4
CAS:<p>CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.</p>Fórmula:C27H45NO3Cor e Forma:SolidPeso molecular:431.65(S)-Terazosin
CAS:<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43
