GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(942 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.948 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(149 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(409 produtos)
- Receptor Endotelina(75 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(32 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(166 produtos)
- Hedgehog/Smoothened(45 produtos)
- Receptor de Histamina(359 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(298 produtos)
- PAFR(11 produtos)
- PKA(49 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5373 produtos de "GPCR/Proteína-G"
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Nelonicline
CAS:<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Fórmula:C17H19N3OSPureza:98%Cor e Forma:SolidPeso molecular:313.42(Iso)-FK-480
CAS:(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.Fórmula:C26H19FN4O2Pureza:98.36% - 99.41%Cor e Forma:SolidPeso molecular:438.45(S)-(-)-Propranolol hydrochloride
CAS:<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。</p>Fórmula:C16H22ClNO2Pureza:99.02% - 99.91%Cor e Forma:SolidPeso molecular:295.8PA-9
CAS:<p>PA-9 is the first small-molecule PAC1 receptor antagonist.</p>Fórmula:C17H18N6O2Pureza:98%Cor e Forma:SolidPeso molecular:338.36PM226
CAS:<p>CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.</p>Fórmula:C22H31NO3Cor e Forma:SolidPeso molecular:357.49AM404
CAS:<p>AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.</p>Fórmula:C26H37NO2Cor e Forma:SolidPeso molecular:395.58S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SCor e Forma:SolidPeso molecular:470.45GSK-345931A
CAS:<p>GSK-345931A is an EP(1) antagonist with CNS uptake in mice/rats, offering strong pain relief in acute and prolonged inflammation.</p>Fórmula:C22H20ClNNaO3Cor e Forma:SolidPeso molecular:404.85AZD-1678
CAS:<p>AZD-1678 is a potent CCR4 receptor antagonist.</p>Fórmula:C11H8Cl2FN3O3SCor e Forma:SolidPeso molecular:352.17Idremcinal
CAS:<p>Idremcinal is a motilin receptor agonist.</p>Fórmula:C39H69NO12Cor e Forma:SolidPeso molecular:743.96CCG-273463
CAS:<p>CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.</p>Fórmula:C26H25BrN4O3Cor e Forma:SolidPeso molecular:521.41Acetylaszonalenin
CAS:<p>Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.</p>Fórmula:C25H25N3O3Cor e Forma:SolidPeso molecular:415.48Pargolol hydrochloride
CAS:<p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>Fórmula:C16H24ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:313.82CCR8 antagonist 2
CAS:<p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>Fórmula:C23H30ClN3O3SCor e Forma:SolidPeso molecular:464.02CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Fórmula:C24H19F3O4Cor e Forma:SolidPeso molecular:428.4ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Fórmula:C25H29BrF3N5OCor e Forma:SolidPeso molecular:552.43SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Fórmula:C17H20BrNO2Cor e Forma:SolidPeso molecular:350.25Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Fórmula:C22H27ClN2Cor e Forma:SolidPeso molecular:354.92A 55453
CAS:<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Fórmula:C25H32N6O3Cor e Forma:SolidPeso molecular:464.56LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Cor e Forma:SolidPeso molecular:326.41FRG8701
CAS:<p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>Fórmula:C22H30N2O4SPureza:98%Cor e Forma:SolidPeso molecular:418.55Naronapride
CAS:<p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>Fórmula:C27H41ClN4O5Cor e Forma:SolidPeso molecular:537.09S-777469
CAS:<p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>Fórmula:C23H27FN2O4Cor e Forma:SolidPeso molecular:414.47CB2 receptor agonist 3
CAS:<p>GP 2A is a selective agonist of CB2 receptor.</p>Fórmula:C24H23Cl2N3OCor e Forma:SolidPeso molecular:440.36BAY-u 9773
CAS:<p>BAY-u9773 is a non-selective CysLT receptor antagonist with similar IC50 for CysLT1 and CysLT2, inhibiting LT responses.</p>Fórmula:C27H36O5SCor e Forma:White OilPeso molecular:472.64Edivoxetine
CAS:<p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>Fórmula:C18H26FNO4Cor e Forma:SolidPeso molecular:339.4ChemR23-IN-1
CAS:<p>ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.</p>Fórmula:C28H29N7O2Cor e Forma:SolidPeso molecular:495.58BGC-20-1531 free base
CAS:<p>BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.</p>Fórmula:C26H24N2O6SCor e Forma:SolidPeso molecular:492.54Ko-3290
CAS:<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Fórmula:C19H25N3O3Pureza:98%Cor e Forma:SolidPeso molecular:343.42GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Fórmula:C28H26N4O2Cor e Forma:SolidPeso molecular:450.53SSTR4 agonist 2
CAS:<p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>Fórmula:C18H24N4OCor e Forma:SolidPeso molecular:312.41ZM 169369
CAS:<p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>Fórmula:C19H20N2SCor e Forma:SolidPeso molecular:308.44RP101442
CAS:<p>RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).</p>Fórmula:C23H22N4O3Cor e Forma:SolidPeso molecular:402.45FR-194921
CAS:<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Fórmula:C23H23N5OCor e Forma:SolidPeso molecular:385.46Methapyrilene
CAS:<p>Methapyrilene is a histamine H1 antagonist with sedative action.</p>Fórmula:C14H19N3SCor e Forma:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Peso molecular:261.39PGN36
CAS:<p>PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).</p>Fórmula:C21H23N3O3Cor e Forma:SolidPeso molecular:365.43S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Fórmula:C16H20ClN3OSCor e Forma:SolidPeso molecular:337.87Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Fórmula:C31H56N2O8SPureza:98%Cor e Forma:SolidPeso molecular:616.85(Rac)-SEP-363856
CAS:<p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>Fórmula:C9H13NOSPureza:98%Cor e Forma:SolidPeso molecular:183.27Neladenoson dalanate HCl
CAS:<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Fórmula:C35H35Cl2N7O4S2Pureza:98%Cor e Forma:SolidPeso molecular:752.73UCSF686
CAS:<p>UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.</p>Fórmula:C14H19N3O2SCor e Forma:SolidPeso molecular:293.38RB-005
CAS:<p>RB-005 is a potent SK1 inhibitor with IC(50) of 3.6 μM, potentially treating proliferative diseases like hypertension and degrades SK1 in human cells.</p>Fórmula:C21H35NOCor e Forma:SolidPeso molecular:317.51S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Fórmula:C21H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:336.43ER819762
CAS:<p>ER819762, an antagonist of the prostaglandin E2 EP4 receptor, inhibits Th1 differentiation and Th17 expansion.</p>Fórmula:C30H39N3O3Cor e Forma:SolidPeso molecular:489.65OSU 6162 hydrochloride
CAS:Dopamine stabilizerFórmula:C15H24ClNO2SPureza:98%Cor e Forma:SolidPeso molecular:317.88Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Fórmula:C20H19N3O4SCor e Forma:SolidPeso molecular:397.45Ro 60-0175 fumarate
CAS:<p>5-HT2 receptor agonist</p>Fórmula:C15H16ClFN2O4Pureza:98%Cor e Forma:SolidPeso molecular:342.75(+/-)-PPCC oxalate
CAS:<p>Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 & 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.</p>Fórmula:C50H60N2O10Cor e Forma:SolidPeso molecular:849.034Quininib
CAS:<p>Quininib inhibits ocular angiogenesis, blocks HMEC-1 tubules, aortic sprouts, and retinal revascularization in OIR mice.</p>Fórmula:C17H13NOPureza:99.81%Cor e Forma:SolidPeso molecular:247.29MS-0022
CAS:<p>MS-0022: SMO antagonist, inhibits Hh signaling in nM-µM ranges, curbs tumor cell growth, and delays tumor progression in vivo.</p>Fórmula:C21H16BrN3OCor e Forma:SolidPeso molecular:406.28Etersalate
CAS:<p>Etersalate inhibits platelet function. It also reduces thromboxane A2 (TXA2) levels.</p>Fórmula:C19H19NO6Pureza:98%Cor e Forma:SolidPeso molecular:357.36Mrgx2 antagonist-1
CAS:Mrgx2 antagonist-1 is a potent antagonist of Mrgx2 (Mas-related Gene X2) and can be used to study Mrgx2-mediated diseases and disorders.Fórmula:C23H26F5N5O3Cor e Forma:SolidPeso molecular:515.48PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Cor e Forma:SolidPeso molecular:554.34T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Fórmula:C56H62N6O8Pureza:98%Cor e Forma:SolidPeso molecular:947.146A331440
CAS:<p>A331440 is an modulator of L-histidine and histamine H3 receptor.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47Remoxipride
CAS:Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.Fórmula:C16H23BrN2O3Pureza:98%Cor e Forma:SolidPeso molecular:371.27UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Fórmula:C15H18N2O2SCor e Forma:SolidPeso molecular:290.38GR-203040 HCl
CAS:<p>GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.</p>Fórmula:C20H26Cl2N6OCor e Forma:SolidPeso molecular:437.37HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:368.4PGD2-IN-1
CAS:<p>PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.</p>Fórmula:C23H23Cl2N3O3Pureza:98.21%Cor e Forma:SolidPeso molecular:460.35Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Fórmula:C29H29F6N3O2Pureza:98.72%Cor e Forma:SolidPeso molecular:565.55Felypressin acetate
CAS:<p>Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.</p>Fórmula:C48H69N13O13S2Pureza:97.06%Cor e Forma:SolidPeso molecular:1100.27KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Fórmula:C26H32N2O4Cor e Forma:SolidPeso molecular:436.54JHW 007 hydrochloride
CAS:<p>JHW 007 hydrochloride is a Dopamine uptake inhibitor.</p>Fórmula:C24H30ClF2NOPureza:98%Cor e Forma:SolidPeso molecular:421.95ADRA1D receptor antagonist 1 HCl
CAS:<p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>Fórmula:C15H14Cl2N4OPureza:98.13%Cor e Forma:SolidPeso molecular:337.2PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Fórmula:C17H22N4Pureza:98%Cor e Forma:SolidPeso molecular:282.38GW848687X
CAS:GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.Fórmula:C24H18ClF2NO3Pureza:98%Cor e Forma:SolidPeso molecular:441.85cis-Epoxysuccinic acid
CAS:<p>cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.</p>Fórmula:C4H4O5Pureza:99.81%Cor e Forma:SolidPeso molecular:132.07Carbinoxamine
CAS:<p>Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.</p>Fórmula:C16H19ClN2OPureza:98%Cor e Forma:LiquidPeso molecular:290.79Flestolol sulfate
CAS:<p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>Fórmula:C15H24FN3O8SCor e Forma:SolidPeso molecular:425.43hA2A/hCA XII modulator 1
CAS:<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Fórmula:C24H19N7O4SCor e Forma:SolidPeso molecular:501.52Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Fórmula:C20H26N4O5SPureza:98%Cor e Forma:SolidPeso molecular:434.51Ibodutant
CAS:Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).Fórmula:C37H48N4O4SPureza:98%Cor e Forma:SolidPeso molecular:644.87Romifidine
CAS:Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Fórmula:C9H9BrFN3Cor e Forma:SolidPeso molecular:258.09SLV-310
CAS:<p>SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.</p>Fórmula:C25H24FN3O2Pureza:99.39%Cor e Forma:SolidPeso molecular:417.48GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Fórmula:C23H26ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.93Cyclazosin HCl
CAS:<p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>Fórmula:C23H28ClN5O4Pureza:99.10%Cor e Forma:SolidPeso molecular:473.95Ono 6240
CAS:<p>Ono 6240 is an antagonist of platelet-activating factor. Ono 6240 prevents airway eosinophilia by inhibiting production of IL-2 and IL-5.</p>Fórmula:C32H63NO6S2Pureza:98%Cor e Forma:SolidPeso molecular:621.98MRS2567
CAS:MRS2567 is a potent P2Y6 nucleotide receptors antagonists.Fórmula:C16H12N2S2Cor e Forma:SolidPeso molecular:296.41Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81(S)-Carvedilol
CAS:<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47Nα-Methylhistamine dihydrochloride
CAS:<p>Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.</p>Fórmula:C6H13Cl2N3Pureza:98%Cor e Forma:SolidPeso molecular:198.094CJB-090 2HCl
CAS:<p>CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.</p>Fórmula:C26H30Cl4N4OCor e Forma:SolidPeso molecular:556.35(R)-Praziquantel
CAS:(R)-Praziquantel is an active enantiomer of praziquantel.Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:312.41SGS518 oxalate
CAS:<p>SGS518 oxalate is a 5-HT6 antagonist.</p>Fórmula:C23H24F2N2O7SPureza:98%Cor e Forma:SolidPeso molecular:510.51S 12024-2
CAS:<p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>Fórmula:C16H26N2O5SPureza:98%Cor e Forma:SolidPeso molecular:358.45Bepafant
CAS:<p>Bepafant: a PAF antagonist with anti-inflammatory properties; induces apoptosis in PTEN-positive NB4, KG1, NB4-MR4 cells, not in PTEN-negative THP1, U937.</p>Fórmula:C23H22ClN5O2SPureza:98%Cor e Forma:SolidPeso molecular:467.97KSCM-5
CAS:<p>KSCM-5 is a sigma receptor ligand.</p>Fórmula:C24H28N2O2Pureza:98%Cor e Forma:SolidPeso molecular:376.49Pronethalol hydrochloride
CAS:<p>β-adrenergic antagonist</p>Fórmula:C15H20ClNOPureza:98%Cor e Forma:SolidPeso molecular:265.78CI-1015
CAS:<p>CI-1015 is a CCK-B receptor antagonist with oral activity.</p>Fórmula:C29H39N3O4Cor e Forma:SolidPeso molecular:493.64Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Fórmula:C25H25NO6Pureza:99.809%Cor e Forma:SolidPeso molecular:435.48Bavisant dihydrochloride
CAS:<p>Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.</p>Fórmula:C19H29Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:402.36CV-3988
CAS:<p>CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).</p>Fórmula:C28H53N2O7PSCor e Forma:SolidPeso molecular:592.775-Nonyloxytryptamine oxalate
CAS:<p>5-HT1B agonist</p>Fórmula:C21H32N2O5Pureza:98%Cor e Forma:SolidPeso molecular:392.49Naminterol
CAS:<p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>Fórmula:C19H26N2O3Pureza:98%Cor e Forma:SolidPeso molecular:330.42Flutonidine
CAS:<p>Flutonidine is an agonist of alpha2-Adrenergic receptor.</p>Fórmula:C10H12FN3Pureza:98%Cor e Forma:SolidPeso molecular:193.22Dihydroalprenolol, (S)-
CAS:<p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>Fórmula:C15H25NO2Pureza:98%Cor e Forma:SolidPeso molecular:251.36Roxindole hydrochloride
CAS:<p>Dopamine D2 autoreceptor agonist</p>Fórmula:C23H27ClN2OPureza:98%Cor e Forma:SolidPeso molecular:382.93(R)-V-0219
<p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>Fórmula:C20H25F3N4O2Cor e Forma:SolidPeso molecular:410.43ADX-10061
CAS:<p>ADX-10061 is a dopamine D1 receptor antagonist.</p>Fórmula:C19H20N2O4Cor e Forma:SolidPeso molecular:340.37PNU-96415E
CAS:dopamine D4 and serotonergic 5-HT2A receptor antagonistFórmula:C21H27Cl2FN2OPureza:98%Cor e Forma:SolidPeso molecular:413.36MRS 1523
CAS:<p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.</p>Fórmula:C23H29NO3SPureza:98%Cor e Forma:SolidPeso molecular:399.55Gastrazole free acid
CAS:Gastrazole is a CCK2 receptor antagonist potentially. It also used for the treatment of pancreatic cancer.Fórmula:C34H34FN5O7Pureza:98%Cor e Forma:SolidPeso molecular:643.66Mepixanox
CAS:Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.Fórmula:C20H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:323.39Diftalone
CAS:<p>Diftalone is an anti-Inflammatory agent.</p>Fórmula:C16H12N2O2Pureza:98%Cor e Forma:SolidPeso molecular:264.28Jmv 390-1
CAS:Jmv 390-1 is an inhibitor of metallopeptidase.Fórmula:C23H35N3O6Pureza:98%Cor e Forma:SolidPeso molecular:449.54UCM710
CAS:<p>UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).</p>Fórmula:C19H34O3Pureza:98%Cor e Forma:SolidPeso molecular:310.47JNJ-26070109
CAS:<p>JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.</p>Fórmula:C23H17BrF2N4O3SPureza:98%Cor e Forma:SolidPeso molecular:547.37Dacopafant
CAS:<p>Dacopafant is an antagonist of platlet activationg factor receptor.</p>Fórmula:C12H11N3OSCor e Forma:SolidPeso molecular:245.3MK-4256
CAS:MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).Fórmula:C27H23FN8OCor e Forma:SolidPeso molecular:494.52BW-A 575C
CAS:<p>BW-A 575C is an inhibitor of ACE.</p>Fórmula:C29H43N5O8Pureza:98%Cor e Forma:SolidPeso molecular:589.68TCV-309 chloride
CAS:TCV-309 chloride is an antagonist of platelet activating factor (PAF).Fórmula:C30H34BrClN4O4Pureza:98%Cor e Forma:SolidPeso molecular:629.97Aplysamine-1
CAS:Aplysamine-1 is an antagonist of histamine H3 receptor.Fórmula:C15H24Br2N2OPureza:98%Cor e Forma:SolidPeso molecular:408.17L 368935
CAS:<p>L 368935 is an antagonist of the cholecystokinin receptor.</p>Fórmula:C27H26N8O2Pureza:98%Cor e Forma:SolidPeso molecular:494.55ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Fórmula:C12H16N8OPureza:98%Cor e Forma:SolidPeso molecular:288.31Nor-SCH-12679 Maleate
CAS:<p>Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.</p>Fórmula:C22H25NO6Pureza:98%Cor e Forma:SolidPeso molecular:399.44Linadryl hydrochloride
CAS:<p>Linadryl hydrochloride may have antihistamine activity.</p>Fórmula:C19H24ClNO2Cor e Forma:SolidPeso molecular:333.855-Carboxamidotryptamine maleate
CAS:<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Fórmula:C15H17N3O5Pureza:99.88%Cor e Forma:SolidPeso molecular:319.31Resomelagon
CAS:<p>Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.</p>Fórmula:C14H14N6O2Cor e Forma:SolidPeso molecular:298.3Dipiproverine
CAS:<p>Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.</p>Fórmula:C20H30N2O2Cor e Forma:SolidPeso molecular:330.46Ipramidil
CAS:<p>Ipramidil (C80-1324) reveals marked dilator activity in the coronary circulation of isolated working hearts.</p>Fórmula:C10H16N4O4Pureza:98%Cor e Forma:SolidPeso molecular:256.26ONO-2952
CAS:<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Fórmula:C22H20ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.86Mirisetron
CAS:<p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>Fórmula:C24H31N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:393.52Setastine
CAS:<p>Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.</p>Fórmula:C22H28ClNOCor e Forma:SolidPeso molecular:357.92Veliflapon
CAS:<p>Veliflapon is an orally active and selective inhibitor of 5-lipoxygenase activating protein (FLAP).</p>Fórmula:C23H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:361.43L 646462
CAS:<p>L 646462 is an antidopaminergic agent.</p>Fórmula:C27H27N3O4Pureza:98%Cor e Forma:SolidPeso molecular:457.52Umespirone
CAS:Umespirone is a potential antipsychotic/anxiolytic drug of the azapirone class. It possesses anxiolytic and antipsychotic properties.Fórmula:C28H40N4O5Pureza:98%Cor e Forma:SolidPeso molecular:512.64PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Cor e Forma:SolidPeso molecular:315.24Alclofenac lysinate
CAS:<p>Alclofenac is an anti-inflammatory agent used in the treatment of rheumatoid arthritis. It also used as an analgesic and an antipyretic.</p>Fórmula:C17H25ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:372.84Substance P Receptor Antagonist 1
CAS:<p>Substance P Receptor Antagonist 1 may aid in treating GI, inflammatory, respiratory, and CNS disorders.</p>Fórmula:C24H29F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:434.49Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Fórmula:C19H24N2OPureza:98%Cor e Forma:SolidPeso molecular:296.41Falintolol
CAS:<p>Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.</p>Fórmula:C12H24N2O2Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:228.33NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Fórmula:C25H27Cl2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:504.47Org41841
CAS:Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.Fórmula:C19H22N4O2S2Pureza:99.46% - 99.92%Cor e Forma:SolidPeso molecular:402.53L748337
CAS:<p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>Fórmula:C26H31N3O5SPureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:497.61PF2562
CAS:<p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>Fórmula:C19H17N5OPureza:98%Cor e Forma:SolidPeso molecular:331.37Dipiproverine hydrochloride
CAS:<p>Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.</p>Fórmula:C20H32Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:403.39SDZ 21009
CAS:<p>β-adrenoceptor and 5-HT1A/1B receptor antagonist</p>Fórmula:C19H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:348.44Adrenaline sulfate
CAS:<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Fórmula:C9H15NO7SCor e Forma:SolidPeso molecular:281.279Verlukast
CAS:<p>Verlukast (MK-0679) is a selective, orally active leukotriene D4 receptor antagonist for use in bronchial asthma research.</p>Fórmula:C26H27ClN2O3S2Pureza:98%Cor e Forma:SolidPeso molecular:515.09Anatibant
CAS:<p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>Fórmula:C34H36Cl2N6O5SPureza:98%Cor e Forma:SolidPeso molecular:711.66OMDM-6
CAS:<p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>Fórmula:C28H42N2O3Pureza:99.66%Cor e Forma:SolidPeso molecular:454.64Acreozast
CAS:<p>Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.</p>Fórmula:C15H14ClN3O6Cor e Forma:SolidPeso molecular:367.74N-Arachidonyldopamine
CAS:<p>N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1</p>Fórmula:C28H41NO3Pureza:97.65%Cor e Forma:SolidPeso molecular:439.63LY 306669
CAS:LY 306669 is an antagonist of leukotriene B4 receptor.Fórmula:C23H29FN4NaO2Cor e Forma:SolidPeso molecular:435.499Pridefine
CAS:<p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>Fórmula:C19H21NPureza:99.15% - 99.66%Cor e Forma:SolidPeso molecular:263.38OPC-14523 hydrochloride
CAS:<p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>Fórmula:C23H29Cl2N3O2Pureza:99.60%Cor e Forma:SolidPeso molecular:450.4Aligeron
CAS:<p>Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit</p>Fórmula:C20H24N2Pureza:99.09% - >99.99%Cor e Forma:SolidPeso molecular:292.42LY 203647
CAS:<p>LY 203647 is a antagonist of leukotriene D4 and E4 receptor.</p>Fórmula:C21H30N8O3Pureza:98%Cor e Forma:SolidPeso molecular:442.51Epanolol
CAS:<p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>Fórmula:C20H23N3O4Pureza:98%Cor e Forma:SolidPeso molecular:369.41Proglumide sodium
CAS:Non-selective cholecystokinin (CCK) antagonistFórmula:C18H26N2NaO4Pureza:98%Cor e Forma:SolidPeso molecular:357.4Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Fórmula:C31H35F6N4O5PPureza:98%Cor e Forma:SolidPeso molecular:688.6A68930
CAS:<p>A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.</p>Fórmula:C16H17NO3Cor e Forma:SolidPeso molecular:271.31Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Fórmula:C18H20ClNPureza:98%Cor e Forma:SolidPeso molecular:285.81Ro 04-6790 dihydrochloride
CAS:<p>Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.</p>Fórmula:C12H18Cl2N6O2SPureza:98%Cor e Forma:SolidPeso molecular:381.28LY 225910
CAS:<p>LY 225910 is a CCK2 receptor antagonist.</p>Fórmula:C27H24BrN3O2Pureza:98%Cor e Forma:SolidPeso molecular:502.4PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.Fórmula:C19H26F2N2O3Pureza:99.44%Cor e Forma:SoildPeso molecular:368.42VUF-10497
CAS:<p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>Fórmula:C18H20ClN5SPureza:98%Cor e Forma:SolidPeso molecular:373.9PD 144418
CAS:<p>PD 144418 displays potential antipsychotic activity.</p>Fórmula:C18H22N2OPureza:98%Cor e Forma:SolidPeso molecular:282.38Rp-cAMPS sodium
CAS:<p>Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.</p>Fórmula:C10H11N5NaO5PSPureza:99.71%Cor e Forma:SolidPeso molecular:367.25Methiothepin maleate
CAS:<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Fórmula:C24H28N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:472.62Amitifadine hydrochloride
CAS:<p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>Fórmula:C11H12Cl3NPureza:98%Cor e Forma:SolidPeso molecular:264.58LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Fórmula:C27H38ClN3OSPureza:98.06%Cor e Forma:SolidPeso molecular:488.13CAY10535
CAS:<p>CAY10535 is a selective TPβ antagonist (IC50 = 99 nM for TPβ vs 1970 nM for TPα), weakly affects platelets (IC50 = 985 nM).</p>Fórmula:C18H21N3O7SCor e Forma:SolidPeso molecular:423.44F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Fórmula:C25H29ClF2N4O5Pureza:98.86%Cor e Forma:SolidPeso molecular:538.97Reversan
CAS:Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).Fórmula:C26H27N5O2Pureza:99.05%Cor e Forma:SolidPeso molecular:441.53L-826266
CAS:<p>L-826266 is an antagonist of EP(1) receptor.</p>Fórmula:C27H21BrClNO4SCor e Forma:SolidPeso molecular:570.88Nexopamil racemate
CAS:<p>Nexopamil racemate（(Rac)-Nexopamil） is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.</p>Fórmula:C24H40N2O3Pureza:98.61%Cor e Forma:SolidPeso molecular:404.59RTI 336
CAS:<p>RTI 336 is used as a chronic brain dopamine transporter (DAT) inhibitor.</p>Fórmula:C24H26Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:429.38Foscarbidopa
CAS:<p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>Fórmula:C10H15N2O7PPureza:96.17% - 97.27%Cor e Forma:SolidPeso molecular:306.21Imnopitant
CAS:<p>Imnopitant is an antagonist of the NK1 receptor [1].</p>Fórmula:C28H28F6N4OCor e Forma:SolidPeso molecular:550.54Zinterol hydrochloride
CAS:<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Fórmula:C19H27ClN2O4SCor e Forma:SolidPeso molecular:414.95ASP7657
CAS:<p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>Fórmula:C28H26F3N3O3Cor e Forma:SolidPeso molecular:509.52E2508
CAS:<p>E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.</p>Fórmula:C36H47N3O7SPureza:98%Cor e Forma:SolidPeso molecular:665.84CCG-224406
CAS:<p>CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.</p>Fórmula:C29H27FN6O5Cor e Forma:SolidPeso molecular:558.56Calhex 231 hydrochloride
CAS:Calhex 231 hydrochloride a potent CaSR negative-conversion modulator that blocks the increase in [3H]inositol phosphate, inhibits mir-208a-mediated .Fórmula:C25H28Cl2N2OPureza:99.36%Cor e Forma:SolidPeso molecular:443.41S-22153
CAS:<p>S22153 is an antagonist of melatonin receptor.</p>Fórmula:C14H17NOSCor e Forma:SolidPeso molecular:247.36GR 128107
CAS:<p>GR 128107 is an antagonist of melatonin receptor.</p>Fórmula:C16H20N2O2Cor e Forma:SolidPeso molecular:272.34PD-156707
CAS:<p>PD-156707 is a selective antagonist of endothelin A receptor.</p>Fórmula:C28H26NaO9Pureza:98%Cor e Forma:SolidPeso molecular:529.4975-HT7 agonist 1
CAS:<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Fórmula:C19H20ClN3Pureza:98.61%Cor e Forma:SolidPeso molecular:325.84RS 15385-197
CAS:<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Fórmula:C18H26N2O3SCor e Forma:SolidPeso molecular:350.48HAMI 3379
CAS:<p>HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.</p>Fórmula:C34H45NO8Pureza:99.75%Cor e Forma:SolidPeso molecular:595.72U-101958 Maleate
CAS:<p>U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.</p>Fórmula:C25H33N3O5Pureza:98%Cor e Forma:SolidPeso molecular:455.55Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53L 651142
CAS:<p>L 651142 is a weak inhibitor of the platelet-activating factor receptor. It is also binding to polymorphonuclear leukocytes.</p>Fórmula:C21H23NO4SCor e Forma:SolidPeso molecular:385.48SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Fórmula:C19H22BrNO2Pureza:98%Cor e Forma:SolidPeso molecular:376.29Abanoquil
CAS:<p>Abanoquil is an antagonist of alpha-1 adrenoceptor.</p>Fórmula:C22H25N3O4Cor e Forma:SolidPeso molecular:395.45JMV3002
CAS:<p>JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.</p>Fórmula:C35H34N6O3Cor e Forma:SolidPeso molecular:586.68AZ-GHS-22
CAS:<p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>Fórmula:C27H33ClN6O5S2Cor e Forma:SolidPeso molecular:621.17LBP-1
CAS:<p>LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.</p>Fórmula:C23H29ClN6O3Cor e Forma:SolidPeso molecular:472.97CI 1020
CAS:<p>endothelin-A receptor (ETA) antagonist</p>Fórmula:C28H26O9Pureza:98%Cor e Forma:SolidPeso molecular:506.5Alniditan
CAS:<p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>Fórmula:C17H26N4OPureza:98%Cor e Forma:SolidPeso molecular:302.41CCR1 antagonist 7
CAS:<p>CCR1 antagonist 7 (compound 16r) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 4 nM [1].</p>Fórmula:C21H24ClN5O3SPureza:98%Cor e Forma:SolidPeso molecular:461.96Seproxetine HCl
CAS:<p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>Fórmula:C16H17ClF3NOPureza:98%Cor e Forma:SolidPeso molecular:331.76MRS2179
CAS:<p>MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.</p>Fórmula:C11H17N5O9P2Cor e Forma:SolidPeso molecular:425.23Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48ADRA1D receptor antagonist 1 free base
CAS:<p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>Fórmula:C15H13ClN4OCor e Forma:SolidPeso molecular:300.74SB-277011 dihydrochloride
CAS:<p>SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.</p>Fórmula:C28H32Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:511.49Levobunolol hydrochloride
CAS:<p>Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。</p>Fórmula:C17H26ClNO3Pureza:98.49% - >99.99%Cor e Forma:SolidPeso molecular:327.85Agroclavine
CAS:<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Fórmula:C16H18N2Cor e Forma:SolidPeso molecular:238.33
