GPCR/Proteína-G
Os inibidores de GPCR/proteínas G são compostos que têm como alvo os receptores acoplados a proteínas G (GPCRs) e as proteínas G associadas, que desempenham papéis críticos na transmissão de sinais do exterior para o interior das células. Esses inibidores são essenciais para estudar as vias de sinalização mediadas por GPCRs, que estão envolvidas em numerosos processos fisiológicos, incluindo percepção sensorial, resposta imunológica e neurotransmissão. Os inibidores de GPCR também são importantes no desenvolvimento de medicamentos, pois muitos agentes terapêuticos têm como alvo esses receptores. Na CymitQuimica, oferecemos uma ampla gama de inibidores de GPCR/proteínas G de alta qualidade para apoiar sua pesquisa em farmacologia, biologia celular e áreas afins.
Subcategorias de "GPCR/Proteína-G"
- Receptor 5-HT(939 produtos)
- Receptor de adenosina(242 produtos)
- Receptor adrenérgico(2.945 produtos)
- Receptor de Bombesina(30 produtos)
- Receptor de Bradicinina(59 produtos)
- CXCR(148 produtos)
- CaSR(32 produtos)
- Receptor de Canabinóides(195 produtos)
- Receptor de Dopamina(407 produtos)
- Receptor Endotelina(76 produtos)
- Receptor GNRH(73 produtos)
- GPCR19(31 produtos)
- GRK(31 produtos)
- GTPase(21 produtos)
- Receptor Glucagon(165 produtos)
- Hedgehog/Smoothened(44 produtos)
- Receptor de Histamina(358 produtos)
- Receptor LPA(21 produtos)
- Receptor de Melatonina(24 produtos)
- Receptor OX(40 produtos)
- Receptor opioide(297 produtos)
- PAFR(11 produtos)
- PKA(48 produtos)
- Receptor S1P(17 produtos)
- SGLT(30 produtos)
- Receptor Sigma(46 produtos)
Exibir 18 mais subcategorias
Foram encontrados 5352 produtos de "GPCR/Proteína-G"
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IRL-3630
CAS:<p>IRL 3460 is an enantiomer.</p>Fórmula:C31H40N4O6SPureza:98%Cor e Forma:SolidPeso molecular:596.74Lisuride maleate
CAS:<p>Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.</p>Fórmula:C24H30N4O5Pureza:99.85%Cor e Forma:SolidPeso molecular:454.52SB 201146
CAS:<p>SB 201146 is a leukotriene B4 antagonist with high affinity.</p>Fórmula:C30H35LiN2O5SCor e Forma:SolidPeso molecular:542.61Parstatin(mouse)
CAS:<p>Peptide inhibits endothelial migration/proliferation (IC50 ~20μM), induces cell cycle arrest, triggers apoptosis, and has cardioprotective effects.</p>Fórmula:C189H326N58O57S3Pureza:98%Cor e Forma:SolidPeso molecular:4419.19Urocortin, rat
CAS:<p>Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.</p>Fórmula:C206H338N62O64Pureza:98%Cor e Forma:SolidPeso molecular:4707.26Nadolol
CAS:<p>Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.</p>Fórmula:C17H27NO4Pureza:99.87% - 99.92%Cor e Forma:White To Off-White Crystalline Powder SolidPeso molecular:309.40GLP-1 receptor agonist 8
CAS:<p>GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.</p>Fórmula:C34H36ClFN6O4Cor e Forma:SolidPeso molecular:647.14PEN (human)
CAS:<p>PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.</p>Fórmula:C97H159N27O32Pureza:98%Cor e Forma:SolidPeso molecular:2215.49WAY-620645
CAS:<p>WAY-620645 is a CCK antagonist with antitumor and analgesic activities.</p>Fórmula:C22H22N4O2Pureza:99.89%Cor e Forma:SolidPeso molecular:374.44HHS-0701
CAS:<p>HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.</p>Fórmula:C20H20N4O3SPureza:97.24%Cor e Forma:SoildPeso molecular:396.46N,N′-Diferuloylputrescine
CAS:<p>N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.</p>Fórmula:C24H28N2O6Pureza:98%Cor e Forma:SolidPeso molecular:440.49SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Fórmula:C54H71N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1074.258hNTS1R agonist-1
<p>Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (</p>Fórmula:C37H62N10O9Pureza:98%Cor e Forma:SolidPeso molecular:790.95[D-Trp34]-Neuropeptide Y Acetate
<p>[D-Trp34]-Neuropeptide Y Acetate is a potent Y5 receptor agonist that increases rat food intake; less potent at Y1, Y2, Y4, Y6.</p>Fórmula:C198H293N55O58Pureza:99.73%Cor e Forma:SoildPeso molecular:4371.78[D-Trp34]-Neuropeptide Y
CAS:<p>Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.</p>Fórmula:C196H289N55O56Pureza:98%Cor e Forma:SolidPeso molecular:4311.77A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Fórmula:C23H25IN4Cor e Forma:SolidPeso molecular:484.38Galanin-Like Peptide (porcine)
CAS:<p>Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.</p>Fórmula:C281H443N81O78Pureza:98%Cor e Forma:SolidPeso molecular:6204.0215(R)-17-phenyl trinor Prostaglandin F2α
CAS:<p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>Fórmula:C23H32O5Cor e Forma:SolidPeso molecular:388.5AD186
<p>AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.</p>Fórmula:C22H28N2Pureza:98%Cor e Forma:SolidPeso molecular:320.47Arotinolol hydrochloride
CAS:<p>Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.</p>Fórmula:C15H22ClN3O2S3Pureza:99.84%Cor e Forma:SolidPeso molecular:408APJ receptor agonist 1
CAS:<p>Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.</p>Fórmula:C31H26ClN3O3Cor e Forma:SolidPeso molecular:524.02Litoxetine HCl
<p>Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.</p>Fórmula:C16H20ClNOPureza:99.56% - 99.75%Cor e Forma:SoildPeso molecular:277.79α-CGRP(human)
CAS:<p>Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.</p>Fórmula:C163H267N51O49S2Pureza:98%Cor e Forma:SolidPeso molecular:3789.33GLP-1 receptor agonist 9 citrate
<p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>Fórmula:C38H39ClFN3O12Pureza:98.76%Cor e Forma:SolidPeso molecular:784.18SR 142948 dihydrochloride
<p>SR 142948 dihydrochloride is a selective oral non-peptide NT antagonist, IC50 <4 nM, with brain penetration and potential for psychiatric research.</p>Fórmula:C39H53Cl2N5O6Cor e Forma:SolidPeso molecular:758.77MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Fórmula:C60H90N20O11SPureza:98%Cor e Forma:SolidPeso molecular:1299.56α-CGRP, rat
CAS:<p>Endogenous neuropeptide, potent vasodilator</p>Fórmula:C162H262N50O52S2Pureza:98%Cor e Forma:SolidPeso molecular:3806.25Secretin, porcine
CAS:<p>Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.</p>Fórmula:C130H220N44O41·xC2H4O2Pureza:98%Cor e Forma:SolidPeso molecular:N/AMethicillin sodium hydrate
CAS:<p>Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.</p>Fórmula:C17H21N2NaO7SCor e Forma:SolidPeso molecular:420.41AMTG-DA1
<p>AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.</p>Fórmula:C101H149IN22O25Cor e Forma:SolidPeso molecular:2197.0109LY 293284
CAS:<p>LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.</p>Fórmula:C19H26N2OCor e Forma:SolidPeso molecular:298.42Ala5-Galanin (2-11)
CAS:<p>Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].</p>Fórmula:C54H81N13O13Pureza:98%Cor e Forma:SolidPeso molecular:1120.3Sibenadet hydrochloride
CAS:<p>Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.</p>Fórmula:C22H29ClN2O5S2Cor e Forma:SolidPeso molecular:501.06Jatrorrhizine hydroxide
CAS:<p>Jatrorrhizine hydroxide: alkaloid from Coptis chinensis; neuroprotective, antimicrobial, antiplasmodial, antioxidant; AChE inhibitor, affects 5-HT/NE uptake.</p>Fórmula:C20H21NO5Cor e Forma:SolidPeso molecular:355.38Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Fórmula:C23H27N5O3Cor e Forma:SolidPeso molecular:421.501Ontazolast
CAS:<p>Ontazolast: a small-molecule LTB4R antagonist targeting asthma and immune disorders.</p>Fórmula:C21H25N3OPureza:99.79%Cor e Forma:SoildPeso molecular:335.44IRL-1620
CAS:<p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>Fórmula:C86H117N17O27Pureza:98%Cor e Forma:SolidPeso molecular:1820.974SB656104
CAS:<p>SB656104 is a bioactive chemical.</p>Fórmula:C25H30ClN3O3SCor e Forma:SolidPeso molecular:488.04Maridebart
CAS:<p>Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].</p>Cor e Forma:LiquidRhazimine
CAS:<p>Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation.</p>Fórmula:C21H22N2O3Cor e Forma:SolidPeso molecular:350.418NF 340
CAS:<p>P2Y11 antagonist</p>Fórmula:C37H30N4Na4O15S4Pureza:98%Cor e Forma:SolidPeso molecular:990.87Val9-Oxytocin
CAS:<p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>Fórmula:C46H72N12O12S2Pureza:98%Cor e Forma:SolidPeso molecular:1049.27Azepexole hydrochloride
CAS:<p>Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic</p>Fórmula:C9H16ClN3OPureza:99.88% - 99.89%Cor e Forma:SoildPeso molecular:217.715(S)-15-methyl Prostaglandin E2
CAS:<p>15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.</p>Fórmula:C21H34O5Cor e Forma:SolidPeso molecular:366.49Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Fórmula:C14H20ClN3SCor e Forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Fórmula:C18H20ClNO4Cor e Forma:SolidPeso molecular:349.81Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21D3R ligand 1
<p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>Fórmula:C27H37NO5Pureza:98%Cor e Forma:SolidPeso molecular:455.59PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Fórmula:C18H20N5O7S2·NH4·75H2OPureza:98%Cor e Forma:SolidPeso molecular:532.09Pentagastrin meglumine
CAS:<p>Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.</p>Fórmula:C44H66N8O14SCor e Forma:SolidPeso molecular:963.11Uroguanylin (human)
CAS:<p>Uroguanylin (human) serves as a natural ligand for the Guanylyl Cyclase C (GCC) receptor in metastatic colorectal cancer tumors and exhibits anti-tumor effects</p>Fórmula:C64H102N18O26S4Pureza:98%Cor e Forma:SolidPeso molecular:1667.86Phoenixin-14
CAS:<p>Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/</p>Fórmula:C75H110N18O20Pureza:98%Cor e Forma:SolidPeso molecular:1583.78PACAP-Related Peptide (PRP), human
<p>PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.</p>Fórmula:C139H229N41O42Pureza:98%Cor e Forma:SolidPeso molecular:3146.57VVZ-149
<p>VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.</p>Cor e Forma:SolidG-Protein antagonist peptide acetate
<p>G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding.</p>Fórmula:C59H68N12O11SPureza:98.06%Cor e Forma:SolidPeso molecular:1153.33(Leu31,Pro34)-Peptide YY (human) (TFA)
<p>"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a derivative of Peptide YY that acts as a</p>Fórmula:C195H296N54O56·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:4292.75 (free base)Kisspeptin-10, rat
CAS:<p>Kisspeptin-10, rat is an Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).</p>Fórmula:C63H83N17O15Pureza:98%Cor e Forma:SolidPeso molecular:1318.44Satavaptan
CAS:<p>Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.</p>Fórmula:C33H45N3O8SCor e Forma:SolidPeso molecular:643.79Guanylin TFA (mouse,rat)
<p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>Fórmula:C60H90N16O22S4·xC2HF3O2Cor e Forma:SolidPeso molecular:1515.71 (free base)PD 142893
CAS:<p>PD 142893 is a functional endothelin-stimulated vasoconstriction antagonist.</p>Fórmula:C50H65N7O10Pureza:98%Cor e Forma:SolidPeso molecular:924.09Antibacterial agent 189
<p>Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.</p>Fórmula:C37H28N4OPeso molecular:544.22631Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Fórmula:C161H274N48O46SPureza:98%Cor e Forma:SolidPeso molecular:3650.29Antidepressant agent 4
<p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>Fórmula:C19H38ClN5O2SCor e Forma:SolidPeso molecular:436.06[Sar9] Substance P
CAS:<p>[Sar9]-Substance P is one of NK-1 receptor agonist. The action of SP on progesterone metabolism was mimicked by the rNK1-specific agonist [Sar-9,Met(O2)11]-SP.</p>Fórmula:C64H100N18O13SPureza:98%Cor e Forma:SolidPeso molecular:1361.66CB2R agonist 2
<p>CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].</p>Pureza:98%Cor e Forma:Odour SolidMibenratide TFA
<p>Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].</p>Pureza:98%Cor e Forma:Odour SolidTamsolusin Hydrochloride
CAS:<p>Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.</p>Fórmula:C20H29ClN2O5SPureza:99.92%Cor e Forma:SoildPeso molecular:444.97Tiaspirone hydrochloride
CAS:<p>Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.</p>Fórmula:C24H33ClN4O2SPureza:99.87%Cor e Forma:SoildPeso molecular:477.06Surfagon
CAS:<p>Surfagon is an effective LHRH agonist.</p>Fórmula:C56H78N16O12Pureza:98%Cor e Forma:SolidPeso molecular:1167.34Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Fórmula:C22H37NO4Cor e Forma:SolidPeso molecular:379.541GRK2i
CAS:<p>GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.</p>Fórmula:C153H256N50O41SPureza:98%Cor e Forma:SolidPeso molecular:3484.08(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:<p>(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].</p>Fórmula:C52H76N14O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1137.38Zebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Fórmula:C58H84N16O15Cor e Forma:SolidPeso molecular:1245.39VU0453379 hydrochloride
<p>VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.</p>Fórmula:C26H35ClN4O2Cor e Forma:SolidPeso molecular:471.03Neurokinin A(4-10)
CAS:<p>Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .</p>Fórmula:C34H54N8O10SPureza:98%Cor e Forma:SolidPeso molecular:766.91(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Fórmula:C14H22N2O3Pureza:98.72%Cor e Forma:SolidPeso molecular:266.34Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Fórmula:C36H49Cl3N6O6SCor e Forma:SolidPeso molecular:800.23Drinabant
CAS:<p>Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.</p>Fórmula:C23H20Cl2F2N2O2SPureza:99.8%Cor e Forma:SolidPeso molecular:497.38Israpafant
CAS:<p>Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.</p>Fórmula:C28H29ClN4SCor e Forma:SolidPeso molecular:489.0715(S)-HpEPE
CAS:<p>15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.456Sigma-1 receptor antagonist 5
<p>Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors</p>Fórmula:C26H27N3OPureza:98%Cor e Forma:SolidPeso molecular:397.51Alosetron-d3
CAS:<p>Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Fórmula:C17H18N4OPureza:98%Cor e Forma:SolidPeso molecular:297.37ACTH (1-17)
CAS:<p>ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.</p>Fórmula:C95H145N29O23SPureza:98%Cor e Forma:SolidPeso molecular:2093.41Neuropeptide Y (22-36)
CAS:<p>Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.</p>Fórmula:C85H139N29O21Pureza:98%Cor e Forma:SolidPeso molecular:1903.19Sarafotoxin S6c
CAS:<p>Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).</p>Fórmula:C103H147N27O37S5Pureza:98%Cor e Forma:SolidPeso molecular:2516EB1002
CAS:<p>EB1002 is a selective NK2R agonist that has demonstrated significant enhancements in the expression levels of genes associated with mitochondrial biogenesis (such as PGC-1α) in obese mice. This suggests that EB1002 promotes energy expenditure by enhancing mitochondrial activity. Additionally, EB1002 has improved insulin sensitivity and glucose-lipid metabolism in mice. Therefore, EB1002 holds potential for research into obesity and type 2 diabetes.</p>Fórmula:C73H124N12O23Cor e Forma:SolidPeso molecular:1537.83[18F]-Labeled L-dopa precursor
CAS:<p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>Fórmula:C35H36N2O7Cor e Forma:SolidPeso molecular:596.67Eledoisin
CAS:<p>Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family</p>Fórmula:C54H85N13O15SPureza:98%Cor e Forma:SolidPeso molecular:1188.4PEN (rat)
CAS:<p>PEN (rat) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.</p>Fórmula:C102H169N27O33Pureza:98%Cor e Forma:SolidPeso molecular:2301.62Vapreotide
CAS:<p>Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).</p>Fórmula:C57H70N12O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1131.38γ-Glu-Abu TFA
<p>Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.</p>Fórmula:C11H17F3N2O7Cor e Forma:SolidPeso molecular:346.26Antidepressant agent 3
<p>Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.</p>Fórmula:C17H30ClN5O2SCor e Forma:SolidPeso molecular:403.97PACAP (1-27), human, ovine, rat TFA
<p>PACAP (1-27) TFA is a pacap-38 fragment and PACAP receptor antagonist with IC50s: 3nm (rat PAC1), 2nm (rat VPAC1), 5nm (human VPAC2).</p>Fórmula:C144H225F3N40O41SPureza:98%Cor e Forma:SolidPeso molecular:3261.68Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Fórmula:C110H161N31O27S2Pureza:98%Cor e Forma:SolidPeso molecular:2413.78GIP/GLP-1 dual receptor agonist-1
CAS:<p>Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.</p>Cor e Forma:SolidMK-0493 HCl
CAS:<p>MK-0493 is a novel, potent, and selective agonist for melanocortin receptor 4 (MC4R).</p>Fórmula:C30H39Cl2F2N3O2Cor e Forma:SolidPeso molecular:582.55Fenoldopam
CAS:<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Fórmula:C16H16ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:305.76Palmitoyl tetrapeptide-20 TFA
<p>Palmitoyl tetrapeptide-20 (PTP20) TFA is a biomimetic peptide and acts as an agonist of α-MSH. It protects follicular melanocytes by boosting catalase expression and activating melanogenesis.</p>Fórmula:C38H70N6O8·xC2HF3O2ZL-1101
<p>ZL-1101 is a human monoclonal antibody (mAb) targeting TNFRSF4/OX40/CD134.</p>Cor e Forma:Odour LiquidBPP-2
<p>BPP-2 is a GHSR ligand containing the element F. By labeling BPP-2 with the isotope 18F, a PET probe targeting GHSR can be produced. The binding affinity (Ki) of 18F-BPP-2 for GHSR is 274 nM.</p>Fórmula:C27H28FN5O2Peso molecular:473.2227Setmelanotide Acetate(920014-72-8 free base)
CAS:<p>Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM</p>Fórmula:C51H72N18O11S2Pureza:99.71%Cor e Forma:SolidPeso molecular:1177.35Relaxin H3 (human) TFA
<p>Relaxin H3 (human) (TFA) is a relaxin peptide that exerts antifibrotic effects through the RXFP1 receptor.</p>Fórmula:C237H374N70O69S6·xC2HF3O2GLP-1R agonist 20
<p>GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.</p>Fórmula:C31H30Cl2F2N4O5Peso molecular:646.15613palm11-PrRP31
<p>Palm11-PrRP31 is a lipid-modified analog of the endogenous appetite-suppressing neuropeptide (PrRP). It functions as a potent dual agonist for GPR10 (EC50 = 39 pM) and NPFF-R2. By mimicking the natural activity of PrRP, palm11-PrRP31 binds to these receptors to reduce food intake. It has potential applications as an anti-obesity agent and is useful in studying neuropeptide and receptor interactions.</p>Fórmula:C181H289N55O46SPeso molecular:4001.16865Angiopeptin
CAS:<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Fórmula:C54H71N11O10S2Cor e Forma:SolidPeso molecular:1098.34SYD5115
<p>SYD5115 is an orally active TSH-R antagonist.</p>Fórmula:C22H32F2N4O3Peso molecular:438.24425Big Gastrin I (human) TFA
<p>BigGastrinI, human (TFA), is a gastrointestinal hormone comprised of 34 amino acids. It can serve as a potential substance in the study of conditions such as cancer, autoimmune diseases, fibrotic diseases, inflammatory diseases, neurological disorders, or cardiovascular diseases.</p>Fórmula:C178H252F3Peso molecular:2446.96712[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Fórmula:C82H120N20O25Cor e Forma:SolidPeso molecular:1785.95Neuropeptide Y (human) free acid
CAS:<p>Neuropeptide Y (human) free acid is the deamidated form of Neuropeptide Y (human, rat, mouse). The amidation of the C-terminal tyrosine in Neuropeptide Y is essential for its function, while the non-amidated form cannot initiate G-protein signaling.</p>Fórmula:C189H284N54O58SPeso molecular:4270.06542RAG8 peptide
<p>RAG8 peptide is an antagonist of protease-activated receptor 4 (PAR 4), which inhibits late-stage platelet activation and reduces thrombosis without altering hemostasis or increasing bleeding risk. It is applicable in atherosclerosis research.</p>Fórmula:C56H98N16O11Peso molecular:1170.7601Azido-FTY720
CAS:<p>Azido-FTY720 (azido-Fingolimod) is an analogue of FTY720, with an azido group for click chemistry reactions. FTY720 is an orally available S1P1R modulator .</p>Fórmula:C19H32N4O2Cor e Forma:SolidPeso molecular:348.49[Lys4] Sarafotoxin S6c
CAS:<p>[Lys4] Sarafotoxin S6c: potent partial endothelin receptor agonist; causes pig coronary contraction, EC50=1.5 nM.</p>Fórmula:C105H153N27O36S5Cor e Forma:SolidPeso molecular:2529.82Cinanserin hydrochloride
CAS:<p>Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.</p>Fórmula:C20H25ClN2OSPureza:99.57%Cor e Forma:SolidPeso molecular:376.94Spantide I TFA
<p>Spantide I TFA is a selective NK1 antagonist (230 nM); much less for NK2 (8150 nM); it modulates cytokines to prevent corneal perforation.</p>Fórmula:C77H109F3N20O15Cor e Forma:SolidPeso molecular:1611.81OXA(17-33) TFA
<p>OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).</p>Fórmula:C81H126F3N23O24Cor e Forma:SolidPeso molecular:1863[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:<p>Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.</p>Fórmula:C50H75N15O10Pureza:98%Cor e Forma:SolidPeso molecular:1046.23Tirzepatide
CAS:<p>Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.</p>Fórmula:C225H348N48O68Pureza:99.52% - 99.99%Cor e Forma:SolidPeso molecular:4813.45Tezusomant
CAS:<p>Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.</p>Fórmula:C120H171N23O32SCor e Forma:SolidPeso molecular:2479.84PF-03382792
CAS:<p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>Fórmula:C23H32FN3O4Pureza:99.64%Cor e Forma:SolidPeso molecular:433.52(R)-CJ 11974
CAS:<p>(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.</p>Fórmula:C31H38N2OPureza:97.15%Cor e Forma:SoildPeso molecular:454.65δ8-THC acetate
CAS:<p>Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.</p>Fórmula:C23H32O3Cor e Forma:SolidPeso molecular:356.5JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23Azaline
CAS:<p>Azaline is a gonadorelin antagonist.</p>Fórmula:C74H106ClN23O12Pureza:98%Cor e Forma:SolidPeso molecular:1545.26MRS 2365
CAS:<p>Highly potent, selective P2Y1 receptor agonist</p>Fórmula:C13H19N5O9P2SPureza:98%Cor e Forma:SolidPeso molecular:483.33Tirzepatide TFA
<p>Tirzepatide TFA, a GIP and GLP-1 agonist, targets type 2 diabetes treatment.</p>Fórmula:C227H349F3N48O70Cor e Forma:SolidPeso molecular:4927.47Neurokinin A(4-10) TFA
<p>Neurokinin A (4-10) TFA is a tachykinin NK 2 receptor agonist [1] .</p>Fórmula:C36H55F3N8O12SCor e Forma:SolidPeso molecular:880.93SBI-810
CAS:<p>SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.</p>Fórmula:C27H34N4O2Cor e Forma:SolidPeso molecular:446.59Clopidogrel-related Compound B hydrochloride
CAS:<p>Clopidogrel Related Compound B is a useful organic compound for research related to life sciences.</p>Fórmula:C16H17Cl2NO2SCor e Forma:SolidPeso molecular:358.28Sarafotoxin S6a
CAS:<p>Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo.</p>Fórmula:C105H156N28O34S5Pureza:98%Cor e Forma:SolidPeso molecular:2514.85des-Gln14-Ghrelin TFA
<p>Des-Gln14-Ghrelin TFA, a ligand for GHSR, boosts [Ca2+]i with an EC50 of 2.4 nM in CHO-GHSR62 cells.</p>Fórmula:C144H238F3N43O42Cor e Forma:SolidPeso molecular:3300.69L 366811
CAS:<p>L 366811 is a potent oxytocin antagonist.</p>Fórmula:C43H56N8O6Cor e Forma:SolidPeso molecular:780.95Lys-[Hyp3]-Bradykinin
CAS:<p>Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.</p>Fórmula:C56H85N17O13Cor e Forma:SolidPeso molecular:1204.38LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Fórmula:C39H43ClN4O9S2Cor e Forma:SolidPeso molecular:811.36CB2 receptor agonist 9
CAS:<p>CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.</p>Fórmula:C16H23N3O2SCor e Forma:SolidPeso molecular:321.44(Pro34)-Peptide YY (human)
CAS:<p>(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .</p>Fórmula:C194H294N54O56Cor e Forma:SolidPeso molecular:4278.73Ici 216140
CAS:<p>ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.</p>Fórmula:C45H65N13O8Cor e Forma:SolidPeso molecular:916.08d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Fórmula:C52H72F3N13O13S2Cor e Forma:SolidPeso molecular:1208.33Amylin (IAPP), feline TFA
<p>Amylin (IAPP), feline TFA: 37-amino acid peptide; inhibits insulin/glucagon; secreted by pancreatic β-cells.</p>Fórmula:C167H271F3N52O56S2Cor e Forma:SolidPeso molecular:4024.47Endothelin 1 (swine, human), Alexa Fluor 488-labeled
<p>Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.</p>Cor e Forma:SolidPeso molecular:2848.4CCR6 inhibitor 1
CAS:<p>CCR6 inhibitor 1 selectively blocks CCR6 (0.45 nM in monkeys, 6 nM in humans), aiding in vitro/vivo disease studies.</p>Fórmula:C24H23F3N4O3SPureza:99.89%Cor e Forma:SolidPeso molecular:504.52GLP-1(9-36)amide TFA
<p>GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.</p>Fórmula:C142H215F3N36O45Cor e Forma:SolidPeso molecular:3203.43Atrial natriuretic factor (1-28) (rat) TFA
<p>ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.</p>Fórmula:C130H206N45F3O41S2Pureza:98%Cor e Forma:SolidPeso molecular:3176.43RFRP-3(human)
CAS:<p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>Fórmula:C45H72N14O10Pureza:98%Cor e Forma:SolidPeso molecular:969.15(S, R)-LSN 3318839
CAS:<p>(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.</p>Fórmula:C26H23Cl2N3O2Pureza:99.57%Cor e Forma:SoildPeso molecular:480.39Semaglutide TFA
<p>Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patients</p>Fórmula:C189H290F3N45O61Pureza:99.69%Cor e Forma:SolidPeso molecular:4225.6482PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Fórmula:C135H214N34O40SPureza:98%Cor e Forma:SolidPeso molecular:2985.44(±)14(15)-EpETE
CAS:<p>(±)14(15)-EpETE is an intestinal microbial lipid metabolite that attenuates cisplatin chemotherapy-induced nausea in rats by inhibiting Substance P release.</p>Fórmula:C20H30O3Cor e Forma:SolidPeso molecular:318.45CCR6 antagonist 1
CAS:<p>CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.</p>Fórmula:C17H12F3NO2Pureza:99.83%Cor e Forma:SoildPeso molecular:319.28SAG dihydrochloride
CAS:<p>SAG dihydrochloride: potent Smo agonist, activates Hedgehog pathway, counters Cyclopamine. EC50=3 nM, Kd=59 nM.</p>Fórmula:C28H30Cl3N3OSPureza:>99.99%Cor e Forma:SoildPeso molecular:562.98Galantide acetate
<p>Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.</p>Fórmula:C106H155N25O28SPureza:97.8% - 97.91%Cor e Forma:SolidPeso molecular:2259.58GLP-1 moiety from Dulaglutide
<p>GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.</p>Fórmula:C149H221N37O49Pureza:98%Cor e Forma:SolidPeso molecular:3314.62Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Fórmula:C27H22F4N4O3SPureza:98.83%Cor e Forma:SolidPeso molecular:558.55H4R antagonist 3
CAS:<p>H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of</p>Fórmula:C19H21ClN4SPureza:98%Cor e Forma:SolidPeso molecular:372.92Xanthine amine congener trihydrochloride
CAS:<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Fórmula:C21H29ClN6O4Pureza:98.81%Cor e Forma:SolidPeso molecular:464.9512-epi Leukotriene B4
CAS:<p>LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.</p>Fórmula:C20H32O4Cor e Forma:SolidPeso molecular:336.47211β-Prostaglandin E2
CAS:<p>11β-PGE2 is the C-11 epimer of PGE2.</p>Fórmula:C20H32O5Cor e Forma:SolidPeso molecular:352.47Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Fórmula:C49H68N18O9S2Pureza:98%Cor e Forma:SolidPeso molecular:1117.31Cetirizine Impurity D
CAS:<p>Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.</p>Fórmula:C30H28Cl2N2Cor e Forma:SolidPeso molecular:487.46Colulintide
CAS:<p>Colulintide is an analog of amylin, utilized in obesity research.</p>Cor e Forma:SolidPG 106 acetate
<p>PG 106 acetate: Selective hMC3 receptor antagonist, IC50=210 nM; inactive on hMC5 and hMC4, EC50=9900 nM.</p>Fórmula:C53H73N13O11Pureza:98.24%Cor e Forma:SolidPeso molecular:1068.23Adenosine 2',5'-diphosphate sodium
CAS:<p>Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.</p>Fórmula:C10H15N5NaO10P2Cor e Forma:SolidPeso molecular:450.192CCR8 antagonist 1
CAS:<p>CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.</p>Fórmula:C26H29N3O5SPureza:99.51%Cor e Forma:SolidPeso molecular:495.59Glucagon receptor antagonists-1
CAS:<p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>Fórmula:C29H34FNO2Pureza:98%Cor e Forma:SolidPeso molecular:447.58Antibiotic Sch 60057
CAS:<p>Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.</p>Fórmula:C45H84O6Cor e Forma:SolidPeso molecular:721.161CCR2 antagonist 1
CAS:<p>CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).</p>Fórmula:C28H32BrF3N2OCor e Forma:SolidPeso molecular:549.47CUR61414 hydrochloride
<p>CUR61414 hydrochloride: potent cell-permeable Hedgehog pathway inhibitor, IC50=100-200 nM, selectively targets Smo (Ki=44 nM), induces cancer cell apoptosis.</p>Fórmula:C31H43ClN4O5Pureza:94.05%Cor e Forma:SolidPeso molecular:587.15SB 258585
CAS:<p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>Fórmula:C18H22IN3O3SPureza:99.8%Cor e Forma:SoildPeso molecular:487.3617-trifluoromethylphenyl trinor Prostaglandin F2α
CAS:<p>A number of 17-phenyl trinor prostaglandin F2α (17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.</p>Fórmula:C24H31F3O5Cor e Forma:SolidPeso molecular:456.502Pasireotide ditrifluoroacetate
<p>Pasireotide is a stable cyclohexapeptide somatostatin mimic.</p>Fórmula:C62H68F6N10O13Pureza:98%Cor e Forma:SolidPeso molecular:1275.25Melanostatin, frog TFA
<p>Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.</p>Pureza:99.23%Cor e Forma:Odour SolidpCPA methyl ester hydrochloride
CAS:<p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>Fórmula:C10H13Cl2NO2Pureza:99.73% - 99.88%Cor e Forma:SolidPeso molecular:250.12Prostaglandin J2
CAS:<p>PGJ2, a PGD2 metabolite, is a DP agonist (Ki: 0.9 nM hDP, 6.6 nM hCRTH2), induces cAMP (EC50: 1.2 nM), oxidative stress, neuronal apoptosis, and neurotoxicity.</p>Fórmula:C20H30O4Cor e Forma:SolidPeso molecular:334.45Substance P(1-7) TFA
CAS:<p>Substance P(1-7) TFA is a fragment of neuropeptide P (SP), with anti-harmful effects, used in neurological disease research.</p>Fórmula:C43H66F3N13O12Pureza:98.23%Cor e Forma:SolidPeso molecular:1014.06Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Fórmula:C191H330N64O53S3Pureza:98%Cor e Forma:SolidPeso molecular:4467.29PACAP-38 (16-38), human, mouse, rat
CAS:<p>PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine production</p>Fórmula:C123H215N39O28SPureza:98%Cor e Forma:SolidPeso molecular:2720.33Substance P(1-7)
CAS:<p>Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.</p>Fórmula:C41H65N13O10Pureza:98%Cor e Forma:SolidPeso molecular:900.04(Ala13)-Apelin-13 acetate
<p>(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier.</p>Fórmula:C65H111N23O18SPureza:98%Cor e Forma:SolidPeso molecular:1534.79Dexbrompheniramine maleate
CAS:<p>Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.</p>Fórmula:C20H23BrN2O4Cor e Forma:SolidPeso molecular:435.318Cagrilintide acetate
<p>.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.</p>Fórmula:C196H316N54O61S2Pureza:99.88%Cor e Forma:SolidPeso molecular:4469.06Dapoxetine
CAS:<p>Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.</p>Fórmula:C21H23NOPureza:99.73%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:305.42Tebufelone
CAS:<p>Tebufelone is a potent NSAID, inhibits CO, has anti-inflammatory and analgesic properties, and blocks lipoxygenase products (IC50 ~20-22 microM).</p>Fórmula:C20H28O2Pureza:99.32%Cor e Forma:SolidPeso molecular:300.44HAEGTFTSD acetate(926018-45-3 free base)
<p>HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from</p>Fórmula:C42H61N11O19Pureza:98%Cor e Forma:SolidPeso molecular:1024.01CB2 receptor agonist 2
CAS:<p>CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.</p>Fórmula:C30H36N2O4Pureza:99.75%Cor e Forma:SolidPeso molecular:488.62[Des-Arg9]-Bradykinin acetate
CAS:<p>[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.</p>Fórmula:C46H65N11O12Pureza:99.05%Cor e Forma:SolidPeso molecular:964.07Thrombin Receptor Activator for Peptide 5 (TRAP-5)
CAS:<p>Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), used in the research of coronary heart disease (CHD).</p>Fórmula:C30H50N8O7Pureza:98%Cor e Forma:SolidPeso molecular:634.77N-0500 HCl
CAS:<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Fórmula:C15H22ClNO2Pureza:98.85% - 99.54%Cor e Forma:SolidPeso molecular:283.79Hemopressin (human, mouse)
CAS:<p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>Fórmula:C50H79N13O12Pureza:98%Cor e Forma:SolidPeso molecular:1054.26HAEGTFT
CAS:<p>HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C33H47N9O12Pureza:98%Cor e Forma:SolidPeso molecular:761.78Donetidine
CAS:<p>Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.</p>Fórmula:C20H25N5O3SPureza:99.32%Cor e Forma:SolidPeso molecular:415.51Vanicoside E
CAS:<p>Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .</p>Fórmula:C53H52O22Cor e Forma:SolidPeso molecular:1040.97CGRP 8-37 (rat)
CAS:<p>CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.</p>Fórmula:C138H224N42O41Pureza:99.28%Cor e Forma:SolidPeso molecular:3127.51KSK67
CAS:<p>KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki</p>Fórmula:C22H27N3O2Pureza:99.11%Cor e Forma:SoildPeso molecular:365.47S1PR1 modulator 1
CAS:<p>S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.</p>Fórmula:C23H24N2O3SPureza:99.69%Cor e Forma:SolidPeso molecular:408.51Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Cor e Forma:White Crystalline SolidPeso molecular:451.6GLP-1(7-36), amide acetate
CAS:<p>GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.</p>Fórmula:C151H230N40O47Pureza:99.89%Cor e Forma:SolidPeso molecular:3357.68GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Fórmula:C165H254N44O55SPureza:98%Cor e Forma:SolidPeso molecular:3766.19IRL-1620 acetate
<p>IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a Ki of 16 pM which is more selective than ETA with a Ki of 19 μM.</p>Fórmula:C88H121N17O29Pureza:96.64%Cor e Forma:SolidPeso molecular:1881Prostaglandin F2α 1,11-lactone
CAS:<p>Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.</p>Fórmula:C20H32O4Pureza:98%Cor e Forma:SolidPeso molecular:336.47Vedaprofen
CAS:<p>Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.</p>Fórmula:C19H22O2Pureza:99.24% - 99.70%Cor e Forma:SolidPeso molecular:282.38PF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Fórmula:C36H50Cl2N4O7SPureza:98.81%Cor e Forma:SolidPeso molecular:753.78
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