PKC
PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
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Cercosporin
CAS:35082-49-6
Cercosporin, produced by the plant pathogen Cercospora kikuchii and the elsinochromes, is a potent photosensitizer …
Formula:
C29H26O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
534.51
Ref: TM-T13605
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Go6976
CAS:136194-77-9
Go6976 is a PKC inhibitor, widely used in research to probe PKC functions in health …
Formula:
C24H18N4O
Purity:
95.89%
Color and Shape:
Off-White To Yellow Solid
Molecular weight:
378.43
Ref: TM-T6515
| 1mg | 84.00 € | ||
| 5mg | 179.00 € | ||
| 10mg | 265.00 € | ||
| 25mg | 450.00 € | ||
| 50mg | 641.00 € | ||
| 100mg | 887.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
HIV-1 protease-IN-10
HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to …
Formula:
C23H40O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
396.56
Ref: TM-T79493
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Protein kinase inhibitor H-7 dihydrochloride
CAS:108930-17-2
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor.
Formula:
C14H19Cl2N3O2S
Purity:
99.54%
Color and Shape:
White Crystalline Solid
Molecular weight:
364.29
Ref: TM-T22831
| 5mg | 49.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 392.00 € | ||
| 500mg | 888.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(±)-1,2-Diolein
CAS:2442-61-7
(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) (1,2-Dioleoyl-rac-glycerol) is a PKC activator. (±)-1,2-Diolein could increases myotubes Ca 2+ influx.
Formula:
C39H72O5
Color and Shape:
Liquid
Molecular weight:
620.99
Ref: TM-T40101
| 25mg | 94.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 344.00 € | ||
| 500mg | 522.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PKC-θ inhibitor
CAS:736048-65-0
PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.
Formula:
C20H25F3N6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.45
Ref: TM-T5423
| 5mg | 255.00 € | ||
| 10mg | 405.00 € | ||
| 1mL*10mM (DMSO) | 276.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ruboxistaurin hydrochloride
CAS:169939-93-9
Ruboxistaurin HCl (LY 333531) selectively inhibits PKCβI/II with IC50 of 4.7/5.9 nM; much less effective …
Formula:
C28H28N4O3·HCl
Purity:
98.44% - 99.22%
Color and Shape:
Solid
Molecular weight:
505.01
Ref: TM-T3689
| 1mg | 71.00 € | ||
| 2mg | 91.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 723.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,023.00 € | ||
| 1mL*10mM (DMSO) | 201.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hispidin
CAS:555-55-5
Hispidin is a polyphenol originally, including antioxidant, anti-inflammatory, and cytoprotective properties
Formula:
C13H10O5
Purity:
99.55%
Color and Shape:
White Crystalline Powder
Molecular weight:
246.22
Ref: TM-T7792
| 1mg | 86.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 287.00 € | ||
| 25mg | 515.00 € | ||
| 50mg | 721.00 € | ||
| 100mg | 980.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Bisindolylmaleimide I
CAS:133052-90-1
Bisindolylmaleimide I (GF109203X) is a potent and highly selective protein kinase C (PKC) inhibitor with …
Formula:
C25H24N4O2
Purity:
98.19% - 99.08%
Color and Shape:
Orange Solid
Molecular weight:
412.48
Ref: TM-T6513
| 5mg | 66.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 460.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Mitoxantrone
CAS:65271-80-9
Mitoxantrone: anthracenedione antibiotic, disrupts DNA/RNA replication, binds to topoisomerase II, less cardiotoxic than doxorubicin.
Formula:
C22H28N4O6
Purity:
97.97% - 98.74%
Color and Shape:
Blue Powder
Molecular weight:
444.48
Ref: TM-T6588
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 70.00 € | ||
| 200mg | 105.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
PKC-θ inhibitor hcl
CAS:2253640-49-0
PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM).
Formula:
C20H26ClF3N6O3
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
490.91
Ref: TM-T5817
| 1mg | 92.00 € | ||
| 2mg | 119.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 619.00 € | ||
| 50mg | 879.00 € | ||
| 100mg | 1,189.00 € | ||
| 500mg | 2,392.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Aurothiomalate sodium
CAS:12244-57-4
Sodium aurothiomalate (Miochrysin) inhibits PKC-ι, TrxR; used as an anti-rheumatic and has anti-tumor properties.
Formula:
C4H6O4S·Au·xNa
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
390.07
Ref: TM-T20168
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 217.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 523.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
TAS-301
CAS:193620-69-8
TAS-301, an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon …
Formula:
C23H19NO3
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
357.4
Ref: TM-T2441
| 5mg | 50.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 261.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
PKC-iota inhibitor 1
CAS:2328094-11-5
PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 …
Formula:
C21H22N6O
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
374.44
Ref: TM-T8764
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 226.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 602.00 € | ||
| 50mg | 860.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,354.00 € | ||
| 1mL*10mM (DMSO) | 238.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Taurochenodeoxycholic Acid
CAS:516-35-8
Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.
Formula:
C26H45NO6S
Purity:
99.69% - 99.86%
Color and Shape:
Solid
Molecular weight:
499.7
Ref: TM-T2A2481
| 25mg | 46.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 123.00 € | ||
| 500mg | 205.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Valrubicin
CAS:56124-62-0
Valrubicin (AD-32) (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) …
Formula:
C34H36F3NO13
Purity:
97.41%
Color and Shape:
Solid
Molecular weight:
723.64
Ref: TM-T7604
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 499.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Go 6983
CAS:133053-19-7
Go 6983 is a pan-PKC inhibitor targeting PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, exhibiting IC50 …
Formula:
C26H26N4O3
Purity:
98.41% - 99.04%
Color and Shape:
Solid
Molecular weight:
442.51
Ref: TM-T6313
| 1mg | 43.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 379.00 € | ||
| 100mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Darovasertib
CAS:1874276-76-2
Darovasertib (LXS196) is a potent PKC inhibitor, orally active, with IC50 of 1.9 nM (PKCα), …
Formula:
C22H23F3N8O
Purity:
99.67% - ≥95%
Color and Shape:
Solid
Molecular weight:
472.47
Ref: TM-T5600
| 1mg | 52.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 733.00 € | ||
| 500mg | 1,523.00 € | ||
| 1mL*10mM (DMSO) | 154.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Taurochenodeoxycholic acid sodium
CAS:6009-98-9
Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).
Formula:
C26H44NNaO6S
Purity:
98.23% - 99.45%
Color and Shape:
White To Off-White Powder
Molecular weight:
521.68
Ref: TM-TN2215
| 100mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
Fasudil hydrochloride
CAS:105628-07-7
Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki …
Formula:
C14H18ClN3O2S
Purity:
100% - ≥95%
Color and Shape:
White Solid
Molecular weight:
327.83
Ref: TM-T3060
| 50mg | 46.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 79.00 € | ||
| 500mg | 99.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 13 Dec 2024
