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PKC

PKC

PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.

Found 102 products of "PKC"

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  • [Ala107]MBP(104-118)
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    [Ala107]MBP(104-118)

    CAS:
    <p>Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).</p>
    Formula:C67H104N20O19
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1493.68

    Ref: TM-TP1887

  • 1-Oleoyl-2-acetyl-sn-glycerol
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    1-Oleoyl-2-acetyl-sn-glycerol

    CAS:
    <p>1-Oleoyl-2-acetyl-sn-glycerol (1-oleoyl-2-acetyl-glycerol) is a PKC activator that induces superoxide production.</p>
    Formula:C23H42O5
    Color and Shape:Solid
    Molecular weight:398.58

    Ref: TM-T40972

  • PKCiota-IN-2
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    PKCiota-IN-2

    CAS:
    <p>PKCiota-IN-2 selectively inhibits PKC-ι (IC50=2.8nM) and also blocks PKC-α, ε (IC50s=71nM, 350nM).</p>
    Formula:C24H21N5O
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:395.46

    Ref: TM-T9863

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    Aurothiomalate tetramer sodium

    <p>Aurothiomalate tetramer sodium, a tetrameric form of Aurothiomalate sodium, functions as an anti-arthritis gold agent. It also acts as a potent and selective inhibitor of the oncogenic PKCι signaling pathway.</p>
    Color and Shape:Odour Solid

    Ref: TM-T201767

  • Bisindolylmaleimide III
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    Bisindolylmaleimide III

    CAS:
    <p>Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively interacts with PKCα or ribosomal S6</p>
    Formula:C23H20N4O2
    Purity:98.6%
    Color and Shape:Solid
    Molecular weight:384.43

    Ref: TM-T77628

  • Lys-arg-ala-lys-ala-lys-thr-thr-lys-lys-arg
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    Lys-arg-ala-lys-ala-lys-thr-thr-lys-lys-arg

    CAS:
    <p>Lys-arg-ala-lys-ala-lys-thr-thr-lys-lys-arg is a protein kinase C substrate.</p>
    Formula:C56H110N22O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1315.61

    Ref: TM-TP2458

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    LY 379196

    <p>LY 379196, a potent PKC-β inhibitor (IC 50: 50 nM for PKC βI and 30 nM for PKC βII), effectively suppresses the proliferation of bovine retinal microvascular endothelial cells (BREC) induced by VEGF, IGF-1, and bFGF. This compound serves as an antiproliferative agent for proliferative retinopathy.</p>
    Formula:C30H34N4O5S
    Color and Shape:Solid
    Molecular weight:562.68

    Ref: TM-T89929

  • CymitQuimica logo
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    (8R)-8-Hydroxyepoxyboetirane A

    <p>(8R)-8-Hydroxyepoxyboetirane A is a neuroactivating compound that interacts with PKCδ-C1B. This compound binds into the PKC enzyme pocket through hydrogen bonds with glycine-253, leucine-251, and threonine-242. It induces the release of NRG1 and promotes the differentiation of neural stem cells into neurons. (8R)-8-Hydroxyepoxyboetirane A holds potential for research into nervous system disorders.</p>
    Color and Shape:Odour Solid

    Ref: TM-T200548

  • PKCδ Peptide Substrate
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    PKCδ Peptide Substrate

    CAS:
    <p>PKCδ Peptide Substrate is a highly specific substrate for the δ-type of Protein kinase C, composed of a sequence that mirrors murine eEF-1α (422-443) and</p>
    Formula:C109H191N35O29S
    Color and Shape:Solid
    Molecular weight:2487.97

    Ref: TM-T76412

  • Protein kinase C α peptide TFA
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    Protein kinase C α peptide TFA

    CAS:
    <p>Protein Kinase C (alpha) Peptide (TFA) is a PKC-α-associated peptide functioning as a lipid-dependent serine/threonine protein kinase.</p>
    Formula:C68H115F3N24O26S
    Color and Shape:Solid
    Molecular weight:1773.85

    Ref: TM-T76388

  • Protein Kinase C (19-31)
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    Protein Kinase C (19-31)

    CAS:
    <p>Protein Kinase C (19-31), a PKC inhibitor derived from PKCa, has a serine at position 25 and tests PKC activity.</p>
    Formula:C67H118N26O16
    Purity:98%
    Color and Shape:Lyophilized Powder
    Molecular weight:1543.82

    Ref: TM-TP1053

  • [Ala113]MBP(104-118)
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    [Ala113]MBP(104-118)

    CAS:
    <p>Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 28 - 62 mM).</p>
    Formula:C67H104N20O19
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1493.68

    Ref: TM-TP1888

  • Protein Kinase C (19-36)
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    Protein Kinase C (19-36)

    CAS:
    <p>Protein Kinase C (19-36) is a pseudosubstrate peptide inhibitor of protein kinase C (PKC), with an IC50 of 0.18 μM.</p>
    Formula:C93H159N35O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2151.48

    Ref: TM-TP1503

  • PKC β pseudosubstrate
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    PKC β pseudosubstrate

    CAS:
    <p>Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM).</p>
    Formula:C177H294N62O38S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3994.84

    Ref: TM-TP1955

  • K-252b
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    K-252b

    CAS:
    <p>K-252b, an indolocarbazole derived from the actinomycete Nocardiopsis, functions as a protein kinase C (PKC) inhibitor.</p>
    Formula:C26H19N3O5
    Purity:98%
    Color and Shape:Ready-To-Use Solution
    Molecular weight:453.45

    Ref: TM-T15637

  • PKC-θ inhibitor
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    PKC-θ inhibitor

    CAS:
    <p>PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.</p>
    Formula:C20H25F3N6O3
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:454.45

    Ref: TM-T5423

  • (±)-1,2-Diolein
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    (±)-1,2-Diolein

    CAS:
    <p>(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) (1,2-Dioleoyl-rac-glycerol) is a PKC activator. (±)-1,2-Diolein could increases myotubes Ca 2+ influx.</p>
    Formula:C39H72O5
    Color and Shape:Solid
    Molecular weight:620.99

    Ref: TM-T40101

  • Protein kinase inhibitor H-7 dihydrochloride
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    Protein kinase inhibitor H-7 dihydrochloride

    CAS:
    <p>Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor.</p>
    Formula:C14H19Cl2N3O2S
    Purity:99.54%
    Color and Shape:White Crystalline Solid
    Molecular weight:364.29

    Ref: TM-T22831

  • Taurochenodeoxycholic Acid
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    Taurochenodeoxycholic Acid

    CAS:
    <p>Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) is one of the main bioactive substances of animals' bile acid.</p>
    Formula:C26H45NO6S
    Purity:99.53% - 99.86%
    Color and Shape:Solid
    Molecular weight:499.7

    Ref: TM-T2A2481

  • HA-100
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    HA-100

    CAS:
    <p>HA-100 is an inhibitor of protein kinase</p>
    Formula:C13H15N3O2S
    Purity:99.44%
    Color and Shape:Pale Yellow Crystalline Solid
    Molecular weight:277.34

    Ref: TM-T7648