PKC
PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
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Iso-H7 dihydrochloride
CAS:140663-38-3
Iso-H7 dihydrochloride is a less potent inhibitor of phosphokinase C than H-7.
Formula:
C14H19Cl2N3O2S
Purity:
99.64%
Color and Shape:
White Crystalline Solid
Molecular weight:
364.29
Ref: TM-T7501
| 2mg | 39.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 283.00 € | ||
| 200mg | 393.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Verbascoside
CAS:61276-17-3
Verbascoside (Kusaginin) is a protein kinase C inhibitor with antimicrobial, anti-inflammatory activities.
Formula:
C29H36O15
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
624.59
Ref: TM-T3375
| 5mg | 63.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 449.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Phorbol 12-myristate 13-acetate
CAS:16561-29-8
Phorbol 12-myristate 13-acetate (PMA) belongs to the phorbol ester group of natural products and is …
Formula:
C36H56O8
Purity:
100% - 99.5%
Color and Shape:
White To Off-White Solid
Molecular weight:
616.83
Ref: TM-TQ0198
| 1mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 201.00 € | ||
| 50mg | 297.00 € | ||
| 100mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Afuresertib hydrochloride
CAS:1047645-82-8
Afuresertib hydrochloride is an inhibitor of Akt kinase (Kis of 0.08/2/2.6 nM for Akt1/Akt2/Akt3 respectively)
Formula:
C18H18Cl3FN4OS
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
463.8
Ref: TM-T7885
| 2mg | 52.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 429.00 € | ||
| 200mg | 556.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
HA-100
CAS:84468-24-6
HA-100 is an inhibitor of protein kinase
Formula:
C13H15N3O2S
Purity:
99.44%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
277.34
Ref: TM-T7648
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 531.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Midostaurin
CAS:120685-11-2
PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.
Formula:
C35H30N4O4
Purity:
100% - 99.56%
Color and Shape:
Solid
Molecular weight:
570.64
Ref: TM-T3211
| 1mg | 51.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 321.00 € | ||
| 100mg | 477.00 € | ||
| 500mg | 1,072.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Daphnetin
CAS:486-35-1
Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR …
Formula:
C9H6O4
Purity:
98.33% - 99.82%
Color and Shape:
Solid
Molecular weight:
178.14
Ref: TM-T2851
| 10mg | 50.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 239.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Chelerythrine
CAS:34316-15-9
1.
Formula:
C21H18NO4
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
348.37
Ref: TM-T6S0052
| 5mg | 54.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 80.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Sotrastaurin
CAS:425637-18-9
Sotrastaurin (AEB071) is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKCα/βI/δ/ε/η/θ).
Formula:
C25H22N6O2
Purity:
98% - 99.43%
Color and Shape:
Solid
Molecular weight:
438.48
Ref: TM-T6278
| 1mg | 49.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 164.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 545.00 € | ||
| 100mg | 776.00 € | ||
| 500mg | 1,542.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Decursin
CAS:5928-25-6
Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.
Formula:
C19H20O5
Purity:
100% - 97.22%
Color and Shape:
Solid
Molecular weight:
328.36
Ref: TM-T3S1416
| 1mg | 42.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 453.00 € | ||
| 100mg | 649.00 € | ||
| 500mg | 1,328.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ζ-Stat
CAS:3316-02-7
ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, …
Formula:
C10H8O10S3
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
384.36
Ref: TM-T35407
| 1mg | 115.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 439.00 € | ||
| 25mg | 721.00 € | ||
| 50mg | 1,019.00 € | ||
| 100mg | 1,361.00 € | ||
| 500mg | 2,732.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Chelerythrine chloride
CAS:3895-92-9
Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the …
Formula:
C21H18ClNO4
Purity:
95% - 99.19%
Color and Shape:
Yellow To Orange Solid
Molecular weight:
383.83
Ref: TM-T3419
| 5mg | 68.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 537.00 € | ||
| 500mg | 1,175.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
R59949
CAS:120166-69-0
R59949 is used as a Diacylglycerol kinase (DGK) inhibitor.
Formula:
C28H25F2N3OS
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
489.58
Ref: TM-T26019
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 293.00 € | ||
| 50mg | 455.00 € | ||
| 100mg | 685.00 € | ||
| 500mg | 1,421.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Taurolithocholic acid sodium salt
CAS:6042-32-6
Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which …
Formula:
C26H44NNaO5S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
505.69
Ref: TM-T4727
| 5mg | 46.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 203.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Desmethylglycitein
CAS:17817-31-1
Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase …
Formula:
C15H10O5
Purity:
97.93%
Color and Shape:
Solid
Molecular weight:
270.24
Ref: TM-TN1299
| 1mg | 175.00 € | ||
| 5mg | 530.00 € | ||
| 10mg | 703.00 € | ||
| 25mg | 1,082.00 € | ||
| 50mg | 1,459.00 € | ||
| 100mg | 1,960.00 € | ||
| 500mg | 3,942.00 € | ||
| 1mL*10mM (DMSO) | 439.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hypocrellin A
CAS:77029-83-5
Hypocrellin A is a natural PKC inhibitor with light-induced antitumor, antifungal and antiviral activities.Cost-effective and …
Formula:
C30H26O10
Purity:
98% - 99.81%
Color and Shape:
Solid
Molecular weight:
546.52
Ref: TM-T5771
| 1mg | 51.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 371.00 € | ||
| 50mg | 541.00 € | ||
| 100mg | 773.00 € | ||
| 500mg | 1,548.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bisindolylmaleimide V
CAS:113963-68-1
Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.
Formula:
C21H15N3O2
Purity:
90%
Color and Shape:
Red Solid
Molecular weight:
341.36
Ref: TM-T7790
| 1mg | 73.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 491.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Staurosporine
CAS:62996-74-1
Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) …
Formula:
C28H26N4O3
Purity:
99.24% - 99.87%
Color and Shape:
Off-White Powder
Molecular weight:
466.53
Ref: TM-T6680
| 1mg | 60.00 € | ||
| 2mg | 85.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 582.00 € | ||
| 500mg | 1,251.00 € | ||
| 1mL*10mM (DMSO) | 107.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
1,2-Dimyristoyl-sn-glycerol
CAS:60562-16-5
1,2-Dimyristoyl-sn-glycerol (1,2-DMG) is able to increase AChE activity by 35-40% at concentrations of 25 micrograms/ml …
Formula:
C31H60O5
Purity:
99.49%
Color and Shape:
White Powder With Lumps
Molecular weight:
512.81
Ref: TM-T22464
| 50mg | 54.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Decursinol angelate
CAS:130848-06-5
Decursinol angelate is anti-tumor, anti-inflammatory, anti-oxidant, hepatoprotective, and inhibits VEGF and cancer cell invasion.
Formula:
C19H20O5
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
328.36
Ref: TM-TN1557
| 5mg | 50.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
